carbamates has been researched along with physostigmine in 77 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 41 (53.25) | 18.7374 |
1990's | 13 (16.88) | 18.2507 |
2000's | 15 (19.48) | 29.6817 |
2010's | 8 (10.39) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Watts, P; Wilkinson, RG | 1 |
Dawson, RM | 2 |
Gatta, F; Marta, M; Pomponi, M | 1 |
Kuhlmann, J; Maelicke, A; Okonjo, KO | 1 |
Boddeke, H; Enz, A; Gray, J; Spiegel, R | 1 |
Anderson, DR; Harris, LW; Lennox, WJ; Solana, RP | 1 |
D'Mello, GD; Sidell, FR | 1 |
Brooks, DP; Cyronak, MJ; DePalma, PD; Karpinski, K; Weinstock, J | 1 |
Bowers, WD; Francesconi, RP; Hubbard, RW; Matthew, CB | 1 |
Arndt, H; Sprengard, M | 1 |
Levin, E; Svensson, LA; Tunek, A | 1 |
Armstrong, DM; Dokla, CP; Thal, LJ | 1 |
Dokla, CP; Thal, LJ | 1 |
Atack, JR; Brossi, A; Rapoport, SI; Yu, QS | 1 |
Albuquerque, EX; Boyne, AF; Brossi, A; Cintra, WM; Deshpande, SS; Kawabuchi, M | 1 |
Annau, Z; Mansour, NA; Shamoo, AE; Valdes, JJ | 1 |
Dawson, RM; Gray, PJ | 1 |
Inns, RH; Leadbeater, L; Rylands, JM | 1 |
Booth, GM; Connor, J; Larsen, JR; Metcalf, RA | 1 |
Stock, K; Westermann, E | 1 |
Mrsulja, BB; Terzić, M; Varagić, VM | 1 |
Pleuvry, BJ; Tobias, MA | 1 |
Czajka, M; Lièvremont, M; Tazieff-Depierre, F | 1 |
Watson, PJ | 1 |
Berry, WK; Davies, DR; Gordon, JJ | 1 |
Tegelström, H; Wahren, H | 1 |
Natoff, IL; Reiff, B | 1 |
Chiou, CY; Wecker, L | 1 |
Bajgar, J; Patocka, J | 1 |
Bentley, GA | 1 |
Kato, G | 1 |
Azmeh, N; Clark, IJ; Wenzel, DG | 1 |
Post, LC | 1 |
Wilson, EB | 1 |
Chinn, C; Weber, LJ | 1 |
Berry, WK; Davies, DR | 1 |
Hashimoto, K; Matsumura, S; Taira, N | 1 |
Winteringham, FP | 1 |
Fowler, KS; Winteringham, FP | 1 |
Overton, DA | 1 |
Benes, J; Hrusovský, J; Nistiar, F | 1 |
Green, AL | 1 |
Hayashi, E; Katsuoka, M; Okudaira, H; Yamada, S | 1 |
Harris, LW; Heyl, WC; Stitcher, DL | 1 |
Borroni, E; Da Prada, M; Damsma, G; Giovacchini, C; Jakob-Rötne, R; Mutel, V | 1 |
Das Gupta, S; Husain, K; Kumar, P; Singh, R; Vijayaraghavan, R | 1 |
Futagawa, H; Kakinuma, Y; Takahashi, H | 2 |
Brossi, A; Greig, NH; Holloway, HW; Yu, Q | 1 |
Brefel-Courbon, C; Freslon, JL; Lazartigues, E; Montastruc, JL; Pelat, M; Rascol, O; Tellioglu, T; Tran, MA | 1 |
Bejar, C; Wang, RH; Weinstock, M | 1 |
Kosasa, T; Kuriya, Y; Ogura, H; Yamanishi, Y | 1 |
Brossi, A; Flippen-Anderson, JL; Greig, NH; Hoffman, B; Holloway, HW; Yu, Q | 1 |
Robert, P | 1 |
Blount, PJ; McDeavitt, JT; Nguyen, CD | 1 |
Tang, XC; Zhao, Q | 1 |
Butler, R; Prabhakaran, P; Warner, J | 1 |
HASSON, A; LIEPIN, LL | 1 |
GOLDBERG, ME; JOHNSON, HE | 1 |
GOLDBERG, ME; JOHNSON, HE; KNAAK, JB | 1 |
DELLABELLA, D; GANDINI, A; PRETI, M | 1 |
Rakonczay, Z | 1 |
Castro, A; Martinez, A | 1 |
Eckert, S; Eyer, P; Mückter, H; Worek, F | 1 |
Alley, GM; Chen, D; Greig, NH; Lahiri, DK; Tweedie, D | 1 |
El Kharbili, M; Fekonja, O; Fournier, D; Stojan, J; Zorec-Karlovsek, M | 1 |
Dantoine, T; Debord, J; Laubarie, C | 1 |
Bumm, R; Eckert, S; Eyer, P; Herkert, NM; Thiermann, H; Weber, G; Worek, F | 1 |
Akaike, A; Fuse, S; Hijikuro, I; Kihara, T; Kunimoto, R; Murugesh, MG; Niidome, T; Okuno, Y; Sugimoto, H; Takahashi, J; Takahashi, T; Tsumura, Y | 1 |
Akaike, A; Fuse, S; Hijikuro, I; Kihara, T; Murugesh, MG; Niidome, T; Sugimoto, H; Takahashi, J; Takahashi, T; Tsumura, Y | 1 |
Joosen, MJ; Smit, AB; van Helden, HP | 1 |
