Page last updated: 2024-08-24

carfentanil and naloxone

carfentanil has been researched along with naloxone in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19905 (16.67)18.7374
1990's7 (23.33)18.2507
2000's5 (16.67)29.6817
2010's10 (33.33)24.3611
2020's3 (10.00)2.80

Authors

AuthorsStudies
Galzi, JL; Goeldner, M; Hirth, C; Ilien, B; Mejean, A; Meunier, JC; Mollereau, C1
Costa, EM; Hoffmann, BB; Loew, GH1
Kreeger, TJ; Seal, US1
Crozier, WC; Dannals, RF; Douglass, KH; Frost, JJ; Links, JM; Mayberg, HS; Ravert, HT; Wagner, HN; Wilson, AA1
Bullock, A; Dannals, RF; Frost, JF; Kuhar, MJ; Leonhardt, S; Lyon, RA; Price, DL; Rydelek, LT; Struble, RG; Titeler, M1
Frost, JJ; Smith, AC; Wagner, HN1
Bice, AN; Dannals, RF; Frost, JJ; Lee, MC; Links, JM; Natarajan, TK; Ravert, HT; Wagner, HN; Wilson, AA; Wong, DF1
Baker, JR; Gatesman, TJ1
Gates, CC; Haigh, JC1
Carpenter, JW; Leith, DE; Shaw, ML1
Dannals, RF; Frost, JJ; Lever, JR; Natarajan, TK; Ravert, HT; Tanada, S; Villemagne, VL; Wagner, HN; Wilson, AA1
Civelek, AC; Dannals, RF; Dixon, RB; Joh, T; Kao, PF; Kim, S; Ravert, HT; Villemagne, VL; Wagner, HN1
Ananthanarayanan, VS; Zhorov, BS1
Frost, JJ1
Dannals, RF; Frost, JJ; Ravert, HT; Villemagne, PS1
Gaynor, JS; Larsen, RS; Moresco, A; Sleeman, JM; Wild, MA1
Stanley, T1
Kuwabara, H; McCaul, ME; Wand, GS; Weerts, EM; Wong, DF; Xu, X1
Krenzelok, EP1
Cole, JB; Nelson, LS1
Batdorf, S; Bixler, D; Ellison, D; Gladden, RM; Gupta, R; Haddy, L; Halpin, J; Kilkenny, M; Massey, J; Sanders, SK1
Bozat-Emre, S; Marshall, SG; Reimer, J; Zhong, C1
Juurlink, DN; Leen, JLS1
Agrawal, A; Alho, H; Crystal, R; Ekblad, L; Helin, S; Hirvonen, J; Johansson, J; Kaasinen, V; Lovró, Z; Pennanen, M; Rajasilta, O; Scheinin, M; Sirén, S; Tuisku, J; Vainio, PJ1
Gill, H; Henderson, G; Kelly, E1
McCranor, BJ; Pierce, SA; Racine, MC; Sciuto, AM; Tressler, J; Tuet, WY; Wong, B1
Bardsley, R1
Arteaga, J; Carlo, DJ; Henderson, BD; Koeppe, RA; Moss, RB; Rodnick, ME; Scott, PJH; Shao, X; Sherman, PS; Sowa, AR; Stauff, J1
Adamowicz, P; Kosmal, W; Kuczyńska, K; Markiewicz, K; Zawilska, JB1
Chen, Y; Di, B; Lai, M; Li, F; Li, X; Qiu, Y; Shen, H; Wei, J; Xu, P1

Reviews

3 review(s) available for carfentanil and naloxone

ArticleYear
PET imaging of the opioid receptor: the early years.
    Nuclear medicine and biology, 2001, Volume: 28, Issue:5

    Topics: Animals; Diprenorphine; Fentanyl; Humans; Naloxone; Receptors, Opioid; Tomography, Emission-Computed

2001
Carfentanil: a narrative review of its pharmacology and public health concerns.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 2019, Volume: 66, Issue:4

