carbamates and anandamide

carbamates has been researched along with anandamide in 151 studies

Research

Studies (151)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (0.66)18.2507
2000's46 (30.46)29.6817
2010's94 (62.25)24.3611
2020's10 (6.62)2.80

Authors

AuthorsStudies
Abood, ME; Aung, MM; Martin, BR; Ng, EW; Razdan, RK1
Duranti, A; Kathuria, S; Mor, M; Park, C; Piersanti, G; Piomelli, D; Plazzi, PV; Rivara, S; Tarzia, G; Tontini, A1
Bátkai, S; Bukoski, RD; Harvey-White, J; Kunos, G; Liu, J; Mackie, K; Offertáler, L; Osei-Hyiaman, D; Pacher, P; Radaeva, S; Rudd, MA1
Duranti, A; Fegley, D; Gaetani, S; Mor, M; Piomelli, D; Tarzia, G; Tontini, A1
Lambert, DM; Okamoto, Y; Sun, YX; Tsuboi, K; Ueda, N; Zhao, LY1
Fegley, D; Gutierrez, T; Hohmann, AG; Piomelli, D; Suplita, RL1
Bambico, FR; Bortolato, M; Campolongo, P; Cassano, T; Cuomo, V; Debonnel, G; Duranti, A; Gobbi, G; Goldberg, SR; Mangieri, R; Mor, M; Morgese, MG; Piomelli, D; Solinas, M; Tarzia, G; Tontini, A; Trezza, V1
Jones, PG; Ramarao, MK; Rogers, KE; Uveges, A; Wang, Y; Xu, J1
Filip, M; McCreary, AC; Przegaliński, E; Zaniewska, M1
Goldberg, SR; Justinova, Z; Solinas, M; Tanda, G1
Nomikos, GG; Panagis, G; Vlachou, S1
Cross-Mellor, SK; Ossenkopp, KP; Parker, LA; Piomelli, D1
Goldberg, SR; Justinova, Z; Makriyannis, A; Piomelli, D; Solinas, M; Tanda, G; Vadivel, SK; Wertheim, CE; Yasar, S1
Ali, N; Chapman, V; Chimenti, M; de Lago, E; Fernandez-Ruiz, J; Kendall, DA; Millns, PJ; Ryland, E1
Ho, WS; Randall, MD1
Lam, FF; Luk, PW; Ng, ES1
Ahn, K; Cravatt, BF; Lichtman, AH; Martin, BR; Naidu, PS; Varvel, SA1
Alajakku, K; Fowler, CJ; Thors, L1
Drysdale, AJ; Pertwee, RG; Platt, B; Ryan, D1
Agrò, AF; Bagetta, G; Bari, M; Cerulli, A; Corasaniti, MT; De Simone, C; Gasperi, V; Maccarrone, M; Morrone, LA; Nucci, C; Tartaglione, R; Terrinoni, A1
Eriksson, J; Fowler, CJ; Thors, L1
Gorzalka, BB; Hill, MN; Morrish, AC1
Herradón, E; López-Miranda, V; Martín, MI1
Kaiser, N; Lutz, B; Monory, K; Moreira, FA1
Cassano, T; Cuomo, V; Giuffrida, A; Morgese, MG1
Fratta, W; Goldberg, SR; Haller, J; Makriyannis, A; Medalie, J; Mikics, E; Piomelli, D; Scherma, M; Tanda, G; Vadivel, SK; Yasar, S1
Castiglioni, C; Di Marzo, V; Guidali, C; Maccarrone, M; Marras, E; Parolaro, D; Perletti, G; Petrosino, S; Realini, N; Rubino, T; Viganó, D1
Cascio, MG; de Novellis, V; De Petrocellis, L; Di Marzo, V; Maione, S; Morera, E; Nalli, M; Ortar, G; Rossi, F; Schiano-Moriello, A; Woodward, DF1
Béquet, F; Desbazeille, M; Le Fur, G; Ludwiczak, P; Maftouh, M; Picard, C; Scatton, B; Uzabiaga, F1
Bilbao, A; Braconi, S; Cannella, N; Ciccocioppo, R; Cippitelli, A; Defonseca, FR; Duranti, A; Piomelli, D; Tontini, A1
Njie, YF; Qiao, Z; Song, ZH; Wang, W; Xiao, Z1
Fowler, CJ; Ghafouri, N1
Aguiar, DC; Guimarães, FS; Lisboa, SF; Resstel, LB1
Barnes, C; Fadda, P; Fattore, L; Fratta, W; Gamaleddin, I; Goldberg, SR; Haller, J; Justinová, Z; Le Foll, B; Medalie, J; Mikics, E; Panlilio, LV; Piomelli, D; Scherma, M; Stroik, J; Tanda, G; Yasar, S1
Haller, VL; Stevens, DL; Welch, SP1
Bortolato, M; Chefer, SI; Clapper, JR; Goldberg, SR; Justinova, Z; King, AR; Mangieri, RA; Mukhin, AG; Piomelli, D; Redhi, GH; Yasar, S1
Butler, RK; Finn, DP; Gavin, AM; Lang, Y; Rea, K1
Billi, S; Farina, M; Franchi, AM; Gervasi, MG; Perez Martinez, S; Rapanelli, M; Ribeiro, ML1
Adriani, W; Laviola, G; Marco, EM; Parolaro, D; Rubino, T; Viveros, MP1
Gardiner, SM; Ho, WS1
Kwiatkowska, M; Limebeer, CL; Litt, DL; Parker, LA; Piomelli, D; Rock, EM1
Benton, VM; Bradshaw, HB; Cravatt, BF; Hu, SS; Masuda, K; O'Dell, DK; Rimmerman, N; Stuart, JM; Walker, JM1
Abdullah, RA; Boger, DL; Cravatt, BF; Kinsey, SG; Lichtman, AH; Long, JZ; O'Neal, ST; Poklis, JL1
Gontinou, C; Karaliota, S; Mavri-Vavayanni, M; Psarra, K; Siafaka-Kapadai, A1
Floresco, SB; Gorzalka, BB; Hill, MN; Hillard, CJ; McLaughlin, RJ; Morrish, AC; Viau, V1
Fowler, CJ; Thors, L1
Booker, L; Burston, JJ; Cravatt, BF; Jin, X; Lichtman, AH; Long, JZ; Nomura, DK; Sim-Selley, LJ; Vann, RE; Walentiny, DM; Wiley, JL1
Galadari, S; Jaligam, V; Oz, M; Petroianu, G; Shippenberg, TS; Shuba, YM1
Burdet, B; De Laurentiis, A; Fernandez-Solari, J; Mohn, C; Rettori, V; Zorrilla Zubilete, MA1
Bernardi, G; Cantarella, C; Castelli, M; Cavasinni, F; Centonze, D; De Chiara, V; Mataluni, G; Musella, A; Rossi, S1
Baufreton, J; Manuel, I; Morera-Herreras, T; Rodriguez-Puertas, R; Ruiz-Ortega, JA; Taupignon, A; Ugedo, L1
Alger, BE; Kim, J1
Bingham, B; Gorzalka, BB; Gray, JM; Hill, MN; Hillard, CJ; Lee, TT; McLaughlin, RJ; Shrestha, L; Viau, V1
Alter, BJ; Burston, JJ; Cravatt, BF; Fowler, CJ; Gereau, RW; McKinney, MK; Pertwee, RG; Ross, RA; Thors, L; Wiley, JL1
Casarotto, PC; Gomes, FV; Guimarães, FS; Resstel, LB1
McMahon, LR; Stewart, JL1
Jain, NS; Manna, SS; Umathe, SN2
Beltrame, JS; Burdet, J; Cella, M; Franchi, AM; Pardo, R; Ribeiro, ML; Sordelli, MS; Zotta, E1
Busquets-Garcia, A; de la Torre, R; Maldonado, R; Ozaita, A; Pastor, A; Puighermanal, E1
Butler, RK; Chapman, V; Doyle, KM; Finn, DP; Ford, GK; Hogan, M; Kelly, JP; Kendall, DA; Roche, M1
Astarita, G; Caprioli, G; Ciccocioppo, R; Cippitelli, A; Duranti, A; Kallupi, M; Piomelli, D; Rodrìguez de Fonseca, F; Sagratini, G; Stopponi, S; Ubaldi, M1
Boczán, J; Czikora, Á; Daragó, A; Édes, I; Lizanecz, E; Papp, Z; Tóth, A1
Bambico, FR; Gobbi, G; Gorzalka, BB; Hill, MN; Hillard, CJ; McLaughlin, RJ; Stuhr, KL1
Bouzin, C; Feron, O; Gallez, B; Hamtiaux, L; Lambert, DM; Masquelier, J; Muccioli, GG1
Dykstra, LA; Miller, LL; Picker, MJ; Schmidt, KT; Umberger, MD1
Buczynski, MW; Chang, JW; Cognetta, AB; Cravatt, BF; Lum, KM; Matthews, ML; Niessen, S; Niphakis, MJ; Parsons, LH; Wang, C1
Harding-Rose, C; Khasabov, S; Khasabova, IA; Paz, J; Seybold, VS; Simone, DA1
Alexander, SP; Barrett, DA; Bennett, AJ; Burston, J; Chapman, V; Kendall, DA; Norris, LM; Okine, BN; Patel, A; Woodhams, S1
Cooper, TB; Hungund, BL; Psychoyos, D; Tejani-Butt, SM; Vinod, KY; Xie, S1
Baranowska-Kuczko, M; Kozłowska, H; MacLean, MR; Malinowska, B1
Bowie, AG; Campbell, VA; Gowran, A; Keating, SE; Noonan, J; Tanveer, R1
Bacigaluppi, M; Bari, M; Brambilla, E; Butti, E; Cambiaghi, M; Cebrian Silla, A; Centonze, D; Comi, G; D'Adamo, P; De Ceglia, R; De Chiara, V; Garcia-Verdugo, JM; Leocani, L; Maccarrone, M; Martino, G; Musella, A; Muzio, L; Quattrini, A; Rossi, S; Teneud, L1
Barker, E; Chester, JA; Cooper, BR; Davisson, VJ; Han, B; Kirchhoff, AM; Wright, R1
Przewlocka, B; Starowicz, K1
Bradshaw, HB; Guindon, J; Hohmann, AG; Lai, Y; Takacs, SM1
Burger, F; Cravatt, B; Galan, K; Lenglet, S; Montecucco, F; Pelli, G; Soehnlein, O; Staub, C; Steffens, S; Thomas, A1
Avraham, HK; Li, H; Makriyannis, A; Seng, S; Vadivel, SK; Whitten, KM; Wood, JT1
Giuffrida, A; Martinez, AA; Seillier, A1
Cristino, L; De Petrocellis, L; Di Marzo, V; Korostynski, M; Makuch, W; Malek, N; Petrosino, S; Przewlocka, B; Slezak, M; Starowicz, K; Zychowska, M1
Burlakova, N; Coicou, L; Harding-Rose, C; Holman, M; Khasabova, IA; Morse, T; Seybold, VS; Simone, DA1
Aliczki, M; Goldberg, SR; Haller, J; Panlilio, LV; Pelczer, KG1
Antunes-Rodrigues, J; Elias, LL; Ruginsk, SG; Uchoa, ET1
Boccella, S; Comelli, F; Costa, B; De Chiaro, M; Di Marzo, V; Guida, F; Maione, S; Morera, E; Ortar, G; Piscitelli, F; Verde, R1
Centonze, D; Laricchiuta, D; Petrosini, L1
Aliczki, M; Balogh, Z; Haller, J; Kantor, S; Pelczer, KG; Spitzer, K1
Abdullah, RA; Imhof, E; Lichtman, AH; Limebeer, CL; Parker, LA; Rock, EM; Wang, K1
Bindila, L; Fleischmann, BK; Lerner, R; Lutz, B; Matthey, M; Wenzel, D; Zimmer, A1
Cinar, R; Godlewski, G; Jourdan, T; Kunos, G; Lin, Y; Liu, J; Ntambi, JM; Xiong, K1
Becker, A; Hoyer, FF; Kebschull, M; Khoury, M; Lerner, R; Lütjohann, D; Lutz, B; Nickenig, G; Schott, H; Slomka, H; Wojtalla, A; Zimmer, A1
Abdullah, RA; Kwilasz, AJ; Lichtman, AH; Negus, SS; Poklis, JL1
Basavarajappa, BS; Nagre, NN; Subbanna, S; Xie, S1
Bystrowska, B; Filip, M; Gawliński, D; Pomierny, B; Smaga, I; Stankowicz, P1
Al Kury, LT; Ali, RM; Galadari, S; Howarth, FC; Oz, M; Rajesh, M; Shuba, YM; Thayyullathil, FT; Yang, KH1
Chavant, F; Duranti, A; Francheteau, M; Gennequin, B; Maccarrone, M; Makriyannis, A; Nader, J; Rapino, C; Solinas, M; Thiriet, N1
Cravatt, BF; Germano, P; Hama, AT; Milne, GT; Pearson, JP; Sagen, J; Varghese, MS1
Bader, M; Brosnihan, KB; Dechend, R; Howlett, AC; McGee, CM; Pulgar, VM; Varagic, J; Yamaleyeva, LM1
Drew, GM; Lau, BK; Mitchell, VA; Vaughan, CW1
Impastato, RA; Katz, PS; Molina, PE; Rogers, EK; Sulzer, JK; Teng, SX1
Abels, C; Chicca, A; Gertsch, J; Nicolussi, S; Rau, M; Rihs, S; Soeberdt, M1
Aguiar, DC; Hott, SC; Moreira, FA; Resstel, LB; Viana, TG1
de Ceballos, ML; Giusto, NM; Martín-Moreno, AM; Pascual, AC; Pasquaré, SJ1
Atsak, P; Campolongo, P; Cuomo, V; Hauer, D; McGaugh, JL; Morena, M; Peloso, A; Ratano, P; Roozendaal, B; Schelling, G; Trabace, L; Trezza, V1
Khasabova, IA; Simone, DA; Uhelski, ML1
Chauvet, C; Duranti, A; Lardeux, MV; Nicolas, C; Solinas, M; Thiriet, N1
Bedse, G; Bellomo, A; Cassano, T; Cifani, C; Duranti, A; Gaetani, S; Lavecchia, MA; Micioni Di Bonaventura, MV; Pace, L; Romano, A; Tempesta, B1
Bastos, JR; Batista, LA; Moreira, FA1
Camargo, LH; Cunha, FQ; Gomes, FV; Guimarães, FS; Joca, SR; Lisboa, SF; Resstel, LB; Silva, AL; Uliana, DL1
Vann, RE; Walentiny, DM; Wiley, JL1
Binkowski, M; Czaja, M; Di Marzo, V; Kolosowska, N; Makuch, W; Malek, N; Morera, E; Mrugala, M; Przewlocka, B; Starowicz, K1
Markert, A; Nozaki, C; Zimmer, A1
Campolongo, P; Cuomo, V; Hill, MN; Manduca, A; Morena, M; Palmery, M; Servadio, M; Trabace, L; Trezza, V; Vanderschuren, LJ1
Krych, L; Moulton, K; Qin, M; Smith, CB; Xia, Z; Zeidler, Z1
Hinz, B; Ivanov, I; Peters, K; Ramer, R; Salamon, A; Wollank, Y1
Kregiel, J; Malek, N; Popik, P; Rygula, R; Starowicz, K1
Congiu, C; Deplano, A; Fowler, CJ; Fredriksson Sundbom, M; Gouveia-Figueira, S; Hashemian, S; Karlsson, J; Onnis, V; Svensson, M1
Cox, CD; Gall, CM; Geschwind, DH; Karsten, CA; Lee, D; Peñagarikano, O; Piomelli, D; Wei, D1
Aguilar, DD; Giuffrida, A; Lodge, DJ1
Gray, JM; Hill, MN; McLaughlin, RJ; Verlezza, S; Walker, CD1
Goldberg, SR; Justinova, Z; Makriyannis, A; Redhi, GH; Scherma, M; Schindler, CW; Vadivel, SK1
Aliczki, M; Baranyi, M; Barna, I; Goldberg, SR; Haller, J; Sperlagh, B; Till, I1
Alapafuja, SO; Bergman, J; Kangas, BD; Leonard, MZ; Makriyannis, A; Nikas, SP; Shukla, VG1
Forget, B; Gamaleddin, I; Goldberg, SR; Guranda, M; Le Foll, B1
Aymerich, MS; Celorrio, M; Echeverry-Alzate, V; Fernández-Suárez, D; Franco, R; Hillard, CJ; López-Moreno, JA; Maldonado, R; Oyarzábal, J; Ramírez, MJ; Rojo-Bustamante, E1
Campolongo, P; Gray, JM; Hill, MN; Leitl, KD; Morena, M; Vecchiarelli, HA1
Abdullah, RA; Cabrera, R; Cravatt, BF; Ghosh, S; Lichtman, AH; Maldonado, RL; Mustafa, M; Niphakis, MJ; Wilkerson, JL1
Barrett, DA; Couch, DG; Karwad, MA; Larvin, M; Lund, JN; O'Sullivan, SE; Sarmad, S; Theophilidou, E; Wright, KL1
Gupta, K; Simone, DA; Uhelski, ML1
Finn, DP; Flannery, LE; Henry, RJ; Kerr, DM; Roche, M1
Genewsky, A; Heinz, DE; Wotjak, CT1
Abouabdellah, A; Bergis, OE; Cohen, C; Dargazanli, G; Fauchey, V; Griebel, G; Lopez-Grancha, M; Pichat, P; Slowinski, F; Stemmelin, J1
Akirav, I; Fidelman, S; Hillard, CJ; Lange, R; Mizrachi Zer-Aviv, T1
Gong, DY; Hai, KR; Jiang, HX; Ke, BW; Liu, J; Ma, G; Yang, Z; Zhou, C1
Cuccurazzu, B; Grilli, M; Nazzaro, C; Parolaro, D; Prini, P; Rubino, T; Tonini, R; Trusel, M; Zamberletti, E1
Cavin, JB; Cravatt, BF; Hill, MN; Keenan, CM; Lau, DJ; Makriyannis, A; Morena, M; Sharkey, KA; Sticht, MA; Vemuri, VK1
Blanco, E; Fernández-Arjona, MDM; Grondona, JM; López-Ávalos, MD; Pavón, FJ; Rivera, P; Rodríguez de Fonseca, F; Serrano, A; Silva-Peña, D; Suárez, J; Vargas, A1
Biernacki, M; Jastrząb, A; Malinowska, B; Remiszewski, P; Skrzydlewska, E; Timoszuk, M; Toczek, M1
Aliczki, M; Balogh, Z; Biro, L; Haller, J; Szente, L; Varga, ZK1
Aguilera-Portillo, G; Colonnello, A; Galván-Arzate, S; Kotlar, I; Pedraza-Chaverri, J; Rangel-López, E; Santamaría, A; Serratos, IN; Túnez, I; Wajner, M1
Correa, FM; Fassini, A; Guimarães, FS; Hartmann, A; Lisboa, SF; Resstel, LB; Scopinho, A1
Campolongo, P; Colucci, P; Hill, MN; Mancini, GF; Morena, M; Palmery, M; Puglisi-Allegra, S; Santori, A; Trezza, V1
Chen, PS; Chu, MC; Lee, CW; Lin, HC; Lu, TY; Wu, HF1
Akirav, I; Maymon, N; Mizrachi Zer-Aviv, T; Sabban, EL1
Carnevali, L; Ferlenghi, F; Mor, M; Rivara, S; Sgoifo, A; Spadoni, G; Statello, R; Vacondio, F1
Angelucci, CB; Ballone, A; Dainese, E; De Fabritiis, G; Dufrusine, B; Fezza, F; Maccarrone, M; Oddi, S; Sabatucci, A; Simonetti, M1
Abohalaka, R; Bozkurt, TE; Nemutlu, E; Onder, SC; Sahin-Erdemli, I1
Baranowska-Kuczko, M; Biernacki, M; Niklińska, GN; Skrzydlewska, E1
Bales, KL; Simmons, TC; Singh, ALK1
Baranowska-Kuczko, M; Biernacki, M; Harasim-Symbor, E; Kasacka, I; Kloza, M; Kozłowska, H; Malinowska, B1
Gordon, RY; Khutsian, SS; Kitchigina, VF; Mikheeva, IB; Shubina, LV1
Armeli, F; Bisogno, T; Businaro, R; Coccurello, R; D'Erme, M; De Caris, MG; Grieco, M; Maccarrone, M; Maggi, E; Mancini, P1