Herkert, NM; Thiermann, H; Worek, F | 1 |
Bala, C; Rotariu, L; Zamfir, LG | 1 |
Beier, RC; Dong, JX; He, YS; Lai, LN; Shen, YD; Sun, YM; Wang, H; Wu, WJ; Xiao, ZL; Xie, X; Xu, ZL; Yang, JY | 1 |
Lilja, AM; Malmsten, L; Marutle, A; Nordberg, A; Ögren, SO; Röjdner, J; Verkhratsky, A; Voytenko, L | 1 |
Dehpour, AR; Moradi, A; Nikoui, V; Ostadhadi, S; Zolfaghari, S | 1 |
4 review(s) available for carbamates and physostigmine
Article | Year |
---|---|
Understanding and managing behavioural symptoms in Alzheimer's disease and related dementias: focus on rivastigmine.
Topics: Acetylcholine; Alzheimer Disease; Carbamates; Cholinesterase Inhibitors; Cognitive Behavioral Therapy; Disease Progression; Donepezil; Galantamine; Humans; Indans; Neuroprotective Agents; Phenylcarbamates; Physostigmine; Piperidines; Rivastigmine; Tacrine; Time Factors; Treatment Outcome | 2002 |
Clinical use of cholinomimetic agents: a review.
Topics: Administration, Oral; Adult; Aged; Alzheimer Disease; Brain Injuries; Carbamates; Clinical Trials as Topic; Cytidine Diphosphate Choline; Donepezil; Female; Follow-Up Studies; Humans; Indans; Injections, Intravenous; Injury Severity Score; Male; Middle Aged; Parasympathomimetics; Phenylcarbamates; Physostigmine; Piperidines; Rivastigmine; Severity of Illness Index; Tacrine; Treatment Outcome | 2002 |
Dementia.
Topics: Alzheimer Disease; Anticonvulsants; Antipsychotic Agents; Carbamates; Donepezil; Galantamine; Ginkgo biloba; Humans; Indans; Nootropic Agents; Phenylcarbamates; Phosphatidylcholines; Physostigmine; Phytotherapy; Piperidines; Rivastigmine; Tacrine; Vitamin E | 2003 |
Novel cholinesterase inhibitors as future effective drugs for the treatment of Alzheimer's disease.
Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Animals; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Clinical Trials as Topic; Drug Delivery Systems; Drug Evaluation, Preclinical; Galantamine; Humans; Physostigmine; Protein Conformation | 2006 |
1 trial(s) available for carbamates and physostigmine
Article | Year |
---|---|
Pharmacologic and clinicopharmacologic properties of SDZ ENA 713, a centrally selective acetylcholinesterase inhibitor.
Topics: Alzheimer Disease; Animals; Carbamates; Cholinesterase Inhibitors; Humans; Male; Phenylcarbamates; Physostigmine; Placebos; Rats; Rivastigmine | 1991 |
72 other study(ies) available for carbamates and physostigmine
Article | Year |
---|---|
The interaction of carbamates with acetylcholinesterase.
Topics: Acetylcholinesterase; Animals; Benzofurans; Carbachol; Carbamates; Cattle; Erythrocytes; Insecticides; Kinetics; Physostigmine; Pyridostigmine Bromide | 1977 |
Carbamylation and decarbamylation of acetylcholinesterase: effect of choline, 3,3-dimethyl-1-butanol and some allosteric effectors.
Topics: Acetylcholinesterase; Allosteric Regulation; Animals; Carbamates; Cattle; Choline; Erythrocytes; Hexanols; Kinetics; Mathematics; Physostigmine | 1978 |
Physostigmine analogs anticholinesterases: effects of the lengthening of the N-carbamic chain on the inhibition kinetics.
Topics: Animals; Carbamates; Cholinesterase Inhibitors; Enzyme Activation; Physostigmine; Protein Conformation; Structure-Activity Relationship; Substrate Specificity | 1992 |
A second pathway of activation of the Torpedo acetylcholine receptor channel.
