Page last updated: 2024-08-17

carbachol and piperidines

carbachol has been researched along with piperidines in 246 studies

Research

Studies (246)

TimeframeStudies, this research(%)All Research%
pre-199037 (15.04)18.7374
1990's109 (44.31)18.2507
2000's71 (28.86)29.6817
2010's28 (11.38)24.3611
2020's1 (0.41)2.80

Authors

AuthorsStudies
Alioto, RL; Eash, JR; Krebs, JB; Mir, GN; Sperow, JW; Yelnosky, J1
Changeux, JP; Kato, G1
Kashima, K; Kataoka, K; Kato, M; Kuriyama, K; Ohkuma, S1
Sastry, BV; Stephan, CC1
Abdallah, EA; Eldefrawi, AT; Eldefrawi, ME; Jett, DA1
Bado, A; Cherifi, Y; Le Romancer, M; Lewin, MJ; Pigeon, C; Reyl-Desmars, F1
Buchan, AM; Kwok, YN; MacLeod, MD; Meloche, RM1
Bado, A; Laigneau, JP; Lewin, MJ; Moizo, L1
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1
Martin, JR1
Barlow, RB; Christophe, J; Renzetti, AR; Tastenoy, M; Waelbroeck, M1
Funakoshi, A; Jimi, A; Kono, A; Tateishi, K; Tsuru, M; Wakasugi, H1
Buyse, MA; Fraeyman, NH; Lefebvre, RA1
Pechnick, RN; Vargas, HM1
Challiss, RA; Nahorski, SR; Whitham, EM1
Courtney, MJ; Nicholls, DG1
Bagetta, G; Constanti, A1
Cheung, CL; De Boer, T; Tonnaer, JA1
Daniel, EE; Janssen, LJ1
Donoff, B; Lad, R; Rangachari, PK1
Alonso, MJ; Arribas, S; Balfagón, G; Marín, J; Salaices, M1
Chiba, S; Furukawa, Y; Nakane, T1
Costa, G; Massi, M; Melchiorre, C; Perfumi, M; Polidori, C; Sajia, A1
Hersey, SJ; Kajimura, M; Sachs, G; Scott, DR; Wilkes, JM1
Benedito, S; García-Sacristán, A; Hernández, M; Prieto, D; Rivera, L1
Richards, MH1
Endou, M1
Aihara, H; Isobe, Y; Muramatsu, M; Otomo, S1
Igata, H; Nishida, T; Okabe, S; Takagi, K1
Yang, CM1
Massi, M; Melchiorre, C; Perfumi, M; Polidori, C; Pompei, PL1
Alger, BE; Pitler, TA1
Harbon, S; Leiber, D; Marc, S1
Fleming, N; Laniyonu, A; Sliwinski-Lis, E1
Bloom, JW; Lai, J; Roeske, WR; Yamamura, HI1
Beinfeld, MC; Brog, JS1
Hanack, C; Herawi, M; Kopp, R; Lambrecht, G; Moser, U; Mutschler, E; Pfeiffer, A; Tacke, R1
Akahane, K; Chiba, S; Furukawa, Y; Karasawa, Y1
Gilani, AU1
Choo, LK; Darroch, SA; Mitchelson, F; Taylor, WC1
Daly, JW; Gusovsky, F; Hollingsworth, EB1
Brown, DR; Chang, EB; Field, M; Wang, NS1
Cohen-Armon, M; Sokolovsky, M1
Cohen-Armon, M; Henis, YI; Kloog, Y; Sokolovsky, M1
Ghataorre, AS; Lambert, DG; Nahorski, SR1
Syed, M; Tokuno, H; Tomita, T1
Diener, M; Knobloch, SF; Rummel, W1
Adeagbo, AS; Magbagbeola, AO1
Fowler, CJ; Thorell, G1
Roger, T; Ruckebusch, Y1
Funakoshi, A; Kitani, K; Miyasaka, K; Shinozaki, H1
Sokolovsky, M; van Koppen, CJ1
Davidesko, D; Doods, HN; Rinner, I; van Charldorp, KJ; van Zwieten, PA1
Cobbin, LB; Gilani, SA1
Bali, JP; Baudiere, B; Giraldo, E; Ladinsky, H; Monferini, E1
Barbieri, RL; Gochberg, J; Ryan, KJ1
Marshall, IG; Parsons, SM; Whitton, PS1
Barenholz, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M; Yechiel, E1
Eglen, RM; Whiting, RL1
Barlow, RB; Shepherd, MK1
Terrar, DA1
Bonta, IL; Saxena, PR1
Eichele, O; Mutschler, E1
Gandiha, A; Marshall, IG1
Fabian, K; Mörsdorf, K; Vahlensieck, W1
Mörsdorf, K; Wengenroth, H1
Aust, G; Van Zwieten, PA1
Thron, CD; Waud, DR1
Madill, HD; Savoie, ML; Stewart, WC1
Baron, B; Kloog, Y1
Frey, HH; Reiche, R1
Bonfilio, AC; Jacoby, HI; Mills, JE; Rasmussen, CR; Scott, MK1
Bartfai, T; Hedlund, B; Lundberg, JM1
Bartfai, T; Hedlund, B; Järv, J1
Coupar, IM; McLean, PG1
Mitchelson, F; Shen, A1
Hackmiller, RC; Jumblatt, JE1
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ1
Bristow, DR; Dupere, JR; Zamani, MR1
Imaizumi, Y; Kawai, T; Masuda, Y; Ryang, S; Tanaka, M; Watanabe, M; Yamahara, NS1
Maggio, R; Nanavati, S; Vogel, Z; Wess, J1
Bertrand, C; Bunnett, NW; Debas, HT; Geppetti, P; Huber, O; Nadel, JA; Pellegrini, CA1
Classen, M; Schaffer, K; Schepp, W; Schusdziarra, V; Wegner, U; Weigert, N1
De Giorgio, R; Giachetti, A; Maggi, CA; Patacchini, R1
Gabelt, BT; Kaufman, PL; Poyer, JF1
Fukui, H; Inagaki, N; Kondou, H1
Ko, FN; Lin, CH; Teng, CM; Wu, YC; Yang, CM1
DelValle, J; Park, J; Yamada, T; Yokotani, K1
Erwin, VG; Radcliffe, RA1
Barzaghi, F; Bonetti, C; Cesana, R; Fortin, M; Galliani, G; Hunt, P; Maggioni, A; Nencioni, A; Parini, C; Toja, E1
Dauphin, F; Hamel, E; Linville, DG1
Bobbin, RP; Erostegui, C; Norris, CH1
Blüml, K; Mutschler, E; Wess, J1
Angeli, P; Bianchi, S; Imeri, L; Mancia, M1
Fisher, L; Hall, S; Pennefather, JN1
Chuang, DM; Fukamauchi, F; Hough, C; Saunders, PA1
Maggio, R; Vogel, Z; Wess, J1
Consolo, S; Garcia Ruiz, AJ; La Porta, C; Ladinsky, H; Zambelli, M1
Fain, JN; Sallés, J; Wallace, MA1
Tonnaer, JA; van Huizen, F1
Shiraishi, K; Takayanagi, I1
Bado, A; Cherifi, Y; Laigneau, JP; Lewin, MJ; Moizo, L1
Gean, PW; Hsu, KS; Huang, CC1
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM1
Sjögren, C; Tobin, G1
Bartolini, A; Galeotti, N; Ghelardini, C; Gualtieri, F; Teodori, E1
De Neef, P; Domenach, V; Vandermeers, A; Vandermeers-Piret, MC; Waelbroeck, M1
de la Vega, MT; Montano, JA; Nunez, A1
Bilezikian, JP; Huber, F; Robinson, RB; Steinberg, SF; Sun, LS; Vulliemoz, Y1
Tobin, G1
Benavente, V; Botey, J; Eseverri, JL; Marin, A1
Buchan, AM; Koop, I; Meloche, RM; Squires, PE1
Gillespie, JI; Slater, BJ; Varma, JS1
Hsu, KS; Huang, CC; Yang, CH1
Arana, R; Bacman, S; Borda, E; Camusso, JJ; Hubscher, O; Sterin-Borda, L1
Onoe, H; Sakai, K1
Murayama, T; Nomura, Y; Yamada, T1
Aronstam, RS; Puhl, HL; Raman, PS; Williams, CL1
Levin, RJ; Przyborski, SA1
Semba, K; White, TD1
Arias-Montaño, JA; de la Vega, MT; Nuñez, A1
Bolton, TB; Zholos, AV1
Hara, Y; Nakaya, H; Tamagawa, M; Watanabe, Y1
Alfonzo, MJ; de Alfonzo, RG; de Becemberg, IL; de Herrera, VN; de Villaroel, SS; Misle, AJ1
Baba, H; Goldstein, PA; Kohno, T; Okamoto, M; Shimoji, K; Yoshimura, M1
Cobuzzi, A; Lai, FM; Spinelli, W1
Komori, S; Nakayama, T; Ohashi, H; Unno, T1
Laurier, LG; Preiksaitis, HG1
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M1
Blumenthal, JA; Carey, HV; Onorato, JJ1
Galas, L; Garnier, M; Lamacz, M; Lenglet, S; Tonon, MC; Vaudry, H1
Chew, CS; Flemström, G; Säfsten, B1
Hiley, CR; White, R1
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S; Rinaldi-Carmona, M1
Harris, D; Kendall, DA; Randall, MD1
Hara, T; Iwanaga, S; Makita, T; Shibata, O; Shibata, S; Sumikawa, K; Tsuda, A1
Braverman, A; Legos, J; Luthin, G; Ruggieri, M; Young, W1
Haapalinna, A; Larson, J; Niittykoski, M; Ruotsalainen, S; Sirviö, J1
Cross, AJ; De Souza, RJ; Green, AR; Misra, A; Murray, TK; Snape, MF; Williams, JL1
Damer, V; Krichevsky, VP; Pagala, MK; Vaydovsky, I; Wise, GJ1
Erickson, KA; Schroeder, A; Zhang, X1
Bernardi, G; Bonci, A; Grillner, P; Mercuri, NB; Svensson, TH1
Baiardi, P; Lucchelli, A; Masoero, E; Santagostino-Barbone, MG; Tonini, M1
Acs, Z; Makara, GB; Némethy, Z1
Arellano, RO; Garay, E; Miledi, R1
Feldman, JL; Shao, XM1
Kouznetsova, M; Nistri, A1
Eglen, RM; Luong, LA; MacLennan, SJ; Martin, GR; Martin, RS; Welsh, NJ1
Lau, WA; Mitchelson, FJ; Pennefather, JN1
Emala, CW; Fehr, JJ; Hirshman, CA1
Andersson, K; Fujiwara, M; Persson, K1
Malomough, A; Naumenko, N; Nikolsky, E; Urazaev, A; Vyskocil, F1
Levendusky, M; Longhurst, PA1
Kim, D; Moore, BA; Vanner, S1
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K1
Hashimoto, S; Iwanaga, S; Makita, T; Saito, M; Shibata, O; Sumikawa, K; Tsuda, A1
Chapple, CR; Chess-Williams, R; Couldwell, C; Sellers, DJ; Yamanishi, T; Yasuda, K1
Barrett, KE; Kahn, ME; Sausville, EA; Senderowicz, A1
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD1
Dohi, S; Ishizawa, Y; Ma, HC; Wang, YF; Yanagidate, F1
Kadota, H; Kuwahara, M; Mikami, H; Nishibata, R; Tsubone, H1
Franco, W; Leite, RS1
Bosmans, JP; Briejer, MR; Heylen, L; Jurzak, M; Leysen, JE; Prins, NH; Schuurkes, JA; Van Daele, P1
Choppin, A; Eglen, RM1
Herzog, M; Liu, J; Scherer, EQ; Scofield, MA; Shimozono, M; Wangemann, P1
Delbro, DS; Giglio, D; Tobin, G1
Fujikawa, T; Kimura, T; Mase, T; Noguchi, K; Numazawa, T; Ohtake, N; Sagara, T; Sagara, Y1
Pérez Leirós, C; Rosignoli, F1
Huang, SC1
Furness, JB; Kumano, K; Kunze, WA; Larsson, H; Murr, E; Vogalis, F1
Braverman, AS; Ruggieri, MR; Tallarida, RJ1
Alger, BE; Isokawa, M; Kim, J; Ledent, C1
Fukumori, R; Goshima, Y; Hagiwara, Y; Kanaya, T; Kubo, T; Okatani, H2
Alsasua, A; Benhamú, B; Girón, R; López-Rodríguez, ML; Martín, MI; Pascual, D1
Choi, KH; Jeon, JH; Kang, TM; Kim, HJ; Kim, IG; Kim, KW; Kim, SJ; Min, KW; Park, KH; So, I; Yang, DK1
Bernardino, CR; Chang, EL; Dartt, DA; Hodges, RR; Horikawa, Y; Rios, JD; Rubin, PA; Shatos, MA; Zoukhri, D1
Borda, E; Busch, L1
Bordi, F; Costa, LG; Dieguez-Acuña, FJ; Guizzetti, M; Madia, F; Vitalone, A; Woods, JS1
BENNETT, PB1
Harada, N; Makita, T; Niwa, M; Saito, M; Shibata, O; Sumikawa, K; Yamaguchi, M; Yoshimura, M1
Caruso, ML; De Ponti, F; Demma, I; Guerra, V; Lorusso, D; Maselli, MA; Pezzolla, F; Piepoli, AL1
Crittenden, EL; García, DM; González, A1
Borroni, B; Cattabeni, F; Colciaghi, F; Di Luca, M; Gardoni, F; Marcello, E; Padovani, A; Zimmermann, M1
Borda, E; Orman, B; Reina, S; Sterin-Borda, L1
Boxberger, M; Choritz, L; Krauss, A; Meissner, S; Rosenthal, R; Stumpff, F; Thieme, H; Wiederholt, M1
Blaha, CD; Miller, AD1
Borda, ES; Orman, B; Reina, S; Sterin-Borda, L1
Izumi, Y; Komori, S; Matsuyama, H; Okamoto, H; Sakamoto, T; Uchiyama, M; Unno, T; Wess, J; Yamada, M1
Alger, BE; Jones, LM; Karnup, SV; Karson, MA; Reich, CG1
Forrest, AS; Ordög, T; Sanders, KM1
Paulose, CS; Renuka, TR; Savitha, B1
Hattori, M; Komori, S; Matsuyama, H; Nishimura, M; Sakamoto, T; Uchiyama, M; Unno, T1
de Groat, WC; Ng, YK; Wu, HY1
Arias-Montaño, JA; Sánchez-Lemus, E1
Miyazu, M; Ohinata, H; Sugawara, R; Takai, A; Takai, Y; Yoshida, A1
Braverman, AS; Ruggieri, MR1
Braeter, M; Hakenberg, OW; Kelly, LU; Ravens, U; Waelbroeck, M; Weiss, A; Wuest, M1
Cao, J; Hashiba, K; Kitazawa, T; Komori, S; Taneike, T; Unno, T; Wess, J; Yamada, M1
Chapple, CR; Chess-Williams, R; Stevens, LA1
Hirose, K; Kaeriyama, S; Muramatsu, A; Nouchi, H; Sato, M; Shigenobu, K; Shimizu, N; Tanaka, H1
De Ridder, D; Gevaert, T; Hutchings, G; Nilius, B; Vandepitte, J; Vriens, J1
Alves, FH; Corrêa, FM; Crestani, CC; Resstel, LB1
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S1
Cloutier, S; Richter, M; Sirois, P1
Finney, SM; Gillespie, JI; Stewart, LH1
Lemtiri-Chlieh, F; Levine, ES1
Andersson, M; Aronsson, P; Delbro, DS; Giglio, D; Haraldsson, B; Tobin, G1
Korolkiewicz, RP; Sein-Anand, J; Sokołowska-Wojdyło, M; Umer, A; Włodarkiewicz, A; Ługowska-Umer, H1
Chen, H; Chen, YH; Li, J; Li, L; Liang, L; Liu, X; Liu, Y; Ma, J; Peng, L; Qi, J; Wu, X; Xiao, J; Xu, J; Yang, Y; Zhang, Y; Zhao, C1
Boone, TB; Lai, HH; Munoz, A; Smith, CP; Somogyi, GT; Szigeti, GP1
Anhê, G; Barbosa, HC; Bordin, S; Borelli, MI; Boschero, AC; Bowe, J; Gagliardino, JJ; Persaud, SJ1
Alves-Faria, P; Amaral, M; Falcão-Reis, F; Leite-Moreira, AF; Rocha-Sousa, A; Saraiva, J1
Atorino, G; Aviello, G; Borrelli, F; Capasso, R; Pagano, E; Romano, B1
Eda, H; Kimura, N; Komada, T; Mikami, T; Naganeo, R; Nakata, E; Nakatani, K; Ohmi, T; Sakakibara, M; Sugimoto, H; Suzuki, K; Toga, T1
Aydin, B; Cabadak, H; Kan, B; Küçükibrahimoğlu, E; Zafer Gören, M1
Choi, S; Choi, SJ; Jun, JY; Kim, SH; Parajuli, SP; So, KY; Sohn, HM; Yeum, CH; Yoon, PJ1
Kaba, H; Takahashi, Y1
Amici, M; Cho, K; Collingridge, GL; Dickinson, BA; Futai, K; Jo, J; Kim, MJ; Lee, YB; Sheng, M; Son, GH; Whitcomb, DJ; Winters, BL1
Haghparast, A; Hassanpour-Ezatti, M; Safari, MS; Taslimi, Z1
Ami, N; Fushiki, H; Koga, K; Ogino, Y; Ohta, H; Ueno, Y1
Boone, TB; Lai, HH; Munoz, A; Smith, CP; Somogyi, GT1
Britton, FC; Koh, SD; O'Driscoll, K; Sanders, KM; Sung, IK; Sung, TS; Zheng, H; Zhu, MH1
Barnes, PJ; Brown, SM; Chana, KK; Donnelly, LE; Fenwick, PS; Koarai, A; Nicholson, AG; Russell, RE; Traves, SL1
Altun, A; Bagcivan, I; Durmus, N; Kaya, T; Sarac, B; Sencan, M; Turan, M1
Chess-Williams, R; Moro, C; Uchiyama, J1
Browning, C; Clark, KL; Connor, HE; Ford, AJ; Hall, DA; Hodgson, ST; Luttmann, MA; Russell, LJ; Saunders, KA; Slack, RJ1
Henry, PJ; Mann, TS; Taylor, SJ1
Kajioka, S; Naito, S; Seki, N; Shahab, N1
Andersson, M; Aronsson, P; Doufish, D; Lampert, A; Tobin, G1
Lograno, MD; Romano, MR1
Barnes, PJ; Brown, SM; Donnelly, LE; Koarai, A; Nicholson, AG; Sturton, RG1
Ambudkar, I; Cotrim, A; Liu, X; Mitchell, J; Mori, Y; Swaim, W; Teos, L; Zheng, C1
Arrighi, N; Bodei, S; Cosciani Cunico, S; Michel, MC; Sigala, S; Simeone, C; Spano, P; Zani, D1
Parajuli, SP; Petkov, GV1
Jackson, MW; Park, K; Park, S1
Andersson, KE; Campeau, L; Füllhase, C; Gratzke, C; Hedlund, P; Hennenberg, M; Sibaev, A; Stief, C; Storr, M1
Deng, J; Li, L; Shi, C; Song, B; Wu, Y; Zhang, X1
de Guzman, G; Freestone, PS; Lipski, J; Wu, XH1
Haghparast, A; Jahangirvand, M; Moradi, M; Pirasteh, AH; Yazdi, F1
Esmaeili, MH; Ezzatpanah, S; Haghparast, A; Reisi, Z2
Brown, RE; McKenna, JT; Yang, C1
Al-Ayed, MSZ1
Agnetta, L; Bermudez, M; Decker, M; Gerwe, H; Holze, J; Irmen, M; Littmann, T; Schramm, S; Tränkle, C; Wolber, G1
Hassanpour, S; Lankarani Mohajer, L; Zendehdel, M1