    Topics: Analgesics, Opioid; Animals; Fentanyl; Humans; Illicit Drugs; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Public Health; Veterinary Drugs

2019
Carfentanil - from an animal anesthetic to a deadly illicit drug.
    Forensic science international, 2021, Volume: 320

    Topics: Analgesics, Opioid; Chromatography, Liquid; Drug Contamination; Drug Overdose; Fentanyl; Forensic Toxicology; Humans; Mass Spectrometry; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Respiratory Insufficiency

2021

Trials

3 trial(s) available for carfentanil and naloxone

ArticleYear
Longer occupancy of opioid receptors by nalmefene compared to naloxone as measured in vivo by a dual-detector system.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1997, Volume: 38, Issue:11

    Topics: Adult; Analgesics, Opioid; Brain; Carbon Radioisotopes; Cross-Over Studies; Female; Fentanyl; Humans; Male; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Time Factors; Tomography, Emission-Computed

1997
PET imaging of human cardiac opioid receptors.
    European journal of nuclear medicine and molecular imaging, 2002, Volume: 29, Issue:10

    Topics: Aged; Carbon Radioisotopes; Feasibility Studies; Female; Fentanyl; Heart; Humans; Indoles; Lung; Male; Middle Aged; Morphinans; Muscle, Skeletal; Myocardium; Naloxone; Radiopharmaceuticals; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Reproducibility of Results; Sensitivity and Specificity; Tissue Distribution; Tomography, Emission-Computed

2002
Intranasal naloxone rapidly occupies brain mu-opioid receptors in human subjects.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:9

    Topics: Administration, Intranasal; Adult; Analgesics, Opioid; Brain; Double-Blind Method; Fentanyl; Healthy Volunteers; Humans; Male; Naloxone; Narcotic Antagonists; Positron-Emission Tomography; Receptors, Opioid, mu; Young Adult

2019

Other Studies

24 other study(ies) available for carfentanil and naloxone

ArticleYear
Photoactivatable opiate derivatives as irreversible probes of the mu-opioid receptor.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Affinity Labels; Animals; Azides; Azo Compounds; Binding Sites; Brain; Chemical Phenomena; Chemistry; Guinea Pigs; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, mu; Structure-Activity Relationship

1990
Opioid agonists binding and responses in SH-SY5Y cells.
    Life sciences, 1992, Volume: 50, Issue:1

    Topics: Alprostadil; Analgesics; Cyclic AMP; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; GTP Phosphohydrolases; Humans; Meperidine; Morphinans; Naloxone; Narcotics; Oxymorphone; Receptors, Opioid; Receptors, Opioid, mu; Tumor Cells, Cultured

1992
Immobilization of gray wolves (Canis lupus) with sufentanil citrate.
    Journal of wildlife diseases, 1990, Volume: 26, Issue:4

    Topics: Anesthetics; Animals; Arousal; Carnivora; Etorphine; Female; Fentanyl; Immobilization; Male; Naloxone; Sufentanil; Xylazine; Yohimbine

1990
Multicompartmental analysis of [11C]-carfentanil binding to opiate receptors in humans measured by positron emission tomography.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1989, Volume: 9, Issue:3

    Topics: Adult; Brain; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Fentanyl; Frontal Lobe; Humans; Kinetics; Male; Naloxone; Occipital Lobe; Receptors, Opioid; Thalamus; Tomography, Emission-Computed

1989
Mu opiate receptors are selectively labelled by [3H]carfentanil in human and rat brain.
    European journal of pharmacology, 1989, Aug-22, Volume: 167, Issue:2

    Topics: Animals; Binding, Competitive; Brain Chemistry; Cerebral Cortex; Diencephalon; Fentanyl; Haloperidol; Humans; In Vitro Techniques; Kinetics; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu

1989
3H-diprenorphine is selective for mu opiate receptors in vivo.
    Life sciences, 1986, Apr-28, Volume: 38, Issue:17

