carbetapentane and dextromethorphan

carbetapentane has been researched along with dextromethorphan in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19902 (15.38)18.7374
1990's5 (38.46)18.2507
2000's4 (30.77)29.6817
2010's1 (7.69)24.3611
2020's1 (7.69)2.80

Authors

AuthorsStudies
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Chen, EC; Chien, HC; Giacomini, KM; Huang, Y; Khuri, N; Liang, X; Sali, A; Stecula, A; Yee, SW1
Agard, DA; Ashworth, A; Barrio-Hernandez, I; Batra, J; Beltrao, P; Bennett, MJ; Bohn, M; Bouhaddou, M; Braberg, H; Broadhurst, DJ; Cai, Y; Cakir, M; Calviello, L; Cavero, DA; Chang, JCJ; Chorba, JS; Craik, CS; d'Enfert, C; Dai, SA; Eckhardt, M; Emerman, M; Fabius, JM; Fletcher, SJ; Floor, SN; Foussard, H; Frankel, AD; Fraser, JS; Fujimori, DG; Ganesan, SJ; García-Sastre, A; Gordon, DE; Gross, JD; Guo, JZ; Haas, K; Haas, P; Hernandez-Armenta, C; Hiatt, J; Huang, XP; Hubert, M; Hüttenhain, R; Ideker, T; Jacobson, M; Jang, GM; Jura, N; Kaake, RM; Kim, M; Kirby, IT; Klippsten, S; Koh, C; Kortemme, T; Krogan, NJ; Kuzuoglu-Ozturk, D; Li, Q; Liboy-Lugo, J; Lin, Y; Liu, X; Liu, Y; Lou, K; Lyu, J; Mac Kain, A; Malik, HS; Mathy, CJP; McGregor, MJ; Melnyk, JE; Memon, D; Meyer, B; Miorin, L; Modak, M; Moreno, E; Mukherjee, S; Naing, ZZC; Noack, J; O'Meara, MJ; O'Neal, MC; Obernier, K; Ott, M; Peng, S; Perica, T; Pilla, KB; Polacco, BJ; Rakesh, R; Rathore, U; Rezelj, VV; Richards, AL; Roesch, F; Rosenberg, OS; Rosenthal, SB; Roth, BL; Roth, TL; Ruggero, D; Safari, M; Sali, A; Saltzberg, DJ; Savar, NS; Schwartz, O; Sharp, PP; Shen, W; Shengjuler, D; Shi, Y; Shoichet, BK; Shokat, KM; Soucheray, M; Stroud, RM; Subramanian, A; Swaney, DL; Taunton, J; Tran, QD; Trenker, R; Tummino, TA; Tutuncuoglu, B; Ugur, FS; Vallet, T; Venkataramanan, S; Verba, KA; Verdin, E; Vignuzzi, M; von Zastrow, M; Wang, HY; Wankowicz, SA; Wenzell, NA; White, KM; Xu, J; Young, JM; Zhang, Z; Zhou, Y1
Annels, SJ; Davies, JA; Ellis, Y1
Apland, JP; Braitman, DJ1
Braitman, DJ; Brennecke, LH; Sparenborg, S1
Klein, M; Musacchio, JM; Santiago, LJ1
Musacchio, JM; Tortella, FC1
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC1
Baragatti, G; Dematteis, M; Gavend, M; Mallaret, M1
Anderson, TR; Andrew, RD1
Cuevas, J; Hall, AA; Herrera, Y; Katnik, C; Pennypacker, KR; Rodriguez, JD; Willing, A1
Ahrens, N; Deisemann, H; Kirchhoff, C; Möller, C; Netzer, R; Schlobohm, I1

Reviews

2 review(s) available for carbetapentane and dextromethorphan

ArticleYear
Allosteric modulation of dextromethorphan binding sites.
    Neuropharmacology, 1987, Volume: 26, Issue:7B

    Topics: Animals; Anticonvulsants; Binding Sites; Cyclopentanes; Dextromethorphan; Levorphanol; Noscapine; Phenytoin; Receptors, Neurotransmitter

1987
Discriminative stimulus properties of dextromethorphan in rats.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 1995, Volume: 49, Issue:10

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Antitussive Agents; Cyclazocine; Cyclopentanes; Dextromethorphan; Dextrorphan; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Male; Morphine; Neuroprotective Agents; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, sigma

