carbamates has been researched along with jzl 184 in 41 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (7.32) | 29.6817 |
2010's | 34 (82.93) | 24.3611 |
2020's | 4 (9.76) | 2.80 |
Authors | Studies |
---|---|
Abdullah, RA; Carlson, BL; Cravatt, BF; Lichtman, AH; Long, JZ; Ramesh, D; Schlosburg, JE | 1 |
Abdullah, RA; Boger, DL; Cravatt, BF; Kinsey, SG; Lichtman, AH; Long, JZ; O'Neal, ST; Poklis, JL | 1 |
Cravatt, BF; Hillard, CJ; Liu, QS; Long, JZ; Pan, B; Sun, D; Wang, W | 1 |
Holtfrerich, A; Lehr, M; Makharadze, T | 1 |
Guindon, J; Hohmann, AG; Spradley, JM | 1 |
Busquets-Garcia, A; de la Torre, R; Maldonado, R; Ozaita, A; Pastor, A; Puighermanal, E | 1 |
Alhamoruni, A; Larvin, M; O'Sullivan, SE; Wright, KL | 1 |
Baldeyroux, B; Hamtiaux, L; Lambert, DM; Lansiaux, A; Matuszak, N; Muccioli, GG; Poupaert, JH | 1 |
Bittles, V; Borazjani, A; Crow, JA; Potter, PM; Ross, MK | 1 |
Bradshaw, HB; Guindon, J; Hohmann, AG; Lai, Y; Takacs, SM | 1 |
Chavant, F; Duranti, A; Francheteau, M; Gennequin, B; Maccarrone, M; Makriyannis, A; Nader, J; Rapino, C; Solinas, M; Thiriet, N | 1 |
Dominguez Aguilar, D; Giuffrida, A; Seillier, A | 1 |
Gunduz, O; Tosun, NC; Ulugol, A | 1 |
Bader, M; Brosnihan, KB; Dechend, R; Howlett, AC; McGee, CM; Pulgar, VM; Varagic, J; Yamaleyeva, LM | 1 |
Drew, GM; Lau, BK; Mitchell, VA; Vaughan, CW | 1 |
Bindila, L; Hoheisel, U; Lerner, R; Lomazzo, E; Lutz, B; Remmers, F; Schwitter, C | 1 |
Bernal-Chico, A; Canedo, M; Manterola, A; Mato, S; Matute, C; Pérez-Samartín, A; Rodríguez-Puertas, R; Victoria Sánchez-Gómez, M | 1 |
Impastato, RA; Katz, PS; Molina, PE; Rogers, EK; Sulzer, JK; Teng, SX | 1 |
Cravatt, BF; Damaj, MI; Gamage, TF; Ignatowska-Jankowska, BM; Lichtman, AH; Muldoon, PP | 1 |
Vann, RE; Walentiny, DM; Wiley, JL | 1 |
Abdullah, R; Cravatt, BF; Ignatowska-Jankowska, B; Lichtman, AH; Mustafa, M; Niphakis, M; Wiley, JL; Wilkerson, JL | 1 |
Bagci, S; Dogrul, A; Gulsen, M; Ilkaya, F; Sakin, YS; Seyrek, M; Ulas, UH | 1 |
Adamson Barnes, NS; Kazantzis, NP; Mitchell, VA; Vaughan, CW | 1 |
Berdan, CA; Burritt, NE; Corkey, BE; Deeney, JT; Erion, KA | 1 |
Akar, A; Cayirli, M; Dogrul, A; Sakin, YS; Seyrek, M; Yesilyurt, O | 1 |
Benini, R; Costa-Ferreira, W; Crestani, CC; Gomes-de-Souza, L; Oliveira, LA; Rodella, P | 1 |
Alves-Silva, J; Batista, EM; Doria, JG; Ferguson, SS; Ferreira-Vieira, TH; Moreira, FA; Ribeiro, FM | 1 |
Barrett, DA; Couch, DG; Karwad, MA; Larvin, M; Lund, JN; O'Sullivan, SE; Sarmad, S; Theophilidou, E; Wright, KL | 1 |
Genewsky, A; Heinz, DE; Wotjak, CT | 1 |
Giuffrida, A; Seillier, A | 1 |
Berardi, A; Campolongo, P; Colucci, P; Hill, MN; Morena, M; Palmery, M; Trezza, V | 1 |
Fehér, Á; Gyertyán, I; Gyires, K; Németh, J; Tóth, VE; Zádori, ZS | 1 |
Arai, AL; Choi, SH; Hallenbeck, J; Kang, B; Mou, Y; Silva, AC; Yen, CC | 1 |
Bedse, G; Bluett, RJ; Gaulden, AD; Kingsley, PJ; Marnett, LJ; Patel, S; Patrick, TA; Plath, N; Romness, NK | 1 |
Aliczki, M; Balogh, Z; Biro, L; Haller, J; Szente, L; Varga, ZK | 1 |
Fukumori, R; Nawata, Y; Yamaguchi, T; Yamamoto, T | 1 |
Banaszkiewicz, I; Biala, G; Kruk-Slomka, M; Slomka, T | 1 |
Cancienne, HL; Edwards, S; Fucich, EA; Gilpin, NW; Middleton, JW; Molina, PE; Stielper, ZF | 1 |
Burrell, BD; Kabeiseman, E; Paulsen, R | 1 |
Abohalaka, R; Bozkurt, TE; Nemutlu, E; Onder, SC; Sahin-Erdemli, I | 1 |
Adelman, J; Akirav, I; Alteba, S; Ben David, G; Doron, R; Hillard, CJ; Mizrachi Zer-Aviv, T; Tenenhaus, A | 1 |
41 other study(ies) available for carbamates and jzl 184
Article | Year |
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Inhibitors of endocannabinoid-metabolizing enzymes reduce precipitated withdrawal responses in THC-dependent mice.
Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Hallucinogens; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoacylglycerol Lipases; Motor Activity; Piperidines; Postural Balance; Psychomotor Performance; Pyrazoles; Rimonabant; Substance Withdrawal Syndrome | 2009 |
Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain.
Topics: Amidohydrolases; Analgesics, Non-Narcotic; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Cold Temperature; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Narcotic Antagonists; Pain; Pain Measurement; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; TRPV Cation Channels | 2009 |
Blockade of 2-arachidonoylglycerol hydrolysis by selective monoacylglycerol lipase inhibitor 4-nitrophenyl 4-(dibenzo[d][1,3]dioxol-5-yl(hydroxy)methyl)piperidine-1-carboxylate (JZL184) Enhances retrograde endocannabinoid signaling.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Electrophysiology; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hydrolysis; Lipase; Mice; Mice, Inbred C57BL; Mice, Knockout; Patch-Clamp Techniques; Piperidines; Purkinje Cells; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Signal Transduction; Synapses | 2009 |
High-performance liquid chromatography assay with fluorescence detection for the evaluation of inhibitors against human recombinant monoacylglycerol lipase.
Topics: Arachidonic Acids; Benzodioxoles; Butyric Acid; Carbamates; Chromatography, High Pressure Liquid; Enzyme Inhibitors; Fluorescent Dyes; Humans; Monoacylglycerol Lipases; Octoxynol; Organophosphonates; Oxadiazoles; Piperidines; Recombinant Proteins; Spectrophotometry, Ultraviolet; Substrate Specificity | 2010 |
Inhibitors of monoacylglycerol lipase, fatty-acid amide hydrolase and endocannabinoid transport differentially suppress capsaicin-induced behavioral sensitization through peripheral endocannabinoid mechanisms.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzodioxoles; Biological Transport; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Endocannabinoids; Male; Monoacylglycerol Lipases; Piperidines; Rats; Rats, Sprague-Dawley; Sensory System Agents | 2010 |
Differential role of anandamide and 2-arachidonoylglycerol in memory and anxiety-like responses.
Topics: Amidohydrolases; Analgesics; Animals; Anti-Anxiety Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Antagonists; Carbamates; Drug Tolerance; Endocannabinoids; Glycerides; Hippocampus; Maze Learning; Mice; Mice, Inbred Strains; Mice, Knockout; Monoacylglycerol Lipases; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Receptors, Cannabinoid; Recognition, Psychology; TOR Serine-Threonine Kinases | 2011 |
Cannabinoids mediate opposing effects on inflammation-induced intestinal permeability.
Topics: Amidohydrolases; Benzamides; Benzodioxoles; Caco-2 Cells; Cannabinoids; Carbamates; Cell Survival; Enzyme Inhibitors; Humans; Indoles; Inflammation; Interferon-gamma; Intestinal Mucosa; Monoacylglycerol Lipases; Permeability; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Tumor Necrosis Factor-alpha | 2012 |
Dual inhibition of MAGL and type II topoisomerase by N-phenylmaleimides as a potential strategy to reduce neuroblastoma cell growth.
