carbamates has been researched along with thiazoles in 234 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 44 (18.80) | 18.7374 |
| 1990's | 17 (7.26) | 18.2507 |
| 2000's | 68 (29.06) | 29.6817 |
| 2010's | 99 (42.31) | 24.3611 |
| 2020's | 6 (2.56) | 2.80 |
| Authors | Studies |
|---|---|
| Thompson, PE; Voigtman, RE | 1 |
| Daniels, PJ; Loebenberg, D; Nafissi, MM; Panitz, E; Waitz, JA | 1 |
| Panitz, E | 1 |
| Alonso, MT; Berenguer, FJ; Elguero, J; Marin, A; Mercedes Martinez, M; Ramon Martinez, A; Valls, N | 1 |
| Lalezari, I; Schwartz, EL | 1 |
| Anderson, WK; Mach, RH | 1 |
| Georgieva, V; Kappas, A; Tziolas, V; Tzoneva, M; Vachkova, R | 1 |
| Cantino, EC; Matsumae, A | 1 |
| Ross, JB | 1 |
| Benz, GW | 2 |
| Dean, RE; Knapp, SE; Presidente, PJ | 1 |
| Reinecke, RK | 1 |
| Kamaly, M; Lalezari, L; Mirchamsy, H; Niloufari, G; Rezvani, N | 1 |
| Berry, WK; Davies, DR; Gordon, JJ | 1 |
| Jannasch, R | 1 |
| Nagase, H | 1 |
| Kistner, TP; Lindsey, JB | 1 |
| Colglazier, ML; Enzie, FD; Kates, KC; Lindahl, IL; Samuelson, G | 1 |
| Horak, IG; Pienaar, I; Snijders, AJ | 1 |
| Colglazier, ML; Enzie, FD; Kates, KC | 3 |
| Hass, DK | 1 |
| Amborski, GF; Bello, TR; Greer, GJ; Torbert, BJ | 1 |
| Prichard, RK | 1 |
| Allen, RW | 1 |
| Farmer, PS; Leung, CC; Lui, EM | 1 |
| Butler, RW; Campbell, WC | 1 |
| Cooper, AJ; Meister, A | 1 |
| Grace, OD; Mitchell, RJ; Sullivan, TW | 1 |
| Blair, LS; Campbell, WC | 1 |
| Gibson, TE; Parfitt, JW | 1 |
| Lämmler, G; Srivastava, VK; Zahner, H | 1 |
| Lalezari, I; Vahdat, A | 1 |
| Aminzhanov, M; Ostrovskiĭ, AN | 1 |
| Pierpoint, WS | 1 |
| Kagan, FE | 1 |
| Klayman, DL; Milne, GW; Senning, A | 1 |
| Vergieva, T | 1 |
| Drudge, JH; Lyons, ET; Tolliver, SC | 2 |
| Antov, G; Ivanova-Chemishanska, L; Khinkova, L; Khristeva, V; Vergieva, T | 1 |
| Anderson, B; Erickson, JW; Gulnik, SV; Liu, B; Mitsuya, H; Suvorov, LI; Yu, B | 1 |
| Blum, MR; Millard, J; Painter, G; Parry, N; Rooney, J; Sadler, BM; St Clair, MH; Tisdale, M | 1 |
| Bialer, M; Johannessen, SI; Kupferberg, HJ; Levy, RH; Loiseau, P; Perucca, E | 1 |
| Service, RF | 1 |
| Chakravarty, S; Danishefsky, SJ; He, L; Horwitz, SB; Inoue, T; Kuduk, SD; Lin, S; Ojima, I | 1 |
| DeFronzo, RA | 1 |
| Feinglos, MN; Hughes, AT; Luna, B | 1 |
| Pregnolato, M; Zampollo, F; Zani, F | 1 |
| Fukami, T; Fukuroda, T; Hata, M; Ihara, M; Ishihara, A; Kanatani, A; Kanno, T; Mase, T; Sakuraba, A; Tanaka, T; Tsuchiya, Y | 1 |
| Smits, P; Tack, CJ | 1 |
| Brillon, D; Brown, DL | 1 |
| Mozersky, RP | 1 |
| Larmore, SS | 1 |
| Bailey, CJ; Nattrass, M | 1 |
| Arimoto, H; Danishefsky, SJ; Horwitz, SB; Kaufman, MD; Martello, LA; McDaid, HM; Meng, D; Pettus, TR; Regl, DL; Smith, AB; Yang, CP | 1 |
| Berger, S; Jovanovic, L; Raskin, P; Ratner, R; Schwartz, S; Woo, V | 1 |
| Füchtenbusch, M; Schatz, H; Standl, E | 1 |
| Blanchard, SG; Furfine, ES; Ittoop, O; Jain, RG; Lenhard, JM; Orband-Miller, LA; Paulik, MA; Weiel, JE | 1 |
| Fisher, A | 1 |
| Carlton, FB | 1 |
| Blackburn, G | 1 |
| Moses, R | 2 |
| Arai-Otsuki, S; Fukami, T; Haga, Y; Hirose, M; Ihara, M; Ishihara, A; Iwaasa, H; Iwama, T; Kanatani, A; Kannoa, T; Keen, SL; Morishima, H; Sakuraba, A | 1 |
| Chang, HE | 1 |
| Laws, A | 1 |
| Boccuzzi, SJ; Fox, J; Kim, J; Shah, AB; Sung, JC; Wogen, J | 1 |
| Adler, AJ; Crabtree, DV; Geng, X; Ojima, I | 1 |
| Calvo Romero, JM; Lima Rodríguez, EM | 1 |
| Pospísilová, Y | 1 |
| Inzucchi, SE | 1 |
| Cizmárik, J; Gyürösiová, L; Hirvonen, J; Laitinen, L; Raiman, J; Sedlárová, E | 1 |
| Kuritzky, L; Quillen, DM | 1 |
| Büche, C; Kassemeyer, HH; Nick, P; Riemann, M | 1 |
| Koivisto, V | 1 |
| Göke, B; Parhofer, KG | 1 |
| Nurse, P; Pardo, M | 1 |
| Bell, CF; Botteman, MF; Braunstein, SN; Devine, ST; Ramsdell, JW; Stephens, JM | 1 |
| Hayashi, Y; Ito, T; Kimura, T; Kiso, Y; Matsumoto, H; Sohma, Y | 1 |
| MANLY, RS; PILLARD, R | 1 |
| Bilello, JA; Drusano, GL; Piliero, PJ; Preston, SL; Stein, DS; Symonds, WT | 1 |
| Anderson, PC; Bailey, M; Beaulieu, P; Bolger, G; Bonneau, P; Bös, M; Cameron, DR; Cartier, M; Cordingley, MG; Faucher, AM; Goudreau, N; Kawai, SH; Kukolj, G; Lagacé, L; Lamarre, D; LaPlante, SR; Llinàs-Brunet, M; Narjes, H; Poupart, MA; Rancourt, J; Sentjens, RE; Simoneau, B; St George, R; Steinmann, G; Thibeault, D; Tsantrizos, YS; Weldon, SM; Yong, CL | 1 |
| Rice, CM | 1 |
| Foster, GD; Khan, SU; Singh, SB | 1 |
| Brennan, DL; Cottrell, KM; Fulghum, JR; Gates, CA; Hsiao, HM; Kwong, AD; Lin, C; Lin, K; Luong, YP; Ma, S; Maxwell, JP; Perni, RB; Rao, BG; Wei, YY | 1 |
| Chankvetadze, B | 1 |
| Wei, L | 1 |
| Britt, SD; Court, JJ; Courtney, LF; Deininger, DD; Farmer, LJ; Gates, CA; Harbeson, SL; Levin, RB; Lin, C; Lin, K; Luong, YP; Moon, YC; O'Malley, ET; Perni, RB; Pitlik, J; Rao, BG; Thomson, JA; Tung, RD; Van Drie, JH; Wei, Y | 1 |
| Bouillaguet, S; Galgano, C; Golay, A; Krejci, I; Lockwood, PE; Wataha, JC | 1 |
| He, W; Huang, PP; Klein, LL; Lu, L; Mo, H; Molla, A; Pilot-Matias, TJ; Pithawalla, R; Randolph, JT; Stewart, KD | 1 |
| Sasseville, D | 1 |
| Bousquet, C; Gingras, R; Lagacé, L; Lamarre, D; Maurice, R; Thibeault, D; White, PW | 1 |
| Bailey, MD; Beaulieu, PL; Brochu, C; Duceppe, JS; Faucher, AM; Ferland, JM; Ghiro, E; Gorys, V; Halmos, T; Kawai, SH; Llinàs-Brunet, M; Poirier, M; Simoneau, B; Tsantrizos, YS | 1 |
| Tsantrizos, YS | 1 |
| Benhamou, Y; Calleja, JL; Chaves, RL; Crönlein, J; Erhardt, A; Forns, X; Hinrichsen, H; Nehmiz, G; Reiser, M; Sentjens, RE; Steinmann, GG; Wedemeyer, H; Yong, CL | 1 |
| Pawlotsky, JM | 1 |
| Lemon, SM; Li, K; Yi, M | 1 |
| Avendano, C; Benhamou, Y; Hinrichsen, H; Nehmiz, G; Reesink, HW; Reiser, M; Riba, N; Steinmann, GG; Wedemeyer, H; Yong, CL | 1 |
| Harino, H; Mori, Y; Senda, T; Shibata, K; Yamaguchi, Y | 1 |
| Girish, C | 1 |
| Anastasiades, I; Georgiadou, A; Giannakou, IO; Karpouzas, DG; Tsiropoulos, NG | 1 |
| Fujimoto, M; Hata, S; Itoh, N; Kuroda, T; Okamura, N; Sakaeda, T; Sakaguchi, G; Ueda, K; Yagami, T | 1 |
| Brennan, DL; Frantz, JD; Fulghum, JR; Gates, CA; Kwong, AD; Lin, C; Lin, K; Luong, YP; Ma, S; Perni, RB; Rao, BG; Wei, YY | 1 |
| Chang, CF; Hsu, JT; Lee, JC; Lien, TW; Yu, MC | 1 |
| Cheng, G; Chisari, FV; Zhong, J | 1 |
| Aukerman, L; Collett, M; Douglas, D; Gao, T; Hashash, A; Hsi, B; Kline, J; Kneteman, NM; Kovelsky, R; Mercer, DF; Ni, ZJ; O'Connell, J; Schiller, D; Tyrrell, DL; Weiner, AJ; Zhu, Q | 1 |
| Benhamou, Y; Calleja, JL; Forns, X; Herrmann, E; Hinrichsen, H; Manns, MP; Nehmiz, G; Reesink, H; Reiser, M; Sarrazin, C; Steinmann, GG; Zeuzem, S | 1 |
| Farina, V; Haddad, N; Tan, J | 1 |
| Härter, G; Kern, P; Manfras, B; Merkle, M; Reuter, S | 1 |
| Dekhtyar, T; Han, L; Koev, G; Lin, CT; Mo, H; Molla, A; Ng, TI; Yan, P | 1 |
| Brenner, M; Donsbach, K; Farina, V; Feng, X; Frutos, RP; Fuchs, V; Gallou, F; Haddad, N; Houpis, IN; Johnson, M; Kreye, P; Nicola, T; Ridges, MD; Samstag, W; Simpson, RD; Smith-Keenan, LL; Spinelli, EM; Tan, J; Vitous, J; Wang, XJ; Wei, X; Winter, E; Xu, J; Xu, Y; Yee, NK; Zhang, L | 1 |
| Aukerman, SL; Garrett, EN; Hollenbach, PW; Mendel, DB; Oei, Y; Patawaran, MB; Weiner, AJ; Zhu, Q | 1 |
| Amrani, N; Bouzidi, M; Cacoub, P; Courcambeck, J; Halfon, P; Jouirou, B; Pèpe, G; Perbost, R; Sabatier, JM | 1 |
| Arslanyolu, M; Chevallet, P; Fehrentz, JA; Kaplancikli, ZA; Martinez, J; Ozdemir, A; Turan-Zitouni, G; Yildiz, MT | 1 |
| De Vos, R; Leroux-Roels, G; Libbrecht, L; Meuleman, P; Roskams, T; Vanwolleghem, T | 1 |
| Bes, M; Cubero, M; Esteban, JI; Esteban, R; Guardia, J; Otero, T; Quer, J; Sauleda, S | 1 |
| Busacca, CA; Farina, V; Han, Z; Hao, MH; Senanayake, CH; Shu, C; Wei, X; Yee, NK; Zeng, X | 1 |
| Glenn, JS; Lin, MZ; Tsien, RY | 1 |
| Gonzàlez-Candelas, F; López-Labrador, FX; Moya, A | 1 |
| Delouvroy, F; Hu, L; Kock, Hd; Lenz, O; Lin, TI; McGowan, D; Nilsson, M; Raboisson, P; Rosenquist, S; Samuelsson, B; Simmen, K; Surleraux, D; Tahri, A; Vendeville, S; Vreken, WV; Wigerinck, P | 1 |
| Bush, KJ; Carroll, SS; DiMuzio, J; Liverton, NJ; Lyle, TA; McCauley, JA; McIntyre, CJ; Nguyen, KT; Olsen, DB; Romano, JJ; Ross, CW; Rudd, MT; Stahlhut, MW; Vacca, JP; Varga, SL | 1 |
| Allen, TM; Berical, A; Berlin, AM; Bihl, F; Birch, C; Birren, BW; Carlson, J; Cerny, A; Chung, RT; Daar, ES; Donfield, SM; Edlin, BR; Fleckenstein, JF; Galagan, JE; Gomperts, ED; Heckerman, D; Henn, MR; Jacobson, IM; Kim, AY; Kleyman, M; Kodira, C; Koehrsen, M; Kuntzen, T; Lake-Bakaar, GV; Lauer, GM; Ledlie, T; Lee, B; Lennon, N; Liu, Z; Madey, MA; Marion, T; McMahon, CM; Nusbaum, C; Park, VM; Reyor, LL; Roberts, AD; Rosen, HR; Schneidewind, A; Schulze Zur Wiesch, J; Spengler, U; Talal, AH; Timm, J; Walker, BD; Xing, Y; Young, SK | 1 |
| Ciaramella, G; Corbau, R; Flores, MV; Strawbridge, J | 1 |
| Dessole, G; Di Francesco, ME; Di Muzio, J; Fiore, F; Koch, U; Monteagudo, E; Nizi, E; Pace, P; Pesci, S; Rowley, M; Summa, V | 1 |
| Aya, T; Cai, J; Chen, AP; Cheng, Y; Cheng, YC; Dutschman, GE; Grill, SP; Gullen, EA; Hamilton, AD; Lindenbach, BD; Tsou, LK | 1 |
| Marquis, M; Massariol, MJ; Thibeault, D; White, PW; Zhao, S | 1 |
| German, P; Hui, J; Jain, A; Kearney, BP; Mathias, AA; Murray, BP; Warren, D; Wei, L; West, S | 1 |
| Deshpande, M; Huang, M; Miller, MD; Mo, H; Murray, B; Qi, X; Rhodes, G; Sun, SC; Wang, K; Wang, Y; Yang, C | 1 |
| Kim, AY; Kluge, SF; Roggendorf, M; Salloum, S; Timm, J | 1 |
| Bester, K; Lamani, X | 1 |
| Vollmar, AM; von Schwarzenberg, K | 1 |
| Gaylarde, CC; John, VM; Loh, K; Shirakawa, MA; Taqueda, ME; Tavares, RG | 1 |
| Chuck, SL; Cohen, C; DeJesus, E; Elion, R; Kearney, BP; Liu, HC; Ramanathan, S; Rashbaum, B; Ruane, P; Shamblaw, D; Warren, DR; Yale, K | 1 |
| Huang, Q; Knight, BL; Pack, FD; Seidler, RW; Stern, JO; Stoltz, JH | 1 |
| Binder, J; Diehl, W; Lingardo, L; Love, R; Maegley, K; Patick, AK; Smith, GJ; Tetangco, S; Weinshank, M | 1 |
| Delang, L; Froeyen, M; Neyts, J; Vliegen, I | 1 |
