carbamates and jzl195

carbamates has been researched along with jzl195 in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (5.26)29.6817
2010's15 (78.95)24.3611
2020's3 (15.79)2.80

Authors

AuthorsStudies
Booker, L; Burston, JJ; Cravatt, BF; Jin, X; Lichtman, AH; Long, JZ; Nomura, DK; Sim-Selley, LJ; Vann, RE; Walentiny, DM; Wiley, JL1
Abdullah, RA; Imhof, E; Lichtman, AH; Limebeer, CL; Parker, LA; Rock, EM; Wang, K1
Anderson, WB; Gould, MJ; Mitchell, VA; Torres, RD; Vaughan, CW1
Dominguez Aguilar, D; Giuffrida, A; Seillier, A1
Bachovchin, DA; Bachovchin, WW; DiMare, M; Golub, TR; Healey, SE; Kiritsy, CP; Koblan, LW; Lai, JH; Li, Y; Liu, Y; Munford, RS; Poplawski, SE; Sanford, DG; Shu, Y; Woznica, I; Wu, W; Zhao, P1
Belluomo, I; Chaouloff, F; Marsicano, G; Matias, I; Pernègre, C1
Vann, RE; Walentiny, DM; Wiley, JL1
Bagci, S; Dogrul, A; Gulsen, M; Ilkaya, F; Sakin, YS; Seyrek, M; Ulas, UH1
Campolongo, P; Cuomo, V; Hill, MN; Manduca, A; Morena, M; Palmery, M; Servadio, M; Trabace, L; Trezza, V; Vanderschuren, LJ1
Adamson Barnes, NS; Kazantzis, NP; Mitchell, VA; Vaughan, CW1
Abdullah, RA; Cravatt, BF; Ho, W; Lichtman, AH; Limebeer, CL; Niphakis, MJ; Parker, LA; Poklis, JL; Rafla, BR; Sharkey, KA; Sticht, MA1
Akar, A; Cayirli, M; Dogrul, A; Sakin, YS; Seyrek, M; Yesilyurt, O1
Amin, R; Andrews, MJ; Czyzyk, TA; Davis, BJ; Haskins, CP; Henderson-Redmond, AN; Mackie, K; Marcus, DJ; Morgan, DJ; Zee, ML1
Crews, FT; Grant, ML; Jones, VM; Khatri, D; Laroche, G; Mukhopadhyay, S; Vetreno, RP1
Dong, H; Han, J; Higashimori, H; Liu, J; Tong, L; Wang, F; Wang, J; Xiong, L; Yang, Y; Zhang, X1
Bedse, G; Bluett, RJ; Gaulden, AD; Kingsley, PJ; Marnett, LJ; Patel, S; Patrick, TA; Plath, N; Romness, NK1
Arango, V; Bakalian, MJ; Cooper, TB; Dong, B; Goyal, A; Mann, JJ; Shah, R; Shilpa, BM; Suckow, RF; Vinod, KY; Xie, S1
Cancienne, HL; Edwards, S; Fucich, EA; Gilpin, NW; Middleton, JW; Molina, PE; Stielper, ZF1
Demartini, C; Francavilla, M; Greco, R; Tassorelli, C; Zanaboni, AM1

Other Studies

19 other study(ies) available for carbamates and jzl195

ArticleYear
Dual blockade of FAAH and MAGL identifies behavioral processes regulated by endocannabinoid crosstalk in vivo.
    Proceedings of the National Academy of Sciences of the United States of America, 2009, Dec-01, Volume: 106, Issue:48

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Carbamates; Carboxylic Ester Hydrolases; Endocannabinoids; Glycerides; Mice; Molecular Structure; Monoacylglycerol Lipases; Motor Activity; Pain Measurement; Piperazines; Piperidines; Polyunsaturated Alkamides

2009
Attenuation of anticipatory nausea in a rat model of contextually elicited conditioned gaping by enhancement of the endocannabinoid system.
    Psychopharmacology, 2014, Volume: 231, Issue:3