Topics: Antineoplastic Agents; Arachidonic Acids; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Cell Proliferation; DNA Topoisomerases, Type II; Endocannabinoids; Etoposide; Glycerides; Humans; Maleimides; Monoacylglycerol Lipases; Neuroblastoma; Oxadiazoles; Piperidines; Topoisomerase II Inhibitors; Tumor Cells, Cultured | 2012 |
Covalent inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by the carbamates JZL184 and URB597.
Topics: Benzamides; Benzodioxoles; Carbamates; Carboxylesterase; Carboxylic Ester Hydrolases; Enzyme Reactivators; Hep G2 Cells; Humans; Kinetics; Monoacylglycerol Lipases; Paraoxon; Phosphorylation; Piperidines; Recombinant Proteins | 2012 |
Alterations in endocannabinoid tone following chemotherapy-induced peripheral neuropathy: effects of endocannabinoid deactivation inhibitors targeting fatty-acid amide hydrolase and monoacylglycerol lipase in comparison to reference analgesics following c
Topics: Amidohydrolases; Analgesics; Animals; Antineoplastic Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoids; Carbamates; Cisplatin; Endocannabinoids; Enzyme Inhibitors; Ganglia, Spinal; Glycerides; Hyperalgesia; Lipid Metabolism; Male; Monoacylglycerol Lipases; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; RNA, Messenger; Spinal Cord; TRPV Cation Channels | 2013 |
Prior stimulation of the endocannabinoid system prevents methamphetamine-induced dopaminergic neurotoxicity in the striatum through activation of CB2 receptors.
Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Central Nervous System Stimulants; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Methamphetamine; Mice, Inbred C57BL; Neostriatum; Neurotoxicity Syndromes; Piperidines; Polyunsaturated Alkamides; Random Allocation; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Tumor Necrosis Factor-alpha; Tyrosine 3-Monooxygenase | 2014 |
The dual FAAH/MAGL inhibitor JZL195 has enhanced effects on endocannabinoid transmission and motor behavior in rats as compared to those of the MAGL inhibitor JZL184.
Topics: Animals; Anti-Anxiety Agents; Benzodioxoles; Carbamates; Endocannabinoids; Male; Motor Activity; Piperazines; Piperidines; Rats; Rats, Wistar | 2014 |
Attenuation of serotonin-induced itch responses by inhibition of endocannabinoid degradative enzymes, fatty acid amide hydrolase and monoacylglycerol lipase.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Camphanes; Carbamates; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Piperidines; Pruritus; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Serotonin | 2015 |
Increased angiotensin II contraction of the uterine artery at early gestation in a transgenic model of hypertensive pregnancy is reduced by inhibition of endocannabinoid hydrolysis.
Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood Pressure; Carbamates; Disease Models, Animal; Endocannabinoids; Female; Glycerides; Humans; Hydrolysis; Hypertension, Pregnancy-Induced; Male; Monoglycerides; Piperidines; Polyunsaturated Alkamides; Pregnancy; Pregnancy, Animal; Rats; Rats, Sprague-Dawley; Rats, Transgenic; Uterine Artery; Vasoconstriction | 2014 |
Endocannabinoid modulation by FAAH and monoacylglycerol lipase within the analgesic circuitry of the periaqueductal grey.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Endocannabinoids; Female; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Monoacylglycerol Lipases; Neurons; Pain; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission | 2014 |
Therapeutic potential of inhibitors of endocannabinoid degradation for the treatment of stress-related hyperalgesia in an animal model of chronic pain.
Topics: Amidohydrolases; Analgesics, Non-Narcotic; Animals; Anxiety; Benzamides; Benzodioxoles; Brain; Carbamates; Chronic Pain; Depression; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Nerve Growth Factor; Piperidines; Stress, Psychological; Uncertainty | 2015 |
Blockade of monoacylglycerol lipase inhibits oligodendrocyte excitotoxicity and prevents demyelination in vivo.
Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Demyelinating Diseases; Monoacylglycerol Lipases; Multiple Sclerosis; Oligodendroglia; Piperidines; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1 | 2015 |
Endocannabinoid degradation inhibition improves neurobehavioral function, blood-brain barrier integrity, and neuroinflammation following mild traumatic brain injury.
Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood-Brain Barrier; Blotting, Western; Brain Injuries; Carbamates; Disease Models, Animal; Endocannabinoids; Glycerides; Immunohistochemistry; Inflammation; Male; Neuroprotective Agents; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Recovery of Function | 2015 |
Differential effects of endocannabinoid catabolic inhibitors on morphine withdrawal in mice.
