Page last updated: 2024-08-17

carbachol and propylbenzilylcholine mustard

carbachol has been researched along with propylbenzilylcholine mustard in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-199014 (46.67)18.7374
1990's15 (50.00)18.2507
2000's1 (3.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Elliott, JM; Tayler, PJ; Young, JM1
Ward, D; Young, JM1
Jafferji, SS; Michell, RH1
Koike, K; Satoh, M; Takayanagi, I1
Choo, LK; Darroch, SA; Gardner, A; Mitchelson, F; Vong, YM1
Koike, K; Saito, K; Satoh, M; Takayanagi, I1
Hisayama, T; Kiuchi, Y; Kumagai, N; Takayanagi, I1
Koike, K; Ohtsuki, H; Saito, K; Satoh, M; Takayanagi, I1
Koike, K; Saito, K; Takayanagi, I1
Harada, M; Kiuchi, Y; Ohtsuki, H; Takayanagi, I1
Hootman, SR; Picado-Leonard, TM1
Gardner, JD; Jensen, RT; Rattan, S; Sutliff, VE1
Brown, JH; Harden, TK; Heng, MM1
Brown, JH; Goldstein, D1
Kagiya, T; Mizushima, A; Uchida, S; Yoshida, H; Zhou, XM1
Hisayama, T; Kumagai, N; Takayanagi, I1
Christophe, J; De Neef, P; Robberecht, P; Waelbroeck, M1
Birdsall, NJ; Burgen, A; Hulme, EC1
Birdsall, NJ; Burgen, AS; Hulme, EC; Wong, EH1
Ringdahl, B1
Haigh, E; Young, JM1
Richards, MH; van Giersbergen, PL1
Baum, BJ; Dai, Y1
Fain, JN; Sallés, J; Wallace, MA1
Ethier, MF; Madison, JM; Samant, N; Schaefer, OP; Yamaguchi, H1
Levin, RJ; Przyborski, SA1
Chidiac, P; Green, MA; Wells, JW1
Hishinuma, S; Hongo, I; Kurokawa, M; Matsumoto, Y; Narita, F1
Hayasaka, M; Horiuchi, K; Satoh, M; Takayanagi, I1
Park, PS; Wells, JW1

Reviews

1 review(s) available for carbachol and propylbenzilylcholine mustard

ArticleYear
[Transition of drug receptor mechanisms].
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 1992, Volume: 28, Issue:2

    Topics: Animals; Calcium; Carbachol; Dioxanes; Muscle Contraction; Phenylephrine; Pilocarpine; Propylbenzilylcholine Mustard; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Muscarinic

1992

Other Studies

29 other study(ies) available for carbachol and propylbenzilylcholine mustard

ArticleYear
Changes in muscarinic ligand binding to intestinal muscle strips produced by pre-exposure to hypotonic conditions.
    The Journal of pharmacy and pharmacology, 1978, Volume: 30, Issue:1

    Topics: Animals; Atropine Derivatives; Binding, Competitive; Carbachol; Guinea Pigs; In Vitro Techniques; Intestine, Small; Kinetics; Ligands; Muscle, Smooth; Osmolar Concentration; Parasympathomimetics; Propylbenzilylcholine Mustard; Receptors, Cholinergic; Receptors, Muscarinic; Trihexyphenidyl

1978
Ligand binding to muscarinic receptors in intact longitudinal muscle strips from guinea-pig intestine.
    British journal of pharmacology, 1977, Volume: 61, Issue:2

    Topics: Animals; Atropine; Atropine Derivatives; Carbachol; Guinea Pigs; In Vitro Techniques; Intestine, Small; Ligands; Muscle, Smooth; Propylbenzilylcholine Mustard; Quaternary Ammonium Compounds; Receptors, Cholinergic; Receptors, Muscarinic

1977
Investigation of the relationship between cell-surface calcium-ion gating and phosphatidylinositol turnover by comparison of the effects of elevated extracellular potassium ion concentration on ileium smooth muscle and pancreas.
    The Biochemical journal, 1976, Nov-15, Volume: 160, Issue:2

    Topics: Animals; Atropine; Calcium; Carbachol; Cell Membrane; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Pancreas; Phosphatidylinositols; Potassium; Propylbenzilylcholine Mustard; Receptors, Drug

1976
Effect of temperature reduction on responsiveness to cholinomimetics in the taenia caeci of the guinea-pig.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Colon; Drug Interactions; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Kinetics; Muscle Contraction; Parasympathomimetics; Phenoxybenzamine; Pirenzepine; Propylbenzilylcholine Mustard; Quinuclidinyl Benzilate; Temperature

1991
Characterization of muscarine receptors in rabbit ciliary body smooth muscle using propylbenzilylcholine mustard.
    General pharmacology, 1991, Volume: 22, Issue:5

    Topics: Animals; Carbachol; Ciliary Body; In Vitro Techniques; Male; Muscle, Smooth; Propylbenzilylcholine Mustard; Rabbits; Receptors, Muscarinic