    Topics: Amidohydrolases; Animals; Anticipation, Psychological; Arachidonic Acids; Brain; Cannabinoid Receptor Antagonists; Carbamates; Endocannabinoids; Enzyme Inhibitors; Glycerides; Indoles; Lithium Chloride; Male; Monoacylglycerol Lipases; Motor Activity; Nausea; Oleic Acids; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant

2014
Actions of the dual FAAH/MAGL inhibitor JZL195 in a murine inflammatory pain model.
    Neuropharmacology, 2014, Volume: 81

    Topics: Amidohydrolases; Analgesics; Analysis of Variance; Animals; Arthritis, Experimental; Benzamides; Benzoxazines; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Morpholines; Motor Activity; Naphthalenes; Pain; Pain Measurement; Piperazines; Piperidines; Pyrazoles; Time Factors

2014
The dual FAAH/MAGL inhibitor JZL195 has enhanced effects on endocannabinoid transmission and motor behavior in rats as compared to those of the MAGL inhibitor JZL184.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 124

    Topics: Animals; Anti-Anxiety Agents; Benzodioxoles; Carbamates; Endocannabinoids; Male; Motor Activity; Piperazines; Piperidines; Rats; Rats, Wistar

2014
A high-throughput, multiplexed assay for superfamily-wide profiling of enzyme activity.
    Nature chemical biology, 2014, Volume: 10, Issue:8

    Topics: Animals; Boronic Acids; Carbamates; Carboxylic Ester Hydrolases; Dipeptidyl-Peptidase IV Inhibitors; Drug Discovery; Enzyme Inhibitors; Female; Glucose Tolerance Test; Glutamates; High-Throughput Screening Assays; Humans; Lipopolysaccharides; Macaca fascicularis; Male; Mice, Inbred C57BL; Nitriles; Oligopeptides; Piperazines; Proline; Serine Proteases; Serine Proteinase Inhibitors

2014
Opposite control of frontocortical 2-arachidonoylglycerol turnover rate by cannabinoid type-1 receptors located on glutamatergic neurons and on astrocytes.
    Journal of neurochemistry, 2015, Volume: 133, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Astrocytes; Carbamates; Endocannabinoids; Enzyme Inhibitors; Glutamic Acid; Glycerides; Hippocampus; Kinetics; Male; Mice; Mice, Knockout; Neurons; Piperazines; Prefrontal Cortex; Receptor, Cannabinoid, CB1

2015
Phenotypic assessment of THC discriminative stimulus properties in fatty acid amide hydrolase knockout and wildtype mice.
    Neuropharmacology, 2015, Volume: 93

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzodioxoles; Brain; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Mice; Mice, Knockout; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rimonabant

2015
The effect of FAAH, MAGL, and Dual FAAH/MAGL inhibition on inflammatory and colorectal distension-induced visceral pain models in Rodents.
    Neurogastroenterology and motility, 2015, Volume: 27, Issue:7

    Topics: Amidohydrolases; Animals; Benzodioxoles; Carbamates; Colon; Cyclohexanols; Inflammation; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Pain Measurement; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Visceral Pain

2015
Distinct roles of the endocannabinoids anandamide and 2-arachidonoylglycerol in social behavior and emotionality at different developmental ages in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2015, Volume: 25, Issue:8

    Topics: Aging; Animals; Anxiety; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Exploratory Behavior; Glycerides; Male; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Rimonabant; Social Behavior

2015
Actions of the dual FAAH/MAGL inhibitor JZL195 in a murine neuropathic pain model.
    British journal of pharmacology, 2016, Volume: 173, Issue:1

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Benzoxazines; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Hyperalgesia; Male; Mice; Monoacylglycerol Lipases; Morpholines; Naphthalenes; Neuralgia; Piperazines; Piperidines

2016
Endocannabinoid regulation of nausea is mediated by 2-arachidonoylglycerol (2-AG) in the rat visceral insular cortex.
    Neuropharmacology, 2016, Volume: 102