Topics: Acetamides; Amidohydrolases; Animals; Avoidance Learning; Benzodioxoles; Carbamates; Conditioning, Psychological; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Monoacylglycerol Lipases; Morphine; Naloxone; Piperidines; Pyridines; Substance Withdrawal Syndrome | 2015 |
Phenotypic assessment of THC discriminative stimulus properties in fatty acid amide hydrolase knockout and wildtype mice.
Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzodioxoles; Brain; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Mice; Mice, Knockout; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rimonabant | 2015 |
Selective monoacylglycerol lipase inhibitors: antinociceptive versus cannabimimetic effects in mice.
Topics: Analgesics; Animals; Benzodioxoles; Biomimetic Materials; Brain; Cannabinoids; Carbamates; Constriction; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Motor Activity; Neuralgia; Piperidines; Succinimides | 2015 |
The effect of FAAH, MAGL, and Dual FAAH/MAGL inhibition on inflammatory and colorectal distension-induced visceral pain models in Rodents.
Topics: Amidohydrolases; Animals; Benzodioxoles; Carbamates; Colon; Cyclohexanols; Inflammation; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Pain Measurement; Piperazines; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Visceral Pain | 2015 |
Actions of the dual FAAH/MAGL inhibitor JZL195 in a murine neuropathic pain model.
Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Benzoxazines; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Hyperalgesia; Male; Mice; Monoacylglycerol Lipases; Morpholines; Naphthalenes; Neuralgia; Piperazines; Piperidines | 2016 |
Inhibition of Monoacylglycerol Lipase Activity Decreases Glucose-Stimulated Insulin Secretion in INS-1 (832/13) Cells and Rat Islets.
Topics: Animals; Benzodioxoles; Biphenyl Compounds; Calcium; Carbamates; Cell Line; Fatty Acids; Fatty Acids, Nonesterified; Glucose; Glycerol; Insulin; Insulin Secretion; Insulin-Secreting Cells; Islets of Langerhans; Kinetics; Lipids; Lipolysis; Male; Monoacylglycerol Lipases; Phospholipids; Piperidines; Rats; Rats, Sprague-Dawley; Succinimides | 2016 |
Systemic and spinal administration of FAAH, MAGL inhibitors and dual FAAH/MAGL inhibitors produce antipruritic effect in mice.
Topics: Amidohydrolases; Animals; Antipruritics; Benzodioxoles; Carbamates; Disease Models, Animal; Endocannabinoids; Injections, Intraperitoneal; Injections, Spinal; Male; Mice; Mice, Inbred BALB C; Monoacylglycerol Lipases; Piperazines; Piperidines; Pruritus; Pyridines; Serotonin | 2016 |
Involvement of endocannabinoid neurotransmission in the bed nucleus of stria terminalis in cardiovascular responses to acute restraint stress in rats.
Topics: Acute Disease; Animals; Benzamides; Benzodioxoles; Carbamates; Cardiovascular System; Dose-Response Relationship, Drug; Endocannabinoids; Male; Piperidines; Pyrazoles; Rats; Rats, Wistar; Restraint, Physical; Septal Nuclei; Stress, Psychological; Structure-Activity Relationship; Synaptic Transmission | 2016 |
Orchestrated activation of mGluR5 and CB1 promotes neuroprotection.
Topics: Animals; Benzamides; Benzodioxoles; Calcium; Carbamates; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Gene Knockdown Techniques; Intracellular Space; Mice, Inbred C57BL; Models, Biological; Neurons; Neuroprotection; Phosphorylation; Piperidines; Presynaptic Terminals; Proto-Oncogene Proteins c-akt; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Synapses | 2016 |
The role of CB
Topics: Amidohydrolases; Arachidonic Acids; Benzamides; Benzodioxoles; Caco-2 Cells; Carbamates; Colorectal Neoplasms; Cytokines; Electric Impedance; Endocannabinoids; Gene Expression Regulation; Glycerides; Humans; Inflammation; Intestinal Mucosa; Intestines; Monoacylglycerol Lipases; Oxygen Consumption; Permeability; Piperidines; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Tissue Culture Techniques | 2017 |
Enhanced anandamide signaling reduces flight behavior elicited by an approaching robo-beetle.
Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Agonists; Carbamates; Diazepam; Endocannabinoids; Fear; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant | 2017 |
The cannabinoid transporter inhibitor OMDM-2 reduces social interaction: Further evidence for transporter-mediated endocannabinoid release.