Reviews

1 review(s) available for carbachol and piperidines

ArticleYear
Pharmacology and second messenger interactions of cloned muscarinic receptors.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Animals; Atropine; Carbachol; Cell Line; Humans; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic; Recombinant Proteins; Second Messenger Systems; Transfection

1991

Trials

1 trial(s) available for carbachol and piperidines

ArticleYear
[Ebastine : treatment of perennial rhinitis in the child].
    Allergie et immunologie, 1996, Volume: 28, Issue:8

    Topics: Adolescent; Butyrophenones; Carbachol; Child; Conjunctivitis, Allergic; Female; Histamine H1 Antagonists; Humans; Male; Nasal Provocation Tests; Piperidines; Rhinitis, Allergic, Perennial; Skin Tests; Treatment Outcome

1996

Other Studies

244 other study(ies) available for carbachol and piperidines

ArticleYear
In vivo antimotility and antidiarrheal activity of lidamidine hydrochloride (WHR-1142A), a novel antidiarrheal agent. Comparison with diphenoxylate and loperamide.
    Arzneimittel-Forschung, 1978, Volume: 28, Issue:8a

    Topics: Amidines; Animals; Antidiarrheals; Carbachol; Charcoal; Cholera Toxin; Diarrhea; Diphenoxylate; Feces; Gastrointestinal Motility; Isonipecotic Acids; Loperamide; Male; Piperidines; Prostaglandins E; Rats; Serotonin; Stomach

1978
Studies on the effect of histrionicotoxin on the monocellular electroplax from Electrophorus electricus and on the binding of (3H)acetylcholine to membrane fragments from Torpedo marmorata.
    Molecular pharmacology, 1976, Volume: 12, Issue:1

    Topics: Alkynes; Animals; Carbachol; Diaphragm; Eels; Electric Organ; Electrophorus; In Vitro Techniques; Phrenic Nerve; Piperidines; Rats; Receptors, Drug; Toxins, Biological

1976
Characterization of muscarinic receptor subtypes on rat pancreatic acini: pharmacological identification by secretory responses and binding studies.
    Digestion, 1992, Volume: 52, Issue:3-4

    Topics: Amylases; Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Male; Pancreas; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Sincalide

1992
Characterization of the subtype of muscarinic receptor coupled to the stimulation of phosphoinositide hydrolysis in 132-1N1 human astrocytoma cells.
    Cellular and molecular biology (Noisy-le-Grand, France), 1992, Volume: 38, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Astrocytoma; Atropine; Carbachol; Diamines; Humans; Hydrolysis; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Tumor Cells, Cultured

1992
Differential effects of paraoxon on the M3 muscarinic receptor and its effector system in rat submaxillary gland cells.
    Journal of biochemical toxicology, 1992,Summer, Volume: 7, Issue:2

    Topics: Animals; Atropine; Binding Sites; Carbachol; Cyclic AMP; Hydrolysis; Male; Paraoxon; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Regression Analysis; Submandibular Gland

1992
Purification of a histamine H3 receptor negatively coupled to phosphoinositide turnover in the human gastric cell line HGT1.
    The Journal of biological chemistry, 1992, Dec-15, Volume: 267, Issue:35

    Topics: Binding Sites; Carbachol; Cholera Toxin; Chromatography, Affinity; Chromatography, Gel; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Antagonists; Humans; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Kinetics; Methylhistamines; Molecular Weight; Phosphatidylinositols; Piperidines; Receptors, Histamine; Receptors, Histamine H3; Stomach Neoplasms; Tumor Cells, Cultured

1992
Muscarinic regulation of somatostatin release from primary cultures of human antral epithelial cells.
    Pharmacology, 1992, Volume: 44, Issue:1

    Topics: Adult; Carbachol; Cells, Cultured; Epithelium; Female; Humans; Male; Methacholine Chloride; Parasympatholytics; Piperidines; Pyloric Antrum; Radioimmunoassay; Receptors, Muscarinic; Somatostatin

1992
Pharmacological characterization of histamine H3 receptors in isolated rabbit gastric glands.
    The American journal of physiology, 1992, Volume: 262, Issue:1 Pt 1

    Topics: Aminopyrine; Animals; Carbachol; Gastric Mucosa; Histamine; Histamine Release; In Vitro Techniques; Male; Methylhistamines; Piperidines; Rabbits; Ranitidine; Receptors, Histamine H1

1992
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992
Pressor response to posterior hypothalamic administration of carbachol is mediated by muscarinic M3 receptor.
    European journal of pharmacology, 1992, Apr-29, Volume: 215, Issue:1

    Topics: Animals; Atropine Derivatives; Blood Pressure; Carbachol; Diamines; Dose-Response Relationship, Drug; Hypothalamus, Posterior; Kinetics; Male; Microinjections; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1992
Inactivation of brain cortex muscarinic receptors by 4-diphenylacetoxy-1-(2-chloroethyl) piperidine mustard.
    Biochemical pharmacology, 1992, Jul-22, Volume: 44, Issue:2

    Topics: Animals; Carbachol; Cerebral Cortex; Diphenylacetic Acids; Muscarinic Antagonists; Myocardium; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1992
Acetylcholine regulates pancreastatin secretion from the human pancreastatin-producing cell line (QGP-1N).
    The Journal of clinical endocrinology and metabolism, 1991, Volume: 73, Issue:1

    Topics: Acetylcholine; Adenoma, Islet Cell; Atropine; Calcimycin; Calcium; Carbachol; Chromogranin A; Gastrin-Releasing Peptide; Humans; Pancreatic Hormones; Pancreatic Neoplasms; Parasympatholytics; Peptides; Piperidines; Pirenzepine; Receptors, Muscarinic; Sincalide; Tumor Cells, Cultured

1991
Study of the muscarinic receptor subtypes in N1E 115 mouse neuroblastoma cells.
    Pharmacological research, 1991, Volume: 23, Issue:1

    Topics: Animals; Carbachol; Cyclic AMP; Cyclic GMP; Indicators and Reagents; Ligands; Mice; Neuroblastoma; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tumor Cells, Cultured

1991
Binding affinity and antimuscarinic activity of sigma and phencyclidine receptor ligands.
    European journal of pharmacology, 1991, Mar-19, Volume: 195, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Cerebral Cortex; Dioxolanes; Guinea Pigs; Haloperidol; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Pentazocine; Phosphatidylinositols; Piperidines; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine; Scopolamine Derivatives

1991
M3 muscarinic cholinoceptors are linked to phosphoinositide metabolism in rat cerebellar granule cells.
    European journal of pharmacology, 1991, Mar-25, Volume: 206, Issue:3

    Topics: Animals; Animals, Newborn; Binding, Competitive; Carbachol; Cerebellum; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Kinetics; Male; Parasympatholytics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Metabotropic receptor-mediated regulation of cytoplasmic free calcium in cultured cerebellar granule cells.
    Biochemical Society transactions, 1991, Volume: 19, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium; Carbachol; Cells, Cultured; Cerebellum; Cycloleucine; Cytoplasm; Ibotenic Acid; Kinetics; N-Methylaspartate; Neurotoxins; Piperidines; Quisqualic Acid; Receptors, Neurotransmitter

1991
Muscarinic inhibition of excitatory neurotransmission in guinea-pig olfactory cortex slices: weak antagonism by M3-muscarinic receptor antagonists.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cerebral Cortex; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Olfactory Bulb; Parasympatholytics; Piperidines; Receptors, Muscarinic; Synaptic Transmission

1991
cGMP formation and phosphoinositide turnover in rat brain slices are mediated by pharmacologically distinct muscarinic acetylcholine receptors.
    European journal of pharmacology, 1991, Jul-12, Volume: 207, Issue:3

    Topics: Animals; Atropine; Brain; Carbachol; Cyclic GMP; Guanylate Cyclase; Hippocampus; Inositol Phosphates; Male; Nitroprusside; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Succinimides

1991
Pre- and postjunctional muscarinic receptors in canine bronchi.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bethanechol Compounds; Bronchi; Carbachol; Dogs; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Functional subtyping of muscarinic receptors on canine esophageal mucosa.
    The American journal of physiology, 1991, Volume: 261, Issue:3 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Amiloride; Animals; Atropine; Carbachol; Chlorides; Dogs; Electric Conductivity; Esophagus; Female; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Mucous Membrane; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Sodium

1991
Presynaptic M2-muscarinic receptors on noradrenergic nerve endings and endothelium-derived M3 receptors in cat cerebral arteries.
    Brain research, 1991, Dec-13, Volume: 567, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Carbachol; Cats; Cerebral Arteries; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptors, Muscarinic; Vasodilation

1991
Anti-muscarinic effect of alinidine on acetylcholine-induced vasodilation in isolated and perfused dog coronary arteries.
    The Tohoku journal of experimental medicine, 1991, Volume: 165, Issue:2

    Topics: Acetylcholine; Animals; Carbachol; Clonidine; Coronary Vessels; Dogs; Female; In Vitro Techniques; Male; Parasympatholytics; Piperidines; Pirenzepine; Vasodilation

1991
The release of atrial natriuretic factor induced by central carbachol injection may be mediated by muscarinic M1 receptors.
    European journal of pharmacology, 1991, Mar-26, Volume: 195, Issue:2

    Topics: Animals; Atrial Natriuretic Factor; Brain; Carbachol; Diamines; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Subcutaneous; Male; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Muscarinic responses of gastric parietal cells.
    The Journal of membrane biology, 1991, Volume: 122, Issue:2

    Topics: Aminopyrine; Animals; Arachidonic Acids; Calcium; Carbachol; Glucose; Image Processing, Computer-Assisted; Ionomycin; N-Methylscopolamine; Parasympatholytics; Parietal Cells, Gastric; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1991
Distribution and function of cholinergic receptors in the sheep detrusor muscle.
    Journal of the autonomic nervous system, 1991, Jun-15, Volume: 34, Issue:2-3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Carbachol; Cholinesterase Inhibitors; Ganglia, Parasympathetic; Male; Muscle Contraction; Muscle, Smooth; Nerve Tissue Proteins; Piperidines; Pirenzepine; Receptors, Muscarinic; Sheep; Tetraisopropylpyrophosphamide; Urinary Bladder

1991
[Pharmacological analysis of drug interactions of disopyramide and its congeners with peripheral muscarinic acetylcholine receptors].
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1991, Volume: 66, Issue:5

    Topics: Animals; Binding, Competitive; Carbachol; Disopyramide; Drug Interactions; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; N-Methylscopolamine; Piperidines; Propylamines; Pyridines; Receptors, Muscarinic; Scopolamine Derivatives