Reviews

1 review(s) available for carbamates and anandamide

ArticleYear
Modulation of neuropathic-pain-related behaviour by the spinal endocannabinoid/endovanilloid system.
    Philosophical transactions of the Royal Society of London. Series B, Biological sciences, 2012, Dec-05, Volume: 367, Issue:1607

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acid; Arachidonic Acids; Behavior; Benzamides; Carbamates; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Glycerides; Humans; Microglia; Neuralgia; Palmitic Acids; Peripheral Nerve Injuries; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Spinal Cord Injuries; TRPV Cation Channels

2012

Other Studies

150 other study(ies) available for carbamates and anandamide

ArticleYear
Unique analogues of anandamide: arachidonyl ethers and carbamates and norarachidonyl carbamates and ureas.
    Journal of medicinal chemistry, 1999, Jun-03, Volume: 42, Issue:11

    Topics: Analgesics, Non-Narcotic; Animals; Arachidonic Acids; Body Temperature; Cannabinoids; Carbamates; Endocannabinoids; Hydrolysis; Ligands; Mice; Motor Activity; Polyunsaturated Alkamides; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Structure-Activity Relationship; Urea

1999
Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors.
    Journal of medicinal chemistry, 2003, Jun-05, Volume: 46, Issue:12

    Topics: Amidohydrolases; Arachidonic Acids; Biological Transport; Biphenyl Compounds; Brain; Carbamates; Drug Design; Endocannabinoids; Enzyme Inhibitors; Esters; Humans; In Vitro Techniques; Models, Molecular; Molecular Conformation; Polyunsaturated Alkamides; Quantitative Structure-Activity Relationship; Tumor Cells, Cultured

2003
Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension.
    Circulation, 2004, Oct-05, Volume: 110, Issue:14

    Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzyl Compounds; Blood Pressure; Camphanes; Carbamates; Dronabinol; Endocannabinoids; Endothelium, Vascular; Hypertension; Male; Models, Cardiovascular; Myocardial Contraction; Myocardium; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred Dahl; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Up-Regulation; Vascular Resistance; Vasodilation; Ventricular Function, Left

2004
Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3'-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 313, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Body Temperature; Brain; Calcium Channel Blockers; Carbamates; Chromatography, High Pressure Liquid; Drug Synergism; Duodenum; Endocannabinoids; Enzyme Inhibitors; Feeding Behavior; Male; Mass Spectrometry; Mice; Mice, Inbred C57BL; Oleic Acids; Polyunsaturated Alkamides; PPAR alpha; Rats; Rats, Wistar

2005
Involvement of N-acylethanolamine-hydrolyzing acid amidase in the degradation of anandamide and other N-acylethanolamines in macrophages.
    Biochimica et biophysica acta, 2005, Oct-01, Volume: 1736, Issue:3

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Brain; Carbamates; Cell Line; Cell Line, Tumor; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Gene Expression; Humans; Kidney; Liver; Lung; Macrophages; Macrophages, Peritoneal; Male; Mice; Mice, Inbred C57BL; Polyunsaturated Alkamides; Rats; Rats, Wistar; U937 Cells