Topics: Animals; Antibodies, Monoclonal; Binding Sites; Bungarotoxins; Carbamates; Cations; Cell Membrane; Cesium; Electric Organ; Ion Channels; Physostigmine; Quaternary Ammonium Compounds; Receptors, Nicotinic; Torpedo; Tubocurarine | 1991 |
Effects of subacute pretreatment with carbamate together with acute adjunct pretreatment against nerve agent exposure.
Topics: Animals; Carbamates; Cholinesterase Inhibitors; Female; Guinea Pigs; Lethal Dose 50; Male; Mice; Organothiophosphorus Compounds; Physostigmine; Scopolamine; Soman; Trihexyphenidyl | 1991 |
A model for carbamate and organophosphate-induced emesis in humans.
Topics: Adolescent; Adult; Animals; Atropine; Behavior, Animal; Callitrichinae; Carbamates; Cholinesterases; Disease Models, Animal; Erythrocytes; Female; Humans; Male; Organophosphorus Compounds; Physostigmine; Species Specificity; Vomiting | 1991 |
Pharmacology of SK&F R-105058 and R-106114, N-ethyl carbamate ester prodrugs of fenoldopam.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Anesthesia; Animals; Benzazepines; Biotransformation; Blood Pressure; Carbamates; Dogs; Female; Fenoldopam; Pentobarbital; Physostigmine; Prodrugs; Renal Circulation; Vascular Resistance; Vasodilator Agents | 1990 |
Chronic vs acute carbamate administration in exercising rats.
Topics: Animals; Body Temperature Regulation; Carbamates; Cholinesterase Inhibitors; Injections, Intravenous; Injections, Subcutaneous; Male; Neuromuscular Junction; Physical Conditioning, Animal; Physostigmine; Rats; Rats, Inbred Strains | 1990 |
Effects of carbamates upon various behavioural parameters in mice.
Topics: Animals; Behavior, Animal; Carbamates; Dose-Response Relationship, Drug; Double-Blind Method; Male; Mice; Motor Activity; Physostigmine; Psychomotor Performance; Pyridostigmine Bromide; Respiration | 1989 |
Hydrolysis of 3H-bambuterol, a carbamate prodrug of terbutaline, in blood from humans and laboratory animals in vitro.
Topics: Adult; Animals; Butyrylcholinesterase; Carbamates; Female; Humans; Hydrolysis; In Vitro Techniques; Kinetics; Male; Mice; Physostigmine; Prodrugs; Rabbits; Rats; Rats, Inbred Strains; Terbutaline | 1988 |
Nucleus basalis magnocellularis lesions: lack of biochemical and immunocytochemical recovery and effect of cholinesterase inhibitors on passive avoidance.
Topics: Acetylcholinesterase; Animals; Avoidance Learning; Basal Ganglia; Brain Mapping; Carbamates; Choline O-Acetyltransferase; Cholinesterase Inhibitors; Ibotenic Acid; Immunohistochemistry; Male; Phenylcarbamates; Physostigmine; Rats; Rats, Inbred F344; Substantia Innominata; Urethane | 1988 |
Effect of cholinesterase inhibitors on Morris water task behavior following lesions of the nucleus basalis magnocellularis.
Topics: Animals; Basal Ganglia; Carbamates; Cholinesterase Inhibitors; Discrimination Learning; Escape Reaction; Ibotenic Acid; Male; Motor Activity; Orientation; Phenylcarbamates; Physostigmine; Rats; Rats, Inbred F344; Reaction Time; Substantia Innominata; Urethane | 1988 |
Carbamate analogues of (-)-physostigmine: in vitro inhibition of acetyl- and butyrylcholinesterase.
Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbamates; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Electrophorus; Humans; Indoles; Physostigmine | 1988 |
Enantiomer (+)physostigmine prevents organophosphate-induced subjunctional damage at the neuromuscular synapse by a mechanism not related to cholinesterase carbamylation.
Topics: Animals; Carbamates; Cholinesterases; Dose-Response Relationship, Drug; Female; Neuromuscular Junction; Organophosphorus Compounds; Physostigmine; Rats; Rats, Inbred Strains; Sarin; Stereoisomerism; Time Factors | 1988 |
Biochemical interactions of carbamates and ecothiophate with the activated conformation of nicotinic acetylcholine receptor.
Topics: Biotransformation; Bungarotoxins; Carbamates; Echothiophate Iodide; Neostigmine; Phencyclidine; Physostigmine; Pyridostigmine Bromide; Receptors, Nicotinic | 1987 |
Kinetic constants for the inhibition of eel and rabbit brain acetylcholinesterase by some organophosphates and carbamates of military significance.
Topics: Animals; Brain; Carbamates; Chemical Warfare Agents; Cholinesterase Inhibitors; Eels; Kinetics; Neostigmine; Organophosphates; Organophosphorus Compounds; Organothiophosphorus Compounds; Physostigmine; Rabbits; Sarin; Soman | 1987 |
Treatment of poisoning by soman.