| Chuck, SL; Cohen, C; Elion, R; Gathe, J; Hawkins, T; Kearney, BP; Liu, HC; Mathias, AA; Shalit, P; Warren, DR | 1 |
| Lampiris, HW | 1 |
| Brussee, J; Heitman, LH; Ijzerman, AP; Kleinau, G; Krause, G | 1 |
| Marchand, C | 1 |
| Andrews, J; German, P; Hepner, M; Kearney, BP; Liu, HC; Mathias, A; Szwarcberg, J | 1 |
| Cheng, AK; DeJesus, E; Gathe, J; Henry, K; Kearney, BP; Molina, JM; Ramanathan, S; Rockstroh, JK; Szwarcberg, J; Wei, X; White, K; Yale, K | 1 |
| Cheng, AK; Cohen, C; DeJesus, E; Gallant, JE; Kearney, BP; Liu, HC; Mills, A; Quirk, E; Sax, PE; Szwarcberg, J; White, K; Wohl, D; Yale, K; Zhong, L; Zolopa, A | 1 |
| Busacca, CA; Campbell, SJ; Gonnella, NC; Jones, PJ; Saha, AK; Senanayake, CH | 1 |
| Debyser, Z; Schrijvers, R | 2 |
| Lepist, EI; Maclennan, K; Murray, B; Phan, TK; Ray, AS; Roy, A; Tong, L | 1 |
| Pommer, P | 1 |
| Maxmen, A | 1 |
| Haberl, A; von Hentig, N | 1 |
| Klibanov, OM; Olin, JL; Spooner, LM | 1 |
| Hussar, DA; Martinez, LN | 1 |
| Breeze, S | 1 |
| Morrow, T | 1 |
| Temesgen, Z | 2 |
| Belavic, JM | 1 |
| Abram, M; Cheng, AK; DeJesus, E; Fordyce, MW; Gathe, J; Henry, K; Molina, JM; Plummer, A; Ramanathan, S; Rockstroh, JK; Szwarcberg, J; Wei, X | 1 |
| Cheng, AK; Cohen, C; DeJesus, E; Gallant, JE; Liu, HC; Mills, A; Plummer, A; Rhee, MS; Sax, PE; Szwarcberg, J; White, KL; Wohl, D; Zolopa, A | 1 |
| Brůčková, L; Imramovský, A; Jampílek, J; Královec, K; Mandíková, J; Pejchal, V; Šimůnek, P; Štěpánková, Š; Trejtnar, F; Vančo, J; Vorčáková, K | 1 |
| Priano, J; Schafer, JJ; Shah, BM; Squires, KE | 1 |
| Cahn, P; Sued, O | 1 |
| Andrade-Villanueva, J; Antunes, F; Arastéh, K; Callebaut, C; Cheng, AK; Chetchotisakd, P; DeJesus, E; Fehr, J; Gallant, JE; Koenig, E; Liu, Y; Moyle, G; Rhee, MS; Rizzardini, G; Szwarcberg, J; Zhong, L | 1 |
| Bruce, RD; Custodio, JM; Friedland, GH; Kearney, BP; Ramanathan, S; Rhee, MS; Wei, LX; Winkle, P | 1 |
| Matsumura, M; Ohtsu, R; Otuka, A; Sakumoto, S; Sanada-Morimura, S; Satoh, M; Takeuchi, H | 1 |
| Beran, RK; Bush, CO; Delaney, WE; Greenstein, AE | 1 |
| Banu, SH; Chandana, KV; Channe Gowda, D; Sharma, A; Suhas, R | 1 |
| Brodbeck, RM; Chandrasena, G; Grenon, M; Hopper, AT; Packiarajan, M; Pu, X; Robichaud, AJ; White, AD; Zorn, S | 1 |
| Cheng, A; Kearney, BP; Koziara, J; Mathias, A; Ramanathan, S; Shen, G; Wei, X | 1 |
| Bam, RA; Birkus, G; Cihlar, T; Hao, J; Lepist, EI; Ray, AS; Stray, KM; Yant, SR | 1 |
| Aldir, I; Horta, A; Serrado, M | 1 |
| Bruce, RD; Custodio, JM; Friedland, GH; Kearney, BP; Ramanathan, S; Rhee, MS; Wei, X; Winkle, P | 1 |
| Perry, CM | 1 |
| Deeks, ED | 1 |
| Dieterich, DT; Martel-Laferrière, V | 1 |
| Asselah, T; Halfon, P; Marcellin, P; Schinazi, R | 1 |
| Andrews, J; Cheng, A; Custodio, JM; Hao, J; Kearney, BP; Lepist, EI; Ling, KH; Ramanathan, S; Ray, AS; Wang, H | 1 |
| Ford, N; Fortunak, J; Hill, A; Khoo, S; Simmons, B | 1 |
| Callebaut, C; Chau, J; Choi, YC; Desai, MC; Hong, A; Lee, MS; Liu, H; Murray, BP; Rhodes, GR; Stray, KM; Strickley, RG; Swaminathan, S; Tong, L; Tsai, LK; Vivian, R; Wang, J; Xu, L | 1 |
| Anwar, MI; Danielson, UH; Ehrenberg, AE; Gustafsson, SS; Schmuck, B; Stenberg, G | 1 |
| Ikeda, A; Irie, S; Ishikawa, T; Kimura, M; Matsuki, S; Nishino, N; Shiomi, M | 1 |
| Akberdin, IR; Clausznitzer, D; Demenkov, PS; Gursky, VV; Ivanisenko, NV; Ivanisenko, VA; Kaderali, L; Kolchanov, NA; Kozlov, KN; Likhoshvai, VA; Mishchenko, EL; Samsonov, AM; Samsonova, MG; Todorov, DI | 1 |
| Hillewaert, V; Hoetelmans, RM; Iterbeke, K; Kakuda, TN; Opsomer, M; Petrovic, R; Timmers, M; Van De Casteele, T | 1 |
| Bannister, R; Birkus, G; Cihlar, T; Hao, J; Huang, J; Huang, Y; Kosaka, A; Lepist, EI; Murray, BP; Ray, AS; Zhang, X | 1 |
| Hsiao, CB; Ma, Q; Sawyer, JR | 1 |
| Ayala-Sims, VA; Fulco, PP | 1 |
| Capetti, A; Rizzardini, G | 1 |
| Antela, A; Domingo, P; Garner, W; Girard, PM; Guyer, B; Henry, K; Markowitz, M; Mills, A; Nguyen, T; Piontkowsky, D; Pozniak, A; Stellbrink, HJ; White, K | 1 |
| Arribas, JR; Di Perri, G; Ebrahimi, R; Gathe, J; Nguyen, T; Pialoux, G; Piontkowsky, D; Reynes, J; Tebas, P; White, K | 1 |
| Hoetelmans, RM; Kakuda, TN; Neujens, M; Opsomer, M; Petrovic, R; Salih, H; Van De Casteele, T | 1 |
| Bruzzone, B; Di Biagio, A; Gustinetti, G; Prinapori, R; Sticchi, L; Taramasso, L; Viscoli, C | 1 |
| Acosta, EP; Delille, C; Larson, KB; Otofokun, I; Wang, K | 1 |
| Hodges, MR; Ottosen, S; Parsley, TB; Patick, AK; Raney, AK; van der Veer, E; van Doorn, LJ; Yang, L; Zeh, K | 1 |
| Abram, ME; Andrade-Villanueva, JF; Beraud, C; Cheng, AK; Fisher, M; Graham, H; Liu, Y; Post, FA; Rhee, MS; Szwarcberg, J; Winston, J | 1 |
| Deuker, MM; Marsh Durban, V; McMahon, M; Phillips, WA | 1 |
| Fisher, M; Raffe, S | 1 |
| Aplin, AE; Cheng, H | 1 |
| Khoo, S; Lewis, J; Nsutebu, EN; Turtle, L | 1 |
| Harirforoosh, S; Moorman, JP; Murrell, DE | 1 |
| Sun, L; Wei, P; Zhou, F; Zhou, Y; Zou, Q | 1 |
| Baša Česnik, H; Bavčar, D; Leskovšek, R; Simončič, A; Stopar, M; Velikonja Bolta, Š | 1 |
| Baeten, JM; Wyatt, C | 1 |
| Andrade-Villanueva, J; Callebaut, C; Cao, H; Cheng, AK; Crofoot, G; Custodio, JM; DeJesus, E; Fordyce, MW; Koenig, E; Martin, H; McCallister, S; Molina, JM; Oka, S; Plummer, A; Podzamczer, D; Post, F; Pozniak, A; Saag, M; Sax, PE; Thompson, M; Trottier, B; Wohl, D; Yin, MT; Zhong, L | 1 |
| Stone, L | 1 |
| da Rocha, MP; de Oliveira, KM; de Souza Rodrigues, M; Dourado, PL; Grisolia, AB; Raposo, JL | 1 |
| Abram, ME; Andrade-Villanueva, JF; Antunes, F; Arastéh, K; Cao, H; Chetchotisakd, P; DeJesus, E; Fehr, J; Gallant, JE; Koenig, E; Liu, HC; Rizzardini, G; Szwarcberg, J | 1 |
| Fujinaga, M; Hatori, A; Ishii, H; Kumata, K; Kurihara, Y; Nengaki, N; Shimoda, Y; Xie, L; Yamasaki, T; Yui, J; Zhang, MR; Zhang, Y | 1 |
| Li, J; Liao, X; Mao, K; Wan, H; Zhang, K; Zhang, X | 1 |
| Bauer, A; Deza, G; Giménez-Arnau, AM; Johnston, GA; Mahler, V; Sanchez-Perez, J; Schuttelaar, ML; Silvestre, JF; Uter, W; Wilkinson, M | 1 |
| Beasley, G; Rossfeld, K; Salama, AK; Turner, MC; Tyler, D | 1 |
| Avsar, E; Bendell, JC; Chatterjee, A; Delord, JP; Demuth, T; Elez, E; Eskens, FALM; Faris, JE; Jaeger, S; Lenz, HJ; Lolkema, MP; Maharry, K; Schellens, JHM; Schuler, M; Sharma, S; Spreafico, A; Tabernero, J; Tan, E; van Geel, RMJM; Wainberg, ZA; Yaeger, R; Yamada, Y; Yoshino, T | 1 |
| Chen, C; Guo, D; Peng, Q; Qian, Y; Wang, Q; Wang, Y; Yang, G; Zhao, H | 1 |
| Lee, JM; Park, JH; Yang, CM; Yoon, JC | 1 |
| Almasio, PL; Barr, E; Bruno, S; Buti, M; Butterton, JR; Dutko, FJ; Fernsler, D; Gao, W; Grandhi, A; Hassanein, TI; Huang, HC; Jancoriene, L; Lawitz, E; Li, JJ; Liu, H; Muellhaupt, B; Nguyen, BT; Pearlman, B; Plank, RM; Robertson, MN; Ruane, PJ; Shepherd, A; Su, FH; Tannenbaum, B; Vierling, JM; Wahl, J; Wan, S; Yeh, WW; Yoshida, EM | 1 |
| Agarwal, K; Barr, E; Ben-Ari, Z; Butterton, JR; Chen, HL; Dutko, FJ; Esteban, R; Fernsler, D; Fitzgerald, B; Foster, GR; Gane, EJ; Gao, W; Gerstoft, J; Grandhi, A; Huang, HC; Laursen, AL; Li, JJ; Liu, H; Nguyen, BT; Pianko, S; Plank, RM; Roberts, SK; Robertson, MN; Su, FH; Thompson, AJ; Wahl, J; Wan, S; Yeh, WW; Zeng, Z; Zeuzem, S; Zuckerman, E | 1 |
| Cai, L; Chen, C; He, Y; Wang, W; Wang, X; Wang, Y; Yang, G; Yu, Y; Zhao, H | 1 |
| Agrawal, S; Asante-Appiah, E; Black, S; Bystol, K; Carr, D; Chase, R; Curry, S; Ferrari, E; Ingravallo, P; Kozlowski, J; Lahser, F; Liu, R; McMonagle, P; Rokosz, L; Tong, L; Yu, W | 1 |
| Ali, E; Jin, R; Li, J; Liao, X; Mao, K; Ren, Z; Wan, H; Zhang, X | 1 |
| Ito, HC; Nakagawa, M; Shiraishi, H; Takamura, N | 1 |
| Anbar, HS; El-Gamal, MI; Jeon, HR; Kwon, D; Lee, BS; Oh, CH; Tarazi, H | 1 |
| Bernards, R; Boelens, MC; Huijberts, SCFA; Opdam, FL | 1 |
| Tsanni, A | 1 |
| da Motta, KP; Domingues, NLC; Luchese, C; Santos, BF; Wilhelm, EA | 1 |
| Akpomiemie, G; Bosch, B; Casas, CP; Ellis, L; Hill, A; Johnstone, H; Owen, A; Simmons, B; Sokhela, S; Venter, WDF; Woods, J | 1 |
35 review(s) available for carbamates and thiazoles
| Article | Year |
|---|---|
[Antiepileptics. 39].
Topics: Acetazolamide; Adrenocorticotropic Hormone; Aminoglutethimide; Anticonvulsants; Barbiturates; Carbamates; Carbamazepine; Dibenzazepines; Epilepsies, Partial; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Glutethimide; Humans; Hydantoins; Methaqualone; Primidone; Succinimides; Thiazines; Thiazoles; Thioridazine; Trimethadione | 1969 |
Pharmacologic therapy for type 2 diabetes mellitus.
Topics: Acarbose; Administration, Oral; Algorithms; Carbamates; Chromans; Diabetes Mellitus, Type 2; Evidence-Based Medicine; Humans; Hypoglycemic Agents; Insulin; Metformin; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Trisaccharides; Troglitazone | 1999 |
The use of insulin secretagogues in the treatment of type 2 diabetes.
Topics: Acarbose; Carbamates; Chromans; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glucagon; Glucagon-Like Peptide 1; Humans; Hypoglycemic Agents; Metformin; Peptide Fragments; Piperidines; Protein Precursors; Risk Factors; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
New drugs for diabetes.
Topics: Carbamates; Chromans; Cyclohexanes; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Insulin Resistance; Metformin; Nateglinide; Phenylalanine; Piperidines; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
New directions in type 2 diabetes mellitus: an update of current oral antidiabetic therapy.
Topics: Carbamates; Chromans; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Metformin; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
New agents for Type 2 diabetes.
Topics: Anti-Obesity Agents; Carbamates; Chromans; Diabetes Mellitus, Type 2; Drug Design; Humans; Hypoglycemic Agents; Insulin Resistance; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
Clinical efficacy of new thiazolidinediones and glinides in the treatment of type 2 diabetes mellitus.
