carbamates and tacrine

carbamates has been researched along with tacrine in 47 studies

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (29.79)18.2507
2000's30 (63.83)29.6817
2010's0 (0.00)24.3611
2020's3 (6.38)2.80

Authors

AuthorsStudies
Glick, D; Loewenstein-Lichtenstein, Y; Nørgaard-Pedersen, B; Schwarz, M; Soreq, H; Zakut, H1
Dowling, MH; Paddle, BM1
Palacios, JM1
Schneider, LS2
Honma, A1
Brefel-Courbon, C; Freslon, JL; Lazartigues, E; Montastruc, JL; Pelat, M; Rascol, O; Tellioglu, T; Tran, MA1
Lacomblez, L1
Derquesné, C1
Dom, R; Lemière, J; Van Gool, D1
Kosasa, T; Kuriya, Y; Matsui, K; Yamanishi, Y2
Kosasa, T; Kuriya, Y; Yamanishi, Y1
Bejar, C; Wang, RH; Weinstock, M1
Burns, A; Page, S; Russell, E1
Stahl, SM1
Dronfield, S; Egan, K; Green, AR; Marsden, CA1
Giacobini, E1
Grutzendler, J; Morris, JC1
Kosasa, T; Kuriya, Y; Ogura, H; Yamanishi, Y1
Hake, AM1
Lampley-Dallas, VT1
Gavrilova, SI; Zharikov, GA1
Winblad, B1
Allain, H; Bentue-Ferrer, D; Lecavorzin, P; Polard, E; Reymann, JM; Tribut, O1
Klein, C; Rabey, JM; Werber, AE1
Robert, P1
Blount, PJ; McDeavitt, JT; Nguyen, CD1
Jann, MW; Shirley, KL; Small, GW1
Ott, BR1
Castro, A; Martinez, A1
Tang, XC; Zhao, Q1
Kamei, H; Nabeshima, T; Noda, Y1
Almkvist, O; Blennow, K; Hellström-Lindahl, E; Nordberg, A; Stefanova, E1
Hartmann, S; Möbius, HJ1
Albuquerque, EX; Christner, C; Fehrenbacher, A; Höffle, A; Jostock, R; Lübbert, H; Ludwig, J; Maelicke, A; Pereira, EF; Radina, M; Samochocki, M; Ullmer, C; Zerlin, M1
Gandelman-Marton, R; Klein, C; Rabey, JM; Werber, EA1
Butler, R; Prabhakaran, P; Warner, J1
Rakonczay, Z1
Fuchsberger, T; Hampel, H; Möller, HJ1
Haen, E; Ibach, B1
Darreh-Shori, T; Flores-Flores, C; Guan, ZZ; Hellström-Lindahl, E; Nordberg, A; Soreq, H1
Bagri, K; Kumar, A; Kumar, P1
Dogan, B; Durdagi, S; Ozten, O; Sonmez, F; Zengin Kurt, B1
Dolezal, R; Gorecki, L; Hepnarova, V; Hrabcova, V; Hrabinova, M; Jun, D; Korabecny, J; Kucera, T; Mezeiova, E; Muckova, L; Pejchal, J; Schmidt, M1

Reviews

19 review(s) available for carbamates and tacrine

ArticleYear
New therapeutic approaches to Alzheimer's disease.
    The Journal of clinical psychiatry, 1996, Volume: 57 Suppl 14

    Topics: Alzheimer Disease; Antioxidants; Carbamates; Cholinergic Agents; Cholinesterase Inhibitors; Cognition Disorders; Donepezil; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine; Trichlorfon

1996
[Therapeutic agents for Alzheimer's disease].
    Nihon Naika Gakkai zasshi. The Journal of the Japanese Society of Internal Medicine, 1998, Jan-10, Volume: 87, Issue:1

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Humans; Indans; Monoamine Oxidase Inhibitors; Neuropeptides; Phenylcarbamates; Piperidines; Receptor, Muscarinic M1; Receptors, Muscarinic; Rivastigmine; Spiro Compounds; Tacrine