1995

Other Studies

11 other study(ies) available for carbetapentane and dextromethorphan

ArticleYear
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Discovery of Competitive and Noncompetitive Ligands of the Organic Cation Transporter 1 (OCT1; SLC22A1).
    Journal of medicinal chemistry, 2017, 04-13, Volume: 60, Issue:7

    Topics: Drug Discovery; HEK293 Cells; Humans; Ligands; Molecular Docking Simulation; Organic Cation Transporter 1; Small Molecule Libraries

2017
A SARS-CoV-2 protein interaction map reveals targets for drug repurposing.
    Nature, 2020, Volume: 583, Issue:7816

    Topics: Animals; Antiviral Agents; Betacoronavirus; Chlorocebus aethiops; Cloning, Molecular; Coronavirus Infections; COVID-19; COVID-19 Drug Treatment; Drug Evaluation, Preclinical; Drug Repositioning; HEK293 Cells; Host-Pathogen Interactions; Humans; Immunity, Innate; Mass Spectrometry; Molecular Targeted Therapy; Pandemics; Pneumonia, Viral; Protein Binding; Protein Biosynthesis; Protein Domains; Protein Interaction Mapping; Protein Interaction Maps; Receptors, sigma; SARS-CoV-2; SKP Cullin F-Box Protein Ligases; Vero Cells; Viral Proteins

2020
Non-opioid antitussives inhibit endogenous glutamate release from rabbit hippocampal slices.
    Brain research, 1991, Nov-15, Volume: 564, Issue:2

    Topics: Animals; Antitussive Agents; Aspartic Acid; Cyclopentanes; Depression, Chemical; Dextromethorphan; Female; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Glycine; Hippocampus; In Vitro Techniques; Male; Potassium; Rabbits

1991
Effects of non-opioid antitussives on epileptiform activity and NMDA responses in hippocampal and olfactory cortex slices.
    Brain research, 1990, Oct-08, Volume: 529, Issue:1-2

    Topics: Animals; Antitussive Agents; Cyclopentanes; Dextromethorphan; Electric Stimulation; Epilepsy; Evoked Potentials; Guinea Pigs; Hippocampus; In Vitro Techniques; Magnesium; N-Methylaspartate; Olfactory Bulb

1990
Prevention of soman neurotoxicity by non-opioid antitussives.
    Neurotoxicology, 1990,Fall, Volume: 11, Issue:3

    Topics: Animals; Anticonvulsants; Antitussive Agents; Cyclopentanes; Dextromethorphan; Guinea Pigs; Male; Necrosis; Nervous System Diseases; Neurons; Soman

1990
Dextromethorphan and carbetapentane: centrally acting non-opioid antitussive agents with novel anticonvulsant properties.
    Brain research, 1986, Sep-24, Volume: 383, Issue:1-2

    Topics: Animals; Anticonvulsants; Antitussive Agents; Cyclopentanes; Dextromethorphan; Drug Synergism; Electroshock; Levorphanol; Male; Phenytoin; Rats; Rats, Inbred Strains; Seizures

1986
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Spreading depression: imaging and blockade in the rat neocortical brain slice.
    Journal of neurophysiology, 2002, Volume: 88, Issue:5

    Topics: Algorithms; Animals; Cortical Spreading Depression; Cyclopentanes; Dextromethorphan; Diagnostic Imaging; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Extracellular Space; Image Processing, Computer-Assisted; In Vitro Techniques; Loperamide; Magnetic Resonance Imaging; Male; Membrane Potentials; Neocortex; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Spiperone

2002
sigma-1 receptor modulation of acid-sensing ion channel a (ASIC1a) and ASIC1a-induced Ca2+ influx in rat cortical neurons.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acid Sensing Ion Channels; Animals; Calcium; Calcium Channels; Cerebral Cortex; Cyclopentanes; Dextromethorphan; Guanidines; Nerve Tissue Proteins; Peptides; Piperazines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Sodium Channels; Spider Venoms; Tetrodotoxin

2008
Effects of common antitussive drugs on the hERG potassium channel current.
    Journal of cardiovascular pharmacology, 2008, Volume: 52, Issue:6

    Topics: Amino Alcohols; Animals; Antitussive Agents; CHO Cells; Codeine; Cricetinae; Cricetulus; Cyclopentanes; Dextromethorphan; Dose-Response Relationship, Drug; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Membrane Potentials; Potassium; Potassium Channel Blockers; Theobromine; Time Factors; Torsades de Pointes; Transfection

2008