Page last updated: 2024-08-17

carbachol and thiophenes

carbachol has been researched along with thiophenes in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19906 (31.58)18.7374
1990's10 (52.63)18.2507
2000's2 (10.53)29.6817
2010's0 (0.00)24.3611
2020's1 (5.26)2.80

Authors

AuthorsStudies
Baron, JH; Barros D'sa, AA; Bloom, SR; Gaskin, RJ; Joffe, SN; Pallone, F; Polak, JM1
Baron, JH; Barros D'sa, AA; Gaskin, R; Girvan, DP; Gribble, JN; Joffe, SN; Melo, AA1
Baron, JH; Barros D'sa, AA; Gaskin, R; Joffe, SN; Polak, JM1
Angeli, P; Brasili, L; Giannella, M; Gualtieri, F; Picchio, MT; Teodori, E1
Angeli, P; Brasili, L; Gualtieri, F; Romanelli, MN; Teodori, E1
Endoh, M; Taira, N; Yanagisawa, T1
Ciccocioppo, R; Cirillo, R; Massi, M; Polidori, C; Pompei, P2
Barg, J; Danenberg, HD; Gurwitz, D; Haring, R; Heldman, E; Marciano, D; Meshulam, H; Pinkas-Kramarski, R; Pittel, Z; Wengier, A1
Fisher, A; Gurwitz, D; Haring, R; Heldman, E; Karton, Y; Pinkas-Kramarski, R; Stein, R1
Baxter, GS; Byrne, C; Ellis, ES; Murphy, OE; Tilford, NS1
Barg, J; Gurwitz, D; Haring, R; Heldman, E; Karton, Y; Marciano, D; Meshulam, H; Pinkas-Kramarski, R; Pittel, Z; Wengier, A1
Fisher, A; Fraser, CM; Gurwitz, D; Haring, R; Heldman, E; Manor, D1
Barg, J; Behar, L; Fisher, A; Ginzburg, I; Gurwitz, D; Sadot, E1
Lasheras, B; Monge, A; Oset, C; Palop, J; PĂ©rez, S1
Endoh, M; Kawabata, Y1
Grove, KL; Smith, MS; Speth, RC1
Iida, H; Inoue, N; Ishida, H; Ishikawa, Y; Yuan, Z1
Isola, M; Isola, R; Loy, F; Masala, C1

Other Studies

19 other study(ies) available for carbachol and thiophenes

ArticleYear
Gastrin, antral g cells, and gastric acid in secretagogue-induced and antihistamine-inhibited duodenal ulcers.
    Scandinavian journal of gastroenterology, 1977, Volume: 12, Issue:1

    Topics: Animals; Carbachol; Duodenal Ulcer; Fluorescent Antibody Technique; Gastric Juice; Gastrins; Histamine H2 Antagonists; Male; Microscopy, Electron; Pentagastrin; Pyloric Antrum; Pyrrolidines; Rats; Rats, Inbred Strains; Secretory Rate; Thiophenes; Time Factors

1977
Proceedings: Secretagogue-produced duodenal ulcers in the rat and their prevention by the gastric secretory inhibitor UK 9040.
    The British journal of surgery, 1975, Volume: 62, Issue:2

    Topics: Animals; Carbachol; Disease Models, Animal; Duodenal Ulcer; Gastric Mucosa; Histamine H1 Antagonists; Pentagastrin; Pyrrolidines; Rats; Thiophenes

1975
Proceedings: Gastrin, G cells, and gastric acid in rats with secretagogue-produced and anti-secretagogue-inhibited duodenal ulcers.
    Gut, 1975, Volume: 16, Issue:5

    Topics: Animals; Carbachol; Duodenal Ulcer; Gastric Mucosa; Gastrins; Pentagastrin; Pyrrolidines; Rats; Thiophenes

1975
Chiral muscarinic agonists possessing a 1,3-oxathiolane nucleus: enantio- and tissue-selectivity on isolated preparations of guinea-pig ileum and atria and of rat urinary bladder.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:3

    Topics: Animals; Binding, Competitive; Carbachol; Guinea Pigs; Heart; Heterocyclic Compounds; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rats; Receptors, Muscarinic; Stereoisomerism; Thiophenes; Urinary Bladder

1988
Enantioselectivity of muscarinic antagonists. 2,2-Dicyclohexyl-5-[(dimethylamino)methyl]-1,3-oxathiolane methiodides and related 3-oxides.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:9

    Topics: Animals; Atrial Function; Carbachol; Chemical Phenomena; Chemistry; Cyclohexanes; Guinea Pigs; Heart Rate; Heterocyclic Compounds; Ileum; Molecular Conformation; Muscarine; Muscle Contraction; Myocardial Contraction; Rats; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Thiophenes; Urinary Bladder

1988
Involvement of cyclic AMP in the positive inotropic effect of OPC-8212, a new cardiotonic agent, on the canine ventricular muscle.
    Japanese journal of pharmacology, 1984, Volume: 36, Issue:3

    Topics: Animals; Atenolol; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Female; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Pyrazines; Quinolines; Stimulation, Chemical; Thiophenes

1984
The selective angiotensin AT1 receptor antagonist LR-B/081 potently inhibits drinking induced by central injection of angiotensin II in rats.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Carbachol; Dose-Response Relationship, Drug; Drinking; Eating; Imidazoles; Injections, Intraventricular; Lethal Dose 50; Losartan; Male; Milk; Pyrimidinones; Rats; Rats, Wistar; Renin-Angiotensin System; Tetrazoles; Thiophenes