    Topics: Animals; Binding, Competitive; Corpus Striatum; Diprenorphine; Fentanyl; Kinetics; Male; Mice; Mice, Inbred ICR; Morphinans; Naloxone; Receptors, Opioid; Receptors, Opioid, mu; Thalamus; Tritium

1986
Simplified detection system for neuroreceptor studies in the human brain.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1986, Volume: 27, Issue:2

    Topics: Binding, Competitive; Brain; Calibration; Carbon Radioisotopes; Electrons; Equipment Design; Fentanyl; Humans; Naloxone; Radioligand Assay; Receptors, Opioid; Scintillation Counting

1986
Use of carfentanil and a ketamine-xylazine mixture to immobilise wild grey seals (Halichoerus grypus).
    The Veterinary record, 1985, Feb-23, Volume: 116, Issue:8

    Topics: Animals; Caniformia; Drug Combinations; Female; Fentanyl; Immobilization; Ketamine; Male; Naloxone; Seals, Earless; Thiazines; Xylazine

1985
Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures.
    Journal of wildlife diseases, 1995, Volume: 31, Issue:1

    Topics: Analgesics, Opioid; Animals; Bison; Diprenorphine; Drug Combinations; Female; Fentanyl; Hypnotics and Sedatives; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Naloxone; Naltrexone; Narcotic Antagonists; Northwest Territories; Piperidines; Tranquilizing Agents; Xylazine

1995
Complications with the use of carfentanil citrate and xylazine hydrochloride to immobilize domestic horses.
    Journal of the American Veterinary Medical Association, 1995, Mar-15, Volume: 206, Issue:6

    Topics: Analgesics, Opioid; Animals; Animals, Domestic; Fentanyl; Horse Diseases; Horses; Hypertension; Immobilization; Naloxone; Naltrexone; Pulmonary Edema; Tachycardia; Xylazine

1995
Comparison of [11C]diprenorphine and [11C]carfentanil in vivo binding to opiate receptors in man using a dual detector system.
    European journal of pharmacology, 1994, May-12, Volume: 257, Issue:1-2

    Topics: Analgesics, Opioid; Binding Sites; Diprenorphine; Dose-Response Relationship, Drug; Fentanyl; Gamma Rays; Humans; Naloxone; Receptors, Opioid; Receptors, Opioid, mu

1994
Homology models of mu-opioid receptor with organic and inorganic cations at conserved aspartates in the second and third transmembrane domains.
    Archives of biochemistry and biophysics, 2000, Mar-01, Volume: 375, Issue:1

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Aspartic Acid; Benzomorphans; Binding Sites; Cations; Cattle; Computer Simulation; Conserved Sequence; Fentanyl; Humans; Ligands; Metals; Models, Molecular; Molecular Sequence Data; Morphine; Naloxone; Narcotic Antagonists; Protein Binding; Protein Structure, Tertiary; Rats; Receptors, Opioid, mu; Sequence Alignment; Sequence Homology, Amino Acid; Structure-Activity Relationship

2000
Use of naloxone to reverse carfentanil citrate-induced hypoxemia and cardiopulmonary depression in Rocky Mountain wapiti (Cervus elaphus nelsoni).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2001, Volume: 32, Issue:1

    Topics: Adrenergic alpha-Agonists; Analgesics, Opioid; Animals; Blood Gas Analysis; Cross-Over Studies; Deer; Electrocardiography; Female; Fentanyl; Heart Rate; Hypoxia; Naloxone; Narcotic Antagonists; Oximetry; Oxygen; Partial Pressure; Respiration; Xylazine

2001
Human immobilization: is the experience in Moscow just the beginning?
    European journal of anaesthesiology, 2003, Volume: 20, Issue:6

    Topics: Adult; Aerosols; Analgesics, Opioid; Fentanyl; Humans; Immobilization; Moscow; Naloxone; Narcotic Antagonists; Terrorism

2003
The relationship between naloxone-induced cortisol and mu opioid receptor availability in mesolimbic structures is disrupted in alcohol dependent subjects.
    Alcohol (Fayetteville, N.Y.), 2012, Volume: 46, Issue:6

