carbamates and jzl 184

carbamates has been researched along with jzl 184 in 41 studies

Research

Studies (41)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (7.32)29.6817
2010's34 (82.93)24.3611
2020's4 (9.76)2.80

Authors

AuthorsStudies
Abdullah, RA; Carlson, BL; Cravatt, BF; Lichtman, AH; Long, JZ; Ramesh, D; Schlosburg, JE1
Abdullah, RA; Boger, DL; Cravatt, BF; Kinsey, SG; Lichtman, AH; Long, JZ; O'Neal, ST; Poklis, JL1
Cravatt, BF; Hillard, CJ; Liu, QS; Long, JZ; Pan, B; Sun, D; Wang, W1
Holtfrerich, A; Lehr, M; Makharadze, T1
Guindon, J; Hohmann, AG; Spradley, JM1
Busquets-Garcia, A; de la Torre, R; Maldonado, R; Ozaita, A; Pastor, A; Puighermanal, E1
Alhamoruni, A; Larvin, M; O'Sullivan, SE; Wright, KL1
Baldeyroux, B; Hamtiaux, L; Lambert, DM; Lansiaux, A; Matuszak, N; Muccioli, GG; Poupaert, JH1
Bittles, V; Borazjani, A; Crow, JA; Potter, PM; Ross, MK1
Bradshaw, HB; Guindon, J; Hohmann, AG; Lai, Y; Takacs, SM1
Chavant, F; Duranti, A; Francheteau, M; Gennequin, B; Maccarrone, M; Makriyannis, A; Nader, J; Rapino, C; Solinas, M; Thiriet, N1
Dominguez Aguilar, D; Giuffrida, A; Seillier, A1
Gunduz, O; Tosun, NC; Ulugol, A1
Bader, M; Brosnihan, KB; Dechend, R; Howlett, AC; McGee, CM; Pulgar, VM; Varagic, J; Yamaleyeva, LM1
Drew, GM; Lau, BK; Mitchell, VA; Vaughan, CW1
Bindila, L; Hoheisel, U; Lerner, R; Lomazzo, E; Lutz, B; Remmers, F; Schwitter, C1
Bernal-Chico, A; Canedo, M; Manterola, A; Mato, S; Matute, C; Pérez-Samartín, A; Rodríguez-Puertas, R; Victoria Sánchez-Gómez, M1
Impastato, RA; Katz, PS; Molina, PE; Rogers, EK; Sulzer, JK; Teng, SX1
Cravatt, BF; Damaj, MI; Gamage, TF; Ignatowska-Jankowska, BM; Lichtman, AH; Muldoon, PP1
Vann, RE; Walentiny, DM; Wiley, JL1
Abdullah, R; Cravatt, BF; Ignatowska-Jankowska, B; Lichtman, AH; Mustafa, M; Niphakis, M; Wiley, JL; Wilkerson, JL1
Bagci, S; Dogrul, A; Gulsen, M; Ilkaya, F; Sakin, YS; Seyrek, M; Ulas, UH1
Adamson Barnes, NS; Kazantzis, NP; Mitchell, VA; Vaughan, CW1
Berdan, CA; Burritt, NE; Corkey, BE; Deeney, JT; Erion, KA1
Akar, A; Cayirli, M; Dogrul, A; Sakin, YS; Seyrek, M; Yesilyurt, O1
Benini, R; Costa-Ferreira, W; Crestani, CC; Gomes-de-Souza, L; Oliveira, LA; Rodella, P1
Alves-Silva, J; Batista, EM; Doria, JG; Ferguson, SS; Ferreira-Vieira, TH; Moreira, FA; Ribeiro, FM1
Barrett, DA; Couch, DG; Karwad, MA; Larvin, M; Lund, JN; O'Sullivan, SE; Sarmad, S; Theophilidou, E; Wright, KL1
Genewsky, A; Heinz, DE; Wotjak, CT1
Giuffrida, A; Seillier, A1
Berardi, A; Campolongo, P; Colucci, P; Hill, MN; Morena, M; Palmery, M; Trezza, V1
Fehér, Á; Gyertyán, I; Gyires, K; Németh, J; Tóth, VE; Zádori, ZS1
Arai, AL; Choi, SH; Hallenbeck, J; Kang, B; Mou, Y; Silva, AC; Yen, CC1
Bedse, G; Bluett, RJ; Gaulden, AD; Kingsley, PJ; Marnett, LJ; Patel, S; Patrick, TA; Plath, N; Romness, NK1
Aliczki, M; Balogh, Z; Biro, L; Haller, J; Szente, L; Varga, ZK1
Fukumori, R; Nawata, Y; Yamaguchi, T; Yamamoto, T1
Banaszkiewicz, I; Biala, G; Kruk-Slomka, M; Slomka, T1
Cancienne, HL; Edwards, S; Fucich, EA; Gilpin, NW; Middleton, JW; Molina, PE; Stielper, ZF1
Burrell, BD; Kabeiseman, E; Paulsen, R1
Abohalaka, R; Bozkurt, TE; Nemutlu, E; Onder, SC; Sahin-Erdemli, I1
Adelman, J; Akirav, I; Alteba, S; Ben David, G; Doron, R; Hillard, CJ; Mizrachi Zer-Aviv, T; Tenenhaus, A1