Topics: Amidohydrolases; Amygdala; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzodioxoles; Benzyl Compounds; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Male; Piperidines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Social Behavior | 2018 |
Enhancing Endocannabinoid Neurotransmission Augments The Efficacy of Extinction Training and Ameliorates Traumatic Stress-Induced Behavioral Alterations in Rats.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Benzoxazines; Cannabinoid Receptor Modulators; Carbamates; Disease Models, Animal; Electroshock; Endocannabinoids; Extinction, Psychological; Glycerides; Male; Morpholines; Naphthalenes; Piperidines; Psychotropic Drugs; Rats, Sprague-Dawley; Social Isolation; Stress Disorders, Post-Traumatic; Synaptic Transmission | 2018 |
Modulation of central endocannabinoid system results in gastric mucosal protection in the rat.
Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Calcitonin Gene-Related Peptide; Carbamates; Catalepsy; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Endocannabinoids; Ethanol; Gastric Mucosa; Gastrointestinal Motility; Hypothermia; Male; Piperidines; Rats; Rats, Wistar; Somatostatin; Stomach Diseases; Superoxide Dismutase | 2018 |
Neuroprotective Effects of MAGL (Monoacylglycerol Lipase) Inhibitors in Experimental Ischemic Stroke.
Topics: Animals; Benzodioxoles; Brain Ischemia; Carbamates; Disease Models, Animal; Enzyme Inhibitors; Male; Monoacylglycerol Lipases; Neuroprotective Agents; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Stroke; Succinimides | 2018 |
Therapeutic endocannabinoid augmentation for mood and anxiety disorders: comparative profiling of FAAH, MAGL and dual inhibitors.
Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Behavior, Animal; Benzodioxoles; Body Temperature; Brain; Carbamates; Endocannabinoids; Female; Locomotion; Male; Maze Learning; Mice, Inbred C57BL; Mice, Inbred ICR; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyridines; Stress, Psychological | 2018 |
Endocannabinoid interactions in the regulation of acquisition of contextual conditioned fear.
Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Brain; Carbamates; Central Nervous System Agents; Conditioning, Psychological; Endocannabinoids; Fear; Glycerides; Male; Motor Activity; Nociception; Piperidines; Polyunsaturated Alkamides; Random Allocation; Rats, Wistar | 2019 |
Inhibition of Monoacylglycerol Lipase Reduces the Reinstatement of Methamphetamine-Seeking and Anxiety-Like Behaviors in Methamphetamine Self-Administered Rats.
Topics: Amidohydrolases; Amphetamine-Related Disorders; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Addictive; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Antagonists; Carbamates; Central Nervous System Stimulants; Male; Maze Learning; Methamphetamine; Monoacylglycerol Lipases; Piperidines; Rats; Rats, Wistar | 2019 |
Effects of Fatty Acid Amide Hydrolase Inhibitors Acute Administration on the Positive and Cognitive Symptoms of Schizophrenia in Mice.
Topics: Amidohydrolases; Animals; Avoidance Learning; Benzamides; Benzodioxoles; Carbamates; Cognition; Dizocilpine Maleate; Enzyme Inhibitors; Injections; Male; Memory; Mice; Motor Activity; Piperidines; Schizophrenia | 2019 |
Endocannabinoid degradation inhibitors ameliorate neuronal and synaptic alterations following traumatic brain injury.
Topics: Amidohydrolases; Animals; Benzamides; Benzodioxoles; Brain Injuries, Traumatic; Carbamates; Electrophysiological Phenomena; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Machine Learning; Male; Monoacylglycerol Lipases; Piperazines; Piperidines; Pyramidal Cells; Rats; Rats, Wistar; Sensorimotor Cortex; Succinimides | 2020 |
Characterization of a monoacylglycerol lipase in the medicinal leech, Hirudo verbana.
Topics: Animals; Benzodioxoles; Carbamates; Cell Membrane; Cloning, Molecular; Endocannabinoids; Enzyme Inhibitors; HEK293 Cells; Humans; Leeches; Monoacylglycerol Lipases; Phylogeny; Piperidines; Succinimides | 2020 |
The effects of fatty acid amide hydrolase and monoacylglycerol lipase inhibitor treatments on lipopolysaccharide-induced airway inflammation in mice.
Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Cytokines; Endocannabinoids; Glycerides; Inflammation; Lipopolysaccharides; Lung; Male; Mice; Monoacylglycerol Lipases; Piperidines; Pneumonia; Polyunsaturated Alkamides; Respiratory Hypersensitivity | 2020 |
Antidepressant-like effects of URB597 and JZL184 in male and female rats exposed to early life stress.
Topics: Age Factors; Animals; Antidepressive Agents; Benzamides; Benzodioxoles; Carbamates; Depression; Female; Male; Piperidines; Rats; Rats, Sprague-Dawley; Social Interaction; Stress, Psychological; Treatment Outcome | 2020 |