Page last updated: 2024-08-17

carbachol and oxotremorine

carbachol has been researched along with oxotremorine in 278 studies

Research

Studies (278)

TimeframeStudies, this research(%)All Research%
pre-1990159 (57.19)18.7374
1990's91 (32.73)18.2507
2000's23 (8.27)29.6817
2010's4 (1.44)24.3611
2020's1 (0.36)2.80

Authors

AuthorsStudies
Chapman, JM; Kosh, JW; Sowell, JW; Tang, Y; Valli, MJ1
Hacksell, U; Nilsson, BM; Vargas, HM1
Chapman, JM; Kosh, JW; Sowell, JW; Tang, Y; Usher, LA; Valli, MJ; Vaughan, CM1
Amstutz, R; Boelsterli, J; Bolliger, G; Floersheim, P; Gammenthaler, H; Gmelin, G; Shapiro, G; Supavilai, P; Walkinshaw, M1
Baumgold, J; Bradbury, BJ; Jacobson, KA; Kammula, U; Paek, R; Zimmet, J1
Kramss, RH; Mangano, RM; Rusinko, A; Trybulski, EJ1
Jenden, DJ; Ringdahl, B; Roch, M1
Ringdahl, B4
Andrews, PR; Craik, DJ; Martin, JL1
Brann, MR; Bräuner-Osborne, H; Ebert, B; Falch, E; Krogsgaard-Larsen, P1
Kramss, RH; Mangano, RM; Trybulski, EJ; Zhang, J1
Abuh, YF; Dunbar, PG; Edgar, MA; El-Assadi, AA; Fang, Z; Huzl, JJ; Liu, Y; Messer, WS; Nagy, PI; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Roknich, S; Sbeih, S; Zhang, H1
Bromidge, SM; Brown, F; Cassidy, F; Clark, MS; Dabbs, S; Hadley, MS; Hawkins, J; Loudon, JM; Naylor, CB; Orlek, BS; Riley, GJ1
Daly, JW; Gupta, TH; Padgett, WL; Pei, XF1
Chen, D; Shan, L; Wang, H; Yang, R; Yun, L; Zhao, R1
Dei, S; Marconi, C; Pedretti, A; Romanelli, MN; Scapecchi, S; Vistoli, G1
Lamble, AP; Lamble, JW1
Gray, DB; Lane, MA; Sastre, A1
Birdsall, NJ; Burgen, AS; Strange, PG1
Makara, GB; Stark, E1
Maayani, S; Sokolovsky, M; Treister, G1
Bianchetti, A; Biraschi, LM; Guarneri, L; Riva, M1
Brezenoff, HE; Buccafusco, JJ1
Aktories, K; Jakobs, KH; Schultz, G1
Bhargava, VK; McKean, CM; Salamy, A2
Hadházy, P; Szerb, JC1
Dudar, JD; Hadházy, P; Szerb, JC1
Ehlert, FJ; Kokka, N1
Staib, AH; Westermann, KH1
Johnson, KG1
Funk, KF; Oelszner, W; Schwarzenfeld, IV; Staib, AH; Westermann, KH1
Lindenboim, L; Pinkas-Kramarski, R; Sokolovsky, M; Stein, R1
Morrison, KJ; Vanhoutte, PM1
Hato, F; Kinoshita, Y; Tominaga, K; Tominaga, M; Yamada, M1
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E1
Joseph, JA; Roth, GS; Yamagami, K1
Mochizuki, D; Shinoda, Y; Sugiyama, S1
Constanti, A; Das, B; Libri, V1
Gies, JP; Haddad, EB1
Dunant, Y; Sierro, CD; Vitus, J1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Althaus, JS; Buxser, SE; Decker, DE; Von Voigtlander, PF1
Gies, JP; Haddad, EB; Landry, Y1
Daniel, EE; Janssen, LJ1
Chilvers, ER; Nahorski, SR; Offer, GJ1
Lovenberg, TW; Mailman, RB; Nichols, DE; Roth, RH1
Aksoy, S; Gibson, VA; McKinney, M; Miller, JH; Nickelson, L1
Fujimoto, S; Matsuda, T1
Ebadi, M; Govitrapong, P; Pujito, PP1
Richards, MH1
Joseph, JA; Kowatch, MA; Maki, T; Roth, GS1
Schimerlik, MI; Tota, MR1
de Pont, JJ; Rodrigues de Miranda, JF; van Ginneken, CA; van Zwam, AJ; Willems, PH1
Costi, A; Marchi, M; Raiteri, M; Volpe, G1
Bagetta, G; Constanti, A1
Ikeda, T; Kojima, T; Shirasu, Y; Takahashi, H; Tsuda, S; Yoshida, M1
Bartolami, S; Guiramand, J; Lenoir, M; Mayat, E; Pujol, R; Récasens, M; Rumigny, JF1
Baum, BJ; He, XJ; Turner, RJ; Wu, XZ1
Ehlert, FJ; Rathbun, BE1
Bartus, RT; Fisher, SK1