Topics: Animals; Antidotes; Atropine; Carbamates; Diazepam; Guinea Pigs; Male; Motor Activity; Organophosphate Poisoning; Parasympatholytics; Phenylpropionates; Physostigmine; Pyridostigmine Bromide; Sarin; Soman; Time Factors | 1985 |
A comparative study of the effects of selective inhibitors on esterase isozymes from the mosquito Anopheles punctipennis.
Topics: Acetates; Aldicarb; Alleles; Animals; Anopheles; Carbamates; Carbaryl; Carbofuran; Cholinesterase Inhibitors; Dichlorvos; Electrophoresis, Polyacrylamide Gel; Esterases; Fonofos; Isoenzymes; Isoflurophate; Naphthols; Organophosphorus Compounds; Paraoxon; Physostigmine; Thiocarbamates | 1973 |
[On the mechanism of action of the lipolytic effect of physostigmine].
Topics: Adipose Tissue; Animals; Blood; Carbamates; Corticosterone; Fatty Acids; Glucose; Hexobarbital; Hypophysectomy; In Vitro Techniques; Lipids; Physostigmine; Rats | 1966 |
The effect of physostigmine and Neostigmine on the concentration of glycogen in the liver of the rat.
Topics: Adrenalectomy; Animals; Atropine; Blood Glucose; Blood Pressure; Carbamates; Epinephrine; Glycogen; Guanethidine; Hexamethonium Compounds; Liver Glycogen; Male; Myocardium; Neostigmine; Phentolamine; Physostigmine; Propranolol; Rats; Reserpine; Sympathetic Nervous System | 1967 |
Comparison of the antinociceptive activities of physostigmine, oxotremorine and morphine in the mouse.
Topics: 5-Hydroxytryptophan; Analgesics; Animals; Brain Chemistry; Carbamates; Depression, Chemical; Dihydroxyphenylalanine; Dopamine; Drug Combinations; Drug Synergism; Female; Fenclonine; Hot Temperature; Male; Methyltyrosines; Mice; Morphine; Nalorphine; Naloxone; Oxotremorine; Physostigmine; Reaction Time; Reserpine; Serotonin; Stimulation, Chemical; Tremorine | 1971 |
[New method of study of substances active on neuromuscular transmission].
Topics: Acetylcholine; Acetylcholinesterase; Amino Alcohols; Ammonium Chloride; Animals; Butyrates; Calcium; Carbamates; Choline; Cholinesterase Inhibitors; Decamethonium Compounds; Diaphragm; Isoflurophate; Mice; Muscles; Neostigmine; Neuromuscular Junction; Physostigmine; Procaine; Propionates; Succinylcholine; Synaptic Transmission; Tetraethylammonium Compounds | 1968 |
Drug receptor sites in the isolated superior cervical ganglion of the rat.
Topics: Acetylcholine; Angiotensin II; Animals; Atropine; Bradykinin; Carbachol; Carbamates; Cholinesterase Inhibitors; Cholinesterases; Female; Ganglia, Autonomic; Hexamethonium Compounds; Histamine; Kinetics; Male; Mecamylamine; Methacholine Compounds; Neurons; Nicotine; Physostigmine; Pilocarpine; Piperazines; Quaternary Ammonium Compounds; Rats; Receptors, Drug; Sensory Receptor Cells; Serotonin; Sympathomimetics; Tubocurarine | 1970 |
Protection of animals against soman (1,2,2-trimethylpropyl methylphosphono-fluoridate) by pretreatment with some other organophosphorus compounds, followed by oxime and atropine.
Topics: Amitriptyline; Animals; Atropine; Bromides; Carbamates; Cholinesterase Inhibitors; Diphosphates; Drug Antagonism; Female; Fluorine; Guinea Pigs; Hydroxamic Acids; Isoflurophate; Lethal Dose 50; Nitrates; Nitrophenols; Nitroso Compounds; Organophosphonates; Organophosphorus Compounds; Orphenadrine; Oximes; Parasympatholytics; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Salicylates; Scopolamine; Species Specificity; Sulfonic Acids; Sulfuric Acids; Thiazoles; Time Factors | 1971 |
The effect of an N-methylcarbamate on esterases from snail, mouse and man studied by starch-gel electrophoresis.
Topics: Acetates; Animals; Carbamates; Electrophoresis, Starch Gel; Enzyme Activation; Esterases; Humans; Insecticides; Isoenzymes; Liver; Mice; Molluscacides; Naphthols; Physostigmine; Protein Conformation; Salicylates; Snails; Species Specificity; Structure-Activity Relationship; Xylenes | 1972 |
Effect of oximes on the acute toxicity of anticholinesterase carbamates.