1998
New therapeutic approaches to cognitive impairment.
    The Journal of clinical psychiatry, 1998, Volume: 59 Suppl 11

    Topics: Aged; Alzheimer Disease; Antioxidants; Carbamates; Cholinesterase Inhibitors; Cognition Disorders; Dementia; Donepezil; Humans; Indans; Monoamine Oxidase Inhibitors; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine; Trichlorfon

1998
Treatment of Alzheimer's disease: an evaluation of the cholinergic approach.
    Acta neurologica Belgica, 1999, Volume: 99, Issue:2

    Topics: Acetylcholine; Alzheimer Disease; Animals; Carbamates; Chemical and Drug Induced Liver Injury; Cholinergic Agents; Cholinergic Fibers; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Double-Blind Method; Drug Evaluation, Preclinical; Humans; Indans; Nootropic Agents; Phenylcarbamates; Piperidines; Randomized Controlled Trials as Topic; Receptors, Cholinergic; Receptors, Muscarinic; Receptors, Nicotinic; Rivastigmine; Tacrine

1999
Cholinesterase inhibitors stabilize Alzheimer's disease.
    Annals of the New York Academy of Sciences, 2000, Volume: 920

    Topics: Alzheimer Disease; Brain; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Cognition; Donepezil; Galantamine; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine; Trichlorfon

2000
Cholinesterase inhibitors for Alzheimer's disease.
    Drugs, 2001, Volume: 61, Issue:1

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Cost-Benefit Analysis; Donepezil; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

2001
Use of cholinesterase inhibitors for treatment of Alzheimer disease.
    Cleveland Clinic journal of medicine, 2001, Volume: 68, Issue:7

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Donepezil; Galantamine; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

2001
[Current strategies of pathogenetic therapy of Alzheimer's disease].
    Vestnik Rossiiskoi akademii meditsinskikh nauk, 2001, Issue:7

    Topics: Aged; Alzheimer Disease; Amino Acids; Aminoquinolines; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Dopamine Agents; Estrogens; Ginkgo biloba; Humans; Indans; Memantine; Monoamine Oxidase Inhibitors; Multicenter Studies as Topic; Neuronal Plasticity; Neuroprotective Agents; Neurotransmitter Agents; Nicergoline; Nootropic Agents; Phenylcarbamates; Phytotherapy; Piperidines; Piracetam; Pyrithioxin; Rivastigmine; Selegiline; Tacrine; Time Factors

2001
[Perspectives for drug treatment in Alzheimer's disease].
    Annales de medecine interne, 2001, Volume: 152, Issue:8

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Donepezil; Drug Therapy, Combination; Galantamine; Humans; Indans; Nootropic Agents; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

2001
Understanding and managing behavioural symptoms in Alzheimer's disease and related dementias: focus on rivastigmine.
    Current medical research and opinion, 2002, Volume: 18, Issue:3

    Topics: Acetylcholine; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Cognitive Behavioral Therapy; Disease Progression; Donepezil; Galantamine; Humans; Indans; Neuroprotective Agents; Phenylcarbamates; Physostigmine; Piperidines; Rivastigmine; Tacrine; Time Factors; Treatment Outcome

2002
Clinical use of cholinomimetic agents: a review.
    The Journal of head trauma rehabilitation, 2002, Volume: 17, Issue:4

    Topics: Administration, Oral; Adult; Aged; Alzheimer Disease; Brain Injuries; Carbamates; Clinical Trials as Topic; Cytidine Diphosphate Choline; Donepezil; Female; Follow-Up Studies; Humans; Indans; Injections, Intravenous; Injury Severity Score; Male; Middle Aged; Parasympathomimetics; Phenylcarbamates; Physostigmine; Piperidines; Rivastigmine; Severity of Illness Index; Tacrine; Treatment Outcome

2002
Clinical pharmacokinetics and pharmacodynamics of cholinesterase inhibitors.
    Clinical pharmacokinetics, 2002, Volume: 41, Issue:10

