Page last updated: 2024-08-17

carbachol and pinacidil

carbachol has been researched along with pinacidil in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.35)18.7374
1990's13 (56.52)18.2507
2000's7 (30.43)29.6817
2010's2 (8.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Karim, OM; Mostwin, JL; Seki, N1
Arch, JR; Bond, J; Buckle, DR; Shaw, DJ; Taylor, JF; Taylor, SG; Ward, JS1
Bang, L; Nielsen-Kudsk, JE1
Lundbeck, F; Sjögren, C1
Charette, L; Garcia, ML; Jones, TR; Kaczorowski, GJ1
Satoh, E; Taira, N; Yanagisawa, T1
MacLeod, KM; Ray, A1
Andersson, KE; Andersson, PO; Fovaeus, M; Malmgren, A; Sjögren, C1
Cohen, ML; Schoepp, DD; Secrest, RJ1
Ishimura, Y; Katoh, I; Masuda, Y; Oka, M; Yoshizumi, M1
Barth, HL; Hempelmann, RG; Mehdorn, HM; Pradel, RH; Ziegler, A1
Belardinelli, L; Song, Y; Srinivas, M1
Horan, P; Leggett, R; Levin, RM; Whitbeck, C1
Hu, GY; Xu, DY; Yuan, YM1
Dick, JM; Lefebvre, RA; Timmermans, JP; Van Geldre, LA1
Dick, JM; Lefebvre, RA; Libert, C; Van Molle, W1
Bolego, C; Cignarella, A; Pinna, C; Puglisi, L; Sanvito, P1
Aishima, M; Ito, Y; Naito, S; Nakano, T; Seki, N; Sueishi, K; Teramoto, N; Tomoda, T; Yonemitsu, Y; Yunoki, T1
Badawi, JK; Bross, S; Ding, A1
Gok, S; Izanli-Paksoy, A; Vural, K1
Adachi, T; Fujisawa, S; Hongoh, M; Ohba, T; Ono, K; Shimbo, T1

Other Studies

23 other study(ies) available for carbachol and pinacidil

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Effect of pinacidil on the membrane electrical activity of guinea pig detrusor muscle.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Glyburide; Guanidines; Guinea Pigs; Membrane Potentials; Muscle, Smooth; Nifedipine; Pinacidil; Urinary Bladder; Vasodilator Agents

1992
The inhibitory effects of cromakalim and its active enantiomer BRL 38227 against various agonists in guinea pig and human airways: comparison with pinacidil and verapamil.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:2

    Topics: Animals; Benzopyrans; Bronchi; Bronchial Spasm; Bronchodilator Agents; Carbachol; Cromakalim; Drug Interactions; Female; Guanidines; Guinea Pigs; Humans; Male; Muscle Contraction; Pinacidil; Potassium Channels; Pyrroles; Stereoisomerism; Trachea; Vasodilator Agents; Verapamil

1992
Smooth muscle relaxation and inhibition of responses to pinacidil and cromakalim induced by phentolamine in guinea-pig isolated trachea.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dinoprost; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Pinacidil; Pyrroles; SRS-A; Trachea

1992
A pharmacological in vitro study of the mouse urinary bladder at the time of acute change in bladder reservoir function after irradiation.
    The Journal of urology, 1992, Volume: 148, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; Electric Stimulation; Guanidines; In Vitro Techniques; Indomethacin; Mice; Muscle Contraction; Muscle, Smooth; Pinacidil; Scopolamine; Urinary Bladder

1992
Selective inhibition of relaxation of guinea-pig trachea by charybdotoxin, a potent Ca(++)-activated K+ channel inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2

    Topics: Aminophylline; Animals; Benzopyrans; Calcium; Carbachol; Charybdotoxin; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Guanidines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nitroprusside; Pinacidil; Potassium Channels; Pyrroles; Scorpion Venoms; Serotonin; Trachea

1990
Specific antagonism by glibenclamide of negative inotropic effects of potassium channel openers in canine atrial muscle.
    Japanese journal of pharmacology, 1990, Volume: 54, Issue:2

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dogs; Female; Glyburide; Guanidines; Heart Atria; Male; Myocardial Contraction; Niacinamide; Nicorandil; Nifedipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1990
Adrenergic-cholinergic interactions in left atria: a study using K+ channel agonists, antagonist and pertussis toxin.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 4-Aminopyridine; Animals; Benzopyrans; Carbachol; Cromakalim; Cyclic AMP; Dogs; Female; Guanidines; Heart; Isoproterenol; Male; Myocardial Contraction; Parasympathetic Nervous System; Pertussis Toxin; Phenylephrine; Pinacidil; Potassium Channels; Pyrroles; Rabbits; Sympathetic Nervous System; Virulence Factors, Bordetella

1990
Effects of cromakalim (BRL 34915) and pinacidil on normal and hypertrophied rat detrusor in vitro.
    The Journal of urology, 1990, Volume: 143, Issue:4

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Electric Stimulation; Female; Guanidines; Hypertrophy; In Vitro Techniques; Muscle Contraction; Pinacidil; Potassium; Pyrroles; Rats; Rats, Inbred Strains; Urinary Bladder; Vasodilator Agents

1990
Comparison of contractions to serotonin, carbamylcholine and prostaglandin F2 alpha in rat stomach fundus.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Animals; Carbachol; Diltiazem; Dinoprost; Gastric Fundus; Guanidines; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Nitrendipine; Nitroglycerin; Phosphatidylinositols; Pinacidil; Rats; Rats, Inbred Strains; Serotonin