1991
H2-receptor antagonism by a novel compound IT-066 assessed from [14C]aminopyrine accumulation in rabbit parietal cells.
    European journal of pharmacology, 1990, Mar-27, Volume: 178, Issue:3

    Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Cimetidine; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Piperidines; Pyridines; Rabbits

1990
[Effects of IT-066, a new histamine H2-receptor antagonist, on gastric acid secretion and experimental gastric ulcers in rats and dogs].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1990, Volume: 95, Issue:5

    Topics: Acetates; Animals; Anti-Ulcer Agents; Carbachol; Depression, Chemical; Dogs; Famotidine; Female; Gastric Acid; Histamine Antagonists; Histamine H2 Antagonists; Male; Pentagastrin; Piperidines; Pyridines; Rats; Rats, Inbred Strains; Stomach Ulcer

1990
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:1

    Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea

1991
Natriuresis, kaliuresis and antidiuresis induced by central carbachol injection are mediated by muscarinic M1 receptors.
    European journal of pharmacology, 1991, Mar-19, Volume: 195, Issue:1

    Topics: Animals; Carbachol; Diamines; Diuresis; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Muscarinic Antagonists; Natriuresis; Piperidines; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Activation of the pharmacologically defined M3 muscarinic receptor depolarizes hippocampal pyramidal cells.
    Brain research, 1990, Nov-26, Volume: 534, Issue:1-2

    Topics: Animals; Carbachol; Evoked Potentials; Hippocampus; In Vitro Techniques; Kinetics; Parasympatholytics; Piperidines; Pirenzepine; Pyramidal Tracts; Rats; Receptors, Muscarinic

1990
Pharmacological evidence for distinct muscarinic receptor subtypes coupled to the inhibition of adenylate cyclase and to the increased generation of inositol phosphates in the guinea pig myometrium.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Cyclic AMP; Female; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Myometrium; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Type C Phospholipases; Uterine Contraction

1990
Muscarinic M3 receptors are coupled to two signal transduction pathways in rat submandibular cells.
    European journal of pharmacology, 1990, Mar-13, Volume: 188, Issue:2-3

    Topics: Animals; Atropine; Carbachol; Cyclic AMP; Parasympatholytics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Signal Transduction; Submandibular Gland

1990
Amplification of the rat M2 muscarinic receptor gene by the polymerase chain reaction: functional expression of the M2 muscarinic receptor.
    Life sciences, 1990, Volume: 47, Issue:12

    Topics: Alkaloids; Amino Acid Sequence; Animals; Base Sequence; Carbachol; Cell Line; Cloning, Molecular; Cyclic AMP; Fibroblasts; Furans; Gene Amplification; Gene Expression; Molecular Sequence Data; Muscarinic Antagonists; Naphthalenes; Phosphatidylinositols; Piperidines; Pirenzepine; Plasmids; Polymerase Chain Reaction; Rats; Receptors, Muscarinic; Transfection

1990
Inhibition of carbachol-induced inositol phosphate accumulation by phencyclidine, phencyclidine-like ligands and sigma agonists involves blockade of the muscarinic cholinergic receptor: a novel dioxadrol-preferring interaction.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Animals; Brain; Carbachol; Culture Techniques; Dibenzocycloheptenes; Dioxolanes; Dizocilpine Maleate; Inositol Phosphates; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sigma Factor; Transcription Factors

1990
Human gastric mucosa expresses glandular M3 subtype of muscarinic receptors.
    Digestive diseases and sciences, 1990, Volume: 35, Issue:12

    Topics: Carbachol; Gastric Mucosa; Humans; In Vitro Techniques; N-Methylscopolamine; Parasympatholytics; Piperazines; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1990
Muscarinic receptor subtypes mediating negative chrono- and inotropic responses in isolated, blood-perfused dog right atria.
    Journal of autonomic pharmacology, 1990, Volume: 10, Issue:1

    Topics: Animals; Atropine; Carbachol; Cardiotonic Agents; Dogs; Electric Stimulation; Female; Heart Atria; Male; Myocardial Contraction; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Vagus Nerve

1990
Comparison of the rate of occupancy of receptors by anti-cholinergic drugs.
    Biochemical Society transactions, 1990, Volume: 18, Issue:2

    Topics: Alkaloids; Animals; Atropine; Carbachol; Furans; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Naphthalenes; Parasympatholytics; Piperidines; Receptors, Cholinergic

1990
Structure-activity relationships of some Galbulimima alkaloids related to himbacine.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Alkaloids; Animals; Carbachol; Electric Stimulation; Furans; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Naphthalenes; Parasympatholytics; Piperidines; Plants, Medicinal; Structure-Activity Relationship

1990
Regulation of phosphatidylinositol turnover in brain synaptoneurosomes: stimulatory effects of agents that enhance influx of sodium ions.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:9

    Topics: Alkaloids; Animals; Batrachotoxins; Brain; Carbachol; Guinea Pigs; In Vitro Techniques; Indolizines; Ion Channels; Magnesium; Male; Norepinephrine; Ouabain; Phosphatidylinositols; Piperidines; Protein Kinase C; Saxitoxin; Scorpion Venoms; Sodium; Synaptosomes; Tetrodotoxin

1986
Secretagogue-induced changes in membrane calcium permeability in chicken and chinchilla ileal mucosa. Selective inhibition by loperamide.
    The Journal of clinical investigation, 1986, Volume: 78, Issue:1

    Topics: Amiloride; Animals; Bombesin; Calcium; Carbachol; Carrier Proteins; Cell Membrane Permeability; Chickens; Chinchilla; Dose-Response Relationship, Drug; Gallopamil; Ileum; Intestinal Mucosa; Loperamide; Neurotensin; Piperidines; Serotonin; Sodium-Hydrogen Exchangers; Substance P; Trifluoperazine

1986
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
    The Journal of biological chemistry, 1986, Sep-25, Volume: 261, Issue:27

    Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1986
Batrachotoxin changes the properties of the muscarinic receptor in rat brain and heart: possible interaction(s) between muscarinic receptors and sodium channels.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:10

    Topics: Aconitine; Animals; Batrachotoxins; Benzilates; Binding, Competitive; Brain; Carbachol; Guanylyl Imidodiphosphate; Ion Channels; Kinetics; Macromolecular Substances; Male; Myocardium; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1985
Muscarinic receptor binding characteristics of a human neuroblastoma SK-N-SH and its clones SH-SY5Y and SH-EP1.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Arecoline; Atropine; Carbachol; Cell Membrane; Humans; Neuroblastoma; Piperidines; Pirenzepine; Receptors, Muscarinic; Tumor Cells, Cultured

1989
Effects of cisapride on isolated guinea pig colon.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cisapride; Colon; Electric Stimulation; Female; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Microelectrodes; Muscle, Smooth; Piperidines; Serotonin; Serotonin Antagonists; Tetrodotoxin

1989
Action of loperamide on neuronally mediated and Ca2+- or cAMP-mediated secretion in rat colon.
    European journal of pharmacology, 1988, Aug-02, Volume: 152, Issue:3

    Topics: Animals; Calcium; Carbachol; Colforsin; Colon; Cyclic AMP; Electric Stimulation; In Vitro Techniques; Intestinal Mucosa; Loperamide; Male; Morphine; Neurons; Piperidines; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil

1988
Pharmacological actions of ifenprodil in the rat isolated anococcygeus muscle.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:11

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Chloride; Carbachol; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperidines; Potassium Chloride; Rats; Vasodilator Agents

1985
Antagonist effects of the enantiomers of 3-PPP towards alpha 1-adrenoceptors coupled to inositol phospholipid breakdown in the rat cerebral cortex.
    Pharmacology & toxicology, 1987, Volume: 60, Issue:5

    Topics: Animals; Antiparkinson Agents; Atropine; Carbachol; Cerebral Cortex; Haloperidol; In Vitro Techniques; Inositol Phosphates; Male; Norepinephrine; Phenoxybenzamine; Piperidines; Prazosin; Raclopride; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Salicylamides; Stereoisomerism; Sugar Phosphates

1987
Prokinetic effects of cisapride, naloxone and parasympathetic stimulation at the equine ileo-caeco-colonic junction.
    Journal of veterinary pharmacology and therapeutics, 1988, Volume: 11, Issue:4

    Topics: Animals; Carbachol; Cecum; Cisapride; Colon; Gastrointestinal Motility; Horses; Ileum; Injections, Intravenous; Metoclopramide; Naloxone; Parasympathomimetics; Pilocarpine; Piperidines

1988
Effects of cisapride on the pancreatic exocrine secretion in rats.
    Gastroenterologia Japonica, 1988, Volume: 23, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cholecystokinin; Cisapride; In Vitro Techniques; Male; Pancreas; Pancreatic Juice; Piperidines; Proglumide; Rats; Rats, Inbred Strains; Serotonin Antagonists

1988
Chemical modification of rat cerebral cortex M1 muscarinic receptors: role of histidyl residues in antagonist and agonist binding.
    Biochemical and biophysical research communications, 1988, Mar-30, Volume: 151, Issue:3

    Topics: Animals; Atropine; Benzilates; Binding Sites; Carbachol; Cerebral Cortex; Diethyl Pyrocarbonate; Histidine; Hydrogen-Ion Concentration; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Synaptosomes

1988
Binding of muscarine receptor antagonists to pig coronary smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:2

    Topics: Animals; Atropine; Carbachol; Coronary Vessels; Heart Atria; In Vitro Techniques; Muscle, Smooth, Vascular; Piperazines; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine; Tritium

1988
Interaction of himbacine with carbachol at muscarinic receptors of heart and smooth muscle.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 290, Issue:1

    Topics: Alkaloids; Animals; Carbachol; Female; Furans; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Naphthalenes; Parasympatholytics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stomach

1987
Characterization of the muscarinic receptor subtype in isolated gastric fundic cells of the rabbit.
    Biochemical pharmacology, 1987, Sep-15, Volume: 36, Issue:18

    Topics: Aminopyrine; Animals; Atropine; Carbachol; Gastric Fundus; Kinetics; Male; N-Methylscopolamine; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives

1987
Nicotine, cotinine, and anabasine inhibit aromatase in human trophoblast in vitro.
    The Journal of clinical investigation, 1986, Volume: 77, Issue:6

    Topics: Anabasine; Androstenedione; Aromatase Inhibitors; Carbachol; Cells, Cultured; Choriocarcinoma; Cotinine; Decamethonium Compounds; Dose-Response Relationship, Drug; Estradiol; Female; Hexamethonium Compounds; Humans; In Vitro Techniques; Kinetics; Microsomes; Nicotine; Piperidines; Placenta; Pregnancy; Pyrrolidinones; Smoking; Succinylcholine; Trophoblasts; Uterine Neoplasms

1986
Reduction of quantal size by vesamicol (AH5183), an inhibitor of vesicular acetylcholine storage.
    Brain research, 1986, Oct-15, Volume: 385, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; In Vitro Techniques; Membrane Potentials; Mice; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Phencyclidine; Piperidines; Receptors, Cholinergic; Synaptic Vesicles

1986
Role of lipids in age-related changes in the properties of muscarinic receptors in cultured rat heart myocytes.
    Biochemistry, 1986, Dec-02, Volume: 25, Issue:24

    Topics: Acetylcholine; Animals; Animals, Newborn; Benzilates; Carbachol; Cells, Cultured; Guanylyl Imidodiphosphate; Kinetics; Liposomes; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic

1986
Determination of the muscarinic receptor subtype mediating vasodilatation.
    British journal of pharmacology, 1985, Volume: 84, Issue:1

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Atropine; Benzodiazepinones; Carbachol; Dogs; Female; Femoral Artery; Gallamine Triethiodide; In Vitro Techniques; Male; Pancuronium; Parasympatholytics; Phenethylamines; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Vasodilation

1985
A search for selective antagonists at M2 muscarinic receptors.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Animals; Atrial Function; Carbachol; Chemical Phenomena; Chemistry; Guinea Pigs; Heart Rate; Ileum; Muscle Contraction; Myocardial Contraction; Piperidines; Receptors, Muscarinic; Structure-Activity Relationship

1985
Influence of SKF-525A congeners, strophanthidin and tissue-culture media on desensitization in frog skeletal muscle.
    British journal of pharmacology, 1974, Volume: 51, Issue:2

    Topics: Animals; Benzilates; Carbachol; Culture Media; Culture Techniques; Diphenylacetic Acids; Electric Stimulation; Kinetics; Membrane Potentials; Microelectrodes; Muscles; Neuromuscular Depolarizing Agents; Oxyphenonium; Piperidines; Proadifen; Rana temporaria; Strophanthidin; Strophanthins

1974
Specific blockade of cardiac muscarinic receptors by pancuronium bromide.
    Archives internationales de pharmacodynamie et de therapie, 1971, Volume: 189, Issue:2

    Topics: Acetylcholine; Androstanes; Animals; Carbachol; Guinea Pigs; Heart; Methacholine Compounds; Neuromuscular Nondepolarizing Agents; Parasympatholytics; Piperidines; Receptors, Drug

1971
[Basic substituted tryptamines and tryptophols. 3. Pharmacologic studies on 1- and 2-position of basic substituted derivatives].
    Archiv der Pharmazie und Berichte der Deutschen Pharmazeutischen Gesellschaft, 1970, Volume: 303, Issue:11

    Topics: Animals; Carbachol; Ethanol; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Indoles; Piperidines; Rats; Scopolamine; Stimulation, Chemical; Sympathomimetics; Tryptamines

1970
Studies on the action of some cholinoceptor agonists on the chick biventer cervicis muscle preparation.
    The International journal of neuroscience, 1973, Volume: 5, Issue:5

    Topics: Acetylcholine; Animals; Carbachol; Chickens; Choline; Cyclohexanols; Decamethonium Compounds; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Electric Stimulation; Ganglionic Stimulants; In Vitro Techniques; Muscle Contraction; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Nicotine; Parasympathomimetics; Physostigmine; Piperidines; Quaternary Ammonium Compounds

1973
[Induction and control of spasmo-analgesia].
    Zeitschrift fur Urologie und Nephrologie, 1971, Volume: 64, Issue:12

    Topics: Analgesics; Antipyrine; Carbachol; Colic; Dioxoles; Humans; Methylamines; Pain; Parasympatholytics; Pentazocine; Piperidines; Sulfonic Acids; Urinary Bladder Diseases

1971
5,5-diphenyl-2-(2'-piperidinoethyl)-1,3-dioxolane-4-one a new drug with potent spasmolytic activity.
    Pharmacology, 1970, Volume: 3, Issue:4

    Topics: Acetylcholine; Animals; Asthma; Atropine; Barium; Blood Pressure; Blood Vessels; Carbachol; Cats; Chlorides; Dioxoles; Guinea Pigs; Heart Rate; Histamine; Ileum; Jejunum; Muscle Contraction; Muscles; Papaverine; Parasympatholytics; Piperidines; Rabbits; Respiration; Vagus Nerve

1970
The influence of 1-[3-(1-cyclohexenyl)-3-phenylpropyl]-1-methylpiperidinium bromide (HOE 019) on gastric secretion in the rat.
    Arzneimittel-Forschung, 1970, Volume: 20, Issue:8