Topics: Carbamates; Cyclohexanes; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Nateglinide; Phenylalanine; Pioglitazone; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones | 2000 |
Therapeutic strategies in Alzheimer's disease: M1 muscarinic agonists.
Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Apoptosis; Carbamates; Cheirogaleidae; Disease Models, Animal; Humans; Muscarinic Agonists; Neuroprotective Agents; Phenylcarbamates; Piperidines; Receptor, Muscarinic M1; Receptors, Muscarinic; Rivastigmine; Signal Transduction; tau Proteins; Thiazoles | 2000 |
Recent advances in the pharmacologic management of diabetes mellitus.
Topics: Acarbose; Administration, Oral; Carbamates; Chromans; Diabetes Mellitus; Drug Overdose; Emergencies; Humans; Hypoglycemic Agents; Insulin; Insulin Lispro; Metformin; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 2000 |
Combination therapy in type 2 diabetes: the role of repaglinide.
Topics: Carbamates; Chromans; Diabetes Mellitus, Type 2; Drug Synergism; Drug Therapy, Combination; Humans; Hypoglycemic Agents; Insulin, Isophane; Metformin; Piperidines; Thiazoles; Thiazolidinediones; Troglitazone | 2001 |
[Objectives and therapeutic strategy in type 2 diabetes mellitus].
Topics: Carbamates; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Humans; Hyperinsulinism; Hypoglycemic Agents; Insulin Resistance; Piperidines; Thiazoles | 2001 |
[News in oral antidiabetic therapy].
Topics: Administration, Oral; Carbamates; Diabetes Mellitus; Humans; Hypoglycemic Agents; Pioglitazone; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones | 2001 |
Oral antihyperglycemic therapy for type 2 diabetes: scientific review.
Topics: Administration, Oral; Biguanides; Blood Glucose; Carbamates; Chromans; Diabetes Mellitus, Type 2; Diet; Drug Therapy, Combination; Enzyme Inhibitors; Exercise; Glycated Hemoglobin; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Metformin; Piperidines; Randomized Controlled Trials as Topic; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 2002 |
Type 2 diabetes management: a comprehensive clinical review of oral medications.
Topics: Benzamides; Carbamates; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Metformin; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones | 2002 |
[Insulin analogs and new oral antidiabetic drugs].
Topics: Administration, Oral; Carbamates; Cyclohexanes; Diabetes Mellitus; Dose-Response Relationship, Drug; Glucose; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Nateglinide; Phenylalanine; Piperidines; Receptors, Cytoplasmic and Nuclear; Thiazoles; Thiazolidinediones; Transcription Factors | 1999 |
Repaglinide in combination therapy.
Topics: Carbamates; Chromans; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Humans; Hypoglycemic Agents; Insulin; Metformin; Pioglitazone; Piperidines; Postprandial Period; Rosiglitazone; Thiazoles; Thiazolidinediones; Treatment Outcome; Troglitazone | 2002 |
Hypersensitivity to preservatives.
Topics: Carbamates; Cosmetics; Formaldehyde; Humans; Hypersensitivity; Nitriles; Parabens; Preservatives, Pharmaceutical; Prevalence; Thiazoles | 2004 |
Targeting apoptosis pathways by natural compounds in cancer: marine compounds as lead structures and chemical tools for cancer therapy.
Topics: Alkaloids; Alkanes; Animals; Anti-Bacterial Agents; Antineoplastic Agents; Apoptosis; Aquatic Organisms; Biological Products; Bryostatins; Carbamates; Cell Proliferation; Depsipeptides; Dioxoles; Drug Screening Assays, Antitumor; Humans; Lactones; Macrolides; Microtubules; Models, Chemical; Neoplasms; Phenanthrolines; Phenazines; Proteasome Endopeptidase Complex; Pyrones; Pyrroles; Quinolines; Spiro Compounds; Steroids; Tetrahydroisoquinolines; Thiazoles; Trabectedin | 2013 |
Elvitegravir: a once-daily, boosted, HIV-1 integrase inhibitor.
Topics: Adenine; Carbamates; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Deoxycytidine; Drug Combinations; Drug Interactions; Drug Resistance, Viral; Drug-Related Side Effects and Adverse Reactions; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Thiazoles | 2012 |
Combinational therapies for HIV: a focus on EVG/COBI/FTC/TDF.
Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Cobicistat; Deoxycytidine; Drug Combinations; Drug Resistance, Multiple, Viral; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles | 2012 |
Safety of pharmacoenhancers for HIV therapy.
Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Dose-Response Relationship, Drug; Drug Discovery; Drug Interactions; Drug Therapy, Combination; HIV Infections; HIV Protease Inhibitors; Humans; Ritonavir; Thiazoles; Treatment Outcome | 2012 |
Elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate single tablet for HIV-1 infection treatment.
Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials, Phase III as Topic; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV Integrase Inhibitors; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles; Viral Load | 2012 |
Cobicistat-boosted elvitegravir-based fixed-dose combination antiretroviral therapy for HIV infection.
Topics: Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Drug Approval; Drug Combinations; Drug Interactions; Drug Resistance, Viral; HIV Infections; HIV Integrase Inhibitors; Humans; Patient Safety; Quinolones; Thiazoles | 2012 |
Cobicistat: a new boost for the treatment of human immunodeficiency virus infection.
Topics: Anti-HIV Agents; Carbamates; Cobicistat; Cytochrome P-450 CYP3A Inhibitors; Drug Combinations; Drug Interactions; Drug Therapy, Combination; Enzyme Inhibitors; HIV Infections; Humans; Ritonavir; Thiazoles | 2013 |
Single-tablet regimens in HIV: does it really make a difference?
Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Administration Schedule; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Nitriles; Organophosphonates; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Rilpivirine; Tablets; Tenofovir; Thiazoles | 2014 |
Elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate single-tablet regimen (Stribild®): a review of its use in the management of HIV-1 infection in adults.
Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV-1; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles | 2014 |
Cobicistat: a review of its use as a pharmacokinetic enhancer of atazanavir and darunavir in patients with HIV-1 infection.
Topics: Atazanavir Sulfate; Carbamates; Cobicistat; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Darunavir; Drug Synergism; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Oligopeptides; Pyridines; Sulfonamides; Thiazoles | 2014 |
Treating HCV in HIV 2013: on the cusp of change.
Topics: Aminoisobutyric Acids; Antiviral Agents; Carbamates; Coinfection; Drug Interactions; Drug Therapy, Combination; Hepacivirus; Hepatitis C; HIV Infections; Humans; Imidazoles; Leucine; Oligopeptides; Proline; Pyrrolidines; Quinolines; Sofosbuvir; Thiazoles; Treatment Outcome; Uridine Monophosphate; Valine | 2014 |
HCV direct-acting antiviral agents: the best interferon-free combinations.
Topics: Aminoisobutyric Acids; Antiviral Agents; Carbamates; Clinical Trials as Topic; Disease Eradication; Drug Discovery; Drug Therapy, Combination; Hepacivirus; Hepatitis C; Heterocyclic Compounds, 3-Ring; Humans; Imidazoles; Interferon-alpha; Isoquinolines; Leucine; Oligopeptides; Polyethylene Glycols; Proline; Protease Inhibitors; Pyrrolidines; Quinolines; Recombinant Proteins; Ribavirin; Simeprevir; Sofosbuvir; Sulfonamides; Thiazoles; Uridine Monophosphate; Valine; Viral Nonstructural Proteins; Virus Replication | 2014 |
Cobicistat : a new opportunity in the treatment of HIV disease?
Topics: Anti-HIV Agents; Carbamates; Clinical Trials as Topic; Cobicistat; Cost-Benefit Analysis; Drug Combinations; Health Care Costs; HIV Infections; Humans; Thiazoles; Treatment Outcome | 2014 |
Which patients have greatest need for elvitegravir/cobicistat/ emtricitabine/tenofovirDF-based therapy?
Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Combinations; Emtricitabine; HIV Infections; HIV-1; Humans; Patents as Topic; Phosphorous Acids; Quinolones; Thiazoles | 2014 |
Pharmacokinetic enhancers in HIV therapeutics.
Topics: Anti-HIV Agents; Carbamates; Cobicistat; Cytochrome P-450 CYP3A Inhibitors; Drug Combinations; Drug Interactions; Drug Therapy, Combination; HIV Protease Inhibitors; Humans; Ritonavir; Thiazoles | 2014 |
The pharmacokinetics, pharmacodynamics and clinical efficacy of elvitegravir + cobicistat + emtricitabine + tenofovir combination therapy for the treatment of HIV.
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; European Union; HIV Infections; HIV-1; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles | 2015 |
Stribild: a review of component characteristics and combination drug efficacy.
Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Drug Synergism; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Organophosphonates; Quinolones; Thiazoles | 2015 |
Can binimetinib, encorafenib and masitinib be more efficacious than currently available mutation-based targeted therapies for melanoma treatment?
Topics: Benzamides; Benzimidazoles; Carbamates; Humans; Melanoma; Mutation; Piperidines; Protein Kinase Inhibitors; Proteomics; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-kit; Pyridines; Skin Neoplasms; Sulfonamides; Thiazoles | 2017 |
30 trial(s) available for carbamates and thiazoles
| Article | Year |
|---|---|
In vitro antiviral activity of 141W94 (VX-478) in combination with other antiretroviral agents.
Topics: Carbamates; Drug Resistance, Microbial; Drug Synergism; Drug Therapy, Combination; Furans; HIV Infections; HIV Protease Inhibitors; Humans; Indinavir; Isoquinolines; Pyridines; Quinolines; Reverse Transcriptase Inhibitors; Ritonavir; Saquinavir; Sulfonamides; Thiazoles; Valine | 1996 |
Repaglinide/troglitazone combination therapy: improved glycemic control in type 2 diabetes.
Topics: Adult; Aged; Biomarkers; Blood Glucose; Carbamates; Chromans; Cross-Over Studies; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Middle Aged; Piperidines; Thiazoles; Thiazolidinediones; Troglitazone | 2000 |
In vitro-in vivo model for evaluating the antiviral activity of amprenavir in combination with ritonavir administered at 600 and 100 milligrams, respectively, every 12 hours.
Topics: Adult; Anti-HIV Agents; Antiviral Agents; Carbamates; Cell Line; Cells, Cultured; Drug Combinations; Female; Furans; HIV Antigens; Humans; Male; Middle Aged; Models, Biological; Protein Binding; Ritonavir; Sulfonamides; T-Lymphocytes; Tetrazolium Salts; Thiazoles; Time Factors | 2003 |
An NS3 protease inhibitor with antiviral effects in humans infected with hepatitis C virus.
Topics: Administration, Oral; Antiviral Agents; Carbamates; Double-Blind Method; Hepacivirus; Hepatitis C; Humans; Macrocyclic Compounds; Male; Polyproteins; Protein Processing, Post-Translational; Quinolines; Serine Proteinase Inhibitors; Thiazoles; Viral Load; Viral Nonstructural Proteins; Viral Proteins | 2003 |
Short-term antiviral efficacy of BILN 2061, a hepatitis C virus serine protease inhibitor, in hepatitis C genotype 1 patients.
Topics: Antiviral Agents; Carbamates; Dose-Response Relationship, Drug; Double-Blind Method; Female; Hepatitis C, Chronic; Humans; Macrocyclic Compounds; Male; Middle Aged; Protease Inhibitors; Quinolines; RNA, Viral; Serine Endopeptidases; Thiazoles; Viral Load | 2004 |
"Strong reasons make strong actions"--The antiviral efficacy of NS3/4A protease inhibitors.
Topics: Antiviral Agents; Carbamates; Double-Blind Method; Drug Resistance, Viral; Hepatitis C, Chronic; Humans; Macrocyclic Compounds; Quinolines; RNA, Viral; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2005 |
Antiviral efficacy of NS3-serine protease inhibitor BILN-2061 in patients with chronic genotype 2 and 3 hepatitis C.
Topics: Administration, Oral; Adult; Carbamates; Double-Blind Method; Drug Administration Schedule; Female; Genotype; Hepacivirus; Hepatitis C, Chronic; Humans; Kinetics; Macrocyclic Compounds; Male; Middle Aged; Pilot Projects; Prospective Studies; Quinolines; Serine Proteinase Inhibitors; Thiazoles; Viral Load; Viral Nonstructural Proteins | 2005 |
Viral kinetics in patients with chronic hepatitis C treated with the serine protease inhibitor BILN 2061.
Topics: Adult; Antiviral Agents; Area Under Curve; Carbamates; Female; Hepacivirus; Hepatitis C, Chronic; Humans; Interferon-alpha; Kinetics; Macrocyclic Compounds; Male; Middle Aged; Models, Biological; Quinolines; RNA, Viral; Serine Proteinase Inhibitors; Thiazoles | 2006 |
Randomized, phase 2 evaluation of two single-tablet regimens elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate versus efavirenz/emtricitabine/tenofovir disoproxil fumarate for the initial treatment of HIV infection.
Topics: Adenine; Adult; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; CD4 Lymphocyte Count; Cobicistat; Cyclopropanes; Deoxycytidine; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Organophosphonates; Patient Compliance; Patient Selection; Quinolones; Tenofovir; Thiazoles; Treatment Outcome | 2011 |
Phase 2 study of cobicistat versus ritonavir each with once-daily atazanavir and fixed-dose emtricitabine/tenofovir df in the initial treatment of HIV infection.
Topics: Adenine; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Carbamates; CD4 Lymphocyte Count; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Administration Schedule; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Ritonavir; RNA, Viral; Tenofovir; Thiazoles; Treatment Outcome | 2011 |
Effect of cobicistat on glomerular filtration rate in subjects with normal and impaired renal function.
Topics: Adult; Carbamates; Cobicistat; Cohort Studies; Creatinine; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Enzyme Inhibitors; Female; Glomerular Filtration Rate; Humans; Kidney; Male; Metabolic Clearance Rate; Placebos; Thiazoles | 2012 |
Co-formulated elvitegravir, cobicistat, emtricitabine, and tenofovir disoproxil fumarate versus ritonavir-boosted atazanavir plus co-formulated emtricitabine and tenofovir disoproxil fumarate for initial treatment of HIV-1 infection: a randomised, double-
Topics: Adenine; Adult; Anti-HIV Agents; Atazanavir Sulfate; Carbamates; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Ritonavir; Tenofovir; Thiazoles | 2012 |
Co-formulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus co-formulated efavirenz, emtricitabine, and tenofovir for initial treatment of HIV-1 infection: a randomised, double-blind, phase 3 trial, analysis of results after 48 weeks.
Topics: Adenine; Adult; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Cobicistat; Cyclopropanes; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Tenofovir; Thiazoles | 2012 |
A randomized, double-blind comparison of coformulated elvitegravir/cobicistat/emtricitabine/tenofovir DF vs ritonavir-boosted atazanavir plus coformulated emtricitabine and tenofovir DF for initial treatment of HIV-1 infection: analysis of week 96 results
Topics: Adenine; Adult; Alanine Transaminase; Anti-HIV Agents; Aspartate Aminotransferases; Atazanavir Sulfate; Bilirubin; Bone Density; Carbamates; Cobicistat; Confidence Intervals; Creatinine; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Ritonavir; RNA, Viral; Tenofovir; Thiazoles; Triglycerides | 2013 |
A randomized double-blind comparison of coformulated elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate versus efavirenz/emtricitabine/tenofovir disoproxil fumarate for initial treatment of HIV-1 infection: analysis of week 96 results.