1991
Guanosine 5'-triphosphate converts some populations of propylbenzilylcholine mustard-sensitive muscarinic cholinoceptor sites to sites resistant to the drug in intestinal smooth muscle.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:3

    Topics: Alkylation; Animals; Carbachol; Female; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Intestinal Mucosa; Intestines; Kinetics; Membranes; Muscle, Smooth; Propylbenzilylcholine Mustard; Proteins; Quinuclidinyl Benzilate; Receptors, Muscarinic

1991
Propylbenzilycholine mustard (PrBCM)-sensitive cholinoceptors and contractile response to partial agonist in guinea pig ileal muscle.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:2

    Topics: Algorithms; Animals; Calcium; Carbachol; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phenoxybenzamine; Pilocarpine; Propylbenzilylcholine Mustard; Receptors, Cholinergic

1991
Propylbenzilylcholine mustard-sensitive and -resistant muscarinic receptors in cardiac muscle.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Carbachol; Drug Resistance; Guinea Pigs; Heart; In Vitro Techniques; Male; Myocardium; Pilocarpine; Propylbenzilylcholine Mustard; Quaternary Ammonium Compounds; Receptors, Muscarinic

1991
Activation of propylbenzilylcholine mustard-sensitive muscarinic cholinoceptors more effectively utilizes cytosolic Ca2+ for contraction in guinea-pig intestinal smooth muscle.
    European journal of pharmacology, 1990, Oct-02, Volume: 187, Issue:1

    Topics: Animals; Calcium; Carbachol; Cytosol; Fura-2; Guinea Pigs; In Vitro Techniques; Intestines; Male; Muscle Contraction; Muscle, Smooth; Propylbenzilylcholine Mustard; Receptors, Cholinergic; Spectrometry, Fluorescence

1990
Effect of proteolytic cleavage on functional properties of muscarinic acetylcholine receptors in rat pancreatic and parotid acinar cells.
    The Biochemical journal, 1985, Nov-01, Volume: 231, Issue:3

    Topics: Amylases; Animals; Carbachol; In Vitro Techniques; Male; Pancreas; Papain; Parotid Gland; Propylbenzilylcholine Mustard; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1985
Characterization of cholinergic receptors mediating pepsinogen secretion from chief cells.
    The American journal of physiology, 1989, Volume: 257, Issue:2 Pt 1

    Topics: Acetylcholine; Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscarine; Pepsinogens; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Scopolamine

1989
Receptor reserve in the calcium-dependent cyclic AMP response of astrocytoma cells to muscarinic receptor stimulation: demonstration by agonist-induced desensitization, receptor inactivation, and phorbol ester treatment.
    Molecular pharmacology, 1986, Volume: 30, Issue:3

    Topics: Astrocytoma; Calcium; Carbachol; Cells, Cultured; Cyclic AMP; Inositol Phosphates; Isoproterenol; Oxotremorine; Phorbols; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Tetradecanoylphorbol Acetate

1986
Differences in muscarinic receptor reserve for inhibition of adenylate cyclase and stimulation of phosphoinositide hydrolysis in chick heart cells.
    Molecular pharmacology, 1986, Volume: 30, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Chick Embryo; Cyclic AMP; Kinetics; Myocardium; Phosphatidylinositols; Propylbenzilylcholine Mustard; Receptors, Muscarinic

1986
Cardiac M2 receptors consist of two different types, both regulated by GTP.
    European journal of pharmacology, 1987, Mar-31, Volume: 135, Issue:3

    Topics: Alkylation; Animals; Carbachol; GTP-Binding Proteins; Guinea Pigs; Heart; In Vitro Techniques; Kinetics; Membranes; Models, Biological; Myocardium; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Sulfhydryl Reagents

1987
Two apparently distinct muscarinic cholinoceptor mechanisms in guinea-pig taenia caecum.
    Japanese journal of pharmacology, 1988, Volume: 46, Issue:4

    Topics: Animals; Atropine; Carbachol; Cecum; Dibenzylchlorethamine; Female; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Myocardium; Phenoxybenzamine; Pilocarpine; Propylbenzilylcholine Mustard; Receptors, Muscarinic

1988
Propylbenzilylcholine mustard is selective for rat heart muscarinic receptors having a low affinity for agonists.
    British journal of pharmacology, 1986, Volume: 88, Issue:1

    Topics: Albumins; Animals; Binding, Competitive; Buffers; Carbachol; Choline; In Vitro Techniques; Membranes; Myocardium; Parasympathomimetics; Propylbenzilylcholine Mustard; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Time Factors

1986
The character of the muscarinic receptors in different regions of the rat brain.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1980, Feb-13, Volume: 207, Issue:1166

    Topics: Animals; Binding Sites; Brain; Carbachol; Mathematics; Oxotremorine; Propylbenzilylcholine Mustard; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1980
The effects of p-chloromercuribenzoate on muscarinic receptors in the cerebral cortex.
    British journal of pharmacology, 1983, Volume: 80, Issue:1