Topics: Animals; Atropine; Carbamates; Cholinesterase Inhibitors; Germ-Free Life; In Vitro Techniques; Lethal Dose 50; Male; Neostigmine; Oximes; Physostigmine; Pyridinium Compounds; Rats; Rats, Inbred Strains | 1973 |
Central cholinomimetic actions of 3, 3-dimethyl-1-butanol carbamate.
Topics: Acetylcholine; Animals; Atropine; Brain; Carbamates; Carbon Isotopes; Dose-Response Relationship, Drug; Drug Interactions; Hydrolysis; In Vitro Techniques; Kinetics; Lethal Dose 50; Mice; Mice, Inbred ICR; Nerve Endings; Nicotine; Parasympathomimetics; Physostigmine; Rats; Rats, Inbred Strains; Seizures; Time Factors | 1973 |
Affinity of human brain acetylcholinesterase to some organophosphates and carbamates in vitro.
Topics: Acetylcholinesterase; Allosteric Regulation; Brain; Carbamates; Carbaryl; Caudate Nucleus; Cholinesterase Inhibitors; Humans; Isoflurophate; Malathion; Naphthalenes; Organophosphorus Compounds; Organothiophosphorus Compounds; Physostigmine; Protein Binding; Structure-Activity Relationship | 1971 |
Pharmacological studies on the hypogastric ganglion of the rat and guinea-pig.
Topics: Animals; Carbamates; Desensitization, Immunologic; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Erythrocytes; Ganglionic Stimulants; Guinea Pigs; Hypogastric Plexus; In Vitro Techniques; Ligation; Male; Methacholine Compounds; Nicotine; Perfusion; Physostigmine; Piperazines; Potassium; Quaternary Ammonium Compounds; Rats; Species Specificity; Tachyphylaxis; Vas Deferens | 1972 |
Acetylcholinesterase. I. A study by nuclear magnetic resonance of the binding of inhibitors to the enzyme.
Topics: Acetylcholinesterase; Animals; Atropine; Binding Sites; Binding, Competitive; Carbamates; Choline; Cholinesterase Inhibitors; Decapodiformes; Deuterium; Gallamine Triethiodide; Kinetics; Magnetic Resonance Spectroscopy; Mathematics; Physostigmine; Protein Binding | 1972 |
Studies on the acute and chronic depressor actions of nicotine in the rat.
Topics: Animals; Blood Pressure; Carbamates; Female; Ganglionic Stimulants; Guanethidine; Hypertension, Renal; Hypotension; Nicotine; Norepinephrine; Physostigmine; Piperazines; Pyrrolidines; Quaternary Ammonium Compounds; Rats; Tachyphylaxis; Tyramine; Vasopressins | 1971 |
Inhibition of cholinesterase by carbamates. A new kinetic approach.
Topics: Acetylcholinesterase; Animals; Carbamates; Cattle; Cholinesterase Inhibitors; Erythrocytes; Kinetics; Mathematics; Methods; Mites; Models, Biological; Physostigmine; Spectrophotometry | 1971 |
The inhibition and reactivation of acetylcholinesterase.
Topics: Acetylcholinesterase; Carbamates; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Neostigmine; Physostigmine; Quaternary Ammonium Compounds; Sulfonic Acids | 1966 |
Role of the adrenals in the pressor response to 1,1-dimethyl-4-phenylpiperazinium iodide (DMPP) in the rat.
Topics: Adrenal Medulla; Adrenalectomy; Animals; Blood Pressure; Bretylium Compounds; Carbamates; Dopamine; Epinephrine; Guanethidine; Norepinephrine; Physostigmine; Piperazines; Pyrrolidines; Quaternary Ammonium Compounds; Rats; Sympathectomy | 1970 |
The use of carbamates and atropine in the protection of animals against poisoning by 1,2,2-trimethylpropyl methylphosphonofluoridate.
Topics: Animals; Atropine; Carbamates; Chickens; Cholinesterase Inhibitors; Dogs; Esters; Female; Fluorine; Guinea Pigs; Male; Mice; Neostigmine; Organophosphate Poisoning; Organophosphonates; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Species Specificity; Time Factors | 1970 |
Excitation of the parasympathetic ganglia of the canine urinary bladder through a muscarinic mechanism.
Topics: Animals; Atropine; Carbamates; Dogs; Female; Ganglia, Autonomic; Ganglionic Stimulants; Guanethidine; Hexamethonium Compounds; Parasympathomimetics; Physostigmine; Piperazines; Quaternary Ammonium Compounds; Stimulation, Chemical; Tetraethylammonium Compounds; Tetrodotoxin; Urinary Bladder | 1971 |
Dilution effects on the measurement of blood cholinesterase inhibition by carbamates.
Topics: Carbamates; Chemical Phenomena; Chemistry; Cholinesterases; Enzymes; Humans; Insecticides; Physostigmine | 1966 |
Substrate and dilution effects on the inhibition of acetylcholinesterase by carbamates.