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Creatinine; Deoxycytidine; Double-Blind Method; Drug Combinations; Efavirenz, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Female; HIV Infections; HIV-1; Humans; Male; Organophosphonates; Oxazines; Quinolones; RNA, Viral; Thiazoles; Treatment Outcome; Young Adult | 2013 |
Cobicistat versus ritonavir as a pharmacoenhancer of atazanavir plus emtricitabine/tenofovir disoproxil fumarate in treatment-naive HIV type 1-infected patients: week 48 results.
Topics: Adenine; Adult; Anti-HIV Agents; Atazanavir Sulfate; Carbamates; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Ritonavir; Tenofovir; Thiazoles; Treatment Outcome; Viral Load | 2013 |
Pharmacokinetics of once-daily boosted elvitegravir when administered in combination with acid-reducing agents.
Topics: Adolescent; Adult; Antacids; Anti-HIV Agents; Area Under Curve; Carbamates; Cobicistat; Cross-Over Studies; Drug Administration Schedule; Drug Interactions; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Quinolones; Thiazoles | 2013 |
Pharmacokinetics of cobicistat boosted-elvitegravir administered in combination with rosuvastatin.
Topics: Adult; Animals; Anti-HIV Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Carbamates; CHO Cells; Cobicistat; Cricetulus; Dogs; Drug Combinations; Drug Interactions; Drug Therapy, Combination; Female; Fluorobenzenes; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Liver-Specific Organic Anion Transporter 1; Madin Darby Canine Kidney Cells; Male; Neoplasm Proteins; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Pyrimidines; Quinolones; Rosuvastatin Calcium; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfonamides; Thiazoles | 2014 |
Effects of a protein-rich drink or a standard meal on the pharmacokinetics of elvitegravir, cobicistat, emtricitabine and tenofovir in healthy Japanese male subjects: a randomized, three-way crossover study.
Topics: Adenine; Adult; Anti-HIV Agents; Asian People; Beverages; Carbamates; Cobicistat; Cross-Over Studies; Deoxycytidine; Dietary Proteins; Drug Combinations; Emtricitabine; Food-Drug Interactions; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Tenofovir; Thiazoles; Young Adult | 2014 |
Pharmacokinetics of darunavir in fixed-dose combination with cobicistat compared with coadministration of darunavir and ritonavir as single agents in healthy volunteers.
Topics: Adult; Biological Availability; Carbamates; Cobicistat; Cross-Over Studies; Cytochrome P-450 CYP3A Inhibitors; Darunavir; Drug Combinations; Female; Healthy Volunteers; HIV Protease Inhibitors; Humans; Male; Middle Aged; Ritonavir; Sulfonamides; Thiazoles; Young Adult | 2014 |
Switching to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of non-nucleoside reverse transcriptase inhibitor with emtricitabine and tenofovir in virologically suppressed adults with HIV (STRATEGY-NNRTI): 48 week r
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Reverse Transcriptase Inhibitors; Tenofovir; Thiazoles; Viral Load | 2014 |
Simplification to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of ritonavir-boosted protease inhibitor with emtricitabine and tenofovir in adults with virologically suppressed HIV (STRATEGY-PI): 48 week results o
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Therapy, Combination; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Protease Inhibitors; Quinolones; Ritonavir; Tenofovir; Thiazoles; Viral Load | 2014 |
Bioequivalence of a darunavir/cobicistat fixed-dose combination tablet versus single agents and food effect in healthy volunteers.
Topics: Administration, Oral; Adolescent; Adult; Carbamates; Cobicistat; Darunavir; Drug Combinations; Drug Monitoring; Female; Food; Healthy Volunteers; Humans; Male; Middle Aged; Sulfonamides; Therapeutic Equivalency; Thiazoles; Young Adult | 2014 |
In vitro antiviral activity and preclinical and clinical resistance profile of miravirsen, a novel anti-hepatitis C virus therapeutic targeting the human factor miR-122.
Topics: 5' Untranslated Regions; Antiviral Agents; Carbamates; Cyclohexanols; Drug Resistance, Viral; Drug Therapy, Combination; Hepacivirus; Hepatitis C, Chronic; Humans; Imidazoles; Macrocyclic Compounds; MicroRNAs; Molecular Targeted Therapy; Mutation; Oligonucleotides; Oligopeptides; Pyrrolidines; Quinolines; Replicon; Thiazoles; Thiophenes; Valine | 2015 |
Tenofovir alafenamide versus tenofovir disoproxil fumarate, coformulated with elvitegravir, cobicistat, and emtricitabine, for initial treatment of HIV-1 infection: two randomised, double-blind, phase 3, non-inferiority trials.
Topics: Adenine; Adult; Alanine; Anti-HIV Agents; Arthralgia; Bone Density; Carbamates; CD4 Lymphocyte Count; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Combinations; Emtricitabine; Female; Headache; HIV Infections; Humans; Kidney; Male; Nausea; Organophosphonates; Quinolones; Respiration Disorders; Sleep Initiation and Maintenance Disorders; Tenofovir; Thiazoles; Treatment Outcome; Viral Load | 2015 |
Brief Report: Cobicistat Compared With Ritonavir as a Pharmacoenhancer for Atazanavir in Combination With Emtricitabine/Tenofovir Disoproxil Fumarate: Week 144 Results.
Topics: Adenine; Adult; Anti-HIV Agents; Atazanavir Sulfate; Carbamates; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Administration Schedule; Drug Synergism; Drug Therapy, Combination; Emtricitabine; Female; HIV Infections; HIV-1; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Ritonavir; RNA, Viral; Tenofovir; Thiazoles; Viral Load | 2015 |
A Phase Ib Dose-Escalation Study of Encorafenib and Cetuximab with or without Alpelisib in Metastatic
Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Carbamates; Cetuximab; Colorectal Neoplasms; Disease-Free Survival; Female; Humans; Male; Maximum Tolerated Dose; Middle Aged; Mutation; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Sulfonamides; Thiazoles | 2017 |
Safety and efficacy of a fixed-dose combination regimen of grazoprevir, ruzasvir, and uprifosbuvir with or without ribavirin in participants with and without cirrhosis with chronic hepatitis C virus genotype 1, 2, or 3 infection (C-CREST-1 and C-CREST-2,
Topics: Adult; Amides; Antiviral Agents; Carbamates; Cyclopropanes; Drug Administration Schedule; Female; Genotype; Hepatitis C, Chronic; Heterocyclic Compounds, 4 or More Rings; Humans; Liver Cirrhosis; Male; Middle Aged; Pyrrolidines; Quinoxalines; Ribavirin; Sulfonamides; Sustained Virologic Response; Thiazoles; Uridine | 2017 |
Safety and efficacy of an 8-week regimen of grazoprevir plus ruzasvir plus uprifosbuvir compared with grazoprevir plus elbasvir plus uprifosbuvir in participants without cirrhosis infected with hepatitis C virus genotypes 1, 2, or 3 (C-CREST-1 and C-CREST
Topics: Adult; Aged; Amides; Antiviral Agents; Benzofurans; Carbamates; Cyclopropanes; Drug Administration Schedule; Drug Combinations; Drug Therapy, Combination; Female; Genotype; Hepatitis C, Chronic; Heterocyclic Compounds, 4 or More Rings; Humans; Imidazoles; Male; Middle Aged; Pyrrolidines; Quinoxalines; Sulfonamides; Sustained Virologic Response; Thiazoles; Uridine; Young Adult | 2017 |
Randomized clinical trial of nitazoxanide or sofosbuvir/daclatasvir for the prevention of SARS-CoV-2 infection.
Topics: Antiviral Agents; Carbamates; COVID-19; Humans; Imidazoles; Nitro Compounds; Pyrrolidines; SARS-CoV-2; Sofosbuvir; South Africa; Thiazoles; Treatment Outcome; Valine | 2022 |
169 other study(ies) available for carbamates and thiazoles
| Article | Year |
|---|---|
Antischistosomal activity of S-2-[[2-(2-thiazolylcarbamoyl) ethyl] amino] ethyl hydrogen thiosulfate in vitro and in vivo.
Topics: Animals; Carbamates; Female; Haplorhini; Macaca mulatta; Male; Mice; Schistosoma mansoni; Schistosomiasis; Schistosomicides; Thiazoles | 1977 |
Anthelmintic activity of tioxidazole (Sch 21480) against gastrointestinal roundworms.
Topics: Animals; Antinematodal Agents; Carbamates; Dogs; Gastrointestinal Diseases; Mice; Nematode Infections; Sheep; Thiazoles | 1978 |
An evaluation of ethyl-6-ethoxybenzothiazole-2-carbamate (Sch 18099) for anthelmintic activity in domestic animals.
Topics: Animals; Animals, Domestic; Anthelmintics; Ascariasis; Carbamates; Chickens; Horses; Nematode Infections; Poultry Diseases; Sheep; Sheep Diseases; Strongyle Infections, Equine; Swine; Swine Diseases; Thiazoles; Trichuriasis | 1977 |
Synthesis and anthelmintic activity of carbamates derived from imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b]thiazole.
Topics: Animals; Anthelmintics; Antinematodal Agents; Caenorhabditis; Carbamates; Imidazoles; Mice; Nematoda; Nematode Infections; Structure-Activity Relationship; Thiadiazoles; Thiazoles | 1992 |
Synthesis and antineoplastic activity of 5-aryl-2,3-dihydropyrrolo[2,1-b]thiazole-6,7-dimethanol 6,7-bis(isopropylcarbamates).
Topics: Carbamates; Cell Division; Cell Survival; Chemical Phenomena; Chemistry; Colonic Neoplasms; Humans; Leukemia, Myeloid; Neoplasms; Pyrroles; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured | 1988 |
Synthesis, chemical reactivity, and antileukemic activity of 5-substituted 6,7-bis(hydroxymethyl)pyrrolo[1,2-c]thiazole biscarbamates and the corresponding sulfoxides and sulfones.
Topics: Animals; Antineoplastic Agents; Carbamates; Leukemia P388; Leukemia, Experimental; Mice; Structure-Activity Relationship; Sulfones; Sulfoxides; Thiazoles | 1987 |
On the genotoxicity of the pesticides Endodan and Kilacar in 6 different test systems.
Topics: Animals; Aspergillus nidulans; Benzyl Alcohols; Benzyl Compounds; Biotransformation; Bone Marrow; Carbamates; Cells, Cultured; Chromosome Aberrations; Cricetinae; Genes, Dominant; Genes, Lethal; Herbicides; Humans; Lymphocytes; Microsomes, Liver; Mutagenicity Tests; Mutagens; Mutation; Rats; Rats, Inbred Strains; Salmonella typhimurium; Sister Chromatid Exchange; Thiazoles | 1985 |
Sensitivity of the spores of Blastocladiella emersonii and related fungi to antibiotics and some other drugs.
Topics: Acridines; Aniline Compounds; Anti-Bacterial Agents; Antifungal Agents; Antimycin A; Carbamates; Chloramphenicol; Chlortetracycline; Coloring Agents; Cycloheximide; Dactinomycin; Fungi; Mercury; Microbial Sensitivity Tests; Mitomycins; Nitrobenzenes; Nystatin; Phenols; Spores; Staphylococcus; Sulfonic Acids; Tetracycline; Thiazoles; Triazines; Urea | 1971 |
Rubber boot dermatitis in Newfoundland: a survey of 30 patients.
Topics: Adult; Aged; Benzene Derivatives; Carbamates; Chromates; Dermatitis Herpetiformis; Dermatitis, Contact; Dermatitis, Exfoliative; Dermatitis, Occupational; Diagnosis, Differential; Eczema; Eczema, Dyshidrotic; Fisheries; Foot Dermatoses; Guanidines; Humans; Hydrocortisone; Hypersensitivity; Leg Dermatoses; Male; Middle Aged; Neurodermatitis; Newfoundland and Labrador; Plastics; Purpura; Quinolines; Rubber; Shoes; Skin Tests; Sulfides; Thiazoles; Trimeprazine; Workers' Compensation | 1969 |
Anthelmintic activities of cambendazole in calves: effect on nematode morphogenesis from ova to the infective larval stage.
Topics: Ancylostomatoidea; Animals; Anthelmintics; Benzimidazoles; Carbamates; Cattle; Cattle Diseases; Female; Hookworm Infections; Larva; Morphogenesis; Nematoda; Nematode Infections; Oesophagostomiasis; Oesophagostomum; Ovum; Thiazoles; Trichostrongyloidea; Trichostrongyloidiasis | 1973 |
Treatment and control of Dictyocaulus viviparus in captive black-tailed deer.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Carbamates; Deer; Dictyocaulus Infections; Feces; Imidazoles; Larva; Nematoda; Oregon; Poaceae; Seasons; Thiazoles; Time Factors | 1973 |
An anthelmintic test for gastro-intestinal nematodes of cattle.
Topics: Ancylostomatoidea; Animals; Anthelmintics; Benzimidazoles; Benzoates; Carbamates; Cattle; Cattle Diseases; Digestive System; Filtration; Hookworm Infections; Larva; Male; Methods; Nematoda; Nematode Infections; Nylons; Oesophagostomiasis; Oesophagostomum; Thiabendazole; Thiazoles; Trichostrongyloidea; Trichostrongyloidiasis | 1972 |
Adverse effect of thiadiazolylcarbamic acid esters on measles and polio viruses in Vero cells. Brief report.
Topics: Animals; Antiviral Agents; Aphthovirus; Carbamates; Cell Line; Chemical Phenomena; Chemistry; Culture Techniques; Cytopathogenic Effect, Viral; Haplorhini; HeLa Cells; Kidney; Measles virus; Poliovirus; Thiazoles; Vaccinia virus; Virus Replication | 1970 |
Protection of animals against soman (1,2,2-trimethylpropyl methylphosphono-fluoridate) by pretreatment with some other organophosphorus compounds, followed by oxime and atropine.
Topics: Amitriptyline; Animals; Atropine; Bromides; Carbamates; Cholinesterase Inhibitors; Diphosphates; Drug Antagonism; Female; Fluorine; Guinea Pigs; Hydroxamic Acids; Isoflurophate; Lethal Dose 50; Nitrates; Nitrophenols; Nitroso Compounds; Organophosphonates; Organophosphorus Compounds; Orphenadrine; Oximes; Parasympatholytics; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Salicylates; Scopolamine; Species Specificity; Sulfonic Acids; Sulfuric Acids; Thiazoles; Time Factors | 1971 |
Studies on fungicides. XXV. Addition reaction of dithiocarbamates to fumaronitrile, bis(alkylthio)maleonitrile, 2,3-dicyano-5,6-dihydro-1,4-dithiin and 4,5-dicyano-2-oxo-1,4-dithiole.
