carbamates and mjn110

carbamates has been researched along with mjn110 in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's11 (68.75)24.3611
2020's5 (31.25)2.80

Authors

AuthorsStudies
Buczynski, MW; Burston, JJ; Byrne, F; Chang, JW; Chapman, V; Cognetta, AB; Cravatt, BF; Niphakis, MJ; Parsons, LH1
Abdullah, RA; Cravatt, BF; Downey, R; Lichtman, AH; Limebeer, CL; Morris, H; Niphakis, MJ; Parker, LA; Rock, EM; Sticht, MA1
Abdullah, R; Cravatt, BF; Ignatowska-Jankowska, B; Lichtman, AH; Mustafa, M; Niphakis, M; Wiley, JL; Wilkerson, JL1
Cravatt, BF; Limebeer, CL; Millett, G; Niphakis, MJ; Parker, LA; Petrie, GN; Rock, EM; Wills, KL1
Abdullah, RA; Akbarali, H; Banks, ML; Cravatt, BF; Dewey, WL; Grim, TW; Lichtman, AH; Mustafa, MA; Niphakis, MJ; Poklis, JL; Wilkerson, JL; Wise, LE1
Berdan, CA; Burritt, NE; Corkey, BE; Deeney, JT; Erion, KA1
Finn, DP; Flannery, LE; Henry, RJ; Kerr, DM; Roche, M1
Bland, ST; Fontenot, J; Ishiki, M; Loetz, EC1
Arai, AL; Choi, SH; Hallenbeck, J; Kang, B; Mou, Y; Silva, AC; Yen, CC1
Cavin, JB; Cravatt, BF; Hill, MN; Keenan, CM; Lau, DJ; Makriyannis, A; Morena, M; Sharkey, KA; Sticht, MA; Vemuri, VK1
Brouillet, A; Chokr, D; Cravatt, BF; Guillou, H; Habib, A; Hegde, P; Le Faouder, P; Le Gall, M; Lettéron, P; Lotersztajn, S; Mabire, M; Mansouri, A; Moreau, R; Pilard, N; Ribeiro-Parenti, L; Siebert, M; Tardelli, M; Trauner, M; Wan, J; Weiss, E1
Baindur, AN; Bass, CE; Cravatt, BF; Feja, M; Leigh, MPK; McGraw, JJ; Wakabayashi, KT1
Cancienne, HL; Edwards, S; Fucich, EA; Gilpin, NW; Middleton, JW; Molina, PE; Stielper, ZF1
BassiriRad, N; Ciccone, HA; Cravatt, BF; Grenald, SA; Largent-Milnes, TM; Niphakis, MJ; Thompson, AL; Vanderah, TW1
Burrell, BD; Kabeiseman, E; Paulsen, R1
Selvaraj, P; Tanaka, M; Wen, J; Zhang, Y1

Other Studies

16 other study(ies) available for carbamates and mjn110

ArticleYear
Evaluation of NHS carbamates as a potent and selective class of endocannabinoid hydrolase inhibitors.
    ACS chemical neuroscience, 2013, Sep-18, Volume: 4, Issue:9

    Topics: Amidohydrolases; Animals; Blood Glucose; Brain; Carbamates; Diabetes Mellitus, Type 2; Diabetic Neuropathies; Drug Evaluation, Preclinical; Endocannabinoids; HEK293 Cells; Humans; Hyperalgesia; Insulin; Liver; Male; Mice; Molecular Structure; Monoacylglycerol Lipases; Nociception; Rats; Rats, Sprague-Dawley; Species Specificity; Structure-Activity Relationship; Succinimides

2013
Effect of selective inhibition of monoacylglycerol lipase (MAGL) on acute nausea, anticipatory nausea, and vomiting in rats and Suncus murinus.
    Psychopharmacology, 2015, Volume: 232, Issue:3

    Topics: Animals; Carbamates; Disease Models, Animal; Female; Male; Monoacylglycerol Lipases; Nausea; Rats; Rats, Sprague-Dawley; Shrews; Succinimides; Vomiting

2015
Selective monoacylglycerol lipase inhibitors: antinociceptive versus cannabimimetic effects in mice.
    The Journal of pharmacology and experimental therapeutics, 2015, Volume: 353, Issue:2

    Topics: Analgesics; Animals; Benzodioxoles; Biomimetic Materials; Brain; Cannabinoids; Carbamates; Constriction; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Motor Activity; Neuralgia; Piperidines; Succinimides

2015
Double Dissociation of Monoacylglycerol Lipase Inhibition and CB1 Antagonism in the Central Amygdala, Basolateral Amygdala, and the Interoceptive Insular Cortex on the Affective Properties of Acute Naloxone-Precipitated Morphine Withdrawal in Rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2016, Volume: 41, Issue:7

    Topics: Amygdala; Analysis of Variance; Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Carbamates; Cerebral Cortex; Conditioning, Operant; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Endocannabinoids; Glycerides; Male; Monoacylglycerol Lipases; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Succinimides

2016
The Selective Monoacylglycerol Lipase Inhibitor MJN110 Produces Opioid-Sparing Effects in a Mouse Neuropathic Pain Model.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Analgesics, Opioid; Animals; Arachidonic Acids; Behavior, Animal; Carbamates; Constriction, Pathologic; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Morphine; Neuralgia; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid, mu; Succinimides

2016
Inhibition of Monoacylglycerol Lipase Activity Decreases Glucose-Stimulated Insulin Secretion in INS-1 (832/13) Cells and Rat Islets.
    PloS one, 2016, Volume: 11, Issue:2