1995
NGF promotes amyloid precursor protein secretion via muscarinic receptor activation.
    Biochemical and biophysical research communications, 1995, Aug-04, Volume: 213, Issue:1

    Topics: Amyloid beta-Protein Precursor; Animals; Carbachol; Cell Differentiation; Cell Membrane; Dose-Response Relationship, Drug; Kinetics; Nerve Growth Factors; Parasympathomimetics; PC12 Cells; Quinuclidines; Rats; Receptors, Muscarinic; Recombinant Proteins; Tetradecanoylphorbol Acetate; Thiophenes; Time Factors; Transfection

1995
NGF-dependent neurotrophic-like effects of AF102B, an M1 muscarinic agonist, in PC12M1 cells.
    Neuroreport, 1995, Feb-15, Volume: 6, Issue:3

    Topics: Animals; Atropine; Carbachol; Cyclic AMP; Nerve Growth Factors; Parasympathomimetics; PC12 Cells; Quinuclidines; Rats; Thiophenes

1995
Mediation by 5-hydroxytryptamine2B receptors of endothelium-dependent relaxation in rat jugular vein.
    British journal of pharmacology, 1995, Volume: 114, Issue:2

    Topics: Animals; Carbachol; Endothelium, Vascular; In Vitro Techniques; Indoles; Jugular Veins; Male; Mianserin; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes; Urea; Yohimbine

1995
Amyloid precursor protein secretion via muscarinic receptors: reduced desensitization using the M1-selective agonist AF102B.
    Biochemical and biophysical research communications, 1994, Aug-30, Volume: 203, Issue:1

    Topics: Amyloid beta-Protein Precursor; Animals; Carbachol; Kinetics; Parasympatholytics; PC12 Cells; Quinuclidines; Receptors, Muscarinic; Recombinant Proteins; Thiophenes; Transfection

1994
Discrete activation of transduction pathways associated with acetylcholine m1 receptor by several muscarinic ligands.
    European journal of pharmacology, 1994, Mar-15, Volume: 267, Issue:1

    Topics: Adenylyl Cyclases; Animals; Arachidonic Acid; Calcium; Carbachol; Cells, Cultured; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Hydrolysis; Phosphatidylinositols; Pilocarpine; Protein Binding; Quinuclidines; Receptors, Cholinergic; Signal Transduction; Thiophenes; Transfection

1994
Activation of m1 muscarinic acetylcholine receptor regulates tau phosphorylation in transfected PC12 cells.
    Journal of neurochemistry, 1996, Volume: 66, Issue:2

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Drug Synergism; Muscarinic Agonists; Nerve Growth Factors; Neurons; PC12 Cells; Phosphorylation; Quinuclidines; Rats; Receptors, Muscarinic; tau Proteins; Thiophenes; Time Factors; Transfection

1996
Functional evidence for the ability of angiotensin AT1 receptor antagonists to cross the blood-brain barrier in rats.
    European journal of pharmacology, 1996, Jul-04, Volume: 307, Issue:3

    Topics: Administration, Oral; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Blood-Brain Barrier; Carbachol; Dose-Response Relationship, Drug; Drinking; Imidazoles; Injections, Intraperitoneal; Injections, Intraventricular; Losartan; Male; Nicotinic Acids; Pyrimidinones; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Tetrazoles; Thiophenes

1996
Synthesis of thiophene carboxamide derivatives as serotonin 5-HT4 receptor agonists.
    Farmaco (Societa chimica italiana : 1989), 1997, Volume: 52, Issue:2

    Topics: Animals; Carbachol; Esophagus; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Muscarinic Agonists; Muscle Relaxation; Muscle, Smooth; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Receptor Agonists; Spectrophotometry, Infrared; Thiophenes

1997
Effects of a novel cardiotonic agent, Org 9731, on force and aequorin light transients in intact ventricular myocardium of the dog: involvement of a cyclic AMP-mediated mechanism and myofibrillar responsiveness to Ca2+ ions.
    Journal of cardiac failure, 1995, Volume: 1, Issue:2

    Topics: Aequorin; Animals; Calcium; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; Hydroxamic Acids; In Vitro Techniques; Male; Muscarinic Agonists; Myocardial Contraction; Myocardium; Myofibrils; Structure-Activity Relationship; Thiophenes

1995
Brain angiotensinergic mediation of enhanced water consumption in lactating rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 282, Issue:3

    Topics: Acrylates; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensins; Animals; Atropine; Brain; Carbachol; Drinking; Female; Imidazoles; Injections, Intraventricular; Lactation; Muscarinic Agonists; Muscarinic Antagonists; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Reference Values; Thiophenes

2002
Effect of SNI-2011 on amylase secretion from parotid tissue in rats and in neuronal nitric oxide synthase knockout mice.
    European journal of pharmacology, 2003, Mar-19, Volume: 464, Issue:2-3

    Topics: Alkaloids; Amylases; Animals; Azepines; Benzoates; Benzylamines; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Chelating Agents; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Gallic Acid; Genotype; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Mice, Knockout; Molsidomine; Muscarinic Agonists; Myosin-Light-Chain Kinase; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Parotid Gland; Penicillamine; Phosphodiesterase Inhibitors; Pilocarpine; Protein Kinase Inhibitors; Pyrroles; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Wistar; Sulfonamides; Thiophenes; Type C Phospholipases

2003
Reactivity of human labial glands in response to cevimeline treatment.
    Anatomical record (Hoboken, N.J. : 2007), 2021, Volume: 304, Issue:12

    Topics: Carbachol; Humans; Lip; Quinuclidines; Salivary Glands; Sjogren's Syndrome; Thiophenes

2021