Topics: Carbamates; Chemical Phenomena; Chemistry; Fungicides, Industrial; Nitriles; Thiazoles; Thiophenes | 1974 |
Efficacy of cambendazole against naturally occurring Nematodirus helvetianus and Cooperia oncophora infections in calves.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Carbamates; Cattle; Cattle Diseases; Feces; Female; Intestine, Small; Male; Parasite Egg Count; Thiazoles; Trichostrongyloidea; Trichostrongyloidiasis | 1974 |
Helminth control in grazing sheep: periodic treatment with levamisole, morantel, cambendazole, and mebendazole.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Benzoates; Carbamates; Cestode Infections; Haemonchiasis; Helminthiasis; Helminthiasis, Animal; Hematocrit; Levamisole; Oesophagostomiasis; Pyrimidines; Sheep; Sheep Diseases; Strongyloidiasis; Thiazoles; Thiophenes; Trichostrongyloidiasis; Trichuriasis | 1974 |
The efficacy of cambendazole against cestode and nematode infestations in sheep and cattle.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Cattle; Cattle Diseases; Cestode Infections; Haemonchiasis; Monieziasis; Nematode Infections; Ostertagiasis; Sheep; Sheep Diseases; Thiazoles; Trichostrongyloidiasis; Trichostrongylosis | 1972 |
Experimental development of a cambendazole-resistant strain of Haemonchus contortus in sheep.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Drug Resistance; Larva; Sheep; Sheep Diseases; Thiazoles; Trichostrongyloidea; Trichostrongyloidiasis | 1973 |
Nippostrongylus brasiliensis: effect of dexamethasone upon anthelmintic efficacy.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Butanes; Carbamates; Dexamethasone; Hookworm Infections; Immunosuppression Therapy; Male; Rats; Thiabendazole; Thiazoles | 1973 |
Procedures for the treatment and prevention of canine heartworm disease.
Topics: Animals; Arsenicals; Carbamates; Dirofilariasis; Dog Diseases; Dogs; Fenthion; Filaricides; Imidazoles; Sulfhydryl Compounds; Thiazoles | 1973 |
Anthelmintic efficacy of cambendazole against gastrointestinal parasites of the horse.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Carbamates; Horse Diseases; Horses; Intestinal Diseases, Parasitic; Nematode Infections; Oxyuriasis; Stomach Diseases; Strongyle Infections, Equine; Strongyloidiasis; Thiazoles | 1973 |
The fumarate reductase reaction of Haemonchus contortus and the mode of action of some anthelmintics.
Topics: Animals; Anthelmintics; Benzimidazoles; Benzoates; Carbamates; Carbon Isotopes; Drug Resistance; Fumarates; Iodine; Mitochondria; Nitrophenols; Oxidoreductases; Pyrimidines; Spectrophotometry; Succinates; Thiabendazole; Thiazoles; Thiophenes; Trichostrongyloidea | 1973 |
Evaluation of paste form of cambendazole and thiabendazole for administration to calves.
Topics: Administration, Oral; Animals; Anthelmintics; Benzimidazoles; Carbamates; Cattle; Cattle Diseases; Feces; Female; Hookworm Infections; Male; Nematode Infections; Oesophagostomiasis; Parasite Egg Count; Thiabendazole; Thiazoles; Trichostrongyloidiasis; Trichuriasis | 1973 |
Preliminary evauation of levamisole, parbendazole, and cambendazole as thysanosomicides in sheep.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Cestode Infections; Female; Imidazoles; Sheep; Sheep Diseases; Thiazoles | 1973 |
Radioprotective thiazolidines from beta-keto esters.
Topics: Animals; Carbamates; Dose-Response Relationship, Drug; Esters; Isomerism; Keto Acids; Lethal Dose 50; Mercaptoethylamines; Mice; Mice, Inbred Strains; Radiation Dosage; Radiation Effects; Radiation-Protective Agents; Spectrophotometry, Infrared; Thiazoles | 1973 |
Efficacy of cambendazole against tapeworm and roundworm infections in lambs.
Topics: Abomasum; Animals; Anthelmintics; Benzimidazoles; Carbamates; Intestine, Large; Intestine, Small; Monieziasis; Nematode Infections; Sheep; Sheep Diseases; Suspensions; Thiazoles | 1973 |
Action of liver glutamine transaminase and L-amino acid oxidase on several glutamine analogs. Preparation and properties of the 4-S, O, and NH analogs of alpha-ketoglutaramic acid.
Topics: Amidohydrolases; Amino Acid Oxidoreductases; Amino Acids, Diamino; Animals; Carbamates; Carboxylic Acids; Chemical Phenomena; Chemistry; Chromatography, Paper; Cysteine; Glutamine; Glyoxylates; Hydrogen Peroxide; Imidazoles; Lactams; Liver; Propionates; Rats; Semicarbazides; Serine; Snakes; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet; Thiazoles; Transaminases; Urea; Venoms | 1973 |
Efficacy of ipronidazole in feed and water against histomoniasis in turkeys 4 to 10 weeks of age.
Topics: Administration, Oral; Animal Feed; Animals; Antifungal Agents; Arsenicals; Carbamates; Nitro Compounds; Nitroimidazoles; Phenylurea Compounds; Poultry Diseases; Protozoan Infections; Thiazoles; Turkeys; Water | 1973 |
Cambendazole-resistant Haemonchus contortus strain in sheep: further experimental development.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Drug Resistance; Sheep; Sheep Diseases; Thiazoles; Trichostrongyloidea; Trichostrongyloidiasis | 1974 |
Chemotherapy of Trichinella spiralis infections (a review).
Topics: Animals; Anthelmintics; Antinematodal Agents; Benzimidazoles; Benzoates; Cadmium; Carbamates; Cycloheptanes; Cyclopentanes; Diethylcarbamazine; Ethanol; Glucocorticoids; Humans; Imidazoles; Insecticides; Levamisole; Metronidazole; Mice; Organophosphorus Compounds; Piperazines; Pyrantel; Tetramisole; Thiabendazole; Thiazoles; Trichinella; Trichinellosis | 1974 |
The action of six anthelmintics against Trichostrongylus axei in lambs.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Coumarins; Imidazoles; Phenothiazines; Pyridines; Pyrimidines; Sheep; Sheep Diseases; Thiazoles; Time Factors; Trichostrongyloidiasis | 1972 |
The efficacy of various anthelmintics against the parasitic larval stages of Ancylostoma caninum in Mastomys natalensis.
Topics: Ancylostoma; Animals; Anthelmintics; Benzene Derivatives; Benzimidazoles; Carbamates; Disease Models, Animal; Larva; Muscles; Organophosphonates; Pyridines; Rats; Thiabendazole; Thiazoles; Thiocyanates | 1970 |
Preparation and antimicrobial activity of N-thiadiazolycarbamic acid esters.
Topics: Bacteria; Carbamates; Chemical Phenomena; Chemistry; Esters; Microbial Sensitivity Tests; Thiazoles | 1971 |
[A test of anthelmintics in nematodiriasis in sheep].
Topics: Animals; Anthelmintics; Carbamates; Insecticides; Naphthalenes; Nematode Infections; Sheep; Sheep Diseases; Thiazoles | 1967 |
Comparative efficacy of levo-tetramisole, parbendazole, and piperazine citrate against some common helminths of turkeys.
Topics: Animals; Anthelmintics; Benzimidazoles; Carbamates; Female; Male; Methods; Nematoda; Piperazines; Poultry Diseases; Thiazoles; Turkeys | 1969 |
The enzymic oxidation of chlorogenic acid and some reactions of the quinone produced.
Topics: Ascorbic Acid; Carbamates; Chlorogenic Acid; Chromatography, Paper; Cysteine; Cystine; In Vitro Techniques; Manometry; Nicotiana; Oxidoreductases; Plants, Toxic; Quinones; Sulfinic Acids; Thiazoles; Thioglycolates | 1966 |
[Synthesis of 3-furfuralrhodanin and its 5-ariliden derivatives].
Topics: Carbamates; Furaldehyde; Thiazoles | 1966 |
The structure of an N-carbamoyl derivative of 2-amino-delta-2-thiazoline. Mass spectrometry of 15N derivatives of 2-amino-delta-2-thiazoline.
Topics: Carbamates; Cyanates; Spectrum Analysis; Thiazoles | 1967 |
[Experimental study of the teratogenicity and embryotoxicity of endodan].
Topics: Abnormalities, Drug-Induced; Animals; Carbamates; Dose-Response Relationship, Drug; Embryo Loss; Embryo, Mammalian; Female; Herbicides; Male; Pregnancy; Rats; Rats, Inbred Strains; Thiazoles; Time Factors | 1984 |
Tioxidazole: evaluation of antiparasitic activity of a micronized formulation in horses by the critical test method.
Topics: Animals; Carbamates; Horse Diseases; Horses; Thiazoles | 1981 |
[Assessment of the potential risk for progeny in work with endodan (experimental studies)].
Topics: Animals; Carbamates; Dose-Response Relationship, Drug; Enzyme Activation; Female; Genes, Dominant; Genes, Lethal; Herbicides; Male; Mutagens; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Reproduction; Risk; Teratogens; Thiazoles | 1981 |
Critical tests of new benzothiazole anthelmintic tioxidazole in the horse.
Topics: Animals; Anthelmintics; Carbamates; Cestode Infections; Diptera; Horse Diseases; Horses; Nematode Infections; Oxyuriasis; Parasitic Diseases; Parasitic Diseases, Animal; Strongyle Infections, Equine; Thiazoles | 1980 |
Kinetic characterization and cross-resistance patterns of HIV-1 protease mutants selected under drug pressure.
Topics: Amino Acid Sequence; Binding Sites; Carbamates; Cloning, Molecular; Drug Resistance, Microbial; HIV Protease; HIV Protease Inhibitors; HIV-1; Indinavir; Isoquinolines; Kinetics; Methylurea Compounds; Mutagenesis, Site-Directed; Oligopeptides; Point Mutation; Pyridines; Quinolines; Recombinant Proteins; Saquinavir; Structure-Activity Relationship; Thiazoles; Valine | 1995 |
Progress report on new antiepileptic drugs: a summary of the Third Eilat Conference.
Topics: Acetamides; Animals; Anticonvulsants; Azetidines; Carbamates; Drug Evaluation, Preclinical; Drugs, Investigational; Epilepsy; Humans; Israel; Levetiracetam; Nipecotic Acids; Phenylenediamines; Piracetam; Product Surveillance, Postmarketing; Randomized Controlled Trials as Topic; Thiazoles; Tiagabine; Triazoles | 1996 |
Tumor-killer made; how does it work?
Topics: Alkanes; Antineoplastic Agents; Carbamates; Computer Simulation; Epothilones; Epoxy Compounds; Lactones; Microtubules; Models, Molecular; Molecular Conformation; Paclitaxel; Pyrones; Thiazoles; Tumor Cells, Cultured | 1996 |
A common pharmacophore for cytotoxic natural products that stabilize microtubules.
Topics: Alkaloids; Alkanes; Antineoplastic Agents, Phytogenic; Carbamates; Computer Graphics; Diterpenes; Epothilones; Epoxy Compounds; Lactones; Magnetic Resonance Spectroscopy; Microtubules; Models, Molecular; Molecular Conformation; Molecular Structure; Paclitaxel; Pyrones; Thiazoles | 1999 |
Antimicrobial and genotoxic activities of N-(2-hydroxyethyl)-1,2-benzisothiazol-3(2H)-thione carbamic esters.
Topics: Anti-Bacterial Agents; Carbamates; DNA; DNA Damage; Microbial Sensitivity Tests; Mutagenicity Tests; Structure-Activity Relationship; Thiazoles | 1999 |
The novel neuropeptide Y Y(1) receptor antagonist J-104870: a potent feeding suppressant with oral bioavailability.
Topics: Administration, Oral; Animals; Binding, Competitive; Biological Availability; Brain; Carbamates; Cell Membrane; CHO Cells; Cricetinae; Feeding Behavior; Hippocampus; Humans; Inhibitory Concentration 50; Injections, Intraventricular; Male; Neuropeptide Y; Rats; Rats, Sprague-Dawley; Rats, Zucker; Receptors, Neuropeptide Y; Thiazoles; Time Factors | 1999 |
Pharmacologic management of diabetes mellitus.
Topics: Carbamates; Chromans; Diabetes Mellitus; Humans; Hypoglycemic Agents; Metformin; Piperidines; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
Managing type 2 diabetes. A look at the newer agents.
Topics: Acarbose; Carbamates; Chromans; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Metformin; Piperidines; Thiazoles; Thiazolidinediones; Troglitazone | 1999 |
Taxol and discodermolide represent a synergistic drug combination in human carcinoma cell lines.
Topics: Alkaloids; Alkanes; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Carbamates; Cell Count; Cell Division; Cell Line; Cytoskeleton; Diterpenes; Dose-Response Relationship, Drug; Drug Synergism; Epothilones; Epoxy Compounds; Flow Cytometry; Humans; Lactones; Lung Neoplasms; Microtubules; Mitosis; Paclitaxel; Pyrones; Thiazoles; Tumor Cells, Cultured | 2000 |
HIV protease inhibitors block adipogenesis and increase lipolysis in vitro.
Topics: Adipocytes; Animals; Azo Compounds; Bexarotene; Carbamates; Carrier Proteins; Cell Differentiation; Cells, Cultured; Coloring Agents; Fatty Acid-Binding Proteins; Furans; HIV Protease Inhibitors; Indinavir; Insulin; Lipolysis; Lipoprotein Lipase; Nelfinavir; Neoplasm Proteins; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Ritonavir; RNA, Messenger; Rosiglitazone; Saquinavir; Stem Cells; Sulfonamides; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Triglycerides | 2000 |
Honing type 2 diabetes treatment.
Topics: Carbamates; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Pioglitazone; Piperidines; Thiazoles; Thiazolidinediones | 2001 |
Different binding sites for the neuropeptide Y Y1 antagonists 1229U91 and J-104870 on human Y1 receptors.
Topics: Alanine; Amino Acid Sequence; Animals; Appetite Depressants; Binding Sites; Binding, Competitive; Carbamates; Humans; Ligands; Microscopy, Fluorescence; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Peptides, Cyclic; Protein Binding; Protein Structure, Tertiary; Rats; Receptors, Neuropeptide Y; Sequence Homology, Amino Acid; Thiazoles | 2001 |
Conference looks at HIV drug resistance.
Topics: Antiviral Agents; Carbamates; CD4 Lymphocyte Count; Drug Resistance, Microbial; Furans; HIV; HIV Infections; HIV Protease Inhibitors; Humans; Indinavir; Isoquinolines; Lamivudine; Pyridines; Quinolines; Ritonavir; Saquinavir; Sulfonamides; Thiazoles; Valine; Viremia; Zalcitabine; Zidovudine | 1995 |
A new era in type 2 diabetes mellitus treatment?
Topics: 1-Deoxynojirimycin; Acarbose; Carbamates; Diabetes Mellitus, Type 2; Glucosamine; Humans; Hypoglycemic Agents; Imino Pyranoses; Multicenter Studies as Topic; Pioglitazone; Piperidines; Randomized Controlled Trials as Topic; Thiazoles; Thiazolidinediones | 2001 |
Utilization of oral hypoglycemic agents in a drug-insured U.S. population.
Topics: Carbamates; Chromans; Cohort Studies; Databases as Topic; Diabetes Mellitus, Type 2; Enzyme Inhibitors; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Insurance, Pharmaceutical Services; Longitudinal Studies; Managed Care Programs; Metformin; Piperidines; Retrospective Studies; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones; Time Factors; Troglitazone; United States | 2001 |
Tubulins in the primate retina: evidence that xanthophylls may be endogenous ligands for the paclitaxel-binding site.
Topics: Alkaloids; Alkanes; Animals; Antineoplastic Agents, Phytogenic; Binding Sites; Carbamates; Carotenoids; Diterpenes; Epothilones; Epoxy Compounds; Haplorhini; Humans; Lactones; Ligands; Lutein; Models, Molecular; Molecular Sequence Data; Paclitaxel; Pyrones; Retina; Thiazoles; Tubulin | 2001 |
Permeability profiles of M-alkoxysubstituted pyrrolidinoethylesters of phenylcarbamic acid across caco-2 monolayers and human skin.