    Topics: Anesthesia; Animals; Atropine; Carbachol; Cyclohexanes; Depression, Chemical; Electric Stimulation; Gastric Acidity Determination; Gastric Juice; Gastric Mucosa; Histamine; Insulin Antagonists; Male; Parasympatholytics; Piperidines; Pylorus; Rats; Secretory Rate; Stimulation, Chemical; Vagus Nerve

1970
The rate of action of atropine.
    The Journal of pharmacology and experimental therapeutics, 1968, Volume: 160, Issue:1

    Topics: Animals; Atropine; Carbachol; Choline; Dibenzylchlorethamine; Guinea Pigs; Heart; Heart Atria; Hexamethonium Compounds; Ileum; In Vitro Techniques; Kinetics; Models, Biological; Perfusion; Physostigmine; Piperidines; Receptors, Drug; Reserpine

1968
Central and peripheral anticholinergic potency of some drugs antagonistic to anticholinesterase poisoning.
    Canadian journal of physiology and pharmacology, 1968, Volume: 46, Issue:4

    Topics: Animals; Antidotes; Atropine; Bradycardia; Carbachol; Central Nervous System; Cholinesterase Inhibitors; Female; Guinea Pigs; Hallucinogens; Heart Rate; Mandelic Acids; Methacholine Compounds; Mice; Parasympatholytics; Peripheral Nerves; Phosphates; Piperidines; Pupil; Quaternary Ammonium Compounds; Rabbits; Scopolamine; Seizures; Trihexyphenidyl

1968
Fatty acid incorporation increases the affinity of muscarinic cholinergic receptors for agonists.
    Biochimica et biophysica acta, 1984, Oct-16, Volume: 801, Issue:3

    Topics: Animals; Benzilates; Carbachol; Cell Membrane; Cerebral Cortex; Cobalt; Fatty Acids; Guanosine Triphosphate; Medulla Oblongata; Piperidines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1984
Antagonism of the 5-HT-induced bronchoconstriction in the cat.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 263, Issue:1

    Topics: Animals; Bronchi; Carbachol; Cats; Clenbuterol; Cyproheptadine; Female; Hemodynamics; Ketanserin; Male; Piperidines; Pregnancy; Serotonin; Serotonin Antagonists; Theophylline

1983
4-(Diphenylmethyl)-1-[(imino)methyl]piperidines as gastric antisecretory agents.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:4

    Topics: Animals; Anti-Ulcer Agents; Binding, Competitive; Carbachol; Female; Gastric Acid; Gastric Emptying; Piperidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1983
Vasoactive intestinal polypeptide enhances muscarinic ligand binding in cat submandibular salivary gland.
    Nature, 1982, Jan-14, Volume: 295, Issue:5845

    Topics: Animals; Benzilates; Binding, Competitive; Carbachol; Cats; Gastrointestinal Hormones; Kinetics; Parasympatholytics; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Submandibular Gland; Vasoactive Intestinal Peptide

1982
Kinetic studies on muscarinic antagonist-agonist competition.
    The Journal of biological chemistry, 1980, Apr-10, Volume: 255, Issue:7

    Topics: Animals; Atropine; Benzilates; Binding, Competitive; Carbachol; Intestine, Small; Kinetics; Male; Muscle, Smooth; Oxotremorine; Parasympatholytics; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1980
5-HT4 receptor antagonist affinities of SB207710, SB205008, and SB203186 in the human colon, rat oesophagus, and guinea-pig ileum peristaltic reflex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: Animals; Carbachol; Colon; Dioxanes; Esophagus; Female; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Indoles; Male; Muscle, Smooth; Peristalsis; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists

1995
Characterization of the muscarine receptor subtype on sympathetic nerve endings in the rat caudal artery.
    European journal of pharmacology, 1994, Feb-03, Volume: 252, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arteries; Atropine; Bis-Trimethylammonium Compounds; Carbachol; Female; In Vitro Techniques; Isoindoles; Male; Muscarinic Antagonists; Muscle, Smooth, Vascular; Nerve Endings; Parasympatholytics; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Sympathetic Nervous System; Tail; Trihexyphenidyl

1994
M2-type muscarinic receptors mediate prejunctional inhibition of norepinephrine release in the human iris-ciliary body.
    Experimental eye research, 1994, Volume: 58, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Carbachol; Child; Ciliary Body; Diamines; Dose-Response Relationship, Drug; Electric Stimulation; Humans; In Vitro Techniques; Iris; Middle Aged; Muscarine; Norepinephrine; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic

1994
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger

1994
An immortalised murine hypothalamic neuronal cell, GT1-7, expresses functional histamine H1 receptors.
    Neuroscience letters, 1994, Aug-29, Volume: 178, Issue:1

    Topics: Animals; Carbachol; Cell Line, Transformed; Dose-Response Relationship, Drug; Glutamic Acid; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Hypothalamus; Inositol Phosphates; Kinetics; Mice; Neurons; Neuropeptide Y; Piperidines; Pyrimidinones; Ranitidine; Receptors, Histamine H1; Serotonin; Substance P; Tritium

1994
Characterization of muscarinic receptors mediating relaxation and contraction in the rat iris dilator muscle.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Alkaloids; Animals; Arecoline; Bethanechol; Carbachol; Diamines; Dose-Response Relationship, Drug; Furans; Ganglia, Parasympathetic; Ganglionectomy; Iris; Male; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1995
Functional role of proline and tryptophan residues highly conserved among G protein-coupled receptors studied by mutational analysis of the m3 muscarinic receptor.
    The EMBO journal, 1993, Volume: 12, Issue:1

    Topics: Acetylcholine; Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Blotting, Northern; Carbachol; Cell Line; Codon; GTP-Binding Proteins; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; N-Methylscopolamine; Parasympatholytics; Piperidines; Proline; Protein Conformation; Rats; Receptors, Muscarinic; Recombinant Proteins; Restriction Mapping; RNA; Scopolamine Derivatives; Transfection; Tryptophan

1993
Tachykinins contract the circular muscle of the human esophageal body in vitro via NK2 receptors.
    Gastroenterology, 1993, Volume: 105, Issue:4

    Topics: Adolescent; Adult; Aged; Atropine; Benzamides; Biphenyl Compounds; Carbachol; Dose-Response Relationship, Drug; Esophagus; Glycopeptides; Humans; Isometric Contraction; Middle Aged; Muscle Contraction; Muscle, Smooth; Neprilysin; Neurokinin A; Neurokinin B; Piperidines; Receptors, Tachykinin; Substance P; Tachykinins; Tetrodotoxin

1993
Functional characterization of a muscarinic receptor stimulating gastrin release from rabbit antral G-cells in primary culture.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Arecoline; Atropine; Benzodiazepinones; Carbachol; Cell Adhesion; Cell Separation; Cells, Cultured; Gastrins; Immunohistochemistry; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Rabbits; Receptors, Muscarinic

1994
Different mechanism of tachykinin NK2 receptor blockade by SR 48968 and MEN 10,627 in the guinea-pig isolated gallbladder and colon.
    European journal of pharmacology, 1994, Dec-12, Volume: 271, Issue:1

    Topics: Amino Acid Sequence; Animals; Benzamides; Binding, Competitive; Carbachol; Colon; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1994
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
    Experimental eye research, 1994, Volume: 59, Issue:6

    Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines

1994
Formation of inositol phosphates mediated by M3 muscarinic receptors in type-1 and type-2 astrocytes from neonatal rat cerebral cortex.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Animals, Newborn; Astrocytes; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Inositol Phosphates; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Signal Transduction; Tubocurarine

1994
Antimuscarinic action of liriodenine, isolated from Fissistigma glaucescens, in canine tracheal smooth muscle.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Antineoplastic Agents, Phytogenic; Aporphines; Binding, Competitive; Carbachol; Cells, Cultured; Cyclic AMP; Diamines; Dogs; Female; Hydrolysis; Inositol Phosphates; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Phosphatidylinositols; Piperidines; Plants, Medicinal; Receptors, Muscarinic; Trachea

1994
Muscarinic M3 receptor-mediated release of gastrin from canine antral G cells in primary culture.
    Digestion, 1995, Volume: 56, Issue:1

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Enterochromaffin Cells; Gastrins; Muscarinic Antagonists; Parasympathetic Nervous System; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Receptor, Muscarinic M3; Receptors, Muscarinic; Stimulation, Chemical

1995
Characterization of neurotensin-stimulated phosphoinositide hydrolysis in brain regions of long sleep and short sleep mice.
    Brain research, 1993, Nov-26, Volume: 629, Issue:1

    Topics: Animals; Brain; Calcium; Carbachol; Cerebellum; Dose-Response Relationship, Drug; Hippocampus; Histamine H1 Antagonists; Hydrolysis; Inositol; Inositol Phosphates; Kinetics; Membrane Lipids; Mesencephalon; Mice; Mice, Inbred Strains; Neurotensin; Nucleus Accumbens; Organ Specificity; Phosphatidylinositols; Phospholipids; Piperidines; Receptors, Neurotensin; Second Messenger Systems; Sleep

1993
New classes of antimuscarinic agents endowed with selective antispasmodic properties. 1-Arylsulfonyl pyrrolidin-2-ones and 2-thiones, 1-arylsulfonyl piperidin-2-ones and 2-thiones and 1-arylsulfonyl hexahydro-2H-azepin-2-one.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:4

    Topics: Animals; Arecoline; Atropine; Azepines; Butylscopolammonium Bromide; Carbachol; Gastric Acid; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pupil; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Scopolamine Derivatives; Sulfones

1994
Cholinergic dilatation and constriction of feline cerebral blood vessels are mediated by stimulation of phosphoinositide metabolism via two different muscarinic receptor subtypes.
    Journal of neurochemistry, 1994, Volume: 63, Issue:2

    Topics: Animals; Carbachol; Cats; Cerebral Arteries; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Inositol Phosphates; Muscarinic Antagonists; Muscle, Smooth, Vascular; Parasympatholytics; Phosphatidylinositols; Pia Mater; Piperidines; Pirenzepine; Receptors, Muscarinic; Vasoconstriction; Vasodilation

1994
In vitro pharmacologic characterization of a cholinergic receptor on outer hair cells.
    Hearing research, 1994, Volume: 74, Issue:1-2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Bungarotoxins; Carbachol; Choline; Cholinergic Antagonists; Curare; Dimethylphenylpiperazinium Iodide; Guinea Pigs; Hair Cells, Auditory, Outer; In Vitro Techniques; Membrane Potentials; Nicotine; Piperidines; Pirenzepine; Quinolizines; Receptors, Cholinergic; Strychnine; Trimethaphan

1994
Insertion mutagenesis as a tool to predict the secondary structure of a muscarinic receptor domain determining specificity of G-protein coupling.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Aug-16, Volume: 91, Issue:17

    Topics: Acetylcholine; Amino Acid Sequence; Animals; Binding Sites; Carbachol; Cell Line; Chlorocebus aethiops; GTP-Binding Proteins; Kinetics; Models, Molecular; Molecular Sequence Data; Mutagenesis, Insertional; N-Methylscopolamine; Phosphatidylinositols; Piperidines; Protein Structure, Secondary; Rats; Receptors, Muscarinic; Recombinant Proteins; Scopolamine Derivatives; Transfection

1994
Selective blockade of different brain stem muscarinic receptor subtypes: effects on the sleep-wake cycle.
    Brain research, 1994, Feb-04, Volume: 636, Issue:1

    Topics: Animals; Brain Stem; Carbachol; Diamines; Electroencephalography; Male; Microinjections; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Polysomnography; Rats; Reticular Formation; Sleep; Wakefulness

1994
Tachykinin receptors in the rat isolated uterus.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Anti-Bacterial Agents; Benzamides; Carbachol; Estradiol; Female; Glycopeptides; Kinetics; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Uterus

1993
Agonist-induced down-regulation and antagonist-induced up-regulation of m2- and m3-muscarinic acetylcholine receptor mRNA and protein in cultured cerebellar granule cells.
    Molecular pharmacology, 1993, Volume: 44, Issue:5

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Cerebellum; Down-Regulation; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; RNA, Messenger; Up-Regulation

1993
Coexpression studies with mutant muscarinic/adrenergic receptors provide evidence for intermolecular "cross-talk" between G-protein-linked receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Apr-01, Volume: 90, Issue:7

    Topics: Acetylcholine; Animals; Carbachol; Cell Line; GTP-Binding Proteins; Kinetics; Models, Structural; N-Methylscopolamine; Parasympatholytics; Phosphatidylinositols; Piperidines; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Recombinant Fusion Proteins; Scopolamine Derivatives; Signal Transduction; Transfection; Yohimbine

1993
Differences between rat dorsal and ventral hippocampus in muscarinic receptor agonist binding and interaction with phospholipase C.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: Alkaloids; Animals; Carbachol; Furans; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Mitochondria; N-Methylscopolamine; Naphthalenes; Oxotremorine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Synaptosomes; Type C Phospholipases

1993
Differential effects of alkylating agents on the multiple muscarinic receptor subtypes linked to activation of phospholipase C by carbachol in rat brain cortical membranes.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Alkylating Agents; Animals; Carbachol; Cerebral Cortex; Enzyme Activation; In Vitro Techniques; Male; Mustard Compounds; Piperidines; Pirenzepine; Propylbenzilylcholine Mustard; Quinolines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Type C Phospholipases

1993
Muscarinic receptor regulation and 2nd messenger responses in rat neocortex cultures.
    Journal of receptor research, 1993, Volume: 13, Issue:1-4

    Topics: Animals; Binding, Competitive; Carbachol; Cells, Cultured; Cerebral Cortex; Down-Regulation; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Second Messenger Systems

1993
Subtype of muscarinic receptors mediating relaxation and contraction in the rat iris dilator smooth muscle.
    General pharmacology, 1993, Volume: 24, Issue:1

    Topics: Alkaloids; Animals; Atropine; Carbachol; Furans; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1993
H3-receptor activation inhibits cholinergic stimulation of acid secretion in isolated rabbit fundic glands.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:3

    Topics: Animals; Carbachol; Cholinergic Antagonists; Gastric Acid; Gastric Fundus; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Methylhistamines; Muscarinic Antagonists; N-Methylscopolamine; Piperidines; Rabbits; Ranitidine; Receptors, Histamine H3; Receptors, Muscarinic; Scopolamine Derivatives

1995
Muscarinic depression of excitatory synaptic transmission mediated by the presynaptic M3 receptors in the rat neostriatum.
    Neuroscience letters, 1995, Sep-08, Volume: 197, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Carbachol; Depression, Chemical; Electric Stimulation; Evoked Potentials; In Vitro Techniques; N-Methylaspartate; Neostriatum; Neurons; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Presynaptic; Synaptic Transmission

1995
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine

1995
In vivo and in vitro effects of muscarinic receptor antagonists on contractions and release of [3H]acetylcholine in the rabbit urinary bladder.
    European journal of pharmacology, 1995, Jul-25, Volume: 281, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; Diamines; Female; Gallamine Triethiodide; Muscarinic Antagonists; Muscle Contraction; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Tritium; Urinary Bladder

1995
S-(-)-ET 126: a potent and selective M1 antagonist in vitro and in vivo.
    Life sciences, 1996, Volume: 58, Issue:12