    Topics: Animals; Benzodioxoles; Biphenyl Compounds; Calcium; Carbamates; Cell Line; Fatty Acids; Fatty Acids, Nonesterified; Glucose; Glycerol; Insulin; Insulin Secretion; Insulin-Secreting Cells; Islets of Langerhans; Kinetics; Lipids; Lipolysis; Male; Monoacylglycerol Lipases; Phospholipids; Piperidines; Rats; Rats, Sprague-Dawley; Succinimides

2016
FAAH, but not MAGL, inhibition modulates acute TLR3-induced neuroimmune signaling in the rat, independent of sex.
    Journal of neuroscience research, 2018, Volume: 96, Issue:6

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acids; Body Temperature; Carbamates; Chemokine CXCL10; Corticosterone; Endocannabinoids; Estradiol; Ethanolamines; Female; Glycerides; Immunologic Factors; Interferons; Male; Monoacylglycerol Lipases; NF-kappa B; Oleic Acids; Palmitic Acids; Poly I-C; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Sex Factors; Signal Transduction; Succinimides; Toll-Like Receptor 3

2018
Monoacylglycerol lipase inhibition alters social behavior in male and female rats after post-weaning social isolation.
    Behavioural brain research, 2018, 04-02, Volume: 341

    Topics: Animals; Carbamates; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Grooming; Male; Monoacylglycerol Lipases; Motor Activity; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Random Allocation; Rats, Sprague-Dawley; Sex Characteristics; Social Behavior; Social Isolation; Succinimides; Weaning

2018
Neuroprotective Effects of MAGL (Monoacylglycerol Lipase) Inhibitors in Experimental Ischemic Stroke.
    Stroke, 2018, Volume: 49, Issue:3

    Topics: Animals; Benzodioxoles; Brain Ischemia; Carbamates; Disease Models, Animal; Enzyme Inhibitors; Male; Monoacylglycerol Lipases; Neuroprotective Agents; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Stroke; Succinimides

2018
Endocannabinoid regulation of homeostatic feeding and stress-induced alterations in food intake in male rats.
    British journal of pharmacology, 2019, Volume: 176, Issue:10

    Topics: Amidohydrolases; Animals; Anorexia; Arachidonic Acids; Carbamates; Duodenum; Eating; Endocannabinoids; Glycerides; Homeostasis; Jejunum; Male; Monoacylglycerol Lipases; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Stress, Psychological; Succinimides

2019
Inhibition of monoacylglycerol lipase, an anti-inflammatory and antifibrogenic strategy in the liver.
    Gut, 2019, Volume: 68, Issue:3

    Topics: Animals; Anti-Inflammatory Agents; Autophagy; Carbamates; Carbon Tetrachloride; Cell Count; Cells, Cultured; Cytokines; Disease Progression; Drug Evaluation, Preclinical; Hydrolases; Inflammation Mediators; Liver; Liver Cirrhosis, Experimental; Macrophages; Male; Mice, Inbred C57BL; Mice, Knockout; Molecular Targeted Therapy; Monoacylglycerol Lipases; Receptor, Cannabinoid, CB2; Succinimides

2019
The novel MAGL inhibitor MJN110 enhances responding to reward-predictive incentive cues by activation of CB1 receptors.
    Neuropharmacology, 2020, 01-01, Volume: 162

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Carbamates; Conditioning, Operant; Cues; Dopaminergic Neurons; Endocannabinoids; GABAergic Neurons; Glycerides; Male; Monoacylglycerol Lipases; Motivation; Neural Inhibition; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Reward; Rimonabant; Succinimides; Sucrose; Ventral Tegmental Area

2020
Endocannabinoid degradation inhibitors ameliorate neuronal and synaptic alterations following traumatic brain injury.
    Journal of neurophysiology, 2020, 02-01, Volume: 123, Issue:2

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Brain Injuries, Traumatic; Carbamates; Electrophysiological Phenomena; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Machine Learning; Male; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyramidal Cells; Rats; Rats, Wistar; Sensorimotor Cortex; Succinimides

2020
The Endocannabinoid System Alleviates Pain in a Murine Model of Cancer-Induced Bone Pain.
    The Journal of pharmacology and experimental therapeutics, 2020, Volume: 373, Issue:2

    Topics: Animals; Bone Neoplasms; Cancer Pain; Carbamates; Cell Line, Tumor; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Female; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Succinimides

2020
Characterization of a monoacylglycerol lipase in the medicinal leech, Hirudo verbana.
    Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology, 2020, Volume: 243-244

    Topics: Animals; Benzodioxoles; Carbamates; Cell Membrane; Cloning, Molecular; Endocannabinoids; Enzyme Inhibitors; HEK293 Cells; Humans; Leeches; Monoacylglycerol Lipases; Phylogeny; Piperidines; Succinimides

2020
The Novel Monoacylglycerol Lipase Inhibitor MJN110 Suppresses Neuroinflammation, Normalizes Synaptic Composition and Improves Behavioral Performance in the Repetitive Traumatic Brain Injury Mouse Model.
    Cells, 2021, 12-08, Volume: 10, Issue:12

    Topics: Animals; Behavior, Animal; Brain Injuries, Traumatic; Carbamates; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Gene Expression Regulation; Humans; Mice; Monoacylglycerol Lipases; Neuroinflammatory Diseases; Neurons; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Succinimides; Synapses

2021