    Topics: Animals; Carbachol; Cerebral Cortex; Chloromercuribenzoates; Drug Interactions; In Vitro Techniques; Oxotremorine; p-Chloromercuribenzoic Acid; Propylbenzilylcholine Mustard; Rats; Receptors, Muscarinic; Tritium

1983
Determination of dissociation constants and relative efficacies of oxotremorine analogs at muscarinic receptors in the guinea-pig ileum by pharmacological procedures.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:1

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Kinetics; Mathematics; Oxotremorine; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Structure-Activity Relationship

1984
Persistent effects of high concentrations of chlorpromazine on 3H-propylbenzilylcholine mustard binding to muscarinic receptors in guinea-pig intestinal muscle strips.
    Archives internationales de pharmacodynamie et de therapie, 1980, Volume: 247, Issue:1

    Topics: Animals; Atropine; Carbachol; Chlorpromazine; Choline; Drug Interactions; Guinea Pigs; In Vitro Techniques; Intestinal Mucosa; Muscle, Smooth; Propylbenzilylcholine Mustard; Receptors, Cholinergic; Receptors, Muscarinic

1980
Human muscarinic receptors expressed in A9L and CHO cells: activation by full and partial agonists.
    British journal of pharmacology, 1995, Volume: 114, Issue:6

    Topics: Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Humans; Mice; Muscarinic Agonists; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Recombinant Proteins; Stimulation, Chemical

1995
Relationship between muscarinic receptor occupancy and response in rat parotid acinar cells.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Kinetics; Male; N-Methylscopolamine; Parasympatholytics; Parotid Gland; Propylbenzilylcholine Mustard; Radioligand Assay; Rats; Rats, Wistar; Receptors, Muscarinic; Scopolamine Derivatives; Time Factors; Tritium

1993
Differential effects of alkylating agents on the multiple muscarinic receptor subtypes linked to activation of phospholipase C by carbachol in rat brain cortical membranes.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Alkylating Agents; Animals; Carbachol; Cerebral Cortex; Enzyme Activation; In Vitro Techniques; Male; Mustard Compounds; Piperidines; Pirenzepine; Propylbenzilylcholine Mustard; Quinolines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Type C Phospholipases

1993
Muscarinic receptor reserve for inhibition of cAMP accumulation in bovine trachealis cells.
    The American journal of physiology, 1996, Volume: 270, Issue:2 Pt 1

    Topics: Animals; Carbachol; Cattle; Cell Separation; Cyclic AMP; Muscarinic Agonists; Phenoxybenzamine; Propylbenzilylcholine Mustard; Quinuclidinyl Benzilate; Receptors, Muscarinic; Trachea

1996
Assessment of receptor reserve during cholinergically induced intestinal secretion in rat jejunum in vitro.
    Acta physiologica Scandinavica, 1996, Volume: 158, Issue:4

    Topics: Animals; Carbachol; In Vitro Techniques; Jejunum; Male; Muscarinic Agonists; Propylbenzilylcholine Mustard; Rats; Receptors, Muscarinic

1996
Cardiac muscarinic receptors. Relationship between the G protein and multiple states of affinity.
    Biochemistry, 1997, Jun-17, Volume: 36, Issue:24

    Topics: Animals; Carbachol; Cell Membrane; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanylyl Imidodiphosphate; Mesocricetus; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Osmolar Concentration; Parasympatholytics; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1997
Contrasting effects of carbachol, McN-A-343 and AHR-602 on Ca(2+)-mobilization and Ca(2+)-influx pathways in taenia caeci.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Binding Sites; Calcium; Carbachol; Cell Membrane; Colon; Extracellular Space; Female; Guinea Pigs; In Vitro Techniques; Ion Transport; Male; Muscarinic Agonists; Propylbenzilylcholine Mustard; Pyrrolidines

1997
Protein kinase C mediates increase of Ca2+ sensitivity for contraction by cholinoceptor partial agonist in ileal longitudinal muscle of guinea pig.
    General pharmacology, 1998, Volume: 30, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Carbachol; Carbazoles; Cholinergic Agents; Coloring Agents; Enzyme Inhibitors; Fura-2; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Maleimides; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Pilocarpine; Propylbenzilylcholine Mustard; Protein Kinase C; Receptors, Cholinergic; Sensitivity and Specificity

1998
Monomers and oligomers of the M2 muscarinic cholinergic receptor purified from Sf9 cells.
    Biochemistry, 2003, Nov-11, Volume: 42, Issue:44

    Topics: Affinity Labels; Animals; Baculoviridae; Carbachol; Cell Line; Chromatography, Ion Exchange; Digitonin; Dimerization; Epitopes; Humans; Oligopeptides; Peptides; Precipitin Tests; Propylbenzilylcholine Mustard; Protein Binding; Proto-Oncogene Proteins c-myc; Quinuclidinyl Benzilate; Radioligand Assay; Receptor, Muscarinic M2; Solubility; Spodoptera

2003