Other Studies

41 other study(ies) available for carbamates and jzl 184

ArticleYear
Inhibitors of endocannabinoid-metabolizing enzymes reduce precipitated withdrawal responses in THC-dependent mice.
    The AAPS journal, 2009, Volume: 11, Issue:2

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Hallucinogens; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoacylglycerol Lipases; Motor Activity; Piperidines; Postural Balance; Psychomotor Performance; Pyrazoles; Rimonabant; Substance Withdrawal Syndrome

2009
Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 330, Issue:3

    Topics: Amidohydrolases; Analgesics, Non-Narcotic; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Cold Temperature; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Narcotic Antagonists; Pain; Pain Measurement; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; TRPV Cation Channels

2009
Blockade of 2-arachidonoylglycerol hydrolysis by selective monoacylglycerol lipase inhibitor 4-nitrophenyl 4-(dibenzo[d][1,3]dioxol-5-yl(hydroxy)methyl)piperidine-1-carboxylate (JZL184) Enhances retrograde endocannabinoid signaling.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Electrophysiology; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hydrolysis; Lipase; Mice; Mice, Inbred C57BL; Mice, Knockout; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Signal Transduction; Synapses

2009
High-performance liquid chromatography assay with fluorescence detection for the evaluation of inhibitors against human recombinant monoacylglycerol lipase.
    Analytical biochemistry, 2010, Apr-15, Volume: 399, Issue:2

    Topics: Arachidonic Acids; Benzodioxoles; Butyric Acid; Carbamates; Chromatography, High Pressure Liquid; Enzyme Inhibitors; Fluorescent Dyes; Humans; Monoacylglycerol Lipases; Octoxynol; Organophosphonates; Oxadiazoles; Piperidines; Recombinant Proteins; Spectrophotometry, Ultraviolet; Substrate Specificity

2010
Inhibitors of monoacylglycerol lipase, fatty-acid amide hydrolase and endocannabinoid transport differentially suppress capsaicin-induced behavioral sensitization through peripheral endocannabinoid mechanisms.
    Pharmacological research, 2010, Volume: 62, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzodioxoles; Biological Transport; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Endocannabinoids; Male; Monoacylglycerol Lipases; Piperidines; Rats; Rats, Sprague-Dawley; Sensory System Agents

2010
Differential role of anandamide and 2-arachidonoylglycerol in memory and anxiety-like responses.
    Biological psychiatry, 2011, Sep-01, Volume: 70, Issue:5

    Topics: Amidohydrolases; Analgesics; Animals; Anti-Anxiety Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Antagonists; Carbamates; Drug Tolerance; Endocannabinoids; Glycerides; Hippocampus; Maze Learning; Mice; Mice, Inbred Strains; Mice, Knockout; Monoacylglycerol Lipases; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Receptors, Cannabinoid; Recognition, Psychology; TOR Serine-Threonine Kinases