    Topics: Acetylcholine; Animals; Atrial Function, Left; Carbachol; Dose-Response Relationship, Drug; Ileum; In Vitro Techniques; Male; Mice; Muscarinic Antagonists; Phenylacetates; Piperidines; Pirenzepine; Rabbits; Rats; Vas Deferens

1996
Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Elapid Venoms; Furans; Gallamine Triethiodide; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Naphthalenes; Oxotremorine; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Protein Binding; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Membranes; Tubocurarine

1996
Carbachol stimulates inositol phosphate formation in rat thalamus slices through muscarinic M3-receptor activation.
    Neuroscience letters, 1996, Jul-26, Volume: 213, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Dose-Response Relationship, Drug; Inositol Phosphates; Male; Muscarinic Agonists; Muscarinic Antagonists; Organ Culture Techniques; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Thalamus; Tritium

1996
Muscarinic receptor heterogeneity in neonatal rat ventricular myocytes in culture.
    Journal of cardiovascular pharmacology, 1996, Volume: 27, Issue:4

    Topics: Animals; Animals, Newborn; Carbachol; Cells, Cultured; Cyclic AMP; GTP-Binding Proteins; Heart Rate; Inositol Phosphates; Muscarinic Agonists; Muscarinic Antagonists; Myocardium; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptors, Muscarinic; Signal Transduction; Stimulation, Chemical; Virulence Factors, Bordetella

1996
Muscarinic receptor subtypes in the submandibular gland and the urinary bladder of the rabbit: in vivo and in vitro functional comparisons of receptor antagonists.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:6

    Topics: Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Muscarinic Antagonists; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Submandibular Gland; Urinary Bladder

1995
Effect of cholinergic agonists on gastrin release from primary cultures of human antral G cells.
    Gastroenterology, 1997, Volume: 112, Issue:2

    Topics: Adult; Antibodies; Bombesin; Calcium; Carbachol; Cells, Cultured; Female; Gastrins; Humans; Male; Methacholine Chloride; Middle Aged; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pyloric Antrum; Somatostatin

1997
Abnormalities in the contractile properties of colonic smooth muscle in idiopathic slow transit constipation.
    The British journal of surgery, 1997, Volume: 84, Issue:2

    Topics: Adolescent; Adult; Aged; Carbachol; Cisapride; Colorectal Neoplasms; Constipation; Female; Gastrointestinal Transit; Humans; Isometric Contraction; Middle Aged; Muscle, Smooth; Piperidines

1997
Carbachol induces inward current in rat neostriatal neurons through a G-protein-coupled mechanism.
    Neuroscience letters, 1997, Mar-14, Volume: 224, Issue:2

    Topics: Animals; Carbachol; Cyclic AMP-Dependent Protein Kinases; GTP-Binding Proteins; Male; Muscarinic Agonists; Neostriatum; Neurons; Patch-Clamp Techniques; Piperidines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1997
Circulating antibodies against rat parotid gland M3 muscarinic receptors in primary Sjögren's syndrome.
    Clinical and experimental immunology, 1996, Volume: 104, Issue:3

    Topics: Adolescent; Adrenergic beta-Agonists; Adult; Animals; Antibodies, Blocking; Atropine; Carbachol; Carbamates; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Female; Humans; Immunoglobulin G; Isoproterenol; Muscarinic Antagonists; Parasympatholytics; Parotid Gland; Phenylcarbamates; Phosphatidylinositols; Piperidines; Pirenzepine; Protease Inhibitors; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Sjogren's Syndrome

1996
Critical role for M3 muscarinic receptors in paradoxical sleep generation in the cat.
    The European journal of neuroscience, 1997, Volume: 9, Issue:3

    Topics: Animals; Carbachol; Cats; Muscarinic Antagonists; Piperidines; Receptors, Muscarinic; Sleep

1997
Muscarinic acetylcholine receptors on rat thymocytes: their possible involvement in DNA fragmentation.
    Japanese journal of pharmacology, 1997, Volume: 73, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Apoptosis; Atropine; Binding, Competitive; Carbachol; DNA Fragmentation; Electrophoresis, Agar Gel; Hydrocortisone; Injections, Subcutaneous; Isotope Labeling; Male; Muscarinic Agonists; Muscarinic Antagonists; Nucleosomes; Oxotremorine; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Thymus Gland

1997
Inhibition of M3 muscarinic acetylcholine receptor-mediated Ca2+ influx and intracellular Ca2+ mobilization in neuroblastoma cells by the Ca2+/calmodulin-dependent protein kinase inhibitor 1-[N,O-bis(5-isoquinolinesulfonyl)-N-methyl-L-trosyl]-4-phenylpipe
    Biochemical pharmacology, 1997, Apr-25, Volume: 53, Issue:8

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Enzyme Inhibitors; Humans; Neuroblastoma; Piperidines; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Tumor Cells, Cultured

1997
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin

1997
M3 muscarinic receptor-mediated enhancement of NMDA-evoked adenosine release in rat cortical slices in vitro.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Atropine; Carbachol; Cerebral Cortex; Diamines; Drug Synergism; In Vitro Techniques; Kinetics; Magnesium; Male; Muscarinic Agonists; Muscarinic Antagonists; N-Methylaspartate; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic

1997
Carbachol-induced inositol phosphate formation in rat striatum is mediated by both M1 and M3 muscarinic receptors.
    Neuroscience letters, 1997, Sep-19, Volume: 233, Issue:2-3

    Topics: Animals; Carbachol; Corpus Striatum; Drug Evaluation, Preclinical; In Vitro Techniques; Inositol Phosphates; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar

1997
Muscarinic receptor subtypes controlling the cationic current in guinea-pig ileal smooth muscle.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Carbachol; Dioxoles; Dose-Response Relationship, Drug; Electric Conductivity; Guinea Pigs; Ileum; In Vitro Techniques; Ion Channels; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth; Patch-Clamp Techniques; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic

1997
Pirmenol inhibits muscarinic acetylcholine receptor-operated K+ current in the guinea pig heart.
    European journal of pharmacology, 1997, Oct-29, Volume: 338, Issue:1

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Atrial Fibrillation; Carbachol; Disopyramide; Electric Stimulation; Guinea Pigs; Heart; Patch-Clamp Techniques; Piperidines; Potassium Channels; Receptors, Muscarinic

1997
Two opposite signal transducing mechanisms regulate a G-protein-coupled guanylyl cyclase.
    Archives of biochemistry and biophysics, 1998, Feb-01, Volume: 350, Issue:1

    Topics: Animals; Carbachol; Cattle; Cell Membrane; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylate Cyclase; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Trachea; Virulence Factors, Bordetella

1998
Muscarinic facilitation of GABA release in substantia gelatinosa of the rat spinal dorsal horn.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Carbachol; Diamines; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Muscarinic Agonists; Neostigmine; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin

1998
Characterization of muscarinic receptors mediating the contraction of the urinary detrusor muscle in cynomolgus monkeys and guinea pigs.
    Life sciences, 1998, Volume: 62, Issue:13

    Topics: Animals; Carbachol; Diamines; Female; Guinea Pigs; Macaca fascicularis; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic; Urinary Bladder

1998
M2 and M3 muscarinic receptors couple, respectively, with activation of nonselective cationic channels and potassium channels in intestinal smooth muscle cells.
    Japanese journal of pharmacology, 1998, Volume: 76, Issue:2

    Topics: Animals; Atropine; Calcium; Carbachol; Guinea Pigs; Male; Muscarinic Agonists; Muscle, Smooth; Piperidines; Pirenzepine; Potassium Channels; Receptors, Muscarinic

1998
Pharmacological and molecular characterization of muscarinic receptors in cat esophageal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carbachol; Cats; Dioxoles; Electric Stimulation; Esophagus; Female; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Piperidines; Polymerase Chain Reaction; Receptors, Muscarinic; RNA, Messenger

1998
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
    Experimental neurology, 1998, Volume: 151, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon

1998
Muscarinic inhibition of substance P induced ion secretion in piglet jejunum.
    Canadian journal of physiology and pharmacology, 1998, Volume: 76, Issue:2

    Topics: Animals; Atropine; Carbachol; Cholinergic Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Gallamine Triethiodide; Histamine; Ion Transport; Jejunum; Mecamylamine; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Substance P; Swine; Time Factors

1998
Pharmacological and functional characterization of muscarinic receptors in the frog pars intermedia.
    Endocrinology, 1998, Volume: 139, Issue:8

    Topics: Acetylcholine; alpha-MSH; Animals; Calcium; Carbachol; Cyclic AMP; Enzyme Inhibitors; Inositol Phosphates; Male; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Pertussis Toxin; Piperidines; Pituitary Gland; Protein-Tyrosine Kinases; Rana ridibunda; Receptors, Muscarinic; Signal Transduction; Virulence Factors, Bordetella

1998
Calcium signaling in cultured human and rat duodenal enterocytes.
    The American journal of physiology, 1998, Volume: 275, Issue:2

    Topics: Animals; Calcium; Carbachol; Cell Adhesion; Cells, Cultured; Dose-Response Relationship, Drug; Duodenum; Extracellular Matrix; Fluorescent Dyes; Fura-2; Humans; Intestinal Mucosa; Male; Parasympatholytics; Piperidines; Rats; Rats, Inbred Lew; Signal Transduction; Sincalide; Vacuoles

1998
The actions of the cannabinoid receptor antagonist, SR 141716A, in the rat isolated mesenteric artery.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Animals; Benzimidazoles; Calcium; Cannabinoids; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Relaxation; Muscle, Smooth, Vascular; Penicillamine; Piperidines; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant

1998
In vitro functional evidence of neuronal cannabinoid CB1 receptors in human ileum.
    British journal of pharmacology, 1998, Volume: 125, Issue:7

    Topics: Adult; Aged; Aged, 80 and over; Benzoxazines; Calcium Channel Blockers; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Female; Humans; Ileum; In Vitro Techniques; Male; Middle Aged; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurons; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tetrodotoxin

1998
Characterization of cannabinoid receptors coupled to vasorelaxation by endothelium-derived hyperpolarizing factor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:1

    Topics: Animals; Benzofurans; Biological Factors; Carbachol; Cyclooxygenase Inhibitors; Endothelium, Vascular; In Vitro Techniques; Indoles; Male; Muscarinic Agonists; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vasodilation

1999
Contractile and phosphatidylinositol responses of rat trachea to anticholinesterase drugs.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1998, Volume: 45, Issue:12

    Topics: Animals; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Dimethylphenylpiperazinium Iodide; Edrophonium; Glucose; Inositol; Inositol Phosphates; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neostigmine; Neuromuscular Blocking Agents; Nicotinic Agonists; Organ Preservation Solutions; Phosphatidylinositols; Piperidines; Pyridostigmine Bromide; Radiopharmaceuticals; Rats; Rats, Wistar; Tetrodotoxin; Trachea; Tritium; Tromethamine

1998
M2 receptors in genito-urinary smooth muscle pathology.
    Life sciences, 1999, Volume: 64, Issue:6-7

    Topics: Animals; Binding Sites; Carbachol; Diamines; Dose-Response Relationship, Drug; Female; Hypertrophy; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Denervation; Muscle, Smooth; Organ Size; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptors, Muscarinic; Spinal Cord Injuries; Urinary Bladder; Urinary Bladder, Neurogenic

1999
Activation of muscarinic M3-like receptors and beta-adrenoceptors, but not M2-like muscarinic receptors or alpha-adrenoceptors, directly modulates corticostriatal neurotransmission in vitro.
    Neuroscience, 1999, Volume: 90, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic Fibers; Animals; Carbachol; Cerebral Cortex; Cholinergic Fibers; Corpus Striatum; Diamines; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Imidazoles; Isoproterenol; Male; Medetomidine; Mice; Mice, Inbred DBA; Muscarinic Agonists; Muscarinic Antagonists; Phenylephrine; Piperidines; Pirenzepine; Pyrrolidinones; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, AMPA; Receptors, Muscarinic; Scopolamine; Synaptic Transmission

1999
A comparative study in rats of the in vitro and in vivo pharmacology of the acetylcholinesterase inhibitors tacrine, donepezil and NXX-066.
    Neuropharmacology, 1999, Volume: 38, Issue:1

    Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbachol; Cholinesterase Inhibitors; Donepezil; Drug Evaluation, Preclinical; Humans; Indans; Indoles; Injections, Intraperitoneal; Isoquinolines; Logistic Models; Male; Physostigmine; Piperidines; Rats; Structure-Activity Relationship; Tacrine; Tumor Cells, Cultured

1999
Function of M3 muscarinic receptors in the rat urinary bladder following partial outlet obstruction.
    The Journal of urology, 1999, Volume: 161, Issue:5

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder Neck Obstruction

1999
Effect of continuous administration of a cholinergic agonist on [3H]4-DAMP binding and m3 mRNA expression in cultured human ciliary muscle cells.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 1999, Volume: 15, Issue:2

    Topics: Carbachol; Cells, Cultured; Cholinergic Agonists; Ciliary Body; Humans; Muscarinic Antagonists; Piperidines; Receptor, Muscarinic M3; Receptors, Muscarinic; RNA, Messenger

1999
Presynaptic muscarinic (M3) receptors reduce excitatory transmission in dopamine neurons of the rat mesencephalon.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Atropine; Carbachol; Diamines; Dicyclomine; Dopamine; Electric Stimulation; Excitatory Postsynaptic Potentials; Mesencephalon; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reaction Time; Receptor, Muscarinic M3; Receptors, Muscarinic; Synaptic Transmission; Tetrodotoxin

1999
Influence of fluoxetine and litoxetine on 5-HT4 receptor-mediated relaxation in the rat isolated oesophagus.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:3

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Drug Interactions; Esophagus; Fenclonine; Fluoxetine; In Vitro Techniques; Indoles; Male; Muscle Relaxation; Muscle, Smooth; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sulfonamides

1999
Effect of cholinergic drugs on the concentration of intracellular free calcium of rat pituitary intermediate lobe cells.
    Brain research bulletin, 1999, Sep-01, Volume: 50, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Atropine; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Cytosol; Female; Male; Melanocytes; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar; Vasodilator Agents

1999
Muscarinic receptor heterogeneity in follicle-enclosed Xenopus oocytes.
    The Journal of physiology, 1999, Dec-01, Volume: 521 Pt 2

    Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Follicle Stimulating Hormone; Gene Expression; Membrane Potentials; Muscarinic Antagonists; Oocytes; Ovarian Follicle; Oxotremorine; Patch-Clamp Techniques; Piperidines; Pirenzepine; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Transcription, Genetic; Tropicamide; Xenopus laevis

1999
Acetylcholine modulates respiratory pattern: effects mediated by M3-like receptors in preBötzinger complex inspiratory neurons.
    Journal of neurophysiology, 2000, Volume: 83, Issue:3

    Topics: Acetylcholine; Animals; Animals, Newborn; Carbachol; Electrophysiology; In Vitro Techniques; Membrane Potentials; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3; Receptors, Muscarinic; Respiratory Mechanics; Synapses; Tetrodotoxin