2005
Endocannabinoids at the spinal level regulate, but do not mediate, nonopioid stress-induced analgesia.
    Neuropharmacology, 2006, Volume: 50, Issue:3

    Topics: Analgesia; Analysis of Variance; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Glycerides; Male; Mass Spectrometry; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Reaction Time; Rimonabant; Serotonin; Spinal Cord; Stress, Psychological; Time Factors

2006
Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis.
    Proceedings of the National Academy of Sciences of the United States of America, 2005, Dec-20, Volume: 102, Issue:51

    Topics: Animals; Antidepressive Agents; Arachidonic Acids; Behavior, Animal; Benzamides; Brain; Cannabinoid Receptor Agonists; Carbamates; Dronabinol; Endocannabinoids; Hydrolysis; Male; Mice; Mice, Inbred C57BL; Neurons; Norepinephrine; Polyunsaturated Alkamides; Rats; Receptors, Cannabinoid; Serotonin

2005
A novel scintillation proximity assay for fatty acid amide hydrolase compatible with inhibitor screening.
    Analytical biochemistry, 2006, Jul-01, Volume: 354, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Binding Sites; Calcium Channel Blockers; Carbamates; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endocannabinoids; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Ligands; Microsomes; Polyunsaturated Alkamides; Scintillation Counting; Wheat Germ Agglutinins

2006
Evaluation of the role of nicotinic acetylcholine receptor subtypes and cannabinoid system in the discriminative stimulus effects of nicotine in rats.
    European journal of pharmacology, 2006, Jul-01, Volume: 540, Issue:1-3

    Topics: Aconitine; Animals; Arachidonic Acids; Azetidines; Benzamides; Benzoxazines; Camphanes; Cannabinoid Receptor Antagonists; Carbamates; Cyclohexanols; Dihydro-beta-Erythroidine; Discrimination Learning; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Male; Mecamylamine; Morpholines; Naphthalenes; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Polyunsaturated Alkamides; Pyrazoles; Pyridines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Nicotinic

2006
Anandamide administration alone and after inhibition of fatty acid amide hydrolase (FAAH) increases dopamine levels in the nucleus accumbens shell in rats.
    Journal of neurochemistry, 2006, Volume: 98, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Calcium; Cannabinoids; Carbamates; Data Interpretation, Statistical; Dopamine; Endocannabinoids; Enzyme Inhibitors; Male; Microdialysis; Nucleus Accumbens; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission; Tetrodotoxin; TRPV Cation Channels

2006
Effects of endocannabinoid neurotransmission modulators on brain stimulation reward.
    Psychopharmacology, 2006, Volume: 188, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzyl Compounds; Brain; Cannabinoid Receptor Modulators; Carbamates; Conditioning, Operant; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Injections, Intraperitoneal; Male; Medial Forebrain Bundle; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Protease Inhibitors; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement Schedule; Reward; Rimonabant; Self Stimulation; Synaptic Transmission

2006
Effects of the FAAH inhibitor, URB597, and anandamide on lithium-induced taste reactivity responses: a measure of nausea in the rat.
    Psychopharmacology, 2007, Volume: 190, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Association Learning; Avoidance Learning; Benzamides; Carbamates; Conditioning, Classical; Dose-Response Relationship, Drug; Endocannabinoids; Injections, Intraperitoneal; Lithium Chloride; Male; Nausea; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Vomiting

2007
The endogenous cannabinoid anandamide produces delta-9-tetrahydrocannabinol-like discriminative and neurochemical effects that are enhanced by inhibition of fatty acid amide hydrolase but not by inhibition of anandamide transport.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Biological Transport, Active; Brain Chemistry; Carbamates; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Furans; Hallucinogens; Injections, Intraperitoneal; Injections, Intravenous; Male; Microdialysis; Nucleus Accumbens; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reinforcement Schedule; TRPV Cation Channels

2007
Effects of inhibition of fatty acid amide hydrolase vs. the anandamide membrane transporter on TRPV1-mediated calcium responses in adult DRG neurons; the role of CB receptors.
    The European journal of neuroscience, 2006, Volume: 24, Issue:12

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Calcium; Capsaicin; Carbamates; Cells, Cultured; Dopamine; Drug Interactions; Endocannabinoids; Fura-2; Furans; Ganglia, Spinal; Male; Membrane Potentials; Membrane Transport Proteins; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2006
Endothelium-dependent metabolism by endocannabinoid hydrolases and cyclooxygenases limits vasorelaxation to anandamide and 2-arachidonoylglycerol.
    British journal of pharmacology, 2007, Volume: 150, Issue:5

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Glycerides; Hydrolases; In Vitro Techniques; Lectins; Lectins, C-Type; Male; Membrane Proteins; Mesenteric Artery, Superior; Organophosphonates; Polyunsaturated Alkamides; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Receptors, Cell Surface; Vasodilation; Vasodilator Agents

2007
Pharmacological characterization of receptor types mediating the dilator action of anandamide on blood vessels of the rat knee joint.
    Life sciences, 2007, Mar-27, Volume: 80, Issue:16

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Blood Vessels; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Flurbiprofen; Hindlimb; Indoles; Joints; Morpholines; Polyunsaturated Alkamides; Pyrazoles; Rats; Regional Blood Flow; TRPV Cation Channels; Vasodilation

2007
Evaluation of fatty acid amide hydrolase inhibition in murine models of emotionality.
    Psychopharmacology, 2007, Volume: 192, Issue:1

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Emotions; Endocannabinoids; Enzyme Inhibitors; Lighting; Maze Learning; Mice; Mice, Knockout; Polyunsaturated Alkamides; Pyridines; Signal Transduction

2007
The 'specific' tyrosine kinase inhibitor genistein inhibits the enzymic hydrolysis of anandamide: implications for anandamide uptake.
    British journal of pharmacology, 2007, Volume: 150, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Brain; Carbamates; Cell Line, Tumor; Endocannabinoids; Genistein; Hydrolysis; Mice; Nystatin; Polyunsaturated Alkamides; Progesterone; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Rats

2007
Interactions of cannabidiol with endocannabinoid signalling in hippocampal tissue.
    The European journal of neuroscience, 2007, Volume: 25, Issue:7

    Topics: Animals; Arachidonic Acids; Benzamides; Calcium; Cannabidiol; Cannabinoid Receptor Modulators; Carbamates; Cells, Cultured; Dronabinol; Endocannabinoids; Estrenes; Glutamic Acid; Glycerides; Hippocampus; Humans; Morpholines; Pertussis Toxin; Phosphodiesterase Inhibitors; Polyunsaturated Alkamides; Pyrazoles; Pyrrolidinones; Rats; Receptor, Cannabinoid, CB1; Signal Transduction

2007
Involvement of the endocannabinoid system in retinal damage after high intraocular pressure-induced ischemia in rats.
    Investigative ophthalmology & visual science, 2007, Volume: 48, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cell Count; Chromatography, High Pressure Liquid; Endocannabinoids; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Hydrolysis; Intraocular Pressure; Male; Ocular Hypertension; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reperfusion Injury; Retinal Diseases; Retinal Ganglion Cells; Retinal Vessels; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Thy-1 Antigens; TRPV Cation Channels

2007
Inhibition of the cellular uptake of anandamide by genistein and its analogue daidzein in cells with different levels of fatty acid amide hydrolase-driven uptake.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: 3T3-L1 Cells; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Biological Transport; Carbamates; Cell Line, Tumor; Dose-Response Relationship, Drug; Endocannabinoids; Genistein; Humans; Hydrogen-Ion Concentration; Hydrolysis; Isoflavones; Male; Mice; Molecular Structure; Polyunsaturated Alkamides; Protein Kinase Inhibitors; Rats; Tritium

2007
Endocannabinoid modulation of male rat sexual behavior.
    Psychopharmacology, 2008, Volume: 198, Issue:4

    Topics: Amidohydrolases; Animals; Appetitive Behavior; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Consummatory Behavior; Dose-Response Relationship, Drug; Ejaculation; Endocannabinoids; Enzyme Inhibitors; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Sexual Behavior, Animal

2008
Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Aorta, Abdominal; Apamin; Arachidonic Acids; Benzamides; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Charybdotoxin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Isoindoles; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sulfonamides; Vasodilation

2007
Reduced anxiety-like behaviour induced by genetic and pharmacological inhibition of the endocannabinoid-degrading enzyme fatty acid amide hydrolase (FAAH) is mediated by CB1 receptors.
    Neuropharmacology, 2008, Volume: 54, Issue:1

    Topics: Amidohydrolases; Analysis of Variance; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Disease Models, Animal; Endocannabinoids; Glycerides; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2008
Anti-dyskinetic effects of cannabinoids in a rat model of Parkinson's disease: role of CB(1) and TRPV1 receptors.
    Experimental neurology, 2007, Volume: 208, Issue:1

    Topics: Amidohydrolases; Animals; Antiparkinson Agents; Arachidonic Acids; Basal Ganglia; Benzamides; Benzoxazines; Cannabinoids; Capsaicin; Carbamates; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Endocannabinoids; Levodopa; Male; Morpholines; Naphthalenes; Oxidopamine; Parkinson Disease, Secondary; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2007
The endogenous cannabinoid anandamide has effects on motivation and anxiety that are revealed by fatty acid amide hydrolase (FAAH) inhibition.
    Neuropharmacology, 2008, Volume: 54, Issue:1

    Topics: Amidohydrolases; Analgesics; Analysis of Variance; Animals; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzoxazines; Carbamates; Conditioning, Operant; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Inhibitors; Male; Morpholines; Motivation; Motor Activity; Naphthalenes; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Time Factors

2008
Role in anxiety behavior of the endocannabinoid system in the prefrontal cortex.
    Cerebral cortex (New York, N.Y. : 1991), 2008, Volume: 18, Issue:6

    Topics: Animals; Anxiety; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Dose-Response Relationship, Drug; Endocannabinoids; Male; Polyunsaturated Alkamides; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1

2008
New N-arachidonoylserotonin analogues with potential "dual" mechanism of action against pain.
    Journal of medicinal chemistry, 2007, Dec-27, Volume: 50, Issue:26

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Biphenyl Compounds; Brain; Calcium; Carbamates; Cell Line; Endocannabinoids; Humans; Hydrolysis; Hyperalgesia; Indoles; Mice; Pain; Pain Measurement; Polyunsaturated Alkamides; Rats; Serotonin; Structure-Activity Relationship; TRPV Cation Channels

2007
CB1 receptor-mediated control of the release of endocannabinoids (as assessed by microdialysis coupled with LC/MS) in the rat hypothalamus.
    The European journal of neuroscience, 2007, Volume: 26, Issue:12

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Cannabinoid Receptor Modulators; Cannabinoids; Carbamates; Chromatography, Liquid; Endocannabinoids; Extracellular Fluid; Glycerides; Hypothalamus; Male; Microdialysis; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Potassium; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Tandem Mass Spectrometry

2007
Increase of brain endocannabinoid anandamide levels by FAAH inhibition and alcohol abuse behaviours in the rat.
    Psychopharmacology, 2008, Volume: 198, Issue:4

    Topics: Adrenergic alpha-Antagonists; Alcohol Drinking; Alcoholism; Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Benzamides; Brain Chemistry; Carbamates; Conditioning, Operant; Cues; Electroshock; Endocannabinoids; Enzyme Inhibitors; Extinction, Psychological; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Recurrence; Reinforcement Schedule; Self Administration; Stress, Psychological; Yohimbine

2008
N-arachidonylethanolamide-induced increase in aqueous humor outflow facility.
    Investigative ophthalmology & visual science, 2008, Volume: 49, Issue:10

    Topics: Amidohydrolases; Animals; Anterior Eye Segment; Aqueous Humor; Arachidonic Acids; Benzamides; Blotting, Western; Camphanes; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Carbamates; Chromatography, Thin Layer; Endocannabinoids; Organ Culture Techniques; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Rimonabant; Swine; Trabecular Meshwork