    Topics: Adult; Alcoholism; Carbon Radioisotopes; Female; Fentanyl; Humans; Hydrocortisone; Hypothalamo-Hypophyseal System; Male; Middle Aged; Naloxone; Narcotic Antagonists; Pituitary-Adrenal System; Positron-Emission Tomography; Receptors, Opioid, mu

2012
Abuse of fentanyl derivatives: History repeating itself.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2017, 04-15, Volume: 74, Issue:8

    Topics: Analgesics, Opioid; Counterfeit Drugs; Fentanyl; History, 20th Century; History, 21st Century; Humans; Illicit Drugs; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; United States

2017
Controversies and carfentanil: We have much to learn about the present state of opioid poisoning.
    The American journal of emergency medicine, 2017, Volume: 35, Issue:11

    Topics: Analgesics, Opioid; Drug Overdose; Fentanyl; Health Knowledge, Attitudes, Practice; Hospital Rapid Response Team; Humans; Law Enforcement; Naloxone; Narcotic Antagonists; North America; Opioid-Related Disorders; Pharmacovigilance; Police; Prescription Drug Misuse

2017
Opioid Overdose Outbreak - West Virginia, August 2016.
    MMWR. Morbidity and mortality weekly report, 2017, Sep-22, Volume: 66, Issue:37

    Topics: Adolescent; Adult; Analgesics, Opioid; Designer Drugs; Disease Outbreaks; Drug Overdose; Emergency Medical Services; Female; Fentanyl; Humans; Male; Middle Aged; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; West Virginia; Young Adult

2017
At-a-glance - Lessons learned from launching the Manitoba Take-Home Naloxone Program.
    Health promotion and chronic disease prevention in Canada : research, policy and practice, 2018, Volume: 38, Issue:6

    Topics: Adolescent; Adult; Analgesics, Opioid; Child; Drug Overdose; Female; Fentanyl; Humans; Male; Manitoba; Naloxone; Narcotic Antagonists; Program Evaluation; Recurrence; Sex Factors; Young Adult

2018
How the complex pharmacology of the fentanyls contributes to their lethality.
    Addiction (Abingdon, England), 2019, Volume: 114, Issue:9

    Topics: Drug Overdose; Fentanyl; Humans; Muscle Rigidity; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid, mu; Respiratory Insufficiency; Respiratory Muscles

2019
Changes in murine respiratory dynamics induced by aerosolized carfentanil inhalation: Efficacy of naloxone and naltrexone.
    Toxicology letters, 2019, Volume: 316

    Topics: Administration, Inhalation; Aerosols; Analgesics, Opioid; Animals; Computer Simulation; Dose-Response Relationship, Drug; Fentanyl; Humans; Lung; Male; Mice; Models, Biological; Naloxone; Naltrexone; Narcotic Antagonists; Plethysmography, Whole Body; Respiration; Respiratory Insufficiency; Risk Assessment

2019
Higher naloxone dosing may be required for opioid overdose.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2019, Oct-30, Volume: 76, Issue:22

    Topics: Adult; Analgesics, Opioid; Cardiopulmonary Resuscitation; Cyanosis; Drug Overdose; Female; Fentanyl; Hospitals, Community; Humans; Male; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Schizophrenia; Substance-Related Disorders

2019
The Effects of Intramuscular Naloxone Dose on Mu Receptor Displacement of Carfentanil in Rhesus Monkeys.
    Molecules (Basel, Switzerland), 2020, Mar-17, Volume: 25, Issue:6

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Female; Fentanyl; Injections, Intramuscular; Macaca mulatta; Naloxone; Positron-Emission Tomography; Receptors, Opioid, mu

2020
Assessment of abuse potential of carfentanil.
    Addiction biology, 2023, Volume: 28, Issue:2

    Topics: Analgesics, Opioid; Animals; Fentanyl; Heroin; Mice; Naloxone; Rats; Substance Withdrawal Syndrome

2023