2000
Facilitation of cholinergic transmission by substance P methyl ester in the mouse hippocampal slice preparation.
    The European journal of neuroscience, 2000, Volume: 12, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Acetylcholine; Action Potentials; Animals; Atropine; Bicuculline; Carbachol; Cholinergic Agonists; Drug Synergism; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Hippocampus; Male; Membrane Potentials; Mice; Patch-Clamp Techniques; Piperidines; Pyramidal Cells; Quinuclidines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Substance P; Tetrodotoxin; Valine

2000
Effects of cannabinoid receptor agonists on neuronally-evoked contractions of urinary bladder tissues isolated from rat, mouse, pig, dog, monkey and human.
    British journal of pharmacology, 2000, Volume: 129, Issue:8

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Atropine; Benzoxazines; Calcium Channel Blockers; Carbachol; Cholinergic Agonists; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Humans; In Vitro Techniques; Macaca fascicularis; Male; Mice; Morpholines; Muscle Contraction; Naphthalenes; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Receptors, Muscarinic; Rimonabant; Species Specificity; Swine; Urinary Bladder

2000
Cholinergic facilitation of neurotransmission to the smooth muscle of the guinea-pig prostate gland.
    British journal of pharmacology, 2000, Volume: 130, Issue:5

    Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Electric Stimulation; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Prostate; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Transmission

2000
Cellular signaling by the potent bronchoconstrictor endothelin-1 in airway smooth muscle.
    Critical care medicine, 2000, Volume: 28, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Azepines; Carbachol; Cholinergic Agonists; Endothelin-1; Female; Inositol Phosphates; Male; Muscle, Smooth; Oligopeptides; Piperidines; Signal Transduction; Swine; Trachea

2000
Nitric oxide-induced cGMP accumulation in the mouse bladder is not related to smooth muscle relaxation.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Animals; Arginine; Carbachol; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Female; In Vitro Techniques; Mice; Mice, Inbred BALB C; Molsidomine; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroarginine; Nitroprusside; Phosphodiesterase Inhibitors; Piperazines; Piperidines; Purines; Quinazolines; Sildenafil Citrate; Sulfones; Urethra; Urinary Bladder

2000
Carbachol and acetylcholine delay the early postdenervation depolarization of muscle fibres through M1-cholinergic receptors.
    Neuroscience research, 2000, Volume: 37, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Carbachol; Culture Techniques; Diaphragm; Male; Membrane Potentials; Muscarinic Agonists; Muscarinic Antagonists; Muscle Denervation; Muscle Fibers, Skeletal; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic

2000
Influence of gender and the oestrous cycle on in vitro contractile responses of the rat urinary bladder to cholinergic stimulation.
    British journal of pharmacology, 2000, Volume: 131, Issue:2

    Topics: Animals; Carbachol; Cholinergic Agonists; Diamines; Electric Stimulation; Estrus; Female; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Sex Characteristics; Time Factors; Urinary Bladder; Uterine Contraction

2000
Neural pathways regulating Brunner's gland secretion in guinea pig duodenum in vitro.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 279, Issue:5

    Topics: Animals; Brunner Glands; Capsaicin; Carbachol; Choline O-Acetyltransferase; Cholinergic Agonists; Cholinergic Fibers; Dimethylphenylpiperazinium Iodide; Duodenum; Electric Stimulation; Female; Ganglia, Sympathetic; Guanethidine; Guinea Pigs; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Neural Pathways; Neurotransmitter Agents; Nicotinic Agonists; Nicotinic Antagonists; Piperidines; Submucous Plexus; Substance P; Sympatholytics; Tetrodotoxin; Vagotomy; Vagus Nerve

2000
The role of M(2)-muscarinic receptors in mediating contraction of the pig urinary bladder in vitro.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzofurans; Binding, Competitive; Carbachol; Diamines; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Membranes; Muscarinic Antagonists; Muscle Contraction; Piperidines; Pyrrolidines; Quinuclidinyl Benzilate; Radioligand Assay; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Swine; Tritium; Urinary Bladder

2000
A dose-response study of anticholinesterase drugs on contractile and phosphatidylinositol responses of rat trachea.
    Anesthesia and analgesia, 2001, Volume: 92, Issue:1

    Topics: Animals; Carbachol; Cholinergic Agents; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Edrophonium; In Vitro Techniques; Inositol Phosphates; Isometric Contraction; Male; Muscarinic Antagonists; Muscle, Smooth; Neostigmine; Phosphatidylinositols; Piperidines; Pyridostigmine Bromide; Rats; Rats, Wistar; Stimulation, Chemical; Trachea

2001
M3 muscarinic receptors but not M2 mediate contraction of the porcine detrusor muscle in vitro.
    Journal of autonomic pharmacology, 2000, Volume: 20, Issue:3

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Swine; Urinary Bladder

2000
Possible mechanisms of diarrheal side effects associated with the use of a novel chemotherapeutic agent, flavopiridol.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2001, Volume: 7, Issue:2

    Topics: Antineoplastic Agents; Carbachol; Chloride Channels; Chlorides; Cholinergic Agonists; Colforsin; Colon; Cyclic AMP; Cyclin-Dependent Kinases; Diarrhea; Epidermal Growth Factor; Flavonoids; Humans; In Vitro Techniques; Intestinal Mucosa; Piperidines

2001
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate

2001
The antinociceptive and sedative effects of carbachol and oxycodone administered into brainstem pontine reticular formation and spinal subarachnoid space in rats.
    Anesthesia and analgesia, 2001, Volume: 92, Issue:5

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Atropine; Behavior, Animal; Carbachol; Cholinergic Agonists; Conscious Sedation; Diamines; Injections, Spinal; Male; Microinjections; Motor Activity; Muscarinic Antagonists; Pain Threshold; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Reticular Formation; Subarachnoid Space

2001
Effect of M2 and M3 muscarinic receptors on airway responsiveness to carbachol in bronchial-hypersensitive (BHS) and bronchial-hyposensitive (BHR) guinea pigs.
    Experimental animals, 2001, Volume: 50, Issue:1

    Topics: Animals; Bronchial Hyperreactivity; Carbachol; Diamines; Gene Expression; Guinea Pigs; Lung; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Trachea

2001
Effects of cholinergic agents on the vasopressin-mediated water transport in the isolated toad bladder.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 129, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Arginine Vasopressin; Atropine; Biological Transport; Bufo marinus; Calcium; Calcium Channel Blockers; Carbachol; Cholinergic Agonists; Cholinergic Antagonists; In Vitro Techniques; Isotonic Solutions; Lanthanum; Osmolar Concentration; Piperidines; Pirenzepine; Urinary Bladder; Vasoconstrictor Agents; Water

2001
The in vitro pharmacological profile of prucalopride, a novel enterokinetic compound.
    European journal of pharmacology, 2001, Jun-29, Volume: 423, Issue:1

    Topics: Acetylcholine; Animals; Benzofurans; Binding, Competitive; Carbachol; Cell Line; CHO Cells; Colon; Cricetinae; Dioxanes; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Female; Gallbladder; Gastrointestinal Agents; Granisetron; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Indoles; Indomethacin; Male; Motilin; Muscle Contraction; Piperidines; Rabbits; Rats; Rats, Wistar; Receptors, Cholecystokinin; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sincalide; Stomach; Sulfonamides; Vasodilator Agents

2001
Pharmacological characterization of muscarinic receptors in mouse isolated urinary bladder smooth muscle.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Acetylcholine; Animals; Carbachol; Diamines; Dioxolanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pilocarpine; Piperidines; Receptors, Muscarinic; Urinary Bladder

2001
Muscarinic receptors control K+ secretion in inner ear strial marginal cells.
    The Journal of membrane biology, 2001, Aug-01, Volume: 182, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Atropine; Calcium; Carbachol; Cholinergic Agonists; Cloning, Molecular; Cyclic AMP; Diamines; Dose-Response Relationship, Drug; Gerbillinae; Isoproterenol; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Stria Vascularis

2001
On the functional role of muscarinic M2 receptors in cholinergic and purinergic responses in the rat urinary bladder.
    European journal of pharmacology, 2001, Oct-12, Volume: 428, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Triphosphate; Animals; Carbachol; Diamines; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Piperidines; Pirenzepine; Purinergic Agonists; Purinergic Antagonists; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptors, Muscarinic; Receptors, Purinergic; Theophylline; Urinary Bladder

2001
Cyclohexylmethylpiperidinyltriphenylpropioamide: a selective muscarinic M(3) antagonist discriminating against the other receptor subtypes.
    Journal of medicinal chemistry, 2002, Feb-14, Volume: 45, Issue:4

    Topics: Acetylcholine; Animals; Bradycardia; Bronchoconstriction; Carbachol; CHO Cells; Cholinergic Agents; Combinatorial Chemistry Techniques; Cricetinae; Dipeptides; Heart Atria; Humans; In Vitro Techniques; Muscarinic Antagonists; Piperidines; Rats; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship

2002
Activation of nitric oxide synthase through muscarinic receptors in rat parotid gland.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: Amylases; Animals; Atropine; Binding, Competitive; Carbachol; Cell Membrane; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Parotid Gland; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Specific Pathogen-Free Organisms

2002
Two classes of endothelin receptors mediating contraction in esophageal muscularis mucosae.
    Regulatory peptides, 2002, May-30, Volume: 105, Issue:3

    Topics: Animals; Atropine; Autoradiography; Azepines; Binding, Competitive; Carbachol; Cell Membrane; Cells, Cultured; Endothelin Receptor Antagonists; Endothelins; Esophagus; Guinea Pigs; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Oligopeptides; Piperidines; Protein Binding; Receptors, Endothelin; Tetrodotoxin; Viper Venoms

2002
Sensitization of enteric reflexes in the rat colon in vitro.
    Autonomic neuroscience : basic & clinical, 2002, Apr-18, Volume: 97, Issue:1

    Topics: Animals; Area Under Curve; Carbachol; Cholinergic Agonists; Colon; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Hexamethonium; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Neurons, Afferent; Nicotinic Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Tachykinin; Serotonin Antagonists; Time Factors

2002
Interaction between muscarinic receptor subtype signal transduction pathways mediating bladder contraction.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2002, Volume: 283, Issue:3

    Topics: Animals; Carbachol; Cholinergic Agents; Denervation; Female; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Second Messenger Systems; Signal Transduction; Urinary Bladder; Urinary Incontinence

2002
Activation of muscarinic acetylcholine receptors enhances the release of endogenous cannabinoids in the hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Dec-01, Volume: 22, Issue:23

    Topics: Animals; Calcium; Cannabinoid Receptor Modulators; Cannabinoids; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Evoked Potentials; GTP-Binding Proteins; Hippocampus; In Vitro Techniques; Interneurons; Male; Mice; Mice, Knockout; Neural Inhibition; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, Metabotropic Glutamate; Receptors, Muscarinic

2002
Cholinergic mechanism in the lateral septal area is involved in the stress-induced blood pressure increase in rats.
    Brain research bulletin, 2003, Jan-30, Volume: 59, Issue:5

    Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Epinephrine; GABA Agonists; Injections, Intraventricular; Male; Muscarinic Antagonists; Muscimol; Norepinephrine; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Restraint, Physical; Septal Nuclei; Stress, Physiological

2003
New benzimidazole derivatives: selective and orally active 5-HT3 receptor antagonists.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: 5-Hydroxytryptophan; Administration, Oral; Animals; Aza Compounds; Behavior, Animal; Benzimidazoles; Carbachol; Diarrhea; Dose-Response Relationship, Drug; Gastric Emptying; Gastrointestinal Motility; In Vitro Techniques; Injections, Intraperitoneal; Injections, Intravenous; Male; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Piperidines; Propane; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Reflex; Serotonin; Serotonin Antagonists

2003
Five subtypes of muscarinic receptors are expressed in gastric smooth muscles of guinea pig.
    Experimental & molecular medicine, 2003, Feb-28, Volume: 35, Issue:1

    Topics: Animals; Base Sequence; Carbachol; Cations; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Guinea Pigs; Ion Channels; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Muscarinic; Stomach

2003
Activation of mitogen-activated protein kinase by cholinergic agonists and EGF in human compared with rat cultured conjunctival goblet cells.
    Investigative ophthalmology & visual science, 2003, Volume: 44, Issue:6

    Topics: Adult; Aged; Aged, 80 and over; Animals; Blotting, Western; Carbachol; Cells, Cultured; Cholinergic Agonists; Conjunctiva; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Goblet Cells; Humans; Male; Middle Aged; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Piperidines; Quinazolines; Rats; Rats, Sprague-Dawley; Time Factors; Tyrphostins

2003
Castration decreases amylase release associated with muscarinic acetylcholine receptor downregulation in rat parotid gland.
    British journal of pharmacology, 2003, Volume: 139, Issue:2

    Topics: Amylases; Animals; Binding, Competitive; Carbachol; Cholinergic Agonists; Down-Regulation; Inositol Phosphates; Male; Orchiectomy; Parotid Gland; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Receptors, Muscarinic

2003
Nuclear factor kappaB activation by muscarinic receptors in astroglial cells: effect of ethanol.
    Neuroscience, 2003, Volume: 120, Issue:4

    Topics: Astrocytes; Astrocytoma; Atropine; Blotting, Western; Carbachol; Cell Line; Cellular Structures; Central Nervous System Depressants; Chelating Agents; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Ethanol; Gallamine Triethiodide; Humans; Muscarinic Antagonists; NF-kappa B; Nicotinic Antagonists; Pertussis Toxin; Piperidines; Receptors, Muscarinic; Thymidine; Time Factors; Tritium

2003
Projections from the caudal part to the rostral part of the lateral septal area mediate blood pressure increase.
    Brain research bulletin, 2003, Sep-30, Volume: 61, Issue:5

    Topics: Animals; Blood Pressure; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Fluorescent Dyes; GABA Agonists; Hypertension; Male; Microinjections; Muscarinic Antagonists; Muscimol; Neural Pathways; Neurons; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Reaction Time; Septum of Brain; Stress, Physiological

2003
Comparison of the effects of drugs on nitrogen narcosis and oxygen toxicity in rats.
    Life sciences (1962), 1962, Volume: 1

    Topics: Animals; Bemegride; Carbachol; Epinephrine; Glutethimide; Hyperoxia; Inert Gas Narcosis; Methamphetamine; Nitrogen; Oxygen; Pentylenetetrazole; Phenacetin; Physostigmine; Piperidines; Rats; Scopolamine

1962
Metoclopramide causes airway smooth muscle relaxation through inhibition of muscarinic M3 receptor in the rat trachea.
    Anesthesia and analgesia, 2004, Volume: 98, Issue:5

    Topics: Animals; Antiemetics; Carbachol; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Metoclopramide; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phosphatidylinositols; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptor, Muscarinic M3; Trachea

2004
Colonic smooth muscle responses in patients with diverticular disease of the colon: effect of the NK2 receptor antagonist SR48968.
    Digestive and liver disease : official journal of the Italian Society of Gastroenterology and the Italian Association for the Study of the Liver, 2004, Volume: 36, Issue:5

    Topics: Aged; Aged, 80 and over; Anesthetics, Local; Atropine; Benzamides; Carbachol; Case-Control Studies; Cholinergic Agonists; Colon, Sigmoid; Colonic Neoplasms; Diverticulitis, Colonic; Electric Stimulation; Female; Humans; In Vitro Techniques; Isometric Contraction; Male; Middle Aged; Muscle, Smooth; Parasympatholytics; Piperidines; Receptors, Neurokinin-2; Stress, Mechanical; Tetrodotoxin