2008
Does the hydrolysis of 2-arachidonoylglycerol regulate its cellular uptake?
    Pharmacological research, 2008, Volume: 58, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Biphenyl Compounds; Cannabinoid Receptor Modulators; Carbamates; Cell Line, Tumor; Endocannabinoids; Glycerides; Humans; Hydrolysis; Polyunsaturated Alkamides

2008
Activation of cannabinoid CB1 receptors in the dorsolateral periaqueductal gray induces anxiolytic effects in rats submitted to the Vogel conflict test.
    European journal of pharmacology, 2008, Sep-28, Volume: 593, Issue:1-3

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Arachidonic Acids; Benzamides; Carbamates; Conflict, Psychological; Data Interpretation, Statistical; Drinking; Endocannabinoids; Enzyme Inhibitors; Male; Pain Measurement; Periaqueductal Gray; Polyunsaturated Alkamides; Rats; Rats, Wistar; Reaction Time; Receptor, Cannabinoid, CB1

2008
Inhibition of anandamide hydrolysis by cyclohexyl carbamic acid 3'-carbamoyl-3-yl ester (URB597) reverses abuse-related behavioral and neurochemical effects of nicotine in rats.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Conditioning, Psychological; Dopamine; Endocannabinoids; Hydrolysis; Male; Motor Activity; Nicotine; Nucleus Accumbens; Polyunsaturated Alkamides; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Reward; Self Administration; Tobacco Use Disorder

2008
Modulation of opioids via protection of anandamide degradation by fatty acid amide hydrolase.
    European journal of pharmacology, 2008, Dec-14, Volume: 600, Issue:1-3

    Topics: Amidohydrolases; Analgesics, Opioid; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Dose-Response Relationship, Drug; Drug Therapy, Combination; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Mice, Inbred ICR; Mice, Knockout; Morphine; Pain; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Receptors, Opioid, kappa

2008
Fatty acid amide hydrolase inhibition heightens anandamide signaling without producing reinforcing effects in primates.
    Biological psychiatry, 2008, Dec-01, Volume: 64, Issue:11

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Brain; Cannabinoid Receptor Modulators; Carbamates; Chromatography, Liquid; Cocaine; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Reinforcement Schedule; Reinforcement, Psychology; Saimiri; Self Administration

2008
Endocannabinoid-mediated enhancement of fear-conditioned analgesia in rats: opioid receptor dependency and molecular correlates.
    Pain, 2008, Volume: 140, Issue:3

    Topics: Amidohydrolases; Amygdala; Analgesia; Animals; Arachidonic Acids; Avoidance Learning; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Conditioning, Psychological; Endocannabinoids; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Fear; Male; Narcotic Antagonists; Neural Inhibition; Pain; Pain Measurement; Polyunsaturated Alkamides; Rats; Receptor, Cannabinoid, CB1; Receptors, Opioid; Signal Transduction

2008
The endocannabinoid system in bull sperm and bovine oviductal epithelium: role of anandamide in sperm-oviduct interaction.
    Reproduction (Cambridge, England), 2009, Volume: 137, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Blotting, Western; Camphanes; Carbamates; Cattle; Endocannabinoids; Epithelium; Fallopian Tubes; Female; Immunohistochemistry; Male; Microscopy, Fluorescence; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Sperm Motility; Sperm-Ovum Interactions; Spermatozoa

2009
Long-term consequences of URB597 administration during adolescence on cannabinoid CB1 receptor binding in brain areas.
    Brain research, 2009, Feb-27, Volume: 1257

    Topics: Aging; Analysis of Variance; Animals; Arachidonic Acids; Autoradiography; Benzamides; Brain; Carbamates; Endocannabinoids; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2009
Acute hypertension reveals depressor and vasodilator effects of cannabinoids in conscious rats.
    British journal of pharmacology, 2009, Volume: 156, Issue:1

    Topics: Acute Disease; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Blood Pressure; Cannabinoids; Carbamates; Consciousness; Endocannabinoids; Hindlimb; Hypertension; Infusions, Intravenous; Injections, Intravenous; Male; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Renal Circulation; Splanchnic Circulation; Vascular Resistance; Vasodilation

2009
The FAAH inhibitor URB-597 interferes with cisplatin- and nicotine-induced vomiting in the Suncus murinus (house musk shrew).
    Physiology & behavior, 2009, Apr-20, Volume: 97, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Cisplatin; Drug Interactions; Endocannabinoids; Female; Male; Nicotine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Shrews; Vomiting

2009
The endocannabinoid anandamide is a precursor for the signaling lipid N-arachidonoyl glycine by two distinct pathways.
    BMC biochemistry, 2009, May-21, Volume: 10

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Brain; Brain Chemistry; Carbamates; Cell Line, Tumor; Endocannabinoids; Glycine; Lipid Metabolism; Male; Metabolic Networks and Pathways; Mice; Mice, Knockout; Oxidation-Reduction; Polyunsaturated Alkamides; Rats; Recombinant Proteins

2009
Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 330, Issue:3

    Topics: Amidohydrolases; Analgesics, Non-Narcotic; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Cold Temperature; Endocannabinoids; Enzyme Inhibitors; Glycerides; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Monoacylglycerol Lipases; Narcotic Antagonists; Pain; Pain Measurement; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; TRPV Cation Channels

2009
Anandamide increases the differentiation of rat adipocytes and causes PPARgamma and CB1 receptor upregulation.
    Obesity (Silver Spring, Md.), 2009, Volume: 17, Issue:10

    Topics: Adipocytes; Adipose Tissue; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Blotting, Western; Carbamates; Cell Differentiation; Cyclooxygenase 2; Endocannabinoids; Enzyme Inhibitors; Flow Cytometry; Indomethacin; Male; Polyunsaturated Alkamides; PPAR gamma; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Reverse Transcriptase Polymerase Chain Reaction; Up-Regulation

2009
Suppression of amygdalar endocannabinoid signaling by stress contributes to activation of the hypothalamic-pituitary-adrenal axis.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:13

    Topics: Amidohydrolases; Amygdala; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Corticosterone; Dronabinol; Drug Interactions; Endocannabinoids; Hypothalamo-Hypophyseal System; Male; Microinjections; Piperidines; Pituitary-Adrenal System; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Restraint, Physical; Signal Transduction; Stress, Psychological

2009
Effect of nitric oxide donors on membrane tritium accumulation of endocannabinoids and related endogenous lipids.
    European journal of pharmacology, 2009, Oct-25, Volume: 621, Issue:1-3

    Topics: Amides; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cell Line; Cell Membrane; Cyclic N-Oxides; Endocannabinoids; Ethanolamines; Free Radical Scavengers; Glycerides; Imidazoles; Lipid Metabolism; Mice; Nitric Oxide; Nitric Oxide Donors; Palmitic Acids; Polyunsaturated Alkamides; Rats; Signal Transduction; Tritium

2009
Dual blockade of FAAH and MAGL identifies behavioral processes regulated by endocannabinoid crosstalk in vivo.
    Proceedings of the National Academy of Sciences of the United States of America, 2009, Dec-01, Volume: 106, Issue:48

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Carbamates; Carboxylic Ester Hydrolases; Endocannabinoids; Glycerides; Mice; Molecular Structure; Monoacylglycerol Lipases; Motor Activity; Pain Measurement; Piperazines; Piperidines; Polyunsaturated Alkamides

2009
The endogenous cannabinoid, anandamide, inhibits dopamine transporter function by a receptor-independent mechanism.
    Journal of neurochemistry, 2010, Volume: 112, Issue:6

    Topics: Alanine; Arachidonic Acids; Benzamides; Calcium; Cannabinoid Receptor Modulators; Carbamates; Cell Line, Transformed; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Inhibitors; Humans; Luminescent Proteins; Microscopy, Confocal; Phenylmethylsulfonyl Fluoride; Polyunsaturated Alkamides; Receptors, Cannabinoid; Receptors, Scavenger; Silicone Elastomers; Time Factors; Transfection; Tritium; Tropanes

2010
The hypothalamic endocannabinoid system participates in the secretion of oxytocin and tumor necrosis factor-alpha induced by lipopolysaccharide.
    Journal of neuroimmunology, 2010, Apr-15, Volume: 221, Issue:1-2

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Enzyme-Linked Immunosorbent Assay; Gene Expression Regulation; Hypothalamus; Indoles; Lipopolysaccharides; Male; Nitric Oxide; Oxytocin; Polyunsaturated Alkamides; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Tumor Necrosis Factor-alpha

2010
Transient receptor potential vanilloid 1 channels control acetylcholine/2-arachidonoylglicerol coupling in the striatum.
    Neuroscience, 2010, May-19, Volume: 167, Issue:3

    Topics: Acetylcholine; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Corpus Striatum; Endocannabinoids; Enzyme Inhibitors; gamma-Aminobutyric Acid; Glycerides; Inhibitory Postsynaptic Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Agonists; Neural Inhibition; Organ Culture Techniques; Polyunsaturated Alkamides; Receptor, Metabotropic Glutamate 5; Receptor, Muscarinic M1; Receptors, Metabotropic Glutamate; Sensory System Agents; Synaptic Transmission; TRPV Cation Channels

2010
Regulation of subthalamic neuron activity by endocannabinoids.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:9

    Topics: Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cerebral Cortex; Dose-Response Relationship, Drug; Dronabinol; Electrophysiology; Endocannabinoids; Globus Pallidus; Immunohistochemistry; Injections, Intraventricular; Male; Microinjections; Neurons; Piperidines; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Subthalamic Nucleus

2010
Reduction in endocannabinoid tone is a homeostatic mechanism for specific inhibitory synapses.
    Nature neuroscience, 2010, Volume: 13, Issue:5

    Topics: Agatoxins; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Carbamates; Conotoxins; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycerides; Hippocampus; Homeostasis; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Morpholines; Naphthalenes; Nerve Net; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Polyamines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Rimonabant; Sodium Channel Blockers; Synapses; Tetrodotoxin

2010
Endogenous cannabinoid signaling is essential for stress adaptation.
    Proceedings of the National Academy of Sciences of the United States of America, 2010, May-18, Volume: 107, Issue:20

    Topics: Adaptation, Physiological; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Corticosterone; Endocannabinoids; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Signal Transduction; Stress, Physiological

2010
Biochanin A, a naturally occurring inhibitor of fatty acid amide hydrolase.
    British journal of pharmacology, 2010, Volume: 160, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Brain; Cannabinoid Receptor Antagonists; Carbamates; Cell Line, Transformed; Chlorocebus aethiops; COS Cells; Drug Interactions; Endocannabinoids; Extracellular Signal-Regulated MAP Kinases; Formaldehyde; Genistein; Humans; Isoflavones; Liver; Mice; Mice, Inbred ICR; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats

2010
Facilitation of CB1 receptor-mediated neurotransmission decreases marble burying behavior in mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2011, Mar-30, Volume: 35, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Carbamates; Drug Interactions; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Morpholines; Motor Activity; Naphthalenes; Obsessive-Compulsive Disorder; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Synaptic Transmission

2011
The fatty acid amide hydrolase inhibitor URB 597: interactions with anandamide in rhesus monkeys.
    British journal of pharmacology, 2011, Volume: 164, Issue:2b

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Discrimination, Psychological; Dronabinol; Drug Interactions; Drug Therapy, Combination; Endocannabinoids; Female; Macaca mulatta; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rimonabant

2011
Involvement of endocannabinoids in antidepressant and anti-compulsive effect of fluoxetine in mice.
    Behavioural brain research, 2011, Sep-30, Volume: 223, Issue:1

    Topics: Animals; Antidepressive Agents; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Compulsive Behavior; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Endocannabinoids; Fluoxetine; Injections, Intraventricular; Male; Mice; Motor Activity; Piperidines; Polyunsaturated Alkamides; Pyrazoles