    Topics: Aging; Alzheimer Disease; Biological Availability; Carbamates; Cholinesterase Inhibitors; Donepezil; Drug Interactions; Half-Life; Humans; Indans; Intestinal Absorption; Liver; Phenylcarbamates; Piperidines; Protein Binding; Rivastigmine; Tacrine; Tissue Distribution

2002
Medical treatment of Alzheimer's disease: past, present, and future.
    Medicine and health, Rhode Island, 2002, Volume: 85, Issue:7

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Forecasting; Galantamine; Humans; Indans; Male; Phenylcarbamates; Piperidines; Prognosis; Rivastigmine; Severity of Illness Index; Tacrine; Treatment Outcome

2002
Peripheral and dual binding site acetylcholinesterase inhibitors: implications in treatment of Alzheimer's disease.
    Mini reviews in medicinal chemistry, 2001, Volume: 1, Issue:3

    Topics: Acetylcholinesterase; Aged; Alzheimer Disease; Binding Sites; Carbamates; Cholinesterase Inhibitors; Donepezil; Drug Design; Humans; Indans; Molecular Conformation; Molecular Structure; Phenylcarbamates; Piperidines; Rivastigmine; Structure-Activity Relationship; Tacrine

2001
[Anti-dementia drugs for Alzheimer disease in present and future].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2002, Volume: 120, Issue:1

    Topics: Acetylcholine; Alzheimer Disease; Amyloid beta-Peptides; Carbamates; Cholinesterase Inhibitors; Donepezil; Drug Design; Galantamine; Humans; Indans; Memantine; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine; tau Proteins

2002
Dementia.
    Clinical evidence, 2003, Issue:9

    Topics: Alzheimer Disease; Anticonvulsants; Antipsychotic Agents; Carbamates; Donepezil; Galantamine; Ginkgo biloba; Humans; Indans; Nootropic Agents; Phenylcarbamates; Phosphatidylcholines; Physostigmine; Phytotherapy; Piperidines; Rivastigmine; Tacrine; Vitamin E

2003
[Current therapy of patients with dementia].
    MMW Fortschritte der Medizin, 2003, May-26, Volume: 145 Suppl 2

    Topics: Activities of Daily Living; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Controlled Clinical Trials as Topic; Dementia; Dementia, Vascular; Donepezil; Dopamine Agents; Female; Galantamine; Ginkgo biloba; Humans; Indans; Male; Memantine; Meta-Analysis as Topic; Multicenter Studies as Topic; Neuroprotective Agents; Nootropic Agents; Phenylcarbamates; Phytotherapy; Piperidines; Placebos; Plant Preparations; Prospective Studies; Rivastigmine; Tacrine; Time Factors

2003
Acetylcholinesterase inhibition in Alzheimer's Disease.
    Current pharmaceutical design, 2004, Volume: 10, Issue:3

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Galantamine; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

2004
Computational Studies on Acetylcholinesterase Inhibitors: From Biochemistry to Chemistry.
    Mini reviews in medicinal chemistry, 2020, Volume: 20, Issue:14

    Topics: Acetylcholinesterase; Alzheimer Disease; Binding Sites; Carbamates; Cholinesterase Inhibitors; Humans; Molecular Docking Simulation; Molecular Dynamics Simulation; Quantitative Structure-Activity Relationship; Tacrine

2020

Trials

2 trial(s) available for carbamates and tacrine

ArticleYear
Cerebral glucose metabolism, cerebrospinal fluid-beta-amyloid1-42 (CSF-Abeta42), tau and apolipoprotein E genotype in long-term rivastigmine and tacrine treated Alzheimer disease (AD) patients.
    Neuroscience letters, 2003, Feb-27, Volume: 338, Issue:2

    Topics: Aged; Alzheimer Disease; Amyloid beta-Peptides; Apolipoprotein E2; Apolipoprotein E4; Apolipoproteins E; Biomarkers; Brain; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Female; Genotype; Glucose; Humans; Male; Middle Aged; Peptide Fragments; Phenylcarbamates; Rivastigmine; Tacrine; tau Proteins

2003
The clinical use of P300 event related potentials for the evaluation of cholinesterase inhibitors treatment in demented patients.
    Journal of neural transmission (Vienna, Austria : 1996), 2003, Volume: 110, Issue:6

