Page last updated: 2024-09-02

carboxyamido-triazole and bms 214662

carboxyamido-triazole has been researched along with bms 214662 in 1 studies

Compound Research Comparison

Studies
(carboxyamido-triazole)
Trials
(carboxyamido-triazole)
Recent Studies (post-2010)
(carboxyamido-triazole)
Studies
(bms 214662)
Trials
(bms 214662)
Recent Studies (post-2010) (bms 214662)
10515224989

Protein Interaction Comparison

ProteinTaxonomycarboxyamido-triazole (IC50)bms 214662 (IC50)
GTPase HRasHomo sapiens (human)0.0013
GTPase KRasHomo sapiens (human)0.7723
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaHomo sapiens (human)0.3617
Protein farnesyltransferase subunit betaHomo sapiens (human)0.0021
Geranylgeranyl transferase type-1 subunit betaHomo sapiens (human)1.8

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Frett, B; Kaiser, CE; Li, HY; Wang, Y1

Reviews

1 review(s) available for carboxyamido-triazole and bms 214662

ArticleYear
Targeting mutant KRAS for anticancer therapeutics: a review of novel small molecule modulators.
    Journal of medicinal chemistry, 2013, Jul-11, Volume: 56, Issue:13

    Topics: Cell Cycle Proteins; Humans; Models, Biological; Molecular Structure; Molecular Targeted Therapy; Mutation; Polo-Like Kinase 1; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; ras Proteins; Signal Transduction; Small Molecule Libraries

2013