2011
Cannabinoids mediate opposing effects on inflammation-induced intestinal permeability.
    British journal of pharmacology, 2012, Volume: 165, Issue:8

    Topics: Amidohydrolases; Benzamides; Benzodioxoles; Caco-2 Cells; Cannabinoids; Carbamates; Cell Survival; Enzyme Inhibitors; Humans; Indoles; Inflammation; Interferon-gamma; Intestinal Mucosa; Monoacylglycerol Lipases; Permeability; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Tumor Necrosis Factor-alpha

2012
Dual inhibition of MAGL and type II topoisomerase by N-phenylmaleimides as a potential strategy to reduce neuroblastoma cell growth.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2012, Feb-14, Volume: 45, Issue:3

    Topics: Antineoplastic Agents; Arachidonic Acids; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Cell Proliferation; DNA Topoisomerases, Type II; Endocannabinoids; Etoposide; Glycerides; Humans; Maleimides; Monoacylglycerol Lipases; Neuroblastoma; Oxadiazoles; Piperidines; Topoisomerase II Inhibitors; Tumor Cells, Cultured

2012
Covalent inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by the carbamates JZL184 and URB597.
    Biochemical pharmacology, 2012, Nov-01, Volume: 84, Issue:9

    Topics: Benzamides; Benzodioxoles; Carbamates; Carboxylesterase; Carboxylic Ester Hydrolases; Enzyme Reactivators; Hep G2 Cells; Humans; Kinetics; Monoacylglycerol Lipases; Paraoxon; Phosphorylation; Piperidines; Recombinant Proteins

2012
Alterations in endocannabinoid tone following chemotherapy-induced peripheral neuropathy: effects of endocannabinoid deactivation inhibitors targeting fatty-acid amide hydrolase and monoacylglycerol lipase in comparison to reference analgesics following c
    Pharmacological research, 2013, Volume: 67, Issue:1

    Topics: Amidohydrolases; Analgesics; Animals; Antineoplastic Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoids; Carbamates; Cisplatin; Endocannabinoids; Enzyme Inhibitors; Ganglia, Spinal; Glycerides; Hyperalgesia; Lipid Metabolism; Male; Monoacylglycerol Lipases; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; RNA, Messenger; Spinal Cord; TRPV Cation Channels

2013
Prior stimulation of the endocannabinoid system prevents methamphetamine-induced dopaminergic neurotoxicity in the striatum through activation of CB2 receptors.
    Neuropharmacology, 2014, Volume: 87

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Central Nervous System Stimulants; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Methamphetamine; Mice, Inbred C57BL; Neostriatum; Neurotoxicity Syndromes; Piperidines; Polyunsaturated Alkamides; Random Allocation; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Tumor Necrosis Factor-alpha; Tyrosine 3-Monooxygenase

2014
The dual FAAH/MAGL inhibitor JZL195 has enhanced effects on endocannabinoid transmission and motor behavior in rats as compared to those of the MAGL inhibitor JZL184.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 124

    Topics: Animals; Anti-Anxiety Agents; Benzodioxoles; Carbamates; Endocannabinoids; Male; Motor Activity; Piperazines; Piperidines; Rats; Rats, Wistar

2014
Attenuation of serotonin-induced itch responses by inhibition of endocannabinoid degradative enzymes, fatty acid amide hydrolase and monoacylglycerol lipase.
    Journal of neural transmission (Vienna, Austria : 1996), 2015, Volume: 122, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Camphanes; Carbamates; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Piperidines; Pruritus; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Serotonin

2015
Increased angiotensin II contraction of the uterine artery at early gestation in a transgenic model of hypertensive pregnancy is reduced by inhibition of endocannabinoid hydrolysis.
    Hypertension (Dallas, Tex. : 1979), 2014, Volume: 64, Issue:3

    Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood Pressure; Carbamates; Disease Models, Animal; Endocannabinoids; Female; Glycerides; Humans; Hydrolysis; Hypertension, Pregnancy-Induced; Male; Monoglycerides; Piperidines; Polyunsaturated Alkamides; Pregnancy; Pregnancy, Animal; Rats; Rats, Sprague-Dawley; Rats, Transgenic; Uterine Artery; Vasoconstriction