    Topics: Acetylcholine; Aged; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Cognition Disorders; Dementia; Donepezil; Electroencephalography; Event-Related Potentials, P300; Female; Humans; Indans; Male; Middle Aged; Phenylcarbamates; Piperidines; Prospective Studies; Reaction Time; Rivastigmine; Tacrine; Treatment Outcome

2003

Other Studies

26 other study(ies) available for carbamates and tacrine

ArticleYear
Genetic predisposition to adverse consequences of anti-cholinesterases in 'atypical' BCHE carriers.
    Nature medicine, 1995, Volume: 1, Issue:10

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Butyrylthiocholine; Carbamates; Cholinesterase Inhibitors; Homozygote; Humans; Male; Pyridostigmine Bromide; Tacrine

1995
Blockade of cardiac nicotinic responses by anticholinesterases.
    General pharmacology, 1996, Volume: 27, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Carbamates; Catecholamines; Cholinesterase Inhibitors; Edrophonium; Female; Guinea Pigs; Heart; Heart Atria; Heart Rate; In Vitro Techniques; Myocardial Contraction; Nicotine; Nicotinic Antagonists; Soman; Tacrine

1996
Alzheimer's disease: new pharmacological perspectives.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18 Suppl B

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Dihydropyridines; Donepezil; Humans; Indans; Muscarinic Agonists; Oximes; Phenylcarbamates; Piperidines; Pyridines; Rivastigmine; Tacrine; Thiadiazoles

1996
Pressor and bradycardic effects of tacrine and other acetylcholinesterase inhibitors in the rat.
    European journal of pharmacology, 1998, Nov-13, Volume: 361, Issue:1

    Topics: Adrenergic Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine; Atropine Derivatives; Blood Pressure; Carbamates; Cardiovascular Agents; Chlorisondamine; Cholinergic Antagonists; Cholinesterase Inhibitors; Diamines; Diastole; Dose-Response Relationship, Drug; Heart Rate; Male; Phenylcarbamates; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Rivastigmine; Systole; Tacrine

1998
[Drug therapy strategies in Alzheimer's disease].
    La Revue du praticien, 1998, Nov-01, Volume: 48, Issue:17

    Topics: Aggression; Alzheimer Disease; Anti-Anxiety Agents; Antidepressive Agents; Antipsychotic Agents; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Cognition Disorders; Depression; Donepezil; Humans; Indans; Mental Disorders; Neuroprotective Agents; Nootropic Agents; Phenylcarbamates; Piperidines; Rivastigmine; Sleep Wake Disorders; Tacrine

1998
[Alzheimer's disease. Foreword].
    La Revue du praticien, 1998, Nov-01, Volume: 48, Issue:17

    Topics: Age Factors; Aged; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Donepezil; Humans; Indans; Neuroprotective Agents; Nootropic Agents; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

1998
Effect of donepezil hydrochloride (E2020) on basal concentration of extracellular acetylcholine in the hippocampus of rats.
    European journal of pharmacology, 1999, Sep-10, Volume: 380, Issue:2-3

    Topics: Acetylcholine; Acetylcholinesterase; Administration, Oral; Animals; Brain; Carbamates; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; Extracellular Space; Hippocampus; Indans; Male; Phenylcarbamates; Piperidines; Rats; Rats, Wistar; Rivastigmine; Tacrine

1999
Effect of donepezil hydrochloride (E2020) on extracellular acetylcholine concentration in the cerebral cortex of rats.
    Japanese journal of pharmacology, 1999, Volume: 81, Issue:2

    Topics: Animals; Benzazepines; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Chromatography, High Pressure Liquid; Donepezil; Electrochemistry; Extracellular Space; Indans; Male; Microdialysis; Nootropic Agents; Peripheral Nervous System; Phenylcarbamates; Piperidines; Rats; Rats, Wistar; Rivastigmine; Tacrine

1999
Effect of rivastigmine on scopolamine-induced memory impairment in rats.
    European journal of pharmacology, 1999, Nov-03, Volume: 383, Issue:3