Topics: Acetylcholinesterase; Carbamates; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Insecticides; Kinetics; Naphthalenes; Physostigmine | 1966 |
State-dependent learning produced by depressant and atropine-like drugs.
Topics: Animals; Atropine; Avoidance Learning; Bemegride; Carbamates; Chlordiazepoxide; Chlorpromazine; Ethanol; Imipramine; Injections, Intraperitoneal; Male; Meprobamate; Pentobarbital; Phenobarbital; Physostigmine; Rats; Scopolamine; Transfer, Psychology; Urethane | 1966 |
[Use of the protozoan Tetrahymena pyriformis in testing for contamination of biological materials with organophosphates and carbamates].
Topics: Carbamates; Cholinesterase Inhibitors; Culture Media; Dichlorvos; Insecticides; Physostigmine; Tetrahymena pyriformis; Trichlorfon | 1981 |
A theoretical kinetic analysis of the protective action exerted by eserine and other carbamate anticholinesterases against poisoning by organophosphorus compounds.
Topics: Animals; Carbamates; Cholinesterase Inhibitors; Drug Resistance; Kinetics; Lethal Dose 50; Models, Biological; Organophosphate Poisoning; Organophosphorus Compounds; Physostigmine | 1983 |
A pharmacological comparison of organophosphorus and carbamate anti-cholinesterase agents on guinea pig ileum.
Topics: Animals; Carbamates; Cholinesterase Inhibitors; Guinea Pigs; Ileum; In Vitro Techniques; Isoflurophate; Male; Muscle Contraction; Muscle, Smooth; Neostigmine; Organophosphorus Compounds; Physostigmine; Radioligand Assay; Time Factors | 1982 |
The effects of pretreatments with carbamates, atropine and mecamylamine on survival and on soman-induced alterations in rat and rabbit brain acetylcholine.
Topics: Acetylcholine; Animals; Atropine; Benactyzine; Brain Chemistry; Carbamates; Male; Mecamylamine; Neostigmine; Organophosphorus Compounds; Physostigmine; Rabbits; Rats; Soman; Time Factors | 1980 |
A novel acetylcholinesterase inhibitor, Ro 46-5934, which interacts with muscarinic M2 receptors.
Topics: Acetylcholine; Alzheimer Disease; Animals; Carbamates; Cholinesterase Inhibitors; Corpus Striatum; Extracellular Space; Humans; Indoles; Muscarinic Antagonists; Physostigmine; Rats; Receptors, Muscarinic; Scopolamine | 1994 |
Rate constants of carbamylation and decarbamylation of acetylcholinesterase for physostigmine and carbaryl in the presence of an oxime.
Topics: Acetylcholinesterase; Animals; Carbamates; Carbaryl; Cattle; Homeostasis; Oximes; Physostigmine | 1994 |
Influence of pretreatment of carbamates on dynamic pulmonary mechanics in rats exposed to sarin aerosols.
Topics: Aerosols; Animals; Carbamates; Male; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Wistar; Respiratory Mechanics; Sarin | 1993 |
Cardiovascular collapse through non-cholinergic mechanism after intravenous injection of N-methylcarbamate insecticide in rabbits.
Topics: Animals; Blood Pressure; Carbamates; Cholinesterase Inhibitors; Electrocardiography; Hypertension; Injections, Intravenous; Insecticides; Male; Norepinephrine; Physostigmine; Propoxur; Rabbits; Receptors, Cholinergic; Shock, Cardiogenic | 1997 |
Syntheses and anticholinesterase activities of (3aS)-N1, N8-bisnorphenserine, (3aS)-N1,N8-bisnorphysostigmine, their antipodal isomers, and other potential metabolites of phenserine.
Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Erythrocytes; Humans; Hydrolysis; In Vitro Techniques; Indoles; Oxidation-Reduction; Phenylcarbamates; Physostigmine; Stereoisomerism; Structure-Activity Relationship | 1998 |
Pressor and bradycardic effects of tacrine and other acetylcholinesterase inhibitors in the rat.
Topics: Adrenergic Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine; Atropine Derivatives; Blood Pressure; Carbamates; Cardiovascular Agents; Chlorisondamine; Cholinergic Antagonists; Cholinesterase Inhibitors; Diamines; Diastole; Dose-Response Relationship, Drug; Heart Rate; Male; Phenylcarbamates; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Rivastigmine; Systole; Tacrine | 1998 |
Gender differences in the effect of rivastigmine on brain cholinesterase activity and cognitive function in rats.
Topics: Animals; Brain; Carbamates; Cholinesterase Inhibitors; Cholinesterases; Female; Male; Memory; Memory Disorders; Muscarinic Antagonists; Muscle, Skeletal; Myocardium; Orchiectomy; Ovariectomy; Phenylcarbamates; Physostigmine; Rats; Rats, Sprague-Dawley; Rivastigmine; Scopolamine; Sex Factors | 2000 |
The role of cholinergic and noncholinergic mechanisms in the cardiorespiratory failure produced by N-methylcarbamate cholinesterase inhibitors in rabbits.