2011
The effect of anandamide on uterine nitric oxide synthase activity depends on the presence of the blastocyst.
    PloS one, 2011, Apr-29, Volume: 6, Issue:4

    Topics: Animals; Arachidonic Acids; Benzamides; Blastocyst; Cannabinoid Receptor Modulators; Carbamates; Embryo Implantation; Endocannabinoids; Female; Immunohistochemistry; Nitric Oxide Synthase; Polymerase Chain Reaction; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Uterus

2011
Differential role of anandamide and 2-arachidonoylglycerol in memory and anxiety-like responses.
    Biological psychiatry, 2011, Sep-01, Volume: 70, Issue:5

    Topics: Amidohydrolases; Analgesics; Animals; Anti-Anxiety Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Antagonists; Carbamates; Drug Tolerance; Endocannabinoids; Glycerides; Hippocampus; Maze Learning; Mice; Mice, Inbred Strains; Mice, Knockout; Monoacylglycerol Lipases; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Receptors, Cannabinoid; Recognition, Psychology; TOR Serine-Threonine Kinases

2011
Fear-induced suppression of nociceptive behaviour and activation of Akt signalling in the rat periaqueductal grey: role of fatty acid amide hydrolase.
    Journal of psychopharmacology (Oxford, England), 2012, Volume: 26, Issue:1

    Topics: Amidohydrolases; Analgesia; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Conditioning, Psychological; Endocannabinoids; Ethanolamines; Exploratory Behavior; Fear; Formaldehyde; Hippocampus; Male; Motor Activity; Nociception; Pain; Periaqueductal Gray; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-akt; Rats; Signal Transduction

2012
Endocannabinoid regulation of acute and protracted nicotine withdrawal: effect of FAAH inhibition.
    PloS one, 2011, Volume: 6, Issue:11

    Topics: Acute Disease; Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Carbamates; Cotinine; Endocannabinoids; Glycerides; Implants, Experimental; Locomotion; Male; Maze Learning; Nicotine; Polyunsaturated Alkamides; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Tobacco Use Cessation Devices; Weight Gain

2011
Endocannabinoid analogues exacerbate marble-burying behavior in mice via TRPV1 receptor.
    Neuropharmacology, 2012, Volume: 62, Issue:5-6

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Cannabinoids; Carbamates; Endocannabinoids; Mice; Motor Activity; Polyunsaturated Alkamides; TRPV Cation Channels

2012
Vascular metabolism of anandamide to arachidonic acid affects myogenic constriction in response to intraluminal pressure elevation.
    Life sciences, 2012, Mar-10, Volume: 90, Issue:11-12

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Arterioles; Benzamides; Benzoxazines; Blood Pressure; Caproates; Capsaicin; Carbamates; Dose-Response Relationship, Drug; Endocannabinoids; Flavanones; Immunohistochemistry; In Vitro Techniques; Indomethacin; Morpholines; Muscle Contraction; Muscle, Smooth, Vascular; Naphthalenes; Polyunsaturated Alkamides; Rats

2012
Prefrontal cortical anandamide signaling coordinates coping responses to stress through a serotonergic pathway.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2012, Volume: 22, Issue:9

    Topics: Action Potentials; Adaptation, Psychological; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Endocannabinoids; Enzyme Inhibitors; Fenclonine; Glycerides; Male; Microinjections; Piperidines; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Serotonergic Neurons; Signal Transduction; Stress, Psychological

2012
The association of N-palmitoylethanolamine with the FAAH inhibitor URB597 impairs melanoma growth through a supra-additive action.
    BMC cancer, 2012, Mar-19, Volume: 12

    Topics: Amides; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cell Death; Cell Line, Tumor; Cell Survival; Disease Models, Animal; Drug Synergism; Endocannabinoids; Ethanolamines; Male; Mass Spectrometry; Melanoma, Experimental; Mice; Mice, Inbred C57BL; Palmitic Acids; Polyunsaturated Alkamides; Random Allocation; Reverse Transcriptase Polymerase Chain Reaction; Skin Neoplasms

2012
Effects of alterations in cannabinoid signaling, alone and in combination with morphine, on pain-elicited and pain-suppressed behavior in mice.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 342, Issue:1

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cyclohexanols; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Morphine; Nociception; Pain; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1

2012
Highly selective inhibitors of monoacylglycerol lipase bearing a reactive group that is bioisosteric with endocannabinoid substrates.
    Chemistry & biology, 2012, May-25, Volume: 19, Issue:5

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Enzyme Inhibitors; Glycerides; HEK293 Cells; Humans; Mice; Mice, Inbred C57BL; Models, Molecular; Monoacylglycerol Lipases; Polyunsaturated Alkamides; Rats; Rats, Wistar

2012
Cannabinoid type-1 receptor reduces pain and neurotoxicity produced by chemotherapy.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, May-16, Volume: 32, Issue:20

    Topics: Activating Transcription Factor 3; Animals; Antineoplastic Agents; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Cells, Cultured; Cisplatin; Disease Models, Animal; Drug Interactions; Endocannabinoids; Enzyme Inhibitors; Ganglia, Spinal; Hyperalgesia; Male; Mice; Mice, Inbred C3H; Morpholines; Motor Activity; Neurites; Neurotoxicity Syndromes; Peripheral Nervous System Diseases; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2012
Lack of effect of chronic pre-treatment with the FAAH inhibitor URB597 on inflammatory pain behaviour: evidence for plastic changes in the endocannabinoid system.
    British journal of pharmacology, 2012, Volume: 167, Issue:3

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Disease Models, Animal; Drug Administration Schedule; Endocannabinoids; Ethanolamines; Inflammation; Male; Oleic Acids; Pain; Palmitic Acids; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Spinal Cord

2012
Dysfunction in fatty acid amide hydrolase is associated with depressive-like behavior in Wistar Kyoto rats.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Brain; Brain-Derived Neurotrophic Factor; Cannabinoid Receptor Modulators; Carbamates; Depressive Disorder; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Frontal Lobe; Genetic Predisposition to Disease; Hippocampus; Male; Phospholipase D; Polyunsaturated Alkamides; Rats; Rats, Inbred WKY; Rats, Wistar; Receptor, Cannabinoid, CB1; Species Specificity; Swimming

2012
Endothelium-dependent mechanisms of the vasodilatory effect of the endocannabinoid, anandamide, in the rat pulmonary artery.
    Pharmacological research, 2012, Volume: 66, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amidohydrolases; Animals; Anisoles; Apamin; Arachidonic Acids; Benzamides; Benzyl Compounds; Cannabinoid Receptor Antagonists; Capsaicin; Carbamates; Charybdotoxin; Cyclohexanes; Endocannabinoids; Endothelium, Vascular; Imidazoles; Indoles; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Chloride; Prostaglandin-Endoperoxide Synthases; Pulmonary Artery; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Epoprostenol; Tetraethylammonium; TRPV Cation Channels; Vasodilation

2012
The endocannabinoid, anandamide, augments Notch-1 signaling in cultured cortical neurons exposed to amyloid-β and in the cortex of aged rats.
    The Journal of biological chemistry, 2012, Oct-05, Volume: 287, Issue:41

    Topics: Aging; Alzheimer Disease; Amyloid beta-Peptides; Amyloid Precursor Protein Secretases; Animals; Arachidonic Acids; Benzamides; Carbamates; Cells, Cultured; Cerebral Cortex; Endocannabinoids; Gene Expression Regulation, Enzymologic; Glycerides; Hippocampus; Male; Membrane Glycoproteins; Neurons; Peptide Fragments; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Notch1; Signal Transduction; Up-Regulation

2012
Subventricular zone neural progenitors protect striatal neurons from glutamatergic excitotoxicity.
    Brain : a journal of neurology, 2012, Volume: 135, Issue:Pt 11

    Topics: 4-Aminopyridine; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Corpus Striatum; Disease Models, Animal; Dronabinol; Endocannabinoids; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Ganciclovir; Glutamic Acid; Lateral Ventricles; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neural Stem Cells; Neuroprotective Agents; Polyunsaturated Alkamides; Stem Cells; Stroke

2012
Quantitative LC-MS/MS analysis of arachidonoyl amino acids in mouse brain with treatment of FAAH inhibitor.
    Analytical biochemistry, 2013, Jan-15, Volume: 432, Issue:2

    Topics: Amidohydrolases; Amino Acids; Animals; Arachidonic Acids; Benzamides; Brain; Carbamates; Chromatography, High Pressure Liquid; Endocannabinoids; Enzyme Inhibitors; gamma-Aminobutyric Acid; Glycerides; Mice; Polyunsaturated Alkamides; Tandem Mass Spectrometry

2013
Alterations in endocannabinoid tone following chemotherapy-induced peripheral neuropathy: effects of endocannabinoid deactivation inhibitors targeting fatty-acid amide hydrolase and monoacylglycerol lipase in comparison to reference analgesics following c
    Pharmacological research, 2013, Volume: 67, Issue:1

    Topics: Amidohydrolases; Analgesics; Animals; Antineoplastic Agents; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoids; Carbamates; Cisplatin; Endocannabinoids; Enzyme Inhibitors; Ganglia, Spinal; Glycerides; Hyperalgesia; Lipid Metabolism; Male; Monoacylglycerol Lipases; Peripheral Nervous System Diseases; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; RNA, Messenger; Spinal Cord; TRPV Cation Channels

2013
Fatty acid amide hydrolase deficiency enhances intraplaque neutrophil recruitment in atherosclerotic mice.
    Arteriosclerosis, thrombosis, and vascular biology, 2013, Volume: 33, Issue:2

    Topics: Amides; Amidohydrolases; Animals; Aorta; Aortic Diseases; Apolipoproteins E; Arachidonic Acids; Atherosclerosis; Benzamides; Carbamates; Cells, Cultured; Chemokine CXCL1; Cholesterol; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Genotype; Inflammation Mediators; Interferon-gamma; Matrix Metalloproteinase 9; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle, Smooth, Vascular; Neutrophil Infiltration; Neutrophils; Oleic Acids; Palmitic Acids; Phenotype; Plaque, Atherosclerotic; Polyunsaturated Alkamides; Spleen; T-Lymphocytes, Regulatory; Time Factors; Tumor Necrosis Factor-alpha

2013
Inhibition of fatty acid amide hydrolase activates Nrf2 signalling and induces heme oxygenase 1 transcription in breast cancer cells.
    British journal of pharmacology, 2013, Volume: 170, Issue:3

    Topics: Active Transport, Cell Nucleus; Amidohydrolases; Antineoplastic Agents; Arachidonic Acids; Benzamides; Breast Neoplasms; Carbamates; Cell Survival; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Induction; Enzyme Inhibitors; Female; Gene Expression Regulation, Neoplastic; Heme Oxygenase-1; Humans; MCF-7 Cells; NF-E2-Related Factor 2; Polyunsaturated Alkamides; RNA Interference; Signal Transduction; Transcription, Genetic; Transfection

2013
Phencyclidine-induced social withdrawal results from deficient stimulation of cannabinoid CB₁ receptors: implications for schizophrenia.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:9

    Topics: Amidohydrolases; Amygdala; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Cyclohexanols; Dose-Response Relationship, Drug; Endocannabinoids; Male; Phencyclidine; Piperidines; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Quinazolinones; Rats; Receptor, Cannabinoid, CB1; Receptor, Cholecystokinin B; Rimonabant; Schizophrenia; Social Behavior

2013
Full inhibition of spinal FAAH leads to TRPV1-mediated analgesic effects in neuropathic rats and possible lipoxygenase-mediated remodeling of anandamide metabolism.
    PloS one, 2013, Volume: 8, Issue:4

