Page last updated: 2024-08-17

carbachol and tiotropium bromide

carbachol has been researched along with tiotropium bromide in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (16.67)29.6817
2010's4 (66.67)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Bartuschat, A; Fischer, O; Fromm, MF; Gmeiner, P; Heinrich, MR; Hofmann, J; Hübner, H; Kaindl, J; Pratsch, G; Rampp, H; Taudte, RV1
Beleta, J; Carcasona, C; Carreño, C; Cortijo, J; Doménech, T; Gavaldà, A; Gras, J; Llenas, J; Miralpeix, M; Morcillo, E; Otal, R; Ramos, I; Reyes, B; Ryder, H; Vilella, D; Viñals, M1
Amari, G; Bassani, F; Battipaglia, L; Bergamaschi, M; Berti, F; Bolzoni, PT; Cacciani, F; Cenacchi, V; Civelli, M; Delcanale, M; Geppetti, PA; Harrison, S; Mannini, F; Pastore, F; Patacchini, R; Petrillo, P; Razzetti, R; Rizzi, A; Rossoni, G; Santoro, E; Scudellaro, R; Villetti, G; Volta, R; Zaniboni, M1
Barnes, PJ; Brown, SM; Donnelly, LE; Koarai, A; Nicholson, AG; Sturton, RG1
Barrett, VJ; Buckley, PT; Burman, M; DeHaas, CJ; Foley, JJ; Hay, DW; Kotzer, CJ; Lainé, DI; Luttmann, MA; Palovich, MR; Rumsey, WL; Salmon, M; Sarau, HM; Schmidt, DB; Slack, RJ; Webb, EF1
Borger, P; Costa, L; Keglowich, L; Lardinois, D; Miglino, N; Roth, M; Tamm, M; Zhong, J1

Other Studies

6 other study(ies) available for carbachol and tiotropium bromide

ArticleYear
Regiospecific Introduction of Halogens on the 2-Aminobiphenyl Subunit Leading to Highly Potent and Selective M3 Muscarinic Acetylcholine Receptor Antagonists and Weak Inverse Agonists.
    Journal of medicinal chemistry, 2020, 04-23, Volume: 63, Issue:8

    Topics: Aminobiphenyl Compounds; Animals; Caco-2 Cells; Drug Inverse Agonism; Halogens; HEK293 Cells; Humans; Male; Molecular Docking Simulation; Muscarinic Agonists; Muscarinic Antagonists; Protein Binding; Protein Structure, Secondary; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3

2020
Characterization of aclidinium bromide, a novel inhaled muscarinic antagonist, with long duration of action and a favorable pharmacological profile.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Administration, Inhalation; Anesthesia; Animals; Bronchi; Bronchoconstriction; Carbachol; CHO Cells; Cricetinae; Cricetulus; Dogs; Guinea Pigs; Heart Rate; Humans; Ipratropium; Male; Muscarinic Agonists; Muscarinic Antagonists; Receptors, Muscarinic; Scopolamine Derivatives; Stimulation, Chemical; Tiotropium Bromide; Trachea; Tropanes

2009
Bronchodilator activity of (3R)-3-[[[(3-fluorophenyl)[(3,4,5-trifluorophenyl)methyl]amino] carbonyl]oxy]-1-[2-oxo-2-(2-thienyl)ethyl]-1-azoniabicyclo[2.2.2]octane bromide (CHF5407), a potent, long-acting, and selective muscarinic M3 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: Acetylcholine; Aged; Anesthesia; Animals; Blood Pressure; Bronchi; Bronchial Spasm; Bronchoconstriction; Bronchoconstrictor Agents; Bronchodilator Agents; Carbachol; Carbamates; CHO Cells; Cricetinae; Cricetulus; Diamines; Guinea Pigs; Heart Atria; Heart Rate; Humans; Kinetics; Male; Middle Aged; Molecular Structure; Muscarinic Antagonists; Myocardial Contraction; Quinuclidines; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Scopolamine Derivatives; Tiotropium Bromide; Trachea; Transfection; Ventricular Function, Left

2010
A role for M(2) and M(3) muscarinic receptors in the contraction of rat and human small airways.
    European journal of pharmacology, 2013, Feb-28, Volume: 702, Issue:1-3

    Topics: Animals; Carbachol; Cholinergic Agonists; Humans; In Vitro Techniques; Lung; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Scopolamine Derivatives; Tiotropium Bromide

2013
Pharmacological characterization of GSK573719 (umeclidinium): a novel, long-acting, inhaled antagonist of the muscarinic cholinergic receptors for treatment of pulmonary diseases.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 345, Issue:2

    Topics: Administration, Inhalation; Animals; Calcium; Carbachol; CHO Cells; Cholinergic Antagonists; Cricetinae; Cricetulus; Guinea Pigs; Kinetics; Lung; Lung Diseases; Mice; Mice, Inbred BALB C; Muscarinic Agonists; Muscarinic Antagonists; Plethysmography; Quinuclidines; Receptor, Muscarinic M3; Receptors, Muscarinic; Scopolamine Derivatives; Tiotropium Bromide

2013
Tiotropium sustains the anti-inflammatory action of olodaterol via the cyclic AMP pathway.
    Pulmonary pharmacology & therapeutics, 2014, Volume: 27, Issue:1

    Topics: Adrenergic beta-2 Receptor Agonists; Adult; Aged; Anti-Inflammatory Agents; Asthma; Benzoxazines; Bronchodilator Agents; Carbachol; Cyclic AMP; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; Fibroblasts; Humans; In Vitro Techniques; Interleukin-1beta; Interleukin-6; Interleukin-8; Male; Middle Aged; Muscarinic Antagonists; Phosphorylation; Scopolamine Derivatives; Signal Transduction; Tiotropium Bromide

2014