carbamates and itraconazole

carbamates has been researched along with itraconazole in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (33.33)29.6817
2010's5 (55.56)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Backman, JT; Neuvonen, M; Neuvonen, PJ; Niemi, M1
Backman, JT; Kajosaari, LI; Laitila, J; Neuvonen, PJ1
Härter, G; Kern, P; Manfras, B; Merkle, M; Reuter, S1
Bode, C1
Chen, W; Gan, J; Gao, L; Hong, Y; Humphreys, WG; Li, W; Rodrigues, AD; Shen, H; Tang, Y; Tian, Y; Zhang, H; Zhang, Y1
Hisaka, A; Ito, K; Kudo, T; Sugiyama, Y1
Mitra, AK; Pal, D; Patel, M; Paturi, DK; Vadlapatla, RK1
Furihata, KI; Kusuhara, H; Maeda, K; Sugiyama, Y; Yoshikado, T1
Ito, S; Iwamoto, K; Kamimura, H; Mizunaga, M; Nakayama, K; Negoro, T; Nishiwaki, M; Nomura, Y; Suemizu, H; Yamazaki, H; Yoneda, N1

Reviews

2 review(s) available for carbamates and itraconazole

ArticleYear
The nasty surprise of a complex drug-drug interaction.
    Drug discovery today, 2010, Volume: 15, Issue:9-10

    Topics: Carbamates; Drug Approval; Drug Evaluation, Preclinical; Drug Industry; Drug Interactions; Drug Therapy, Combination; Gemfibrozil; Humans; Itraconazole; Models, Biological; Piperidines

2010
Clinically relevant drug-drug interactions between antiretrovirals and antifungals.
    Expert opinion on drug metabolism & toxicology, 2014, Volume: 10, Issue:4

    Topics: AIDS-Related Opportunistic Infections; Alkynes; Anti-Retroviral Agents; Antifungal Agents; Benzoxazines; Carbamates; Cyclopropanes; Drug Interactions; Drug Monitoring; Echinocandins; Furans; HIV Infections; HIV Protease Inhibitors; Humans; Itraconazole; Mycoses; Organophosphates; Pyrimidines; Ritonavir; Sulfonamides; Triazoles; Voriconazole

2014

Trials

1 trial(s) available for carbamates and itraconazole

ArticleYear
Effects of gemfibrozil, itraconazole, and their combination on the pharmacokinetics and pharmacodynamics of repaglinide: potentially hazardous interaction between gemfibrozil and repaglinide.
    Diabetologia, 2003, Volume: 46, Issue:3

    Topics: Adult; Antifungal Agents; Area Under Curve; Aryl Hydrocarbon Hydroxylases; Biotransformation; Blood Glucose; C-Peptide; Carbamates; Cross-Over Studies; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Interactions; Female; Gemfibrozil; Half-Life; Humans; Hypoglycemic Agents; Hypolipidemic Agents; Insulin; Itraconazole; Male; Piperidines

2003

Other Studies

6 other study(ies) available for carbamates and itraconazole

ArticleYear
Metabolism of repaglinide by CYP2C8 and CYP3A4 in vitro: effect of fibrates and rifampicin.
    Basic & clinical pharmacology & toxicology, 2005, Volume: 97, Issue:4

    Topics: Aryl Hydrocarbon Hydroxylases; Bezafibrate; Carbamates; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Interactions; Fenofibrate; Gemfibrozil; Humans; Hypoglycemic Agents; In Vitro Techniques; Itraconazole; Microsomes, Liver; Midazolam; Paclitaxel; Piperidines; Quercetin; Rifampin

2005
In vitro activities of itraconazole, methiazole, and nitazoxanide versus Echinococcus multilocularis larvae.
    Antimicrobial agents and chemotherapy, 2006, Volume: 50, Issue:9

    Topics: Animals; Antiparasitic Agents; Benzimidazoles; Carbamates; Echinococcus multilocularis; Gerbillinae; Itraconazole; Larva; Nitro Compounds; Thiazoles

2006
Repaglinide-gemfibrozil drug interaction: inhibition of repaglinide glucuronidation as a potential additional contributing mechanism.
    British journal of clinical pharmacology, 2010, Volume: 70, Issue:6

    Topics: Biotransformation; Carbamates; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Gemfibrozil; Glucuronides; Glucuronosyltransferase; Hepatocytes; Humans; Hypoglycemic Agents; Hypolipidemic Agents; Itraconazole; Microsomes, Liver; Piperidines

2010
Analysis of the repaglinide concentration increase produced by gemfibrozil and itraconazole based on the inhibition of the hepatic uptake transporter and metabolic enzymes.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:2

    Topics: Area Under Curve; Aryl Hydrocarbon Hydroxylases; Biotransformation; Carbamates; Computer Simulation; Cytochrome P-450 CYP2C8; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Enzyme Inhibitors; Gemfibrozil; Glucuronides; Humans; Hypoglycemic Agents; Itraconazole; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Biological; Nonlinear Dynamics; Organic Anion Transporters; Piperidines

2013
Quantitative Analyses of the Influence of Parameters Governing Rate-Determining Process of Hepatic Elimination of Drugs on the Magnitudes of Drug-Drug Interactions via Hepatic OATPs and CYP3A Using Physiologically Based Pharmacokinetic Models.
    Journal of pharmaceutical sciences, 2017, Volume: 106, Issue:9

    Topics: Adult; Bosentan; Carbamates; Computer Simulation; Cytochrome P-450 CYP3A; Drug Interactions; Hepatobiliary Elimination; Humans; Itraconazole; Liver; Male; Models, Biological; Organic Anion Transporters; Pharmaceutical Preparations; Piperidines; Rifampin; Sulfonamides; Young Adult

2017
Predicted values for human total clearance of a variety of typical compounds with differently humanized-liver mouse plasma data.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:4

    Topics: Acetamides; Albuterol; Animals; Carbamates; Chromatography, Liquid; Diazepam; Diclofenac; Digitoxin; Humans; Itraconazole; Ketoprofen; Liver; Metabolic Clearance Rate; Mice; Mice, Transgenic; Naproxen; Pharmaceutical Preparations; Phenytoin; Piperidines; Pravastatin; Pyrimidines; Quinidine; Tandem Mass Spectrometry; Telmisartan; Terfenadine; Verapamil

2020