Topics: Administration, Cutaneous; Algorithms; Caco-2 Cells; Carbamates; Chemical Phenomena; Chemistry, Physical; Chromatography, High Pressure Liquid; Esters; Humans; In Vitro Techniques; Iontophoresis; Molecular Weight; Permeability; Skin Absorption; Solubility; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles | 2002 |
Cytoskeletal responses during early development of the downy mildew of grapevine (Plasmopara viticola).
Topics: Actins; Bridged Bicyclo Compounds, Heterocyclic; Carbamates; Cell Polarity; Cytoplasmic Vesicles; Cytoskeleton; Oomycetes; Spores, Fungal; Thiazoles; Thiazolidines; Time Factors; Tubulin; Vitis | 2002 |
[Glinides and glitazones in diabetes treatment. Are they really effective?].
Topics: Carbamates; Cyclohexanes; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Humans; Hypoglycemic Agents; Insulin; Nateglinide; Phenylalanine; Pioglitazone; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones; Treatment Outcome | 2002 |
Equatorial retention of the contractile actin ring by microtubules during cytokinesis.
Topics: Actins; Anaphase; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Carbamates; Cell Cycle Proteins; Cell Division; Cell Nucleus; Cytoskeletal Proteins; Interphase; Microtubule-Organizing Center; Microtubules; Mitosis; Mutation; Recombinant Fusion Proteins; Schizosaccharomyces; Schizosaccharomyces pombe Proteins; Temperature; Thiazoles; Thiazolidines; Tubulin | 2003 |
Economic model of first-line drug strategies to achieve recommended glycaemic control in newly diagnosed type 2 diabetes mellitus.
Topics: Carbamates; Cohort Studies; Decision Trees; Diabetes Mellitus, Type 2; Direct Service Costs; Drug Costs; Drug Therapy, Combination; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Managed Care Programs; Markov Chains; Metformin; Models, Economic; Piperidines; Rosiglitazone; Thiazoles; Thiazolidinediones; United States | 2003 |
Development of water-soluble prodrugs of the HIV-1 protease inhibitor KNI-727: importance of the conversion time for higher gastrointestinal absorption of prodrugs based on spontaneous chemical cleavage.
Topics: Animals; Area Under Curve; Biological Availability; Carbamates; Cyclization; Drug Design; Duodenum; Furans; Half-Life; HIV Protease Inhibitors; Imides; Intestinal Absorption; Male; Organophosphates; Prodrugs; Rats; Rats, Sprague-Dawley; Solubility; Structure-Activity Relationship; Sulfonamides; Thiazoles; Water | 2003 |
INHIBITION OF GLYCOLYSIS BY ORGANIC SULFUR DERIVATIVES.
Topics: Antimetabolites; Carbamates; Carbohydrate Metabolism; Esters; Glycolysis; Pharmacology; Saliva; Sulfites; Sulfur; Thiazines; Thiazoles; Thiourea | 1965 |
Virology: fresh assault on hepatitis C.
Topics: Antiviral Agents; Carbamates; Clinical Trials as Topic; Drug Design; Hepacivirus; Hepatitis C; Humans; Macrocyclic Compounds; Quinolines; Serine Proteinase Inhibitors; Thiazoles; Viral Load; Viral Nonstructural Proteins | 2003 |
Microwave-assisted extraction for the simultaneous determination of thiamethoxam, imidacloprid, and carbendazim residues in fresh and cooked vegetable samples.
Topics: Benzimidazoles; Carbamates; Chromatography, High Pressure Liquid; Hot Temperature; Imidazoles; Microwaves; Neonicotinoids; Nitro Compounds; Oxazines; Pesticide Residues; Thiamethoxam; Thiazoles; Vegetables | 2004 |
In vitro resistance studies of hepatitis C virus serine protease inhibitors, VX-950 and BILN 2061: structural analysis indicates different resistance mechanisms.
Topics: Amino Acids; Aspartic Acid; Binding Sites; Carbamates; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Genes, Dominant; Hepacivirus; Inhibitory Concentration 50; Kinetics; Macrocyclic Compounds; Models, Chemical; Models, Molecular; Mutation; Oligopeptides; Plasmids; Protein Structure, Tertiary; Quinolines; Serine Proteinase Inhibitors; Thiazoles; Time Factors; Viral Nonstructural Proteins | 2004 |
Enantioseparation in capillary chromatography and capillary electrochromatography using polysaccharide-type chiral stationary phases.
Topics: Carbamates; Cellulose; Chromatography; Electrophoresis, Capillary; Molecular Conformation; Molecular Structure; Phenylcarbamates; Polysaccharides; Silanes; Stereoisomerism; Thalidomide; Thiazoles; Thiazolidines | 2004 |
[Review of recent research on hepatitis C therapy for 54th annual meeting of the American association for the study of liver diseases].
Topics: Carbamates; Hepatitis C; Humans; Interferon-alpha; Interferons; Macrocyclic Compounds; Oligonucleotides, Antisense; Quinolines; RNA-Dependent RNA Polymerase; Serum Albumin; Serum Albumin, Human; Thiazoles; Viral Hepatitis Vaccines | 2004 |
Inhibitors of hepatitis C virus NS3.4A protease 2. Warhead SAR and optimization.
Topics: Carbamates; Hepacivirus; Macrocyclic Compounds; Quinolines; Serine Endopeptidases; Serine Proteinase Inhibitors; Structure-Activity Relationship; Thiazoles; Viral Nonstructural Proteins | 2004 |
Cytotoxicity and sealing properties of four classes of endodontic sealers evaluated by succinic dehydrogenase activity and confocal laser scanning microscopy.
Topics: Analysis of Variance; Animals; BALB 3T3 Cells; Carbamates; Coloring Agents; Composite Resins; Dental Bonding; Dental Cements; Dental Leakage; Epoxy Resins; Fluorescent Dyes; Humans; Lipopolysaccharides; Materials Testing; Mice; Microscopy, Confocal; Polyesters; Rhodamines; Root Canal Filling Materials; Root Canal Obturation; Succinate Dehydrogenase; Surface Properties; Tetrazolium Salts; Thiazoles; Time Factors | 2004 |
Hepatitis C drug being developed.
Topics: Carbamates; Drug Resistance, Viral; Hepacivirus; Hepatitis C; Humans; Macrocyclic Compounds; Quinolines; Thiazoles; Treatment Outcome; Viral Load | 2004 |
Mutations conferring resistance to a potent hepatitis C virus serine protease inhibitor in vitro.
Topics: Amino Acid Sequence; Amino Acid Substitution; Carbamates; Cloning, Molecular; Drug Resistance, Viral; Genotype; Hepacivirus; Macrocyclic Compounds; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Phenotype; Quinolines; Replicon; RNA, Viral; Serine Proteinase Inhibitors; Thiazoles; Transcription, Genetic; Transfection; Viral Plaque Assay | 2004 |
Sensitivity of NS3 serine proteases from hepatitis C virus genotypes 2 and 3 to the inhibitor BILN 2061.
Topics: Amino Acid Sequence; Antiviral Agents; Binding Sites; Carbamates; Escherichia coli; Genotype; Hepacivirus; Humans; Kinetics; Macrocyclic Compounds; Microbial Sensitivity Tests; Models, Molecular; Molecular Sequence Data; Mutation; Quinolines; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2004 |
Synthesis of BILN 2061, an HCV NS3 protease inhibitor with proven antiviral effect in humans.
Topics: Antiviral Agents; Carbamates; Hepacivirus; Humans; Macrocyclic Compounds; Molecular Structure; Protease Inhibitors; Quinolines; Thiazoles; Viral Nonstructural Proteins | 2004 |
The design of a potent inhibitor of the hepatitis C virus NS3 protease: BILN 2061--from the NMR tube to the clinic.
Topics: Carbamates; Drug Design; Hepacivirus; Hepatitis C; Humans; In Vitro Techniques; Macrocyclic Compounds; Models, Molecular; Nuclear Magnetic Resonance, Biomolecular; Quinolines; Serine Proteinase Inhibitors; Static Electricity; Thiazoles; Viral Nonstructural Proteins | 2004 |
Hepatitis C: it's a long way to new therapy, it's a long way to go...
Topics: Antiviral Agents; Carbamates; Drug Resistance, Viral; Hepacivirus; Hepatitis C; Humans; Macrocyclic Compounds; Quinolines; Thiazoles | 2004 |
Monitoring of antifouling booster biocides in water and sediment from the port of Osaka, Japan.
Topics: Antinematodal Agents; Carbamates; Diuron; Environmental Monitoring; Geologic Sediments; Japan; Paint; Pesticide Residues; Seawater; Ships; Thiabendazole; Thiazoles; Triazines; Water Pollutants, Chemical | 2005 |
Use of placebo: is it a boon or bane?
Topics: Antiviral Agents; Carbamates; Clinical Trials as Topic; Ethics, Clinical; Hepacivirus; Hepatitis C, Chronic; Humans; Macrocyclic Compounds; Placebos; Protease Inhibitors; Quinolines; Serine Endopeptidases; Thiazoles | 2005 |
Factors affecting the efficacy of non-fumigant nematicides for controlling root-knot nematodes.
Topics: Animals; Carbamates; Larva; Nematoda; Organophosphorus Compounds; Organothiophosphorus Compounds; Ovum; Pesticide Residues; Pesticides; Seedlings; Soil; Solanum lycopersicum; Thiazoles; Thiazolidines | 2005 |
S-2474, a novel nonsteroidal anti-inflammatory drug, rescues cortical neurons from human group IIA secretory phospholipase A(2)-induced apoptosis.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Apoptosis; Carbamates; Cell Count; Cell Size; Cells, Cultured; Cerebral Cortex; Chromatin; Cyclic S-Oxides; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Group II Phospholipases A2; Humans; In Situ Nick-End Labeling; Indolizines; Neurons; Phospholipases A; Rats; Rats, Sprague-Dawley; Tetrazolium Salts; Thiazoles | 2005 |
In vitro studies of cross-resistance mutations against two hepatitis C virus serine protease inhibitors, VX-950 and BILN 2061.
Topics: Amino Acid Substitution; Amino Acids; Aspartic Acid; Binding Sites; Carbamates; Drug Resistance, Viral; Genes, Dominant; Hepacivirus; Humans; In Vitro Techniques; Inhibitory Concentration 50; Kinetics; Macrocyclic Compounds; Models, Chemical; Models, Molecular; Mutation; Oligopeptides; Quinolines; Replicon; RNA, Viral; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2005 |
High-throughput cell-based screening for hepatitis C virus NS3/4A protease inhibitors.
Topics: Alkaline Phosphatase; Antiviral Agents; Carbamates; Carrier Proteins; Cell Line; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Genes, Reporter; Green Fluorescent Proteins; Hepacivirus; Humans; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Plasmids; Quinolines; Recombinant Fusion Proteins; Scintillation Counting; Serine Proteinase Inhibitors; Thiazoles; Transfection; Viral Nonstructural Proteins; Viral Proteins | 2005 |
Inhibition of dsRNA-induced signaling in hepatitis C virus-infected cells by NS3 protease-dependent and -independent mechanisms.
Topics: Active Transport, Cell Nucleus; Carbamates; Cell Line, Tumor; Gene Expression Regulation, Viral; Hepacivirus; Humans; I-kappa B Kinase; Interferon Regulatory Factor-3; Interferon-beta; Interferon-Stimulated Gene Factor 3; Macrocyclic Compounds; Promoter Regions, Genetic; Protease Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Quinolines; Response Elements; RNA, Double-Stranded; Signal Transduction; Thiazoles; Viral Nonstructural Proteins | 2006 |
Anti-HCV therapies in chimeric scid-Alb/uPA mice parallel outcomes in human clinical application.
Topics: Analysis of Variance; Animals; Antiviral Agents; Base Sequence; Carbamates; Disease Models, Animal; Hepacivirus; Hepatitis C; Hepatitis C Antibodies; Humans; Interferon alpha-2; Interferon-alpha; Macrocyclic Compounds; Mice; Mice, SCID; Molecular Sequence Data; Oncogene Proteins, Fusion; Probability; Quinolines; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Viral; Sensitivity and Specificity; Thiazoles; Treatment Outcome | 2006 |
Convergent synthesis of the quinolone substructure of BILN 2061 via carbonylative Sonogashira coupling/cyclization.
Topics: Alkynes; Carbamates; Catalysis; Cyclization; Hydrocarbons, Iodinated; Macrocyclic Compounds; Molecular Structure; Palladium; Quinolines; Quinolones; Stereoisomerism; Thiazoles | 2006 |
In vitro activities of itraconazole, methiazole, and nitazoxanide versus Echinococcus multilocularis larvae.
Topics: Animals; Antiparasitic Agents; Benzimidazoles; Carbamates; Echinococcus multilocularis; Gerbillinae; Itraconazole; Larva; Nitro Compounds; Thiazoles | 2006 |
Antiviral interactions of an HCV polymerase inhibitor with an HCV protease inhibitor or interferon in vitro.
Topics: Antiviral Agents; Carbamates; Cell Line; Drug Synergism; Enzyme Inhibitors; Hepacivirus; Humans; Inhibitory Concentration 50; Interferon-alpha; Macrocyclic Compounds; Microbial Sensitivity Tests; Quinolines; RNA-Dependent RNA Polymerase; Serine Proteinase Inhibitors; Thiazoles | 2007 |
Efficient large-scale synthesis of BILN 2061, a potent HCV protease inhibitor, by a convergent approach based on ring-closing metathesis.
Topics: Antiviral Agents; Carbamates; Chromatography, High Pressure Liquid; Cyclization; Hepacivirus; Macrocyclic Compounds; Molecular Structure; Protease Inhibitors; Quinolines; Thiazoles | 2006 |
Novel robust hepatitis C virus mouse efficacy model.
Topics: Animals; Antiviral Agents; Carbamates; Cell Line, Tumor; Disease Models, Animal; Drug Evaluation, Preclinical; Female; Hepacivirus; Hepatitis C; Humans; Interferon-alpha; Macrocyclic Compounds; Mice; Mice, Inbred BALB C; Mice, Nude; Mice, SCID; Quinolines; Thiazoles; Virus Replication | 2006 |
Resistance of hepatitis C virus to NS3-4A protease inhibitors: mechanisms of drug resistance induced by R155Q, A156T, D168A and D168V mutations.
Topics: Binding Sites; Carbamates; Drug Resistance, Viral; Hepacivirus; Macrocyclic Compounds; Models, Molecular; Point Mutation; Quinolines; Serine Endopeptidases; Thiazoles; Viral Nonstructural Proteins | 2006 |
Synthesis and antibacterial activity of tert-butyl [1-benzyl-2[(4-aryl-2-thiazolyl)hydrazono]ethyl]carbamate derivatives.
Topics: Animals; Anti-Bacterial Agents; Artemia; Bacillus cereus; Carbamates; Enterococcus faecalis; Escherichia coli; Hydrazones; Lethal Dose 50; Microbial Sensitivity Tests; Thiazoles | 2007 |
Ultra-rapid cardiotoxicity of the hepatitis C virus protease inhibitor BILN 2061 in the urokinase-type plasminogen activator mouse.