    Topics: Animals; Arachidonic Acids; Carbamates; Cerebral Cortex; Endocannabinoids; Glycerides; Nausea; Neurons; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Receptor, Cannabinoid, CB1

2016
Systemic and spinal administration of FAAH, MAGL inhibitors and dual FAAH/MAGL inhibitors produce antipruritic effect in mice.
    Archives of dermatological research, 2016, Volume: 308, Issue:5

    Topics: Amidohydrolases; Animals; Antipruritics; Benzodioxoles; Carbamates; Disease Models, Animal; Endocannabinoids; Injections, Intraperitoneal; Injections, Spinal; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Piperazines; Piperidines; Pruritus; Pyridines; Serotonin

2016
Mice Expressing a "Hyper-Sensitive" Form of the Cannabinoid Receptor 1 (CB1) Are Neither Obese Nor Diabetic.
    PloS one, 2016, Volume: 11, Issue:8

    Topics: Amino Acid Substitution; Animals; Body Weight; Carbamates; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Dronabinol; Eating; Glucose Tolerance Test; Male; Mice, Mutant Strains; Obesity; Piperazines; Receptor, Cannabinoid, CB1

2016
Acute Ethanol Inhibition of Adult Hippocampal Neurogenesis Involves CB1 Cannabinoid Receptor Signaling.
    Alcoholism, clinical and experimental research, 2018, Volume: 42, Issue:4

    Topics: Animals; Binge Drinking; Cannabinoids; Carbamates; Caspase 3; Cell Death; Cell Proliferation; Doublecortin Domain Proteins; Doublecortin Protein; Drug Interactions; Endocannabinoids; Ethanol; Hippocampus; Ki-67 Antigen; Male; Microtubule-Associated Proteins; Neurogenesis; Neuropeptides; Piperazines; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant

2018
Long-term depression induced by endogenous cannabinoids produces neuroprotection via astroglial CB
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2019, Volume: 39, Issue:6

    Topics: Animals; Astrocytes; Cannabinoids; Carbamates; Long-Term Synaptic Depression; Mice; Neuroprotection; Piperazines; Receptor, Cannabinoid, CB1; Receptors, Glutamate; Rodentia; Stroke

2019
Therapeutic endocannabinoid augmentation for mood and anxiety disorders: comparative profiling of FAAH, MAGL and dual inhibitors.
    Translational psychiatry, 2018, 04-26, Volume: 8, Issue:1

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Behavior, Animal; Benzodioxoles; Body Temperature; Brain; Carbamates; Endocannabinoids; Female; Locomotion; Male; Maze Learning; Mice, Inbred C57BL; Mice, Inbred ICR; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyridines; Stress, Psychological

2018
Dual pharmacological inhibitor of endocannabinoid degrading enzymes reduces depressive-like behavior in female rats.
    Journal of psychiatric research, 2020, Volume: 120

    Topics: Amidohydrolases; Animals; Behavior, Animal; Brain-Derived Neurotrophic Factor; Carbamates; Depression; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Female; Monoacylglycerol Lipases; Piperazines; Rats; Rats, Inbred WKY; Signal Transduction; Ventral Striatum

2020
Endocannabinoid degradation inhibitors ameliorate neuronal and synaptic alterations following traumatic brain injury.
    Journal of neurophysiology, 2020, 02-01, Volume: 123, Issue:2

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Brain Injuries, Traumatic; Carbamates; Electrophysiological Phenomena; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Machine Learning; Male; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyramidal Cells; Rats; Rats, Wistar; Sensorimotor Cortex; Succinimides

2020
Dual Inhibition of FAAH and MAGL Counteracts Migraine-like Pain and Behavior in an Animal Model of Migraine.
    Cells, 2021, 09-26, Volume: 10, Issue:10

    Topics: Animals; Behavior, Animal; Carbamates; Disease Models, Animal; Endocannabinoids; Hyperalgesia; Male; Migraine Disorders; Pain; Piperazines; Rats, Sprague-Dawley

2021