    Topics: Animals; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Corpus Striatum; Drug Therapy, Combination; Hippocampus; Male; Maze Learning; Memory; Muscarinic Antagonists; Muscle, Skeletal; Phenylcarbamates; Rats; Rats, Sprague-Dawley; Rivastigmine; Scopolamine; Tacrine

1999
New drugs for Alzheimer's disease.
    The British journal of psychiatry : the journal of mental science, 1999, Volume: 174

    Topics: Alzheimer Disease; Carbamates; Donepezil; Humans; Indans; Nootropic Agents; Phenylcarbamates; Piperidines; Practice Guidelines as Topic; Rivastigmine; Tacrine

1999
Inhibitory effect of orally administered donepezil hydrochloride (E2020), a novel treatment for Alzheimer's disease, on cholinesterase activity in rats.
    European journal of pharmacology, 2000, Feb-18, Volume: 389, Issue:2-3

    Topics: Administration, Oral; Alzheimer Disease; Animals; Benzazepines; Brain; Carbamates; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; Indans; Learning; Male; Memory; Phenylcarbamates; Piperidines; Rats; Rats, Wistar; Rivastigmine; Tacrine

2000
The new cholinesterase inhibitors for Alzheimer's disease, Part 1: their similarities are different.
    The Journal of clinical psychiatry, 2000, Volume: 61, Issue:10

    Topics: Aged; Alzheimer Disease; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Donepezil; Galantamine; Humans; Indans; Phenylcarbamates; Piperidines; Receptors, Nicotinic; Rivastigmine; Tacrine

2000
Comparison of donepezil-, tacrine-, rivastigmine- and metrifonate-induced central and peripheral cholinergically mediated responses in the rat.
    Journal of psychopharmacology (Oxford, England), 2000, Volume: 14, Issue:3

    Topics: Animals; Body Temperature; Carbamates; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; Hypothermia; Indans; Lacrimal Apparatus; Male; Phenylcarbamates; Piperidines; Rats; Rivastigmine; Saliva; Tacrine; Tremor; Trichlorfon

2000
Comparison of inhibitory activities of donepezil and other cholinesterase inhibitors on acetylcholinesterase and butyrylcholinesterase in vitro.
    Methods and findings in experimental and clinical pharmacology, 2000, Volume: 22, Issue:8

    Topics: Acetylcholinesterase; Alzheimer Disease; Aminoquinolines; Animals; Benzazepines; Brain; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Donepezil; In Vitro Techniques; Indans; Inhibitory Concentration 50; Male; Phenylcarbamates; Physostigmine; Piperidines; Rats; Rivastigmine; Tacrine; Time Factors

2000
Medications for the treatment of Alzheimer's disease.
    The Journal of the Oklahoma State Medical Association, 2001, Volume: 94, Issue:8

    Topics: Alzheimer Disease; Antioxidants; Carbamates; Cholinesterase Inhibitors; Donepezil; Estrogen Replacement Therapy; Humans; Indans; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine

2001
Maintaining functional and behavioral abilities in Alzheimer disease.
    Alzheimer disease and associated disorders, 2001, Volume: 15 Suppl 1

    Topics: Aged; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Galantamine; Humans; Indans; Neuropsychological Tests; Nootropic Agents; Phenylcarbamates; Piperidines; Rivastigmine; Tacrine; Treatment Outcome

2001
Galantamine: new preparation. The fourth cholinesterase inhibitor for Alzheimer's disease.
    Prescrire international, 2001, Volume: 10, Issue:56

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; France; Galantamine; Indans; Tacrine; Treatment Outcome

2001
Evaluation of cholinergic treatment in demented patients by P300 evoked related potentials.
    Neurologia i neurochirurgia polska, 2001, Volume: 35 Suppl 3

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Analysis of Variance; Carbamates; Cholinesterase Inhibitors; Cognition; Donepezil; Evaluation Studies as Topic; Event-Related Potentials, P300; Female; Humans; Indans; Male; Middle Aged; Neuropsychological Tests; Phenylcarbamates; Piperidines; Reaction Time; Rivastigmine; Sensitivity and Specificity; Severity of Illness Index; Tacrine