Topics: Administration, Oral; Animals; Antiviral Agents; Carbamates; Drug Evaluation, Preclinical; Heart Diseases; Hepacivirus; Hepatitis C; Humans; Liver; Liver Transplantation; Macrocyclic Compounds; Mice; Mice, SCID; Mice, Transgenic; Mitochondria, Heart; Mitochondrial Swelling; Models, Animal; Myocytes, Cardiac; Protease Inhibitors; Quinolines; Thiazoles; Time Factors; Transplantation, Heterologous; Urokinase-Type Plasminogen Activator; Viral Load; Viral Nonstructural Proteins | 2007 |
Naturally occurring NS3-protease-inhibitor resistant mutant A156T in the liver of an untreated chronic hepatitis C patient.
Topics: Adult; Amino Acid Sequence; Base Sequence; Carbamates; DNA, Viral; Drug Resistance, Viral; Genes, Viral; Hepacivirus; Hepatitis C, Chronic; Humans; Liver; Macrocyclic Compounds; Male; Molecular Sequence Data; Oligopeptides; Point Mutation; Proline; Quinolines; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serine Endopeptidases; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2008 |
RCM macrocyclization made practical: an efficient synthesis of HCV protease inhibitor BILN 2061.
Topics: Carbamates; Cyclization; Hepacivirus; Macrocyclic Compounds; Protease Inhibitors; Quinolines; Thiazoles | 2008 |
A drug-controllable tag for visualizing newly synthesized proteins in cells and whole animals.
Topics: Animals; Carbamates; Cell Line; Drosophila melanogaster; Epitopes; Humans; Macrocyclic Compounds; Methods; Neurons; Protease Inhibitors; Protein Biosynthesis; Quinolines; Rats; Recombinant Fusion Proteins; Synapses; Thiazoles; Viral Nonstructural Proteins | 2008 |
Mapping natural polymorphisms of hepatitis C virus NS3/4A protease and antiviral resistance to inhibitors in worldwide isolates.
Topics: Amino Acid Sequence; Antiviral Agents; Carbamates; Carrier Proteins; Drug Resistance, Viral; Global Health; Hepacivirus; Hepatitis C; Humans; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Microbial Sensitivity Tests; Molecular Sequence Data; Oligopeptides; Polymorphism, Genetic; Proline; Protease Inhibitors; Quinolines; Sequence Alignment; Thiazoles; Viral Nonstructural Proteins; Viral Proteins | 2008 |
Discovery of novel potent and selective dipeptide hepatitis C virus NS3/4A serine protease inhibitors.
Topics: Administration, Oral; Animals; Antiviral Agents; Carbamates; Combinatorial Chemistry Techniques; Dogs; Liver; Macrocyclic Compounds; Molecular Structure; Quinolines; Rats; Serine Proteinase Inhibitors; Structure-Activity Relationship; Sulfonamides; Thiazoles; Viral Nonstructural Proteins | 2008 |
Bismacrocyclic inhibitors of hepatitis C NS3/4a protease.
Topics: Antiviral Agents; Carbamates; Carrier Proteins; Hepacivirus; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Protease Inhibitors; Quinolines; Structure-Activity Relationship; Thiazoles; Viral Nonstructural Proteins; Viral Proteins | 2008 |
Naturally occurring dominant resistance mutations to hepatitis C virus protease and polymerase inhibitors in treatment-naïve patients.
Topics: Antiviral Agents; Carbamates; Cohort Studies; Drug Resistance, Viral; Female; Genetic Testing; Hepacivirus; Hepatitis C; Humans; Macrocyclic Compounds; Male; Mutation; Oligopeptides; Phenylthiourea; Phylogeny; Proline; Protease Inhibitors; Quinolines; Thiazoles; Viral Load; Viral Nonstructural Proteins | 2008 |
HCV-NS3 inhibitors: determination of their kinetic parameters and mechanism.
Topics: Amino Acid Substitution; Antiviral Agents; Carbamates; Drug Resistance, Viral; Genotype; Half-Life; Hepacivirus; Humans; Kinetics; Macrocyclic Compounds; Models, Biological; Mutation; Oligopeptides; Proline; Quinolines; Recombinant Proteins; Serine Endopeptidases; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2009 |
Novel macrocyclic inhibitors of hepatitis C NS3/4A protease featuring a 2-amino-1,3-thiazole as a P4 carbamate replacement.
Topics: Animals; Carbamates; Carrier Proteins; Catalytic Domain; Dogs; Hepacivirus; Humans; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Models, Molecular; Protease Inhibitors; Rats; Thiazoles; Viral Nonstructural Proteins; Viral Proteins | 2009 |
A novel class of meso-tetrakis-porphyrin derivatives exhibits potent activities against hepatitis C virus genotype 1b replicons in vitro.
Topics: Antiviral Agents; Carbamates; Cell Line; DNA, Mitochondrial; Dose-Response Relationship, Drug; Drug Discovery; Drug Resistance, Viral; Drug Synergism; Genotype; Hepacivirus; Humans; Interferon alpha-2; Interferon-alpha; Macrocyclic Compounds; Mesoporphyrins; Quinolines; Recombinant Proteins; Replicon; RNA, Viral; Structure-Activity Relationship; Thiazoles; Viral Nonstructural Proteins | 2010 |
Protease and helicase activities of hepatitis C virus genotype 4, 5, and 6 NS3-NS4A proteins.
Topics: Amino Acid Sequence; Antiviral Agents; Carbamates; Carrier Proteins; Cloning, Molecular; DNA; Genotype; Hepacivirus; Humans; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Molecular Sequence Data; Protease Inhibitors; Quinolines; RNA; RNA Helicases; Thiazoles; Viral Nonstructural Proteins; Viral Proteins | 2010 |
Pharmacokinetics and pharmacodynamics of GS-9350: a novel pharmacokinetic enhancer without anti-HIV activity.
Topics: Adolescent; Adult; Anti-HIV Agents; Anti-Retroviral Agents; Carbamates; Cobicistat; Cohort Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Female; Humans; Isoenzymes; Male; Midazolam; Middle Aged; Pharmaceutical Preparations; Thiazoles; Young Adult | 2010 |
Estimation of inhibitory quotient using a comparative equilibrium dialysis assay for prediction of viral response to hepatitis C virus inhibitors.
Topics: Antiviral Agents; Blood Proteins; Carbamates; Cell Line; Comparative Effectiveness Research; Dialysis; Hepacivirus; Hepatitis C; Humans; Inhibitory Concentration 50; Macrocyclic Compounds; Membranes, Artificial; Oligopeptides; Phenylthiourea; Plasma; Proline; Protease Inhibitors; Protein Binding; Quinolines; RNA, Viral; Thiazoles; Viral Load | 2011 |
The resistance mutation R155K in the NS3/4A protease of hepatitis C virus also leads the virus to escape from HLA-A*68-restricted CD8 T cells.
Topics: Amino Acid Substitution; Antiviral Agents; Carbamates; Carrier Proteins; CD8-Positive T-Lymphocytes; Drug Resistance, Viral; Epitopes, T-Lymphocyte; Hepacivirus; HLA-A Antigens; Humans; Intracellular Signaling Peptides and Proteins; Macrocyclic Compounds; Mutation, Missense; Quinolines; Thiazoles; Viral Nonstructural Proteins; Viral Proteins; Virus Replication | 2010 |
Determination of biocides as well as some biocide metabolites from facade run-off waters by solid phase extraction and high performance liquid chromatographic separation and tandem mass spectrometry detection.
Topics: Acetonitriles; Carbamates; Chromatography, High Pressure Liquid; Disinfectants; Methanol; Phenylurea Compounds; Sensitivity and Specificity; Solid Phase Extraction; Styrene; Tandem Mass Spectrometry; Thiazoles; Triazines; Vinyl Compounds; Water; Water Pollutants, Chemical | 2010 |
Climate as the most important factor determining anti-fungal biocide performance in paint films.
Topics: Benzimidazoles; Biofilms; Carbamates; Cladosporium; Climate; Disinfectants; Environmental Monitoring; Environmental Pollutants; Fungi; Fungicides, Industrial; Paint; Thiazoles | 2010 |
A twenty-eight-day mechanistic time course study in the rhesus monkey with hepatitis C virus protease inhibitor BILN 2061.
Topics: Administration, Oral; Animals; Antiviral Agents; Biomarkers; Carbamates; Cardiotoxins; Drug Evaluation, Preclinical; Female; Hepacivirus; Macaca mulatta; Macrocyclic Compounds; Male; Mitochondrial Swelling; Myocytes, Cardiac; Protease Inhibitors; Quinolines; Serine Proteases; Thiazoles; Viral Nonstructural Proteins | 2011 |
Development of hepatitis C virus chimeric replicons for identifying broad spectrum NS3 protease inhibitors.
Topics: Animals; Antiviral Agents; Base Sequence; Binding Sites; Carbamates; Cell Line; Cloning, Molecular; Fluorescence Resonance Energy Transfer; Genetic Variation; Genetic Vectors; Genotype; Hepacivirus; Humans; Macrocyclic Compounds; Microbial Sensitivity Tests; Oligopeptides; Phylogeny; Protease Inhibitors; Quinolines; Replicon; Sequence Analysis, Protein; Thiazoles; Viral Nonstructural Proteins; Virus Replication | 2011 |
Comparative study of the genetic barriers and pathways towards resistance of selective inhibitors of hepatitis C virus replication.
Topics: Antiviral Agents; Carbamates; Cell Line; Drug Resistance, Viral; Hepacivirus; Humans; Macrocyclic Compounds; Mutagenesis, Site-Directed; Mutation; Oligopeptides; Phenotype; Quinolines; Replicon; Thiazoles; Transfection; Virus Replication | 2011 |
Determination of different putative allosteric binding pockets at the lutropin receptor by using diverse drug-like low molecular weight ligands.
Topics: Allosteric Site; Animals; Benzamides; Binding Sites; Carbamates; CHO Cells; Cricetinae; Ligands; Models, Molecular; Protein Binding; Protein Structure, Secondary; Pyrimidines; Receptors, LH; Terphenyl Compounds; Thiazoles; Thiophenes | 2012 |
The elvitegravir Quad pill: the first once-daily dual-target anti-HIV tablet.
Topics: Adenine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Clinical Trials as Topic; Deoxycytidine; Drug Administration Schedule; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Organophosphonates; Quinolones; Tablets; Thiazoles | 2012 |
Probing the cation binding modes of macrocyclic HCV protease inhibitor BILN 2061 by multinuclear NMR.
Topics: Antiviral Agents; Binding Sites; Carbamates; Cations; Macrocyclic Compounds; Magnetic Resonance Spectroscopy; Metals, Alkali; Metals, Alkaline Earth; Molecular Structure; Protease Inhibitors; Quinolines; Thiazoles; Transition Elements; Viral Nonstructural Proteins | 2012 |
Cobicistat boosts the intestinal absorption of transport substrates, including HIV protease inhibitors and GS-7340, in vitro.
Topics: Adenine; Alanine; Caco-2 Cells; Carbamates; Cobicistat; HIV Protease Inhibitors; Humans; Intestinal Absorption; Tenofovir; Thiazoles | 2012 |
[A single tablet against HIV: new combination preparation improves therapy].
Topics: Adenine; Alkynes; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Benzoxazines; Carbamates; CD4 Lymphocyte Count; Clinical Trials, Phase III as Topic; Cobicistat; Cyclopropanes; Deoxycytidine; Double-Blind Method; Drug Combinations; Drug Resistance, Viral; Emtricitabine; Glomerular Filtration Rate; HIV Infections; Humans; Oligopeptides; Organophosphonates; Pyridines; Quinolones; Randomized Controlled Trials as Topic; Ritonavir; Tenofovir; Thiazoles; Viral Load | 2012 |
Generic HIV drugs will widen US treatment net.
Topics: Adenine; Anti-HIV Agents; Budgets; Carbamates; Cost-Benefit Analysis; Deoxycytidine; Drug Combinations; Drug Costs; Drugs, Generic; Efavirenz, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Federal Government; Humans; Organophosphonates; Oxazines; Patents as Topic; Quinolones; Thiazoles; United States | 2012 |
FDA approves new 4-drug once-a-day HIV treatment.
Topics: Adenine; Carbamates; Cobicistat; Deoxycytidine; Drug Administration Schedule; Drug Approval; Drug Combinations; Emtricitabine; HIV Infections; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles; United States; United States Food and Drug Administration | 2012 |
A 4-drug combination (Stribild) for HIV.
Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials as Topic; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Approval; Drug Combinations; Drug Interactions; Drug Resistance, Multiple, Viral; Emtricitabine; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Tenofovir; Thiazoles; United States; United States Food and Drug Administration | 2012 |
Elvitegravir/cobicistat, mirabegron, and linaclotide.
Topics: Acetanilides; Adenine; Anti-Retroviral Agents; Carbamates; Constipation; Deoxycytidine; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; HIV-1; Humans; Organophosphonates; Peptides; Quinolones; Thiazoles; Urinary Bladder, Overactive | 2012 |
Novel HIV-1 treatment Stribild™ gains regulatory approval.
Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Thiazoles | 2012 |
Improved adherence expected with new HIV combo treatment.
Topics: Adenine; Aged; Aged, 80 and over; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Combinations; Drug Labeling; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV Infections; Humans; Medication Adherence; Middle Aged; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Thiazoles; United States | 2012 |
Drug updates and approvals: 2012 in review.
Topics: Acetanilides; Adenine; Antibodies, Monoclonal, Humanized; Benzazepines; Carbamates; Cobicistat; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; Emtricitabine; Fatty Alcohols; Humans; Mifepristone; Nicotinic Acids; Nurse Practitioners; Organophosphonates; Phosphatidylglycerols; Prednisone; Proteins; Pyrimidines; Quinolones; Ranibizumab; Tenofovir; Thiazoles; United States; United States Food and Drug Administration | 2013 |
Synthesis and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase inhibitors.
Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cell Line, Tumor; Cell Survival; Cholinesterase Inhibitors; Halogenation; Hep G2 Cells; Humans; Molecular Docking Simulation; Structure-Activity Relationship; Thiazoles | 2013 |
Boosting HIV treatment options: good news, new challenges.
Topics: Adenine; Anti-HIV Agents; Atazanavir Sulfate; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV Infections; HIV Protease Inhibitors; Humans; Male; Oligopeptides; Organophosphonates; Pyridines; Ritonavir; Tenofovir; Thiazoles | 2013 |
The pharmacokinetic and pharmacodynamic interactions between buprenorphine/naloxone and elvitegravir/cobicistat in subjects receiving chronic buprenorphine/naloxone treatment.
Topics: Adult; Anti-Retroviral Agents; Area Under Curve; Buprenorphine; Carbamates; Cobicistat; Drug Interactions; Female; HIV Infections; HIV Seronegativity; Humans; Male; Middle Aged; Naloxone; Narcotic Antagonists; Opioid-Related Disorders; Quinolones; Thiazoles | 2013 |
Cobicistat, a pharmacoenhancer for HIV treatments.
Topics: Anti-HIV Agents; Carbamates; Cobicistat; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Drug Therapy, Combination; Enzyme Inhibitors; HIV Infections; Humans; Thiazoles | 2013 |
Insecticide susceptibilities in populations of two rice planthoppers, Nilaparvata lugens and Sogatella furcifera, immigrating into Japan in the period 2005-2012.
Topics: Animals; Carbamates; Female; Hemiptera; Imidazoles; Insecticide Resistance; Insecticides; Introduced Species; Japan; Neonicotinoids; Nitro Compounds; Organothiophosphates; Oryza; Pyrazoles; Pyrethrins; Thiazoles | 2014 |
Hepatitis C viral entry inhibitors prolong viral suppression by replication inhibitors in persistently-infected Huh7 cultures.