    Topics: Amides; Amidohydrolases; Analgesia; Animals; Arachidonate 15-Lipoxygenase; Arachidonic Acids; Benzamides; Calcium Signaling; Carbamates; Diterpenes; Endocannabinoids; Ethanolamines; Flavanones; Glycerides; HEK293 Cells; Humans; Hyperalgesia; Injections, Spinal; Lipoxygenase Inhibitors; Male; Neuralgia; Oleic Acids; Palmitic Acids; Polyunsaturated Alkamides; Posterior Horn Cells; Rats; Rats, Wistar; Sciatic Nerve; Spinal Cord; TRPV Cation Channels

2013
Increased anandamide uptake by sensory neurons contributes to hyperalgesia in a model of cancer pain.
    Neurobiology of disease, 2013, Volume: 58

    Topics: Animals; Arachidonic Acids; Benzamides; Brain Neoplasms; Cannabinoid Receptor Antagonists; Carbamates; Cells, Cultured; Coculture Techniques; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Fibrosarcoma; Fluorescent Dyes; Ganglia, Spinal; Hyperalgesia; Indoles; Lactones; Male; Mice; Mice, Inbred C3H; Pain; Pain Threshold; Polyunsaturated Alkamides; Sensory Receptor Cells; Statistics, Nonparametric; Tritium

2013
The effects of anandamide signaling enhanced by the FAAH inhibitor URB597 on coping styles in rats.
    Psychopharmacology, 2013, Volume: 230, Issue:3

    Topics: Adaptation, Psychological; Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Endocannabinoids; Male; Maze Learning; Polyunsaturated Alkamides; Rats; Rats, Wistar; Signal Transduction

2013
Anandamide modulates the neuroendocrine responses induced by extracellular volume expansion.
    Clinical and experimental pharmacology & physiology, 2013, Volume: 40, Issue:10

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Endocannabinoids; Gene Expression Regulation; Infusions, Intraventricular; Male; Median Eminence; Neuroprotective Agents; Nitrates; Oxytocin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; RNA, Messenger; Saline Solution, Hypertonic; Vasopressins

2013
Piperazinyl carbamate fatty acid amide hydrolase inhibitors and transient receptor potential channel modulators as "dual-target" analgesics.
    Pharmacological research, 2013, Volume: 76

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Carbamates; Edema; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Pain; Pain Measurement; Polyunsaturated Alkamides; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2013
Effects of endocannabinoid and endovanilloid systems on aversive memory extinction.
    Behavioural brain research, 2013, Nov-01, Volume: 256

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Endocannabinoids; Enzyme Inhibitors; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Male; Memory; Mice, Inbred C57BL; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Social Dominance; Stress, Psychological; Time Factors; TRPV Cation Channels

2013
Effects of the fatty acid amide hydrolase inhibitor URB597 on coping behavior under challenging conditions in mice.
    Psychopharmacology, 2014, Volume: 231, Issue:3

    Topics: Adaptation, Psychological; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Electrodes, Implanted; Electroencephalography; Electromyography; Electroshock; Endocannabinoids; Enzyme Inhibitors; Escape Reaction; Freezing Reaction, Cataleptic; Male; Mice, Inbred Strains; Motor Activity; Polyunsaturated Alkamides; Restraint, Physical; Sleep; Stress, Psychological

2014
Attenuation of anticipatory nausea in a rat model of contextually elicited conditioned gaping by enhancement of the endocannabinoid system.
    Psychopharmacology, 2014, Volume: 231, Issue:3

    Topics: Amidohydrolases; Animals; Anticipation, Psychological; Arachidonic Acids; Brain; Cannabinoid Receptor Antagonists; Carbamates; Endocannabinoids; Enzyme Inhibitors; Glycerides; Indoles; Lithium Chloride; Male; Monoacylglycerol Lipases; Motor Activity; Nausea; Oleic Acids; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant

2014
Endocannabinoid anandamide mediates hypoxic pulmonary vasoconstriction.
    Proceedings of the National Academy of Sciences of the United States of America, 2013, Nov-12, Volume: 110, Issue:46

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Blotting, Western; Carbamates; Chromatography, Liquid; DNA Primers; Endocannabinoids; Hypertension, Pulmonary; Hypoxia; Immunohistochemistry; Lung; Mice; Mice, Knockout; Myocytes, Smooth Muscle; Polyunsaturated Alkamides; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Vasoconstriction

2013
Monounsaturated fatty acids generated via stearoyl CoA desaturase-1 are endogenous inhibitors of fatty acid amide hydrolase.
    Proceedings of the National Academy of Sciences of the United States of America, 2013, Nov-19, Volume: 110, Issue:47

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Carbamates; Endocannabinoids; Fatty Acids, Monounsaturated; Feedback, Physiological; Insulin Resistance; Liver; Male; Mice; Mice, Inbred C57BL; Obesity; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Stearoyl-CoA Desaturase

2013
Inhibition of endocannabinoid-degrading enzyme fatty acid amide hydrolase increases atherosclerotic plaque vulnerability in mice.
    Journal of molecular and cellular cardiology, 2014, Volume: 66

    Topics: Amidohydrolases; Animals; Apolipoproteins E; Arachidonic Acids; Benzamides; Carbamates; Cell Movement; Diet, High-Fat; Dietary Fats; Endocannabinoids; Enzyme Inhibitors; Gene Expression; Macrophages; Mice; Mice, Knockout; Neutrophils; Plaque, Atherosclerotic; Polyunsaturated Alkamides; Superoxides

2014
Effects of the fatty acid amide hydrolase inhibitor URB597 on pain-stimulated and pain-depressed behavior in rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:2

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Brain; Carbamates; Conditioning, Operant; Depression; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Implantable Neurostimulators; Injections, Intraperitoneal; Lactic Acid; Male; Pain; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Self Administration

2014
Elevation of endogenous anandamide impairs LTP, learning, and memory through CB1 receptor signaling in mice.
    Hippocampus, 2014, Volume: 24, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Calcium-Calmodulin-Dependent Protein Kinase Type 4; Carbamates; Cyclic AMP Response Element-Binding Protein; Endocannabinoids; Glycerides; Learning; Long-Term Potentiation; Male; MAP Kinase Signaling System; Maze Learning; Memory; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphorylation; Polyunsaturated Alkamides; Protein Processing, Post-Translational; Receptor, Cannabinoid, CB1; Spatial Memory

2014
Antidepressants and changes in concentration of endocannabinoids and N-acylethanolamines in rat brain structures.
    Neurotoxicity research, 2014, Volume: 26, Issue:2

    Topics: Acetylcysteine; Amides; Amidohydrolases; Animals; Antidepressive Agents; Arachidonic Acids; Benzamides; Brain; Carbamates; Citalopram; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Expectorants; Glycerides; Imipramine; Male; Oleic Acids; Palmitic Acids; Polyunsaturated Alkamides; Rats, Wistar; Thiazepines

2014
Effects of endogenous cannabinoid anandamide on cardiac Na⁺/Ca²⁺ exchanger.
    Cell calcium, 2014, Volume: 55, Issue:5

    Topics: Animals; Arachidonic Acids; Benzamides; Calcium Channel Blockers; Carbamates; Cells, Cultured; Endocannabinoids; HEK293 Cells; Humans; Male; Microscopy, Confocal; Myocytes, Cardiac; Patch-Clamp Techniques; Polyunsaturated Alkamides; Rats; Rats, Wistar; Sodium-Calcium Exchanger

2014
Prior stimulation of the endocannabinoid system prevents methamphetamine-induced dopaminergic neurotoxicity in the striatum through activation of CB2 receptors.
    Neuropharmacology, 2014, Volume: 87

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Cannabinoid Receptor Modulators; Carbamates; Central Nervous System Stimulants; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Methamphetamine; Mice, Inbred C57BL; Neostriatum; Neurotoxicity Syndromes; Piperidines; Polyunsaturated Alkamides; Random Allocation; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Tumor Necrosis Factor-alpha; Tyrosine 3-Monooxygenase

2014
Fatty acid amide hydrolase (FAAH) inhibitors exert pharmacological effects, but lack antinociceptive efficacy in rats with neuropathic spinal cord injury pain.
    PloS one, 2014, Volume: 9, Issue:5

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Brain; Carbamates; Endocannabinoids; Enzyme Inhibitors; Hindlimb; Male; Morpholines; Naphthalenes; Neuralgia; Pain Measurement; Pain Threshold; Piperidines; Polyunsaturated Alkamides; Pyridines; Rats, Sprague-Dawley; Spinal Cord; Spinal Cord Injuries; Treatment Outcome

2014
Increased angiotensin II contraction of the uterine artery at early gestation in a transgenic model of hypertensive pregnancy is reduced by inhibition of endocannabinoid hydrolysis.
    Hypertension (Dallas, Tex. : 1979), 2014, Volume: 64, Issue:3

    Topics: Amidohydrolases; Angiotensin II; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood Pressure; Carbamates; Disease Models, Animal; Endocannabinoids; Female; Glycerides; Humans; Hydrolysis; Hypertension, Pregnancy-Induced; Male; Monoglycerides; Piperidines; Polyunsaturated Alkamides; Pregnancy; Pregnancy, Animal; Rats; Rats, Sprague-Dawley; Rats, Transgenic; Uterine Artery; Vasoconstriction

2014
Endocannabinoid modulation by FAAH and monoacylglycerol lipase within the analgesic circuitry of the periaqueductal grey.
    British journal of pharmacology, 2014, Volume: 171, Issue:23

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Endocannabinoids; Female; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Monoacylglycerol Lipases; Neurons; Pain; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission

2014
Endocannabinoid degradation inhibition improves neurobehavioral function, blood-brain barrier integrity, and neuroinflammation following mild traumatic brain injury.
    Journal of neurotrauma, 2015, Mar-01, Volume: 32, Issue:5

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Blood-Brain Barrier; Blotting, Western; Brain Injuries; Carbamates; Disease Models, Animal; Endocannabinoids; Glycerides; Immunohistochemistry; Inflammation; Male; Neuroprotective Agents; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Recovery of Function

2015
Correlating FAAH and anandamide cellular uptake inhibition using N-alkylcarbamate inhibitors: from ultrapotent to hyperpotent.
    Biochemical pharmacology, 2014, Dec-15, Volume: 92, Issue:4

    Topics: Amidohydrolases; Arachidonic Acids; Carbamates; Cell Line, Tumor; Endocannabinoids; Humans; Magnetic Resonance Spectroscopy; Polyunsaturated Alkamides; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship

2014
Anti-aversive role of the endocannabinoid system in the periaqueductal gray stimulation model of panic attacks in rats.
    Psychopharmacology, 2015, Volume: 232, Issue:9

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Male; N-Methylaspartate; Panic Disorder; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2015
Normal aging in rats and pathological aging in human Alzheimer's disease decrease FAAH activity: modulation by cannabinoid agonists.
    Experimental gerontology, 2014, Volume: 60

    Topics: Aged; Aged, 80 and over; Aging; Alzheimer Disease; Amidohydrolases; Amyloid beta-Peptides; Animals; Arachidonic Acids; Benzamides; Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoids; Carbamates; Case-Control Studies; Cerebral Cortex; Endocannabinoids; Enzyme Inhibitors; Female; Frontal Lobe; Humans; In Vitro Techniques; Male; Middle Aged; Morpholines; Naphthalenes; Polyunsaturated Alkamides; Rats; Rats, Wistar; Synaptosomes

2014
Endogenous cannabinoid release within prefrontal-limbic pathways affects memory consolidation of emotional training.
    Proceedings of the National Academy of Sciences of the United States of America, 2014, Dec-23, Volume: 111, Issue:51

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Avoidance Learning; Benzamides; Carbamates; Emotions; Endocannabinoids; Glycerides; Limbic System; Memory; Polyunsaturated Alkamides; Prefrontal Cortex; Rats; Receptor, Cannabinoid, CB1

2014
Inhibition of anandamide hydrolysis attenuates nociceptor sensitization in a murine model of chemotherapy-induced peripheral neuropathy.
    Journal of neurophysiology, 2015, Mar-01, Volume: 113, Issue:5