2014
Endocannabinoid modulation by FAAH and monoacylglycerol lipase within the analgesic circuitry of the periaqueductal grey.
    British journal of pharmacology, 2014, Volume: 171, Issue:23

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Endocannabinoids; Female; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Monoacylglycerol Lipases; Neurons; Pain; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission

2014
Therapeutic potential of inhibitors of endocannabinoid degradation for the treatment of stress-related hyperalgesia in an animal model of chronic pain.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:2

    Topics: Amidohydrolases; Analgesics, Non-Narcotic; Animals; Anxiety; Benzamides; Benzodioxoles; Brain; Carbamates; Chronic Pain; Depression; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Nerve Growth Factor; Piperidines; Stress, Psychological; Uncertainty

2015
Blockade of monoacylglycerol lipase inhibits oligodendrocyte excitotoxicity and prevents demyelination in vivo.
    Glia, 2015, Volume: 63, Issue:1

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Demyelinating Diseases; Monoacylglycerol Lipases; Multiple Sclerosis; Oligodendroglia; Piperidines; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1

2015
Endocannabinoid degradation inhibition improves neurobehavioral function, blood-brain barrier integrity, and neuroinflammation following mild traumatic brain injury.
    Journal of neurotrauma, 2015, Mar-01, Volume: 32, Issue:5

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood-Brain Barrier; Blotting, Western; Brain Injuries; Carbamates; Disease Models, Animal; Endocannabinoids; Glycerides; Immunohistochemistry; Inflammation; Male; Neuroprotective Agents; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Recovery of Function

2015
Differential effects of endocannabinoid catabolic inhibitors on morphine withdrawal in mice.
    Drug and alcohol dependence, 2015, Jan-01, Volume: 146

    Topics: Acetamides; Amidohydrolases; Animals; Avoidance Learning; Benzodioxoles; Carbamates; Conditioning, Psychological; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Monoacylglycerol Lipases; Morphine; Naloxone; Piperidines; Pyridines; Substance Withdrawal Syndrome

2015
Phenotypic assessment of THC discriminative stimulus properties in fatty acid amide hydrolase knockout and wildtype mice.
    Neuropharmacology, 2015, Volume: 93

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzodioxoles; Brain; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Mice; Mice, Knockout; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rimonabant

2015
Selective monoacylglycerol lipase inhibitors: antinociceptive versus cannabimimetic effects in mice.
    The Journal of pharmacology and experimental therapeutics, 2015, Volume: 353, Issue:2

    Topics: Analgesics; Animals; Benzodioxoles; Biomimetic Materials; Brain; Cannabinoids; Carbamates; Constriction; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Motor Activity; Neuralgia; Piperidines; Succinimides

2015
The effect of FAAH, MAGL, and Dual FAAH/MAGL inhibition on inflammatory and colorectal distension-induced visceral pain models in Rodents.
    Neurogastroenterology and motility, 2015, Volume: 27, Issue:7

    Topics: Amidohydrolases; Animals; Benzodioxoles; Carbamates; Colon; Cyclohexanols; Inflammation; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Pain Measurement; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Visceral Pain

2015
Actions of the dual FAAH/MAGL inhibitor JZL195 in a murine neuropathic pain model.
    British journal of pharmacology, 2016, Volume: 173, Issue:1

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Benzoxazines; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Hyperalgesia; Male; Mice; Monoacylglycerol Lipases; Morpholines; Naphthalenes; Neuralgia; Piperazines; Piperidines

2016
Inhibition of Monoacylglycerol Lipase Activity Decreases Glucose-Stimulated Insulin Secretion in INS-1 (832/13) Cells and Rat Islets.
    PloS one, 2016, Volume: 11, Issue:2

    Topics: Animals; Benzodioxoles; Biphenyl Compounds; Calcium; Carbamates; Cell Line; Fatty Acids; Fatty Acids, Nonesterified; Glucose; Glycerol; Insulin; Insulin Secretion; Insulin-Secreting Cells; Islets of Langerhans; Kinetics; Lipids; Lipolysis; Male; Monoacylglycerol Lipases; Phospholipids; Piperidines; Rats; Rats, Sprague-Dawley; Succinimides