2004
Activation of muscarinic acetylcholine receptors elicits pigment granule dispersion in retinal pigment epithelium isolated from bluegill.
    BMC neuroscience, 2004, Jul-13, Volume: 5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Arecoline; Atropine; Carbachol; Colforsin; Cyclic AMP; Cytoplasmic Granules; Light; Muscarinic Agonists; Muscarinic Antagonists; Perciformes; Pigment Epithelium of Eye; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Retinal Pigments; Second Messenger Systems; Tropicamide

2004
Acetylcholinesterase inhibitors increase ADAM10 activity by promoting its trafficking in neuroblastoma cell lines.
    Journal of neurochemistry, 2004, Volume: 90, Issue:6

    Topics: Acetylcholinesterase; ADAM Proteins; ADAM10 Protein; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Atropine; Blotting, Western; Brefeldin A; Bungarotoxins; Carbachol; Cell Differentiation; Cell Fractionation; Cell Line, Tumor; Cholinergic Agonists; Cholinesterase Inhibitors; Donepezil; Drug Interactions; Embryo, Mammalian; Enzyme-Linked Immunosorbent Assay; Fluorescent Antibody Technique; Humans; Indans; Membrane Proteins; Metalloendopeptidases; Microscopy, Confocal; Muscarinic Antagonists; Neuroblastoma; Physostigmine; Piperidines; Protein Synthesis Inhibitors; Protein Transport; Tretinoin

2004
Signal transduction underlying carbachol-induced PGE2 generation and cox-1 mRNA expression of rat brain.
    Neuropharmacology, 2005, Volume: 48, Issue:5

    Topics: Animals; Carbachol; Cholinergic Agonists; Cyclic GMP; Cyclooxygenase 1; Dinoprostone; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Frontal Lobe; Gene Expression Regulation; Male; Membrane Proteins; Models, Biological; Muscarinic Antagonists; Nitric Oxide Synthase; Phosphatidylinositols; Piperidines; Pirenzepine; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction

2005
Stimulation of cannabinoid (CB1) and prostanoid (EP2) receptors opens BKCa channels and relaxes ocular trabecular meshwork.
    Experimental eye research, 2005, Volume: 80, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adult; Aged; Animals; Benzoxazines; Calcium; Calcium Channel Blockers; Cannabinoids; Carbachol; Cattle; Cells, Cultured; Cholinergic Agonists; Cyclic AMP; Cyclohexanols; Endothelin-1; Humans; In Vitro Techniques; Ion Channel Gating; Middle Aged; Morpholines; Naphthalenes; Patch-Clamp Techniques; Peptides; Piperidines; Potassium Channels, Calcium-Activated; Prostanoic Acids; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Prostaglandin E; Stimulation, Chemical; Trabecular Meshwork

2005
Midbrain muscarinic receptor mechanisms underlying regulation of mesoaccumbens and nigrostriatal dopaminergic transmission in the rat.
    The European journal of neuroscience, 2005, Volume: 21, Issue:7

    Topics: Animals; Carbachol; Cholinergic Agonists; Dopamine; Drug Interactions; Electrochemistry; Electrodes; Male; Muscarinic Antagonists; Nucleus Accumbens; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Scopolamine; Substantia Nigra; Synaptic Transmission; Ventral Tegmental Area

2005
Neuronal nitric oxide synthase activity in rat urinary bladder detrusor: participation in M3 and M4 muscarinic receptor function.
    Autonomic & autacoid pharmacology, 2005, Volume: 25, Issue:3

    Topics: Animals; Carbachol; Cholinergic Agonists; Cyclic GMP; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nitric Oxide Synthase Type I; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Tritium; Tropicamide; Urinary Bladder

2005
M(2) and M(3) muscarinic receptor-mediated contractions in longitudinal smooth muscle of the ileum studied with receptor knockout mice.
    British journal of pharmacology, 2005, Volume: 146, Issue:1

    Topics: Animals; Calcium Channel Blockers; Carbachol; Cholinergic Agonists; Diamines; Female; Ileum; In Vitro Techniques; Male; Mice; Mice, Knockout; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nicardipine; Pertussis Toxin; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3

2005
Regulation of IPSP theta rhythm by muscarinic receptors and endocannabinoids in hippocampus.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Action Potentials; Amino Acids; Animals; Cannabinoid Receptor Modulators; Carbachol; Cholinergic Agonists; Endocannabinoids; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Neural Inhibition; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spectrum Analysis; Synapses; Theta Rhythm; Time Factors; Xanthenes

2005
Neural regulation of slow-wave frequency in the murine gastric antrum.
    American journal of physiology. Gastrointestinal and liver physiology, 2006, Volume: 290, Issue:3

    Topics: Acetylcholine; Androstenes; Animals; Atropine; Benzamides; Benzimidazoles; Carbachol; Electric Stimulation; Electrophysiology; Enteric Nervous System; Female; Gastric Emptying; Male; Mice; Mice, Inbred BALB C; Mice, Inbred Strains; Motor Neurons; Muscle Contraction; Myenteric Plexus; Neostigmine; Piperidines; Pyloric Antrum; Tetrodotoxin

2006
Muscarinic M1 and M3 receptor binding alterations in pancreas during pancreatic regeneration of young rats.
    Endocrine research, 2005, Volume: 31, Issue:4

    Topics: Animals; Atropine; Carbachol; Cholinergic Agonists; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Muscarinic Antagonists; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Regeneration

2005
Characterization of muscarinic receptor-mediated cationic currents in longitudinal smooth muscle cells of mouse small intestine.
    Journal of pharmacological sciences, 2006, Volume: 100, Issue:3

    Topics: Animals; Carbachol; Cations; Cholinergic Agonists; Diamines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Guinea Pigs; In Vitro Techniques; Intestine, Small; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Mice; Muscarinic Antagonists; Myocytes, Smooth Muscle; Pertussis Toxin; Piperidines; Pyrrolidinones; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Type C Phospholipases

2006
Muscarinic regulation of neonatal rat bladder spontaneous contractions.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2006, Volume: 291, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Calcium Channel Agonists; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Diamines; Electric Stimulation; Muscle Contraction; Muscle Hypertonia; Muscle, Smooth; Parasympatholytics; Peptides; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder

2006
M1 muscarinic receptors contribute to, whereas M4 receptors inhibit, dopamine D1 receptor-induced [3H]-cyclic AMP accumulation in rat striatal slices.
    Neurochemical research, 2006, Volume: 31, Issue:4

    Topics: Alkaloids; Animals; Benzazepines; Carbachol; Cholinergic Agonists; Corpus Striatum; Cyclic AMP; Dopamine Agonists; Furans; Male; Muscarinic Antagonists; N-Methylscopolamine; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Protein Kinase C; Radioligand Assay; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Receptors, Dopamine D1

2006
Agonist and antagonist sensitivity of non-selective cation channel currents evoked by muscarinic receptor stimulation in bovine ciliary muscle cells.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:3

    Topics: Animals; Atropine; Barium; Carbachol; Cattle; Cells, Cultured; Ciliary Body; Dose-Response Relationship, Drug; Membrane Potentials; Microscopy, Fluorescence; Muscarinic Agonists; Muscarinic Antagonists; Muscle Cells; Patch-Clamp Techniques; Piperidines; Pirenzepine; Receptor, Muscarinic M3; TRPC Cation Channels

2006
Regulation of bladder muscarinic receptor subtypes by experimental pathologies.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:3

    Topics: Age Factors; Animals; Benzofurans; Carbachol; Denervation; Disease Models, Animal; Electric Stimulation; Female; Gene Expression Regulation; Humans; Hypertrophy; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pyrrolidines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; RNA, Messenger; Urinary Bladder; Urinary Bladder Neck Obstruction; Urinary Bladder, Neurogenic

2006
Propiverine and metabolites: differences in binding to muscarinic receptors and in functional models of detrusor contraction.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 374, Issue:2

    Topics: Animals; Benzilates; Binding, Competitive; Calcium; Carbachol; Cell Line; Cells, Cultured; CHO Cells; Cholinergic Antagonists; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Electric Stimulation; Epithelial Cells; Humans; Molecular Structure; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Potassium Chloride; Receptors, Muscarinic; Urinary Bladder

2006
Functional roles of muscarinic M2 and M3 receptors in mouse stomach motility: studies with muscarinic receptor knockout mice.
    European journal of pharmacology, 2007, Jan-12, Volume: 554, Issue:2-3

    Topics: Animals; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Female; Gastric Emptying; Gastric Fundus; Genotype; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Physostigmine; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Stomach

2007
Human idiopathic and neurogenic overactive bladders and the role of M2 muscarinic receptors in contraction.
    European urology, 2007, Volume: 52, Issue:2

    Topics: Adult; Aged; Benzofurans; Carbachol; Diamines; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Pyrrolidines; Receptors, Muscarinic; Urinary Bladder; Urinary Bladder, Neurogenic; Urinary Bladder, Overactive

2007
Muscarinic receptor subtypes mediating positive and negative inotropy in the developing chick ventricle.
    Journal of pharmacological sciences, 2007, Volume: 103, Issue:1

    Topics: Action Potentials; Alkaloids; Animals; Carbachol; Chick Embryo; Dose-Response Relationship, Drug; Furans; Heart Ventricles; Myocardial Contraction; Naphthalenes; Piperidines; Pirenzepine; Receptors, Muscarinic

2007
TRPV1 is involved in stretch-evoked contractile changes in the rat autonomous bladder model: a study with piperine, a new TRPV1 agonist.
    Neurourology and urodynamics, 2007, Volume: 26, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Indicators and Reagents; Mechanotransduction, Cellular; Muscle Contraction; Piperidines; Polyunsaturated Alkamides; Pressure; Rats; Rats, Wistar; Ruthenium Red; Stress, Mechanical; TRPV Cation Channels; Urinary Bladder

2007
Cardiovascular effects of carbachol microinjected into the bed nucleus of the stria terminalis of the rat brain.
    Brain research, 2007, Apr-27, Volume: 1143

    Topics: Animals; Arginine Vasopressin; Atropine; Blood Pressure; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Heart Rate; Male; Microinjections; Muscarinic Antagonists; Nicotinic Antagonists; Pentolinium Tartrate; Piperidines; Rats; Rats, Wistar; Septal Nuclei

2007
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection

2007
Endothelin, PAF and thromboxane A2 in allergic pulmonary hyperreactivity in mice.
    Prostaglandins, leukotrienes, and essential fatty acids, 2007, Volume: 76, Issue:5

    Topics: Animals; Antihypertensive Agents; Bronchial Hyperreactivity; Carbachol; Endothelin B Receptor Antagonists; Endothelin-1; Endothelins; Male; Mice; Mice, Inbred BALB C; Oligopeptides; Ovalbumin; Peptide Fragments; Phospholipid Ethers; Piperidines; Platelet Activating Factor; Platelet Aggregation Inhibitors; Prostaglandin Endoperoxides, Synthetic; Receptor, Endothelin B; Thromboxane A2

2007
Cholinergic activation of phasic activity in the isolated bladder: possible evidence for M3- and M2-dependent components of a motor/sensory system.
    BJU international, 2007, Volume: 100, Issue:3

    Topics: Animals; Arecoline; Benzofurans; Carbachol; Cholinergic Agonists; Female; Guinea Pigs; Muscarinic Agonists; Piperidines; Pyrrolidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder; Urination

2007
Lack of depolarization-induced suppression of inhibition (DSI) in layer 2/3 interneurons that receive cannabinoid-sensitive inhibitory inputs.
    Journal of neurophysiology, 2007, Volume: 98, Issue:5

    Topics: Action Potentials; Animals; Animals, Newborn; Benzoxazines; Calcium; Cannabinoids; Carbachol; Cerebral Cortex; Cholinergic Agonists; Dose-Response Relationship, Radiation; Electric Stimulation; In Vitro Techniques; Interneurons; Mice; Morpholines; Naphthalenes; Neural Inhibition; Piperidines; Pyramidal Cells; Pyrazoles; Rimonabant

2007
Changes in muscarinic receptors in the toad urothelial cell line TBM-54 following acrolein treatment.
    Clinical and experimental pharmacology & physiology, 2008, Volume: 35, Issue:2

    Topics: Acrolein; Animals; Blotting, Western; Bufo marinus; Carbachol; Cell Line; Diamines; Dose-Response Relationship, Drug; Extracellular Fluid; Hydrogen-Ion Concentration; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Receptors, Muscarinic; Urinary Bladder; Urothelium

2008
Endothelin receptor blockers protect against ischemia/reperfusion impairment of gastrointestinal motility in rats.
    Pharmacological research, 2008, Volume: 57, Issue:6

    Topics: Anesthesia, Inhalation; Anesthetics, Inhalation; Animals; Carbachol; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin Receptor Antagonists; Endothelin-1; Ether; Evans Blue; Gastrointestinal Motility; Male; Muscarinic Agonists; Oligopeptides; Peptides, Cyclic; Piperidines; Pyridines; Rats; Rats, Wistar; Reperfusion Injury; Surgical Procedures, Operative; Tetrazoles

2008
Refractoriness of the sheep superior vena cava myocardial sleeve.
    Experimental biology and medicine (Maywood, N.J.), 2008, Volume: 233, Issue:11

    Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Diamines; Electrophysiologic Techniques, Cardiac; In Vitro Techniques; Microelectrodes; Muscarinic Antagonists; Myocardium; Myocytes, Cardiac; Piperidines; Refractometry; Sheep; Tropicamide; Vasodilator Agents; Vena Cava, Superior

2008
Activation of cholinergic receptors blocks non-adrenergic non-cholinergic contractions in the rat urinary bladder.
    Brain research bulletin, 2008, Dec-16, Volume: 77, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Antineoplastic Agents; Atropine; Calcium Channel Agonists; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Electric Stimulation; Female; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Physostigmine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Suramin; Urinary Bladder

2008
Islet neogenesis-associated protein signaling in neonatal pancreatic rat islets: involvement of the cholinergic pathway.
    The Journal of endocrinology, 2008, Volume: 199, Issue:2

    Topics: Animals; Animals, Newborn; Antigens, Neoplasm; Biomarkers, Tumor; Carbachol; Carrier Proteins; Immunoblotting; In Vitro Techniques; Insulin; Islets of Langerhans; Lectins, C-Type; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Pancreatitis-Associated Proteins; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Piperidines; Proto-Oncogene Proteins c-akt; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Ribosomal Protein S6 Kinases, 70-kDa; Signal Transduction; TOR Serine-Threonine Kinases

2008
ETB2 receptor subtype stimulation relaxes the iris sphincter muscle.
    Physiological research, 2009, Volume: 58, Issue:6

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Endothelin-1; Endothelins; Enzyme Inhibitors; In Vitro Techniques; Indomethacin; Iris; Male; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oligopeptides; Peptide Fragments; Peptides; Piperidines; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Rabbits; Receptor, Endothelin A; Receptor, Endothelin B; Viper Venoms

2009
Inhibitory effect of quercetin on rat trachea contractility in vitro.
    The Journal of pharmacy and pharmacology, 2009, Volume: 61, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antioxidants; Benzamides; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phentolamine; Piperidines; Propranolol; Quercetin; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Trachea