1989
Effects of the potassium channel openers cromakalim and pinacidil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
    Biochemical pharmacology, 1994, May-18, Volume: 47, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Barium; Benzopyrans; Bradykinin; Calcimycin; Calcium; Carbachol; Catecholamines; Cattle; Cells, Cultured; Cromakalim; Guanidines; Histamine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes

1994
Effects of potassium channel openers in isolated human cerebral arteries.
    Neurosurgery, 1995, Volume: 37, Issue:6

    Topics: Benzopyrans; Calcium Channel Blockers; Carbachol; Cerebral Arteries; Cromakalim; Culture Techniques; Dose-Response Relationship, Drug; Endothelium, Vascular; Guanidines; Humans; Iloprost; Nifedipine; Nimodipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1995
Nonspecific inhibition of adenosine-activated K+ current by glibenclamide in guinea pig atrial myocytes.
    The American journal of physiology, 1996, Volume: 271, Issue:6 Pt 2

    Topics: Action Potentials; Adenosine; Animals; Atrial Function; Carbachol; Electric Conductivity; Glyburide; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Myocardium; Pinacidil; Potassium; Reaction Time

1996
Correlation of EGTA and calcium-blocking agents on the response of the bladder to in vitro ischemia.
    Pharmacology, 1999, Volume: 58, Issue:3

    Topics: Animals; Calcium Channel Blockers; Carbachol; Chelating Agents; Diltiazem; Egtazic Acid; Electric Stimulation; In Vitro Techniques; Ischemia; Male; Muscle Contraction; Muscle, Smooth; Pinacidil; Potassium Channels; Rabbits; Reperfusion; Urinary Bladder

1999
Pinacidil suppression on 5-HT3 receptor-mediated contraction of guinea pig ileum in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1998, Volume: 19, Issue:1

    Topics: Animals; Carbachol; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Pinacidil; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1998
Investigation of the interaction between nitric oxide and vasoactive intestinal polypeptide in the guinea-pig gastric fundus.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Adenine; Adrenergic beta-Agonists; Animals; Atrial Natriuretic Factor; Carbachol; Colforsin; Cyclic AMP; Dexamethasone; Electric Stimulation; Enzyme Inhibitors; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Isoproterenol; Molsidomine; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitroarginine; Nitroprusside; Pinacidil; Tetrodotoxin; Thionucleotides; Vasoactive Intestinal Peptide

2000
Antisense knockdown of inducible nitric oxide synthase inhibits the relaxant effect of VIP in isolated smooth muscle cells of the mouse gastric fundus.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Amidines; Animals; Arginine; Benzylamines; Carbachol; Cell Size; DNA, Antisense; Enzyme Inhibitors; Female; Fluorescein-5-isothiocyanate; Gastric Fundus; Glyburide; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscle Relaxation; Muscle, Smooth; Nitrates; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitrites; Nitroarginine; Pinacidil; Tumor Necrosis Factor-alpha; Vasoactive Intestinal Peptide; Vasodilator Agents

2001
Effect of the ATP-sensitive potassium channel opener ZM226600 on cystometric parameters in rats with ligature-intact, partial urethral obstruction.
    European journal of pharmacology, 2005, May-23, Volume: 516, Issue:1

    Topics: Adenosine Triphosphate; Amides; Animals; Benzophenones; Blood Pressure; Carbachol; Dose-Response Relationship, Drug; Female; Heart Rate; In Vitro Techniques; Muscle Contraction; Pinacidil; Potassium Channels; Rats; Rats, Sprague-Dawley; Time Factors; Urethral Obstruction; Urinary Bladder

2005
Actions of ZD0947, a novel ATP-sensitive K+ channel opener, on membrane currents in human detrusor myocytes.
    British journal of pharmacology, 2006, Volume: 149, Issue:5

    Topics: ATP-Binding Cassette Transporters; Carbachol; Diazoxide; Dihydropyridines; Dose-Response Relationship, Drug; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Gliclazide; Glyburide; Humans; Immunochemistry; In Vitro Techniques; Membrane Potentials; Muscle Relaxation; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors; Urinary Bladder

2006
Inhibitory effects of different ATP-sensitive potassium channel openers on electrically generated and carbachol-induced contractions of porcine and human detrusor muscle.
    Fundamental & clinical pharmacology, 2008, Volume: 22, Issue:1

    Topics: Aged; Amides; Animals; Benzophenones; Carbachol; Cromakalim; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Minoxidil; Muscle Contraction; Muscle, Smooth; Pinacidil; Potassium Channels; Swine; Urinary Bladder

2008
Contribution of RhoA kinase and protein kinase C to weak relaxant effect of pinacidil on carbachol-induced contractions in sensitized guinea-pig trachealis.
    Archives of pharmacal research, 2009, Volume: 32, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine; Animals; Benzophenanthridines; Bronchodilator Agents; Carbachol; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; KATP Channels; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ovalbumin; Pinacidil; Protein Kinase C; rhoA GTP-Binding Protein; Trachea

2009
In vitro effect of nicorandil on the carbachol-induced contraction of the lower esophageal sphincter of the rat.
    Journal of pharmacological sciences, 2016, Volume: 131, Issue:4

    Topics: Animals; Carbachol; Diazoxide; Dose-Response Relationship, Drug; Esophageal Sphincter, Lower; Glyburide; In Vitro Techniques; KATP Channels; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nicorandil; Oxadiazoles; Peptides; Pinacidil; Potassium; Quinoxalines; Rats

2016