2016
Systemic and spinal administration of FAAH, MAGL inhibitors and dual FAAH/MAGL inhibitors produce antipruritic effect in mice.
    Archives of dermatological research, 2016, Volume: 308, Issue:5

    Topics: Amidohydrolases; Animals; Antipruritics; Benzodioxoles; Carbamates; Disease Models, Animal; Endocannabinoids; Injections, Intraperitoneal; Injections, Spinal; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Piperazines; Piperidines; Pruritus; Pyridines; Serotonin

2016
Involvement of endocannabinoid neurotransmission in the bed nucleus of stria terminalis in cardiovascular responses to acute restraint stress in rats.
    British journal of pharmacology, 2016, Volume: 173, Issue:19

    Topics: Acute Disease; Animals; Benzamides; Benzodioxoles; Carbamates; Cardiovascular System; Dose-Response Relationship, Drug; Endocannabinoids; Male; Piperidines; Pyrazoles; Rats; Rats, Wistar; Restraint, Physical; Septal Nuclei; Stress, Psychological; Structure-Activity Relationship; Synaptic Transmission

2016
Orchestrated activation of mGluR5 and CB1 promotes neuroprotection.
    Molecular brain, 2016, 08-20, Volume: 9, Issue:1

    Topics: Animals; Benzamides; Benzodioxoles; Calcium; Carbamates; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Gene Knockdown Techniques; Intracellular Space; Mice, Inbred C57BL; Models, Biological; Neurons; Neuroprotection; Phosphorylation; Piperidines; Presynaptic Terminals; Proto-Oncogene Proteins c-akt; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Synapses

2016
The role of CB
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2017, Volume: 31, Issue:8

    Topics: Amidohydrolases; Arachidonic Acids; Benzamides; Benzodioxoles; Caco-2 Cells; Carbamates; Colorectal Neoplasms; Cytokines; Electric Impedance; Endocannabinoids; Gene Expression Regulation; Glycerides; Humans; Inflammation; Intestinal Mucosa; Intestines; Monoacylglycerol Lipases; Oxygen Consumption; Permeability; Piperidines; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Tissue Culture Techniques

2017
Enhanced anandamide signaling reduces flight behavior elicited by an approaching robo-beetle.
    Neuropharmacology, 2017, Volume: 126

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Agonists; Carbamates; Diazepam; Endocannabinoids; Fear; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2017
The cannabinoid transporter inhibitor OMDM-2 reduces social interaction: Further evidence for transporter-mediated endocannabinoid release.
    Neuropharmacology, 2018, 03-01, Volume: 130

    Topics: Amidohydrolases; Amygdala; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzodioxoles; Benzyl Compounds; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Male; Piperidines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Social Behavior

2018
Enhancing Endocannabinoid Neurotransmission Augments The Efficacy of Extinction Training and Ameliorates Traumatic Stress-Induced Behavioral Alterations in Rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2018, Volume: 43, Issue:6

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Benzoxazines; Cannabinoid Receptor Modulators; Carbamates; Disease Models, Animal; Electroshock; Endocannabinoids; Extinction, Psychological; Glycerides; Male; Morpholines; Naphthalenes; Piperidines; Psychotropic Drugs; Rats, Sprague-Dawley; Social Isolation; Stress Disorders, Post-Traumatic; Synaptic Transmission

2018
Modulation of central endocannabinoid system results in gastric mucosal protection in the rat.
    Brain research bulletin, 2018, Volume: 139

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Calcitonin Gene-Related Peptide; Carbamates; Catalepsy; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Endocannabinoids; Ethanol; Gastric Mucosa; Gastrointestinal Motility; Hypothermia; Male; Piperidines; Rats; Rats, Wistar; Somatostatin; Stomach Diseases; Superoxide Dismutase

2018
Neuroprotective Effects of MAGL (Monoacylglycerol Lipase) Inhibitors in Experimental Ischemic Stroke.
    Stroke, 2018, Volume: 49, Issue:3