Topics: Animals; Aorta, Thoracic; Atropine; Bronchodilator Agents; Carbamates; Cardiovascular System; Cholinesterase Inhibitors; Heart Arrest; Male; Muscle Contraction; Papillary Muscles; Physostigmine; Propoxur; Rabbits; Receptors, Cholinergic; Respiration, Artificial | 2000 |
Comparison of inhibitory activities of donepezil and other cholinesterase inhibitors on acetylcholinesterase and butyrylcholinesterase in vitro.
Topics: Acetylcholinesterase; Alzheimer Disease; Aminoquinolines; Animals; Benzazepines; Brain; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Donepezil; In Vitro Techniques; Indans; Inhibitory Concentration 50; Male; Phenylcarbamates; Physostigmine; Piperidines; Rats; Rivastigmine; Tacrine; Time Factors | 2000 |
Methyl analogues of the experimental Alzheimer drug phenserine: synthesis and structure/activity relationships for acetyl- and butyrylcholinesterase inhibitory action.
Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Crystallography, X-Ray; Erythrocytes; Humans; Models, Molecular; Molecular Conformation; Physostigmine; Structure-Activity Relationship | 2001 |
Effects of huperzine A on acetylcholinesterase isoforms in vitro: comparison with tacrine, donepezil, rivastigmine and physostigmine.
Topics: Acetylcholinesterase; Alkaloids; Animals; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Corpus Striatum; Donepezil; Hippocampus; Indans; Isoenzymes; Kinetics; Male; Phenylcarbamates; Physostigmine; Piperidines; Rats; Rats, Sprague-Dawley; Rivastigmine; Sesquiterpenes; Tacrine | 2002 |
REVERSIBLE INHIBITION OF ELECTRIC-ORGAN CHOLINESTERASE BY CURARE AND CURARE-LIKE AGENTS.
Topics: Acetylcholine; Animals; Carbamates; Choline; Cholinesterases; Curare; Decamethonium Compounds; Eels; Electric Organ; Electrophysiological Phenomena; Electrophysiology; Enzyme Inhibitors; Gallamine Triethiodide; Humans; Metabolism; Muscle Relaxants, Central; Physostigmine; Research; Succinylcholine | 1963 |
POTENTIATION OF CHLORPROMAZINE-INDUCED BEHAVIOURAL CHANGES BY ANTICHOLINESTERASE AGENTS.
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Behavior, Animal; Carbamates; Chlorpromazine; Cholinesterase Inhibitors; Cholinesterases; Enzyme Inhibitors; Pharmacology; Physostigmine; Rats; Research | 1964 |
INFLUENCE OF SKF525-A ON THE BEHAVIORAL AND ANTICHOLINESTERASE EFFECTS OF CERTAIN CARBAMATES.
Topics: Amino Acids; Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Carbamates; Cholinesterase Inhibitors; Pharmacology; Physostigmine; Proadifen; Rats; Research | 1964 |
THE MECHANISM OF THE PRESSOR RESPONSES TO PHYSOSTIGMINE IN THE RAT AND THEIR MODIFICATION BY MEBUTAMATE AND AMYLOBARBITONE.
Topics: Ammonium Compounds; Amobarbital; Animals; Antihypertensive Agents; Barbiturates; Blood Pressure; Carbamates; Cats; Electric Stimulation; Hexamethonium Compounds; Humans; Hypogastric Plexus; Male; Nicotine; Pharmacology; Physostigmine; Pilocarpine; Quaternary Ammonium Compounds; Rats; Research; Splanchnic Nerves; Spleen; Urethane; Vas Deferens | 1964 |
Potencies and selectivities of inhibitors of acetylcholinesterase and its molecular forms in normal and Alzheimer's disease brain.
Topics: Acetylcholinesterase; Alzheimer Disease; Benzazepines; Brain; Butyrylcholinesterase; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Edrophonium; Humans; In Vitro Techniques; Phenylcarbamates; Physostigmine; Rivastigmine; Tacrine; Trichlorfon | 2003 |
Kinetic analysis of the protection afforded by reversible inhibitors against irreversible inhibition of acetylcholinesterase by highly toxic organophosphorus compounds.
Topics: Acetylcholinesterase; Algorithms; Alkaloids; Carbamates; Cholinesterase Inhibitors; Cholinesterase Reactivators; Dose-Response Relationship, Drug; Erythrocytes; Humans; Kinetics; Organophosphorus Compounds; Paraoxon; Physostigmine; Pyridostigmine Bromide; Sesquiterpenes; Time Factors | 2006 |
Differential effects of two hexahydropyrroloindole carbamate-based anticholinesterase drugs on the amyloid beta protein pathway involved in Alzheimer's disease.
Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Butyrylcholinesterase; Carbamates; Cell Line; Cell Survival; Cholinesterase Inhibitors; Humans; Indoles; Molecular Structure; Neurons; Physostigmine; Pyrroles | 2007 |
Inhibition and protection of cholinesterases by methanol and ethanol.
Topics: Alcohols; Animals; Carbamates; Chemistry; Cholinesterase Inhibitors; Cholinesterases; Ethanol; Fluorides; Horses; Kinetics; Methanol; Models, Chemical; Phosphates; Phosphorylation; Physostigmine; Substrate Specificity | 2007 |
Microcalorimetric study of the inhibition of butyrylcholinesterase by carbamates.
Topics: Animals; Butyrylcholinesterase; Calorimetry; Carbamates; Cholinesterase Inhibitors; Horses; Kinetics; Neostigmine; Phenylcarbamates; Physostigmine; Rivastigmine | 2008 |
Identical kinetics of human erythrocyte and muscle acetylcholinesterase with respect to carbamate pre-treatment, residual activity upon soman challenge and spontaneous reactivation after withdrawal of the inhibitors.
Topics: Acetylcholinesterase; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Enzyme Activation; Erythrocytes; Humans; Kinetics; Muscle, Skeletal; Physostigmine; Pyridostigmine Bromide; Soman | 2008 |
Design, synthesis, evaluation and QSAR analysis of N(1)-substituted norcymserine derivatives as selective butyrylcholinesterase inhibitors.
Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Drug Design; Humans; Neuroprotective Agents; Physostigmine; Quantitative Structure-Activity Relationship | 2010 |
Design, synthesis and evaluation of carbamate-modified (-)-N(1)-phenethylnorphysostigmine derivatives as selective butyrylcholinesterase inhibitors.
Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbamates; Cholinesterase Inhibitors; Drug Design; Humans; Neuroprotective Agents; Physostigmine; Structure-Activity Relationship | 2010 |
Treatment efficacy in a soman-poisoned guinea pig model: added value of physostigmine?
Topics: Animals; Atropine; Brain; Carbamates; Chemical Warfare Agents; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Electroencephalography; Guinea Pigs; Male; Models, Animal; Obidoxime Chloride; Parasympatholytics; Physostigmine; Seizures; Soman; Time Factors; Treatment Outcome | 2011 |
In vitro kinetic interactions of pyridostigmine, physostigmine and soman with erythrocyte and muscle acetylcholinesterase from different species.
Topics: Acetylcholinesterase; Animals; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Interactions; Erythrocytes; Female; Guinea Pigs; Humans; In Vitro Techniques; Kinetics; Macaca mulatta; Male; Muscle, Skeletal; Physostigmine; Pyridostigmine Bromide; Soman; Species Specificity; Swine | 2011 |
Acetylcholinesterase biosensor for carbamate drugs based on tetrathiafulvalene-tetracyanoquinodimethane/ionic liquid conductive gels.
Topics: Acetylcholinesterase; Animals; Biosensing Techniques; Carbamates; Cholinesterase Inhibitors; Dielectric Spectroscopy; Electrophorus; Enzymes, Immobilized; Gels; Heterocyclic Compounds; Imidazoles; Ionic Liquids; Neostigmine; Nitriles; Physostigmine; Thiocholine | 2013 |
Surface display and bioactivity of Bombyx mori acetylcholinesterase on Pichia pastoris.
Topics: Acetylcholinesterase; Animals; Bombyx; Carbamates; Enzyme Activation; Organophosphorus Compounds; Physostigmine; Pichia; Recombinant Fusion Proteins; Saccharomyces cerevisiae Proteins | 2013 |
Neural Stem Cell Transplant-Induced Effect on Neurogenesis and Cognition in Alzheimer Tg2576 Mice Is Inhibited by Concomitant Treatment with Amyloid-Lowering or Cholinergic α7 Nicotinic Receptor Drugs.
Topics: alpha7 Nicotinic Acetylcholine Receptor; Alzheimer Disease; Amyloid beta-Peptides; Animals; Astrocytes; Carbamates; Cell Proliferation; Cognition; Doublecortin Protein; Female; Hippocampus; Humans; Male; Maze Learning; Memory; Mice; Nerve Regeneration; Neural Stem Cells; Neurogenesis; Nicotinic Agonists; Physostigmine; Quinuclidines; Stem Cell Transplantation | 2015 |
Cromakalim, a Potassium Channel Opener, Ameliorates the Organophosphate and Carbamate-Induced Seizure in Mice.
Topics: Animals; Anticonvulsants; Carbamates; Cromakalim; Dichlorvos; Dose-Response Relationship, Drug; Glyburide; Male; Mice; Organophosphate Poisoning; Physostigmine; Potassium Channels; Seizures | 2018 |