Topics: Antiviral Agents; Carbamates; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Viral; Drug Synergism; Hepacivirus; Hepatocytes; Humans; Imidazoles; Macrocyclic Compounds; Pyrrolidines; Quinolines; Thiazoles; Time Factors; Valine; Viral Load; Virus Internalization; Virus Replication | 2013 |
tert-Butyl 1,5-bis(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)-1,5-dioxopentan-2-ylcarbamate urea/thiourea derivatives as potent H+/K(+)-ATPase inhibitors.
Topics: Animals; Anti-Ulcer Agents; Carbamates; Gastric Mucosa; Glutamic Acid; H(+)-K(+)-Exchanging ATPase; Proton Pump Inhibitors; Sheep; Thiazoles; Thiourea; Urea | 2013 |
Fused thiazolyl alkynes as potent mGlu5 receptor positive allosteric modulators.
Topics: Alkynes; Allosteric Regulation; Amides; Carbamates; Humans; Protein Binding; Receptor, Metabotropic Glutamate 5; Structure-Activity Relationship; Thiazoles | 2013 |
Evaluation of the effect of cobicistat on the in vitro renal transport and cytotoxicity potential of tenofovir.
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cell Line; Cobicistat; Drug Interactions; Humans; In Vitro Techniques; Kidney; Male; Multidrug Resistance-Associated Proteins; Organic Anion Transport Protein 1; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Organic Cation Transporter 2; Organophosphonates; Tenofovir; Thiazoles | 2013 |
[ First integrase inhibitor based single tablet regimen].
Topics: Adenine; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Deoxycytidine; Drug Approval; Drug Combinations; Emtricitabine; HIV Infections; HIV Integrase Inhibitors; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles; Treatment Outcome | 2013 |
Investigation of the interactions between methadone and elvitegravir-cobicistat in subjects receiving chronic methadone maintenance.
Topics: Adult; Anti-HIV Agents; Area Under Curve; Carbamates; Cobicistat; Drug Interactions; Female; Humans; Male; Methadone; Middle Aged; Narcotics; Opiate Substitution Treatment; Opioid-Related Disorders; Quinolones; Thiazoles | 2013 |
Cobicistat + elvitegravir + emtricitabine + tenofovir. Two new drugs, but no progress.
Topics: Acquired Immunodeficiency Syndrome; Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Therapy, Combination; Emtricitabine; HIV-1; Humans; Organophosphonates; Quinolones; Tenofovir; Thiazoles | 2013 |
Minimum costs for producing hepatitis C direct-acting antivirals for use in large-scale treatment access programs in developing countries.
Topics: Aminoisobutyric Acids; Anti-HIV Agents; Antiviral Agents; Carbamates; Developing Countries; Drug Industry; Drug Therapy, Combination; Health Services Accessibility; Hepacivirus; Hepatitis C; Heterocyclic Compounds, 3-Ring; Humans; Imidazoles; Leucine; Oligopeptides; Proline; Pyrrolidines; Quinolines; Ribavirin; Simeprevir; Sofosbuvir; Sulfonamides; Thiazoles; Uridine Monophosphate; Valine | 2014 |
Structure-activity relationships of diamine inhibitors of cytochrome P450 (CYP) 3A as novel pharmacoenhancers. Part II: P2/P3 region and discovery of cobicistat (GS-9350).
Topics: Carbamates; Cobicistat; Cytochrome P-450 CYP3A Inhibitors; Diamines; Enzyme Activation; Molecular Structure; Structure-Activity Relationship; Thiazoles | 2014 |
Accounting for strain variations and resistance mutations in the characterization of hepatitis C NS3 protease inhibitors.
Topics: Antiviral Agents; Carbamates; Cloning, Molecular; Cyclopropanes; Drug Resistance, Viral; Escherichia coli; Gene Expression; Genetic Variation; Genotype; Hepacivirus; Isoindoles; Lactams; Lactams, Macrocyclic; Macrocyclic Compounds; Mutation; Oligopeptides; Proline; Protease Inhibitors; Protein Structure, Tertiary; Quinolines; Recombinant Proteins; Sulfonamides; Thiazoles; Viral Nonstructural Proteins | 2014 |
A new stochastic model for subgenomic hepatitis C virus replication considers drug resistant mutants.
Topics: Antiviral Agents; Carbamates; Drug Resistance, Viral; Hepacivirus; Macrocyclic Compounds; Models, Statistical; Oligopeptides; Polymorphism, Single Nucleotide; Proline; Protease Inhibitors; Quinolines; Replicon; RNA, Viral; Stochastic Processes; Thiazoles; Viral Nonstructural Proteins; Virus Replication | 2014 |
Contribution of the organic anion transporter OAT2 to the renal active tubular secretion of creatinine and mechanism for serum creatinine elevations caused by cobicistat.
Topics: Animals; Biological Transport, Active; Carbamates; Cell Line; Cells, Cultured; CHO Cells; Cimetidine; Cobicistat; Creatinine; Cricetulus; Dogs; HEK293 Cells; Humans; Kidney Tubules; Kinetics; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Organic Cation Transporter 2; Recombinant Proteins; Thiazoles | 2014 |
Single-tablet, once-daily treatment regimens for HIV.
Topics: Adenine; Alkynes; Anti-HIV Agents; Benzoxazines; Carbamates; Cobicistat; Cyclopropanes; Cytochrome P-450 CYP3A Inhibitors; Deoxycytidine; Drug Combinations; Emtricitabine; HIV Infections; HIV Integrase Inhibitors; HIV Reverse Transcriptase; Humans; Nitriles; Organophosphonates; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Rilpivirine; Tenofovir; Thiazoles | 2014 |
Sustained virological response after taking crushed elvitegravir-cobicistat-emtricitabine-tenofovir tablets.
Topics: Adenine; Adult; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Organophosphonates; Powders; Quinolones; Tablets; Tenofovir; Thiazoles; Viral Load | 2014 |
Switching STRATEGIES in HIV treatment.
Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Organophosphonates; Protease Inhibitors; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Tenofovir; Thiazoles | 2014 |
Elvitegravir/cobicistat/emtricitabine/tenofovir DF in HIV-infected patients with mild-to-moderate renal impairment.
Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Cohort Studies; Deoxycytidine; Emtricitabine; Female; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Renal Insufficiency; Tenofovir; Thiazoles; Treatment Outcome | 2015 |
PI3'-kinase inhibition forestalls the onset of MEK1/2 inhibitor resistance in BRAF-mutated melanoma.
Topics: Animals; Carbamates; Cell Line, Tumor; Cell Proliferation; Humans; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Signaling System; Melanoma; Melanoma, Experimental; Mice; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; PTEN Phosphohydrolase; Random Allocation; Sulfonamides; Thiazoles | 2015 |
Game of isoforms: PI3K β-sparing inhibitor is coming.
Topics: Animals; Carbamates; Humans; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Melanoma; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Sulfonamides; Thiazoles | 2015 |
A case of iatrogenic adrenal suppression after co-administration of cobicistat and fluticasone nasal drops.
Topics: Adrenal Insufficiency; Adrenocorticotropic Hormone; Adult; Androstadienes; Carbamates; Cobicistat; Drug Interactions; Enzyme Inhibitors; Fluticasone; Humans; Hydrocortisone; Iatrogenic Disease; Male; Thiazoles | 2014 |
Drug combo beneficial in colorectal cancer.
Topics: Antibodies, Monoclonal, Humanized; Antineoplastic Combined Chemotherapy Protocols; Carbamates; Cetuximab; Colorectal Neoplasms; Humans; Sulfonamides; Thiazoles | 2015 |
Liquid Chromatographic Separation and Thermodynamic Investigation of Mirabegron Enantiomers on a Chiralpak AY-H Column.
Topics: Acetanilides; Amylose; Carbamates; Chromatography, High Pressure Liquid; Ethanol; Limit of Detection; Linear Models; Reproducibility of Results; Stereoisomerism; Thermodynamics; Thiazoles | 2015 |
Integrated pest management of "Golden Delicious" apples.
Topics: Acaricides; Biphenyl Compounds; Carbamates; Crops, Agricultural; Crosses, Genetic; European Union; Food Contamination; Food Quality; Fruit; Fungicides, Industrial; Guidelines as Topic; Humans; Insecticides; Malus; Neonicotinoids; Niacinamide; Nitro Compounds; Oxazines; Pest Control; Pesticide Residues; Pyrazoles; Pyridines; Risk Assessment; Slovenia; Strobilurins; Thiamethoxam; Thiazines; Thiazoles | 2015 |
Tenofovir alafenamide for HIV infection: is less more?
Topics: Adenine; Alanine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV Infections; Humans; Male; Organophosphonates; Quinolones; Tenofovir; Thiazoles | 2015 |
Infectious disease: New HIV-1 prodrug shows promise in phase III trials.
Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Female; HIV Infections; Humans; Male; Organophosphonates; Quinolones; Thiazoles | 2015 |
The influence of industrial and agricultural waste on water quality in the Água Boa stream (Dourados, Mato Grosso do Sul, Brazil).
Topics: Agriculture; Benzimidazoles; Brazil; Carbamates; Chlorophyll; Chlorophyll A; Drug Resistance, Bacterial; Environmental Monitoring; Escherichia coli; Humans; Industrial Waste; Industry; Metals; Neonicotinoids; Nitro Compounds; Oxazines; Pseudomonas; Rivers; Thiamethoxam; Thiazoles; Water Microbiology; Water Pollutants, Chemical; Water Pollution; Water Quality | 2015 |
N-(3,4-Dimethylisoxazol-5-yl)piperazine-4-[4-(2-fluoro-4-[(11)C]methylphenyl)thiazol-2-yl]-1-carboxamide: A promising positron emission tomography ligand for fatty acid amide hydrolase.
Topics: Amidohydrolases; Animals; Benzamides; Brain; Carbamates; Carbon Radioisotopes; Humans; Ligands; Mice; Molecular Structure; Piperazines; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Thiazoles; Tissue Distribution | 2016 |
Insecticide resistance monitoring and correlation analysis of insecticides in field populations of the brown planthopper Nilaparvata lugens (stål) in China 2012-2014.
Topics: Animals; Carbamates; China; Chlorpyrifos; Guanidines; Hemiptera; Imidazoles; Insecticide Resistance; Insecticides; Neonicotinoids; Nitro Compounds; Oxazines; Pyrazoles; Pyrethrins; Pyridines; Thiadiazines; Thiamethoxam; Thiazines; Thiazoles | 2016 |
Contact allergy to preservatives: ESSCA* results with the baseline series, 2009-2012.
Topics: Adolescent; Adult; Aged; Anti-Infective Agents; Carbamates; Dermatitis, Allergic Contact; Europe; Female; Formaldehyde; Humans; Male; Middle Aged; Nitriles; Preservatives, Pharmaceutical; Prevalence; Retrospective Studies; Thiazoles; Young Adult | 2017 |
Mixture toxicity of four commonly used pesticides at different effect levels to the epigeic earthworm, Eisenia fetida.
Topics: Animals; Carbamates; China; Chlorpyrifos; Drug Synergism; Environmental Monitoring; Guanidines; Models, Theoretical; Neonicotinoids; Oligochaeta; Pesticides; Soil Pollutants; Thiazoles; Toluidines | 2017 |
Hepatitis C virus impairs natural killer cell activity via viral serine protease NS3.
Topics: Carbamates; Cell Line; Cell Survival; Coculture Techniques; Down-Regulation; Hepacivirus; Hepatitis C; Humans; Interferon-gamma; Interleukin-12; K562 Cells; Killer Cells, Natural; Macrocyclic Compounds; Microscopy, Confocal; Natural Cytotoxicity Triggering Receptor 1; Natural Cytotoxicity Triggering Receptor 3; Quinolines; Recombinant Proteins; Serine Proteinase Inhibitors; Thiazoles; Viral Nonstructural Proteins | 2017 |
Combined effects of four pesticides and heavy metal chromium (Ⅵ) on the earthworm using avoidance behavior as an endpoint.
Topics: Animals; Avoidance Learning; Carbamates; Chlorpyrifos; Chromium; Drug Synergism; Guanidines; Metals, Heavy; Neonicotinoids; Oligochaeta; Pesticides; Soil Pollutants; Thiazoles; Toluidines | 2018 |
Topics: Amides; Antiviral Agents; Carbamates; Cell Line, Tumor; Cyclopropanes; Drug Resistance, Viral; Drug Therapy, Combination; Genotype; Hepacivirus; Hepatitis C, Chronic; Heterocyclic Compounds, 4 or More Rings; Humans; Protease Inhibitors; Pyrrolidines; Quinoxalines; Replicon; Sulfonamides; Thiazoles; Uridine; Viral Nonstructural Proteins | 2018 |
Characterization of nitenpyram resistance in Nilaparvata lugens (Stål).
Topics: Animals; Carbamates; Guanidines; Hemiptera; Insect Proteins; Insecticide Resistance; Neonicotinoids; Nitro Compounds; Pyrethrins; Pyridines; Pyrimidinones; RNA Interference; Thiazoles | 2019 |
Combined impact of pesticides and other environmental stressors on animal diversity in irrigation ponds.
Topics: Animals; Biodiversity; Carbamates; Ecosystem; Environmental Monitoring; Introduced Species; Invertebrates; Pesticides; Ponds; Thiazoles; Vertebrates | 2020 |
Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies.
Topics: Antineoplastic Agents; Carbamates; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Imidazoles; Melanoma; Molecular Dynamics Simulation; Oximes; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Quantitative Structure-Activity Relationship; Sorafenib; Sulfonamides; Thiazoles; Vemurafenib | 2020 |
Mutational profiles associated with resistance in patients with BRAFV600E mutant colorectal cancer treated with cetuximab and encorafenib +/- binimetinib or alpelisib.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzimidazoles; Biomarkers, Tumor; Carbamates; Cetuximab; Cohort Studies; Colorectal Neoplasms; DNA Mutational Analysis; Drug Resistance, Neoplasm; Female; Humans; Male; Middle Aged; Mutation; Proto-Oncogene Proteins B-raf; Retrospective Studies; Sulfonamides; Thiazoles | 2021 |
African scientists race to test COVID drugs - but face major hurdles.
Topics: Africa; Amides; Amodiaquine; Artesunate; Atazanavir Sulfate; Carbamates; Clinical Trials as Topic; COVID-19; COVID-19 Drug Treatment; COVID-19 Vaccines; Cytidine; Drug Approval; Drug Evaluation, Preclinical; Drug Repositioning; Drug Therapy, Combination; Humans; Hydroxylamines; Imidazoles; Ivermectin; Naphthyridines; Nitro Compounds; Pregnenediones; Pyrazines; Pyrrolidines; Ritonavir; Sample Size; Thiazoles; Valine; World Health Organization | 2021 |
Target enzymes in oxaliplatin-induced peripheral neuropathy in Swiss mice: A new acetylcholinesterase inhibitor as therapeutic strategy.
Topics: Adenosine Triphosphatases; Analgesics; Animals; Anxiety; Benzoates; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Cognitive Dysfunction; Disease Models, Animal; Female; Hippocampus; Indoles; Male; Mice; Oxaliplatin; Oxidative Stress; Peripheral Nervous System Diseases; Spinal Cord; Thiadiazoles; Thiazoles | 2022 |