2009
In vitro and in vivo pharmacological characterization of PF-01354082, a novel partial agonist selective for the 5-HT(4) receptor.
    European journal of pharmacology, 2009, May-01, Volume: 609, Issue:1-3

    Topics: Administration, Oral; Animals; Benzimidazoles; Carbachol; Cell Line; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Esophagus; Gastrointestinal Motility; Humans; Indoles; Kidney; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Sensitivity and Specificity; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Receptor Agonists; Time Factors

2009
Muscarinic receptor-mediated nitric oxide release in a K562 erythroleukaemia cell line.
    Autonomic & autacoid pharmacology, 2009, Volume: 29, Issue:3

    Topics: Arginine; Carbachol; Chromatography, High Pressure Liquid; Citrulline; Dose-Response Relationship, Drug; Humans; K562 Cells; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nitric Oxide; Nitric Oxide Synthase; Piperidines; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; RNA; Tropicamide

2009
Carbachol regulates pacemaker activities in cultured interstitial cells of Cajal from the mouse small intestine.
    Molecules and cells, 2009, May-31, Volume: 27, Issue:5

    Topics: Animals; Anti-Inflammatory Agents; Biological Clocks; Calcium; Calcium-Transporting ATPases; Carbachol; Cation Transport Proteins; Cells, Cultured; Diamines; Flufenamic Acid; Guanosine Diphosphate; Intestine, Small; Membrane Potentials; Mice; Mice, Inbred BALB C; Neuromuscular Depolarizing Agents; Patch-Clamp Techniques; Piperidines; Plant Roots; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Thapsia; Thapsigargin; Thionucleotides

2009
Muscarinic receptor type 1 (M1) stimulation, probably through KCNQ/Kv7 channel closure, increases spontaneous GABA release at the dendrodendritic synapse in the mouse accessory olfactory bulb.
    Brain research, 2010, Jun-21, Volume: 1339

    Topics: Alkaloids; Animals; Anticonvulsants; Calcium; Calcium Channel Blockers; Calcium Channels, R-Type; Carbachol; Carbamates; Cholinergic Agonists; Dendrites; Diclofenac; Excitatory Amino Acid Antagonists; Furans; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; KCNQ Potassium Channels; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Naphthalenes; Nimodipine; Olfactory Bulb; Patch-Clamp Techniques; Phenylenediamines; Piperidines; Pirenzepine; Potassium Channel Blockers; Receptor, Muscarinic M1; Receptors, Glutamate; Synapses

2010
Muscarinic receptors induce LTD of NMDAR EPSCs via a mechanism involving hippocalcin, AP2 and PSD-95.
    Nature neuroscience, 2010, Volume: 13, Issue:10

    Topics: Acetylcholine; Adaptor Protein Complex 2; Animals; Biophysics; Calcium; Carbachol; Cholinergic Agonists; Disks Large Homolog 4 Protein; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agents; Excitatory Postsynaptic Potentials; Hippocalcin; Hippocampus; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Long-Term Synaptic Depression; Male; Membrane Proteins; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Protein Transport; Quinolones; Rats; Receptors, Muscarinic; Receptors, N-Methyl-D-Aspartate; RNA Interference; Synapses; Two-Hybrid System Techniques

2010
Chemical stimulation of the lateral hypothalamus induces conditioned place preference in rats: Involvement of OX1 and CB1 receptors in the ventral tegmental area.
    Behavioural brain research, 2011, Feb-02, Volume: 217, Issue:1

    Topics: Animals; Benzoxazoles; Carbachol; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Male; Naphthyridines; Neural Pathways; Orexin Receptors; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor Cross-Talk; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Urea; Ventral Tegmental Area

2011
Selective M3 muscarinic receptor antagonist inhibits small-cell lung carcinoma growth in a mouse orthotopic xenograft model.
    Journal of pharmacological sciences, 2011, Volume: 116, Issue:1

    Topics: Animals; Antineoplastic Agents; Calcium Signaling; Carbachol; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dipeptides; Dose-Response Relationship, Drug; Female; Humans; Lung Neoplasms; Mice; Mice, Inbred ICR; Mice, SCID; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Receptor, Muscarinic M3; Small Cell Lung Carcinoma; Tumor Burden; Xenograft Model Antitumor Assays

2011
Plasticity of non-adrenergic non-cholinergic bladder contractions in rats after chronic spinal cord injury.
    Brain research bulletin, 2011, Aug-10, Volume: 86, Issue:1-2

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Carbachol; Cholinergic Agonists; Female; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neuronal Plasticity; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Spinal Cord Injuries; Urinary Bladder

2011
Muscarinic activation of Ca2+-activated Cl- current in interstitial cells of Cajal.
    The Journal of physiology, 2011, Sep-15, Volume: 589, Issue:Pt 18

    Topics: Animals; Atropine; Carbachol; Chloride Channels; Green Fluorescent Proteins; Interstitial Cells of Cajal; Intestine, Small; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Models, Animal; Muscarinic Agonists; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Receptors, Muscarinic

2011
Expression of muscarinic receptors by human macrophages.
    The European respiratory journal, 2012, Volume: 39, Issue:3

    Topics: Carbachol; Cells, Cultured; Choline O-Acetyltransferase; Humans; Interleukin-6; Interleukin-8; Leukocytes, Mononuclear; Leukotriene B4; Macrophages; Membrane Transport Proteins; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pulmonary Disease, Chronic Obstructive; Receptors, Muscarinic; RNA; Smoking; Vesicular Acetylcholine Transport Proteins

2012
Effects of cannabinoid agonists on sheep sphincter of oddi in vitro.
    Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.], 2011, Volume: 11, Issue:4

    Topics: Analgesics; Animals; Arachidonic Acids; Benzoxazines; Camphanes; Cannabinoid Receptor Agonists; Cannabinoids; Carbachol; Cyclic GMP; Male; Morpholines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; NG-Nitroarginine Methyl Ester; Organ Culture Techniques; Piperidines; Pyrazoles; Rimonabant; Sheep; Sphincter of Oddi

2011
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
    Urology, 2011, Volume: 78, Issue:6

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium

2011
Pharmacological characterization of GSK1004723, a novel, long-acting antagonist at histamine H(1) and H(3) receptors.
    British journal of pharmacology, 2011, Volume: 164, Issue:6

    Topics: Allergens; Animals; Benzazepines; Binding, Competitive; Bronchi; Bronchial Provocation Tests; Bronchoconstriction; Carbachol; Cell Line; CHO Cells; Cricetinae; Cricetulus; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H3 Antagonists; Humans; In Vitro Techniques; Niacinamide; Ovalbumin; Phthalazines; Piperidines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H3; Recombinant Proteins; Rhinitis, Allergic, Perennial; Transfection

2011
Influence of influenza A infection on capsaicin-induced responses in murine airways.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:2

    Topics: Animals; Biphenyl Compounds; Bronchoalveolar Lavage Fluid; Capsaicin; Carbachol; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Indomethacin; Inflammation; Influenza A virus; Isoproterenol; Leukocytes; Male; Mice; Mice, Inbred BALB C; Models, Biological; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Orthomyxoviridae Infections; Piperidines; Prostaglandin Antagonists; Respiratory Mucosa; Specific Pathogen-Free Organisms; Substance P; Trachea; TRPV Cation Channels; Xanthones

2012
Functional role of muscarinic receptor subtypes in calcium sensitization and their contribution to rho-kinase and protein kinase C pathways in contraction of human detrusor smooth muscle.
    Urology, 2012, Volume: 79, Issue:5

    Topics: Amides; Calcium; Carbachol; Enzyme Inhibitors; Humans; In Vitro Techniques; Indoles; Maleimides; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxants, Central; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Protein Kinase C; Pyridines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; rho-Associated Kinases; Signal Transduction; Urinary Bladder

2012
Muscarinic receptor subtypes involved in urothelium-derived relaxatory effects in the inflamed rat urinary bladder.
    Autonomic neuroscience : basic & clinical, 2012, Sep-25, Volume: 170, Issue:1-2

    Topics: Animals; Carbachol; Cyclophosphamide; Cystitis; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Synthase; Nitroarginine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder; Urothelium

2012
Signaling cross-talk between cannabinoid and muscarinic systems actives Rho-kinase and increases the contractile responses of the bovine ciliary muscle.
    European journal of pharmacology, 2013, Feb-28, Volume: 702, Issue:1-3

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Carbachol; Cattle; Cholinergic Agonists; Ciliary Body; Endocannabinoids; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Polyunsaturated Alkamides; Protein Kinase C; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Muscarinic M3; rho-Associated Kinases

2013
A role for M(2) and M(3) muscarinic receptors in the contraction of rat and human small airways.
    European journal of pharmacology, 2013, Feb-28, Volume: 702, Issue:1-3

    Topics: Animals; Carbachol; Cholinergic Agonists; Humans; In Vitro Techniques; Lung; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Scopolamine Derivatives; Tiotropium Bromide

2013
Loss of TRPM2 function protects against irradiation-induced salivary gland dysfunction.
    Nature communications, 2013, Volume: 4

    Topics: Acinar Cells; Animals; Benzamides; Calcium; Carbachol; Cell Line; Cell Survival; Enzyme Inhibitors; Humans; Hydrogen Peroxide; Ion Channel Gating; Mice; Mice, Inbred C57BL; Piperidines; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Radiation Injuries; Saliva; Salivary Glands; Salivation; Submandibular Gland; TRPM Cation Channels; X-Rays

2013
Different muscarinic receptor subtypes modulate proliferation of primary human detrusor smooth muscle cells via Akt/PI3K and map kinases.
    Pharmacological research, 2013, Volume: 74

    Topics: Aged; Atropine; Benzofurans; Carbachol; Cell Proliferation; Cells, Cultured; Cholinergic Agonists; Gene Expression; Humans; Male; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Myocytes, Smooth Muscle; Phosphatidylinositol 3-Kinases; Piperidines; Pirenzepine; Proto-Oncogene Proteins c-akt; Pyrrolidines; Receptors, Muscarinic; RNA, Messenger; Urinary Bladder

2013
Activation of muscarinic M3 receptors inhibits large-conductance voltage- and Ca2+-activated K+ channels in rat urinary bladder smooth muscle cells.
    American journal of physiology. Cell physiology, 2013, Jul-15, Volume: 305, Issue:2

    Topics: Amphotericin B; Animals; Carbachol; Cholinergic Agonists; Diamines; Evoked Potentials; Gene Expression Regulation; Large-Conductance Calcium-Activated Potassium Channels; Male; Membrane Potentials; Muscarinic Antagonists; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3; Urinary Bladder

2013
The inhibitory effects of antimuscarinic autoantibodies in the sera of primary Sjogren syndrome patients on the gastrointestinal motility.
    Molecular immunology, 2013, Volume: 56, Issue:4

    Topics: Animals; Autoantibodies; Carbachol; Cholinergic Agonists; Colon; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; Humans; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Sjogren's Syndrome; Stomach

2013
Bladder function in a cannabinoid receptor type 1 knockout mouse.
    BJU international, 2014, Volume: 113, Issue:1

    Topics: Animals; Cannabinoid Receptor Antagonists; Carbachol; Female; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Urinary Bladder; Urination; Urodynamics

2014
Expression and function of muscarinic subtype receptors in bladder interstitial cells of cajal in rats.
    Urology journal, 2014, Jul-08, Volume: 11, Issue:3

    Topics: Action Potentials; Animals; Atropine; Calcium Channels; Carbachol; Cholinergic Agonists; Diamines; Interstitial Cells of Cajal; Male; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder

2014
Excitatory drive from the Subthalamic nucleus attenuates GABAergic transmission in the Substantia Nigra pars compacta via endocannabinoids.
    European journal of pharmacology, 2015, Nov-15, Volume: 767

    Topics: Animals; Carbachol; Chromones; Dopaminergic Neurons; Electric Stimulation; Endocannabinoids; Excitatory Postsynaptic Potentials; GABAergic Neurons; Inhibitory Postsynaptic Potentials; Pars Compacta; Pars Reticulata; Piperidines; Pyrazoles; Rats; Rimonabant; Subthalamic Nucleus; Synaptic Transmission

2015
Functional interaction between OX2 and CB1 receptors in the ventral tegmental area and the nucleus accumbens in response to place preference induced by chemical stimulation of the lateral hypothalamus.
    Pharmacology, biochemistry, and behavior, 2015, Volume: 139, Issue:Pt A

    Topics: Animals; Carbachol; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Synergism; Hypothalamic Area, Lateral; Isoquinolines; Male; Microinjections; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Piperidines; Pyrazoles; Pyridines; Rats; Receptor, Cannabinoid, CB1; Reward; Stimulation, Chemical; Ventral Tegmental Area

2015
Functional interaction between orexin-1 and CB1 receptors in the periaqueductal gray matter during antinociception induced by chemical stimulation of the lateral hypothalamus in rats.
    European journal of pain (London, England), 2016, Volume: 20, Issue:10

    Topics: Animals; Benzoxazoles; Carbachol; Disease Models, Animal; Hypothalamic Area, Lateral; Male; Microinjections; Naphthyridines; Orexin Receptors; Orexins; Pain; Pain Measurement; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Stimulation, Chemical; Urea

2016
Role of orexin-2 and CB1 receptors within the periaqueductal gray matter in lateral hypothalamic-induced antinociception in rats.
    Behavioural pharmacology, 2017, Volume: 28, Issue:1

    Topics: Animals; Carbachol; Disease Models, Animal; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Isoquinolines; Male; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pain; Periaqueductal Gray; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2017
Intrinsic membrane properties and cholinergic modulation of mouse basal forebrain glutamatergic neurons in vitro.
    Neuroscience, 2017, 06-03, Volume: 352

    Topics: Action Potentials; Animals; Animals, Genetically Modified; Animals, Newborn; Basal Forebrain; Benzamides; Calcium Channel Blockers; Carbachol; Cholinergic Agents; Electric Stimulation; Glutamates; Luminescent Proteins; Lysine; Mice; Neurons; Patch-Clamp Techniques; Piperidines; Pyrimidines; Red Fluorescent Protein; Sodium Channel Blockers; Tetrodotoxin; Vesicular Glutamate Transport Protein 2

2017
Relaxant effect of ghrelin on guinea pig isolated tracheal smooth muscle: role of epithelial NO and PGE
    Pflugers Archiv : European journal of physiology, 2018, Volume: 470, Issue:6

    Topics: Animals; Carbachol; Dinoprostone; Ghrelin; Guinea Pigs; Histamine; Indomethacin; Male; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Piperidines; Quinazolinones; Respiratory Mucosa; Trachea

2018
Novel BQCA- and TBPB-Derived M
    ChemMedChem, 2019, 07-17, Volume: 14, Issue:14

    Topics: Benzimidazoles; Carbachol; Drug Partial Agonism; HEK293 Cells; Humans; Ligands; Molecular Docking Simulation; Muscarinic Agonists; Piperidines; Quinolines; Receptor, Muscarinic M1

2019
Central muscarinic receptor subtypes (M1 and M3) involved in carbacol-induced hypophagia in neonatal broiler chicken.
    The International journal of neuroscience, 2020, Volume: 130, Issue:2

    Topics: Animals; Animals, Newborn; Behavior, Animal; Carbachol; Chickens; Disease Models, Animal; Eating; Injections, Intraventricular; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M3

2020