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Cisplatin; Endocannabinoids; Hydrolysis; Indoles; Male; Mice; Morpholines; Nerve Fibers, Unmyelinated; Nociception; Nociceptors; Peripheral Nervous System Diseases; Polyunsaturated Alkamides; Pyrazoles; Skin

2015
Chronic stimulation of the tone of endogenous anandamide reduces cue- and stress-induced relapse in rats.
    The international journal of neuropsychopharmacology, 2014, Dec-05, Volume: 18, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Endocannabinoids; Enzyme Inhibitors; Male; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Recurrence; Self Administration; Stress, Physiological; Yohimbine

2014
Inhibition of anandamide hydrolysis enhances noradrenergic and GABAergic transmission in the prefrontal cortex and basolateral amygdala of rats subjected to acute swim stress.
    Journal of neuroscience research, 2015, Volume: 93, Issue:5

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Basolateral Nuclear Complex; Benzamides; Carbamates; Chromatography, High Pressure Liquid; Disease Models, Animal; Endocannabinoids; Extracellular Fluid; gamma-Aminobutyric Acid; Male; Microdialysis; Norepinephrine; Polyunsaturated Alkamides; Prefrontal Cortex; Rats; Rats, Wistar; Stress, Psychological; Swimming

2015
Role of endocannabinoid signalling in the dorsolateral periaqueductal grey in the modulation of distinct panic-like responses.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:3

    Topics: Animals; Arachidonic Acids; Benzamides; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Escape Reaction; Male; Maze Learning; Panic Disorder; Periaqueductal Gray; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Signal Transduction

2015
Increased Contextual Fear Conditioning in iNOS Knockout Mice: Additional Evidence for the Involvement of Nitric Oxide in Stress-Related Disorders and Contribution of the Endocannabinoid System.
    The international journal of neuropsychopharmacology, 2015, Jan-24, Volume: 18, Issue:8

    Topics: Animals; Arachidonic Acids; Benzamides; Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Conditioning, Psychological; Endocannabinoids; Enzyme Inhibitors; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Hippocampus; Indazoles; Male; Mice, Inbred C57BL; Mice, Knockout; Morpholines; Naphthalenes; Nitric Oxide; Nitric Oxide Synthase Type II; Polyunsaturated Alkamides; Prefrontal Cortex; Pyrazoles; Receptor, Cannabinoid, CB1; RNA, Messenger; Stress, Psychological

2015
Phenotypic assessment of THC discriminative stimulus properties in fatty acid amide hydrolase knockout and wildtype mice.
    Neuropharmacology, 2015, Volume: 93

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzodioxoles; Brain; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Enzyme Inhibitors; Glycerides; Male; Mice; Mice, Knockout; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rimonabant

2015
A multi-target approach for pain treatment: dual inhibition of fatty acid amide hydrolase and TRPV1 in a rat model of osteoarthritis.
    Pain, 2015, Volume: 156, Issue:5

    Topics: Activating Transcription Factor 3; Amidohydrolases; Anilides; Animals; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Cinnamates; Disease Models, Animal; Endocannabinoids; Ganglia, Spinal; Gene Expression; Hyperalgesia; Inflammation; Interleukin-6; Lumbar Vertebrae; Male; Osteoarthritis; Pain; Pain Management; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2015
Inhibition of FAAH reduces nitroglycerin-induced migraine-like pain and trigeminal neuronal hyperactivity in mice.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2015, Volume: 25, Issue:8

    Topics: Amidohydrolases; Analgesics; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Inhibitors; Hyperalgesia; Male; Mice, Inbred C57BL; Mice, Knockout; Migraine Disorders; Monoacylglycerol Lipases; Nitroglycerin; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Touch; Trigeminal Nuclei

2015
Distinct roles of the endocannabinoids anandamide and 2-arachidonoylglycerol in social behavior and emotionality at different developmental ages in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2015, Volume: 25, Issue:8

    Topics: Aging; Animals; Anxiety; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Carbamates; Endocannabinoids; Exploratory Behavior; Glycerides; Male; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats, Sprague-Dawley; Rimonabant; Social Behavior

2015
Endocannabinoid-mediated improvement on a test of aversive memory in a mouse model of fragile X syndrome.
    Behavioural brain research, 2015, Sep-15, Volume: 291

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Avoidance Learning; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Fragile X Mental Retardation Protein; Fragile X Syndrome; Male; Memory; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Propofol; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, GABA-A; Social Behavior

2015
Inhibition of FAAH confers increased stem cell migration via PPARα.
    Journal of lipid research, 2015, Volume: 56, Issue:10

    Topics: Adipose Tissue; Amides; Amidohydrolases; Arachidonic Acids; Benzamides; Carbamates; Cell Movement; Cells, Cultured; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Glycerides; Humans; Mesenchymal Stem Cells; Oleic Acids; Palmitic Acids; Polyunsaturated Alkamides; PPAR alpha; Receptor, Cannabinoid, CB1; Serotonin

2015
Anandamide mediates cognitive judgement bias in rats.
    Neuropharmacology, 2016, Volume: 101

    Topics: Acoustic Stimulation; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Bias; Calcium Channel Blockers; Carbamates; Cognition; Conditioning, Psychological; Cues; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Judgment; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats

2016
Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor.
    PloS one, 2015, Volume: 10, Issue:9

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acid; Arachidonic Acids; Benzamides; Brain; Carbamates; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Endocannabinoids; Flurbiprofen; Humans; Hydrolysis; Interferon-gamma; Ionomycin; Isoenzymes; Lipid Metabolism; Lipopolysaccharides; Male; Mice; Polyunsaturated Alkamides; Prostaglandins; RAW 264.7 Cells; Stereoisomerism

2015
Endocannabinoid signaling mediates oxytocin-driven social reward.
    Proceedings of the National Academy of Sciences of the United States of America, 2015, Nov-10, Volume: 112, Issue:45

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Autism Spectrum Disorder; Benzamides; Benzodiazepines; Camphanes; Carbamates; Clozapine; Cocaine; Endocannabinoids; Immunohistochemistry; Infusions, Intraventricular; Lipids; Male; Mice; Mice, Inbred C57BL; Nucleus Accumbens; Oxytocin; Piperazines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Reward; Signal Transduction; Social Behavior

2015
THC and endocannabinoids differentially regulate neuronal activity in the prefrontal cortex and hippocampus in the subchronic PCP model of schizophrenia.
    Journal of psychopharmacology (Oxford, England), 2016, Volume: 30, Issue:2

    Topics: Animals; Arachidonic Acids; Benzamides; Carbamates; Disease Models, Animal; Dronabinol; Endocannabinoids; Hippocampus; Male; Phencyclidine; Polyunsaturated Alkamides; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Schizophrenia; Up-Regulation

2016
Inhibition of anandamide hydrolysis dampens the neuroendocrine response to stress in neonatal rats subjected to suboptimal rearing conditions.
    Stress (Amsterdam, Netherlands), 2016, Volume: 19, Issue:1

    Topics: Adrenocorticotropic Hormone; Amidohydrolases; Animals; Animals, Newborn; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Corticosterone; Endocannabinoids; Hydrolysis; Hypothalamus; Male; Neurosecretory Systems; Paraventricular Hypothalamic Nucleus; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stress, Physiological; Stress, Psychological

2016
Self-administration of the anandamide transport inhibitor AM404 by squirrel monkeys.
    Psychopharmacology, 2016, Volume: 233, Issue:10

    Topics: Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Cocaine; Dose-Response Relationship, Drug; Dronabinol; Drug-Seeking Behavior; Endocannabinoids; Male; Nicotine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Reinforcement, Psychology; Reward; Rimonabant; Saimiri; Self Administration

2016
The effects anandamide signaling in the prelimbic cortex and basolateral amygdala on coping with environmental stimuli in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:10

    Topics: Adaptation, Psychological; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Basolateral Nuclear Complex; Benzamides; Carbamates; Endocannabinoids; Glycerides; Male; Polyunsaturated Alkamides; Prefrontal Cortex; Rats; Rats, Wistar; Signal Transduction

2016
Comparisons of Δ9-Tetrahydrocannabinol and Anandamide on a Battery of Cognition-Related Behavior in Nonhuman Primates.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Animals; Arachidonic Acids; Attention; Behavior, Animal; Benzamides; Carbamates; Cognition; Discrimination Learning; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Learning; Male; Memory, Short-Term; Motivation; Piperidines; Polyunsaturated Alkamides; Psychomotor Performance; Pyrazoles; Reversal Learning; Rimonabant; Saimiri

2016
Attenuation of cue-induced reinstatement of nicotine seeking by URB597 through cannabinoid CB1 receptor in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:10

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Antagonists; Carbamates; Cues; Drug-Seeking Behavior; Endocannabinoids; Male; Nicotine; Piperidines; Polyunsaturated Alkamides; PPAR alpha; Pyrazoles; Rats; Rats, Long-Evans; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Tobacco Use Disorder

2016
Fatty acid amide hydrolase inhibition for the symptomatic relief of Parkinson's disease.
    Brain, behavior, and immunity, 2016, Volume: 57

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Agonists; Carbamates; Disease Models, Animal; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Parkinsonian Disorders; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2

2016
Emotional arousal state influences the ability of amygdalar endocannabinoid signaling to modulate anxiety.
    Neuropharmacology, 2016, Volume: 111

    Topics: Animals; Anxiety; Arachidonic Acids; Arousal; Basolateral Nuclear Complex; Benzamides; Cannabinoid Receptor Agonists; Carbamates; Corticosterone; Emotions; Endocannabinoids; Epinephrine; Glycerides; Male; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Signal Transduction

2016
The endocannabinoid hydrolysis inhibitor SA-57: Intrinsic antinociceptive effects, augmented morphine-induced antinociception, and attenuated heroin seeking behavior in mice.
    Neuropharmacology, 2017, 03-01, Volume: 114

    Topics: Acetamides; Analgesics; Analgesics, Opioid; Animals; Arachidonic Acid; Arachidonic Acids; Carbamates; Carrageenan; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Endocannabinoids; Glycerides; Heroin; Hydrolysis; Hyperalgesia; Inflammation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Neuralgia; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Sciatic Nerve; Self Administration

2017
The role of CB
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2017, Volume: 31, Issue:8

    Topics: Amidohydrolases; Arachidonic Acids; Benzamides; Benzodioxoles; Caco-2 Cells; Carbamates; Colorectal Neoplasms; Cytokines; Electric Impedance; Endocannabinoids; Gene Expression Regulation; Glycerides; Humans; Inflammation; Intestinal Mucosa; Intestines; Monoacylglycerol Lipases; Oxygen Consumption; Permeability; Piperidines; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Tissue Culture Techniques

2017
Sensitization of C-fiber nociceptors in mice with sickle cell disease is decreased by local inhibition of anandamide hydrolysis.
    Pain, 2017, Volume: 158, Issue:9

    Topics: Anemia, Sickle Cell; Animals; Arachidonic Acids; Benzamides; Carbamates; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Evoked Potentials; Hemoglobins; Humans; Hydrolysis; Hyperalgesia; Indoles; Male; Mice; Mice, Transgenic; Morpholines; Nerve Fibers, Unmyelinated; Nociceptors; Pain Threshold; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2

2017
FAAH, but not MAGL, inhibition modulates acute TLR3-induced neuroimmune signaling in the rat, independent of sex.
    Journal of neuroscience research, 2018, Volume: 96, Issue:6

    Topics: Amides; Amidohydrolases; Animals; Arachidonic Acids; Body Temperature; Carbamates; Chemokine CXCL10; Corticosterone; Endocannabinoids; Estradiol; Ethanolamines; Female; Glycerides; Immunologic Factors; Interferons; Male; Monoacylglycerol Lipases; NF-kappa B; Oleic Acids; Palmitic Acids; Poly I-C; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Sex Factors; Signal Transduction; Succinimides; Toll-Like Receptor 3