2001
Effects of huperzine A on acetylcholinesterase isoforms in vitro: comparison with tacrine, donepezil, rivastigmine and physostigmine.
    European journal of pharmacology, 2002, Nov-29, Volume: 455, Issue:2-3

    Topics: Acetylcholinesterase; Alkaloids; Animals; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Corpus Striatum; Donepezil; Hippocampus; Indans; Isoenzymes; Kinetics; Male; Phenylcarbamates; Physostigmine; Piperidines; Rats; Rats, Sprague-Dawley; Rivastigmine; Sesquiterpenes; Tacrine

2002
Tolerability of memantine in combination with cholinesterase inhibitors in dementia therapy.
    International clinical psychopharmacology, 2003, Volume: 18, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Carbamates; Cholinesterase Inhibitors; Dementia; Donepezil; Dose-Response Relationship, Drug; Drug Therapy, Combination; Excitatory Amino Acid Antagonists; Humans; Indans; Memantine; Middle Aged; Phenylcarbamates; Piperidines; Product Surveillance, Postmarketing; Rivastigmine; Surveys and Questionnaires; Tacrine; Treatment Outcome

2003
Galantamine is an allosterically potentiating ligand of neuronal nicotinic but not of muscarinic acetylcholine receptors.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:3

    Topics: Allosteric Regulation; Animals; Carbamates; Cells, Cultured; Cholinesterase Inhibitors; Donepezil; Galantamine; Humans; Indans; Mice; Neurons; Phenylcarbamates; Piperidines; Receptors, Muscarinic; Receptors, Nicotinic; Recombinant Fusion Proteins; Rivastigmine; Tacrine; Trichlorfon

2003
Potencies and selectivities of inhibitors of acetylcholinesterase and its molecular forms in normal and Alzheimer's disease brain.
    Acta biologica Hungarica, 2003, Volume: 54, Issue:2

    Topics: Acetylcholinesterase; Alzheimer Disease; Benzazepines; Brain; Butyrylcholinesterase; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Edrophonium; Humans; In Vitro Techniques; Phenylcarbamates; Physostigmine; Rivastigmine; Tacrine; Trichlorfon

2003
Anticholinesterases in Alzheimer's disease: a modest effect on moderately severe disease.
    Prescrire international, 2003, Volume: 12, Issue:68

    Topics: Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; France; Galantamine; Humans; Indans; Piperidines; Product Surveillance, Postmarketing; Randomized Controlled Trials as Topic; Tacrine; Treatment Outcome

2003
Long-lasting acetylcholinesterase splice variations in anticholinesterase-treated Alzheimer's disease patients.
    Journal of neurochemistry, 2004, Volume: 88, Issue:5

    Topics: Acetylcholinesterase; Aged; Alternative Splicing; Alzheimer Disease; Blotting, Western; Carbamates; Centrifugation, Density Gradient; Cerebrospinal Fluid; Cerebrospinal Fluid Proteins; Cholinesterase Inhibitors; Cognition Disorders; Female; Humans; Isoenzymes; Male; Middle Aged; Neuroprotective Agents; Neuropsychological Tests; Parietal Lobe; Phenylcarbamates; Rivastigmine; Tacrine; Time

2004
Synthesis, molecular docking and molecular dynamics studies of novel tacrine-carbamate derivatives as potent cholinesterase inhibitors.
    Bioorganic chemistry, 2021, Volume: 115

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Structure; Structure-Activity Relationship; Tacrine

2021
Non-covalent acetylcholinesterase inhibitors: In vitro screening and molecular modeling for novel selective insecticides.
    Toxicology in vitro : an international journal published in association with BIBRA, 2022, Volume: 85

    Topics: Acetylcholinesterase; Animals; Anopheles; Butyrylcholinesterase; Carbamates; Carbofuran; Cholinesterase Inhibitors; Humans; Insecticides; Mosquito Vectors; Organophosphates; Tacrine

2022