    Topics: Animals; Benzodioxoles; Brain Ischemia; Carbamates; Disease Models, Animal; Enzyme Inhibitors; Male; Monoacylglycerol Lipases; Neuroprotective Agents; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Stroke; Succinimides

2018
Therapeutic endocannabinoid augmentation for mood and anxiety disorders: comparative profiling of FAAH, MAGL and dual inhibitors.
    Translational psychiatry, 2018, 04-26, Volume: 8, Issue:1

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Behavior, Animal; Benzodioxoles; Body Temperature; Brain; Carbamates; Endocannabinoids; Female; Locomotion; Male; Maze Learning; Mice, Inbred C57BL; Mice, Inbred ICR; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyridines; Stress, Psychological

2018
Endocannabinoid interactions in the regulation of acquisition of contextual conditioned fear.
    Progress in neuro-psychopharmacology & biological psychiatry, 2019, 03-02, Volume: 90

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Brain; Carbamates; Central Nervous System Agents; Conditioning, Psychological; Endocannabinoids; Fear; Glycerides; Male; Motor Activity; Nociception; Piperidines; Polyunsaturated Alkamides; Random Allocation; Rats, Wistar

2019
Inhibition of Monoacylglycerol Lipase Reduces the Reinstatement of Methamphetamine-Seeking and Anxiety-Like Behaviors in Methamphetamine Self-Administered Rats.
    The international journal of neuropsychopharmacology, 2019, 02-01, Volume: 22, Issue:2

    Topics: Amidohydrolases; Amphetamine-Related Disorders; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Addictive; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Antagonists; Carbamates; Central Nervous System Stimulants; Male; Maze Learning; Methamphetamine; Monoacylglycerol Lipases; Piperidines; Rats; Rats, Wistar

2019
Effects of Fatty Acid Amide Hydrolase Inhibitors Acute Administration on the Positive and Cognitive Symptoms of Schizophrenia in Mice.
    Molecular neurobiology, 2019, Volume: 56, Issue:11

    Topics: Amidohydrolases; Animals; Avoidance Learning; Benzamides; Benzodioxoles; Carbamates; Cognition; Dizocilpine Maleate; Enzyme Inhibitors; Injections; Male; Memory; Mice; Motor Activity; Piperidines; Schizophrenia

2019
Endocannabinoid degradation inhibitors ameliorate neuronal and synaptic alterations following traumatic brain injury.
    Journal of neurophysiology, 2020, 02-01, Volume: 123, Issue:2

    Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Brain Injuries, Traumatic; Carbamates; Electrophysiological Phenomena; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Machine Learning; Male; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyramidal Cells; Rats; Rats, Wistar; Sensorimotor Cortex; Succinimides

2020
Characterization of a monoacylglycerol lipase in the medicinal leech, Hirudo verbana.
    Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology, 2020, Volume: 243-244

    Topics: Animals; Benzodioxoles; Carbamates; Cell Membrane; Cloning, Molecular; Endocannabinoids; Enzyme Inhibitors; HEK293 Cells; Humans; Leeches; Monoacylglycerol Lipases; Phylogeny; Piperidines; Succinimides

2020
The effects of fatty acid amide hydrolase and monoacylglycerol lipase inhibitor treatments on lipopolysaccharide-induced airway inflammation in mice.
    Pulmonary pharmacology & therapeutics, 2020, Volume: 62

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Cytokines; Endocannabinoids; Glycerides; Inflammation; Lipopolysaccharides; Lung; Male; Mice; Monoacylglycerol Lipases; Piperidines; Pneumonia; Polyunsaturated Alkamides; Respiratory Hypersensitivity

2020
Antidepressant-like effects of URB597 and JZL184 in male and female rats exposed to early life stress.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2020, Volume: 39

    Topics: Age Factors; Animals; Antidepressive Agents; Benzamides; Benzodioxoles; Carbamates; Depression; Female; Male; Piperidines; Rats; Rats, Sprague-Dawley; Social Interaction; Stress, Psychological; Treatment Outcome

2020