2018
Enhanced anandamide signaling reduces flight behavior elicited by an approaching robo-beetle.
    Neuropharmacology, 2017, Volume: 126

    Topics: Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Avoidance Learning; Behavior, Animal; Benzamides; Benzodioxoles; Cannabinoid Receptor Agonists; Carbamates; Diazepam; Endocannabinoids; Fear; Male; Mice, Inbred C57BL; Monoacylglycerol Lipases; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2017
The selective reversible FAAH inhibitor, SSR411298, restores the development of maladaptive behaviors to acute and chronic stress in rodents.
    Scientific reports, 2018, 02-05, Volume: 8, Issue:1

    Topics: Acute Disease; Amides; Amidohydrolases; Animals; Anti-Anxiety Agents; Anxiety Disorders; Arachidonic Acids; Cannabinoid Receptor Agonists; Carbamates; Chronic Disease; Dioxanes; Endocannabinoids; Enzyme Inhibitors; Ethanolamines; Female; Gene Expression; Male; Mice; Oleic Acids; Palmitic Acids; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Receptors, Cannabinoid; Stress, Psychological

2018
Chronic treatment with URB597 ameliorates post-stress symptoms in a rat model of PTSD.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2018, Volume: 28, Issue:5

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Basolateral Nuclear Complex; Benzamides; Benzoxazines; CA1 Region, Hippocampal; Cannabinoid Receptor Antagonists; Carbamates; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Extinction, Psychological; Glycerides; Male; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reflex, Startle; Stress Disorders, Post-Traumatic

2018
Inhibition of Fatty Acid Amide Hydrolase Improves Depressive-Like Behaviors Independent of Its Peripheral Antinociceptive Effects in a Rat Model of Neuropathic Pain.
    Anesthesia and analgesia, 2019, Volume: 129, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Carbamates; Depression; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Feeding Behavior; Glycerides; Hippocampus; Locomotion; Male; Neuralgia; Neurogenesis; Pain Threshold; Polyunsaturated Alkamides; Rats, Wistar; Receptor, Cannabinoid, CB1; Signal Transduction; Swimming

2019
Adult Cellular Neuroadaptations Induced by Adolescent THC Exposure in Female Rats Are Rescued by Enhancing Anandamide Signaling.
    The international journal of neuropsychopharmacology, 2018, 11-01, Volume: 21, Issue:11

    Topics: Adaptation, Psychological; Animals; Arachidonic Acids; Benzamides; Carbamates; Dentate Gyrus; Depression; Dronabinol; Endocannabinoids; Female; Marijuana Abuse; Neurogenesis; Neuronal Plasticity; Polyunsaturated Alkamides; Prefrontal Cortex; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Sexual Maturation; Signal Transduction; Synapses; Tissue Culture Techniques

2018
Endocannabinoid regulation of homeostatic feeding and stress-induced alterations in food intake in male rats.
    British journal of pharmacology, 2019, Volume: 176, Issue:10

    Topics: Amidohydrolases; Animals; Anorexia; Arachidonic Acids; Carbamates; Duodenum; Eating; Endocannabinoids; Glycerides; Homeostasis; Jejunum; Male; Monoacylglycerol Lipases; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Stress, Psychological; Succinimides

2019
Pharmacological blockade of fatty acid amide hydrolase (FAAH) by URB597 improves memory and changes the phenotype of hippocampal microglia despite ethanol exposure.
    Biochemical pharmacology, 2018, Volume: 157

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Chemokines; Cytokines; Dentate Gyrus; Endocannabinoids; Enzyme Inhibitors; Ethanol; Gene Expression; Glial Fibrillary Acidic Protein; Hippocampus; Male; Memory; Memory, Long-Term; Memory, Short-Term; Microglia; Nitric Oxide Synthase Type II; Phenotype; Polyunsaturated Alkamides; Rats, Wistar; Receptors, Chemokine

2018
Hypertension and chronic inhibition of endocannabinoid degradation modify the endocannabinoid system and redox balance in rat heart and plasma.
    Prostaglandins & other lipid mediators, 2018, Volume: 138

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Carbamates; Desoxycorticosterone Acetate; Endocannabinoids; Glycerides; Heart; Hypertension; Male; Myocardium; Oxidation-Reduction; Oxidative Stress; Polyunsaturated Alkamides; Rats, Inbred SHR; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2

2018
Endocannabinoid interactions in the regulation of acquisition of contextual conditioned fear.
    Progress in neuro-psychopharmacology & biological psychiatry, 2019, 03-02, Volume: 90

    Topics: Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Brain; Carbamates; Central Nervous System Agents; Conditioning, Psychological; Endocannabinoids; Fear; Glycerides; Male; Motor Activity; Nociception; Piperidines; Polyunsaturated Alkamides; Random Allocation; Rats, Wistar

2019
Anandamide Reduces the Toxic Synergism Exerted by Quinolinic Acid and Glutaric Acid in Rat Brain Neuronal Cells.
    Neuroscience, 2019, 03-01, Volume: 401

    Topics: Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Agonists; Carbamates; Cell Survival; Cells, Cultured; Cerebral Cortex; Drug Synergism; Endocannabinoids; Female; Glutarates; Male; Neurons; Piperidines; Polyunsaturated Alkamides; Pregnancy; Pyrazoles; Quinolinic Acid; Rats; Rats, Inbred WF; Receptors, Cannabinoid

2019
Role of the endocannabinoid system in the dorsal hippocampus in the cardiovascular changes and delayed anxiety-like effect induced by acute restraint stress in rats.
    Journal of psychopharmacology (Oxford, England), 2019, Volume: 33, Issue:5

    Topics: Amidohydrolases; Animals; Anxiety; Arachidonic Acids; Arterial Pressure; Behavior, Animal; Benzamides; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbamates; Disease Models, Animal; Endocannabinoids; Heart Rate; Hippocampus; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Restraint, Physical; Skin Temperature; Stress, Psychological

2019
Anandamide modulation of circadian- and stress-dependent effects on rat short-term memory.
    Psychoneuroendocrinology, 2019, Volume: 108

    Topics: Animals; Arachidonic Acids; Arousal; Benzamides; Carbamates; Circadian Rhythm; Corticosterone; Emotions; Endocannabinoids; Male; Memory, Short-Term; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Stress, Psychological

2019
Targeting the inhibition of fatty acid amide hydrolase ameliorate the endocannabinoid-mediated synaptic dysfunction in a valproic acid-induced rat model of Autism.
    Neuropharmacology, 2020, 01-01, Volume: 162

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Autism Spectrum Disorder; Benzamides; Carbamates; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Female; Long-Term Synaptic Depression; Neuronal Plasticity; Polyunsaturated Alkamides; Prefrontal Cortex; Pregnancy; Prenatal Exposure Delayed Effects; Protein Transport; Rats; Receptors, AMPA; Receptors, Metabotropic Glutamate; Social Behavior; Valproic Acid

2020
Neuropeptide Y and cannabinoids interaction in the amygdala after exposure to shock and reminders model of PTSD.
    Neuropharmacology, 2020, 01-01, Volume: 162

    Topics: Amygdala; Animals; Arachidonic Acids; Arousal; Basolateral Nuclear Complex; Behavior, Animal; Benzamides; Carbamates; Depression; Disease Models, Animal; Endocannabinoids; Extinction, Psychological; Neuropeptide Y; Polyunsaturated Alkamides; Rats; Receptor, Cannabinoid, CB1; Receptors, Neuropeptide Y; Reflex, Startle; Social Behavior; Stress Disorders, Post-Traumatic

2020
Antidepressant-like effects of pharmacological inhibition of FAAH activity in socially isolated female rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2020, Volume: 32

    Topics: Amidohydrolases; Animals; Antidepressive Agents; Arachidonic Acids; Biphenyl Compounds; Brain-Derived Neurotrophic Factor; Carbamates; Endocannabinoids; Enzyme Activation; Female; Hippocampus; Polyunsaturated Alkamides; Rats; Social Isolation

2020
The endocannabinoid hydrolase FAAH is an allosteric enzyme.
    Scientific reports, 2020, 02-10, Volume: 10, Issue:1

    Topics: Allosteric Regulation; Allosteric Site; Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Biocatalysis; Carbamates; Catalytic Domain; Drug Design; Endocannabinoids; Enzyme Assays; Humans; Hydrolysis; Kinetics; Molecular Dynamics Simulation; Mutation; Polyunsaturated Alkamides; Protein Subunits; Rats

2020
The effects of fatty acid amide hydrolase and monoacylglycerol lipase inhibitor treatments on lipopolysaccharide-induced airway inflammation in mice.
    Pulmonary pharmacology & therapeutics, 2020, Volume: 62

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Benzodioxoles; Carbamates; Cytokines; Endocannabinoids; Glycerides; Inflammation; Lipopolysaccharides; Lung; Male; Mice; Monoacylglycerol Lipases; Piperidines; Pneumonia; Polyunsaturated Alkamides; Respiratory Hypersensitivity

2020
The FAAH Inhibitor URB597 Modulates Lipid Mediators in the Brain of Rats with Spontaneous Hypertension.
    Biomolecules, 2020, 07-10, Volume: 10, Issue:7

    Topics: Animals; Arachidonic Acids; Benzamides; Brain; Carbamates; Disease Models, Animal; Endocannabinoids; Hypertension; Injections, Intraperitoneal; Male; Malondialdehyde; Oxidation-Reduction; Phospholipids; Polyunsaturated Alkamides; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, G-Protein-Coupled

2020
Effects of systemic endocannabinoid manipulation on social and exploratory behavior in prairie voles (Microtus ochrogaster).
    Psychopharmacology, 2021, Volume: 238, Issue:1

    Topics: Animals; Anxiety; Arachidonic Acids; Arvicolinae; Behavior, Animal; Benzamides; Carbamates; Endocannabinoids; Exploratory Behavior; Female; Male; Maze Learning; Nucleus Accumbens; Pair Bond; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Oxytocin; Social Behavior

2021
Beneficial Changes in Rat Vascular Endocannabinoid System in Primary Hypertension and under Treatment with Chronic Inhibition of Fatty Acid Amide Hydrolase by URB597.
    International journal of molecular sciences, 2021, May-02, Volume: 22, Issue:9

    Topics: Acetylcholine; Amidohydrolases; Animals; Aorta; Arachidonic Acids; Benzamides; Carbamates; Endocannabinoids; Essential Hypertension; Hypertension; Male; Mesenteric Arteries; Nitroprusside; Polyunsaturated Alkamides; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Cannabinoid; Vasoconstriction; Vasodilation

2021
Kainate-Induced Degeneration of Hippocampal Neurons. Protective Effect of Activation of the Endocannabinoid System.
    Bulletin of experimental biology and medicine, 2021, Volume: 171, Issue:3

    Topics: Animals; Arachidonic Acids; Autophagosomes; Benzamides; CA3 Region, Hippocampal; Carbamates; Dentate Gyrus; Endocannabinoids; Endoplasmic Reticulum; Excitatory Amino Acid Agonists; Golgi Apparatus; Kainic Acid; Lysosomes; Male; Microscopy, Electron; Necrosis; Nerve Degeneration; Polyunsaturated Alkamides; Pyramidal Cells; Rats; Rats, Wistar; Status Epilepticus

2021
Fatty Acid Amide Hydrolase (FAAH) Inhibition Modulates Amyloid-Beta-Induced Microglia Polarization.
    International journal of molecular sciences, 2021, Jul-19, Volume: 22, Issue:14

    Topics: Alzheimer Disease; Amidohydrolases; Amyloid beta-Peptides; Animals; Arachidonic Acids; Benzamides; Carbamates; Cell Line; Cell Movement; Cell Polarity; Cytokines; Cytoskeleton; Disease Models, Animal; Endocannabinoids; Mice; Microglia; Polyunsaturated Alkamides

2021