Nezu, E; Yoneyama, T; Yoshimura, K1
Cohen-Armon, M; Sokolovsky, M1
Pappano, AJ; Tajima, T; Tsuji, Y; Yuen, J1
Baumgold, J; Fishman, PH1
Fertel, R; Hadjiconstantinou, M; Neff, NH; Qu, ZX1
Arrang, JM; Gulat-Marnay, C; Lafitte, A; Schwartz, JC1
Henis, YI; Moscona-Amir, E; Sokolovsky, M1
Luthin, GR; Manning, DR; Matesic, DF; Wolfe, BB1
Lang, U; Walland, A1
Matsumoto, K; Pappano, AJ1
Marchi, M; Raiteri, M1
Drews, U; Oettling, G; Schmidt, H2
Gil, DW; Wolfe, BB1
Imaizumi, T; Misaki, N; Mizushima, A; Osugi, T; Tatebayashi, Y; Uchida, S; Yoshida, H; Zhou, XM1
Flynn, DD; Palermo, N; Suarez, A1
Good, DM; Small, RC1
Boselli, C; Kenakin, T1
Boddeke, HW; Doods, HN; Rondas, AA; Thörig, L; van Haeringen, NJ; van Zwieten, PA1
Borasio, PG; Capuzzo, A; Fabbri, E1
Ashkenazi, A; Capon, DJ; Peralta, EG; Peterson, GL; Ramachandran, J; Schimerlik, MI; Winslow, JW1
Baraban, JM; Heller, WA; Snyder, SH; Worley, PF1
Chen, WY; Wince, LC1
Pinkas-Kramarski, R; Sokolovsky, M; Stein, R1
Alger, BE; McCarren, M; Pitler, TA1
Ek, B; Nahorski, S1
Critchett, DJ; Joseph, JA; Lippa, AS1
Costa, E; Eva, C2
Baux, G; Fossier, P; Poulain, B; Tauc, L1
Dalton, TK; Hunt, WA; Joseph, JA1
Anderson, W; Dickinson, KE; Hirschowitz, BI; Matsumoto, H; Pruitt, RE; Uemura, N1
Baraban, JM; Huganir, RL; Stratton, KR; Worley, PF1
Amstutz, R; Jenden, DJ; Karlén, B; Ringdahl, B; Roch, M1
Cantin, M; Garcia, R; Gutkowska, J; Lachance, D; Thibault, G1
Limas, C; Limas, CJ1
Heisler, S1
Gjörstrup, P; Hjalmarson, A; Jacobsson, B; Ransnäs, L; Sjögren, CG1
Brown, JH; Harden, TK; Heng, MM1
Chuang, DM; Xu, J1
DeGeorge, JJ; Lapetina, EG; McCarthy, KD; Morell, P1
Channell, SL; Iversen, SD; Lalies, MD; Salamone, JD1
Alger, BE; Baraban, JM; McCarren, M; Snyder, SH; Worley, PF1
Crain, B; Crain, SM; Makman, MH2
Aronstam, RS; Narayanan, TK1
Bertrand, C; Gies, JP; Landry, Y1
Anthony, BL; Aronstam, RS; Dennison, RL; Narayanan, TK1
Lüllmann, H; Mohr, K; Pfeffer, J1
Galron, R; Sokolovsky, M1
Erwin, VG; Jones, BC; Korte, A1
Amstutz, R; Closse, A; Ringdahl, B1
Camus, J; Christophe, J; De Neef, P; Fourmy, D; Pradayrol, L; Robberecht, P; Scemama, JL; Tastenoy, M; Vaysse, N; Waelbroeck, M1
Band, LC; Bitran, D; Clemens, LG; Holmes, GM; Hull, EM; Pehek, EA; Warner, RK1
Fujii, AM; Homcy, CJ; Lee, DL; Longabaugh, JP; Schwarz, KR; Vatner, DE; Vatner, SF1
Abdel-Latif, AA; Honkanen, RE1
Crain, SM; Makman, MH1
Gies, JP; Landry, Y1
Sokolovsky, M; van Koppen, CJ1
Dutar, P; Nicoll, RA1
Adem, A; Nordberg, A; Sabbagh, M1
Constanti, A; Williams, SH2
Hynie, S1
Stojić, D; Terzić, M1
Bonaventure, N; Jardon, B; Rudolf, G; Wioland, N1
Collins, SM; Crankshaw, DJ1
Markowicz, ME; Ringdahl, B1
Christophe, J; Gillard, M; Waelbroeck, M1
Bartfai, T; Hedlund, B1
Collins, AC; Marks, MJ; Romm, E1
Green, RD; Hosey, MM; Kwatra, MM; Leung, E; Maan, AC; McMahon, KK; Ptasienski, J1
Pittaluga, A; Raiteri, M1
Clemens, LG; Richmond, G1
Anthony, BL; Aronstam, RS1
Horváth, E; Spencer, DG; Traber, J; Van Rooijen, LA1
Chien, JL; Warren, JR1
Baker, SP; Posner, P1
Johnston, CI; Leung, E; Woodcock, EA1
Barenholz, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M; Yechiel, E1
Bering, B; Müller, WE1
Cubeddu, LX; James, MK1
Luthin, GR; Wolfe, BB1
Henry, PJ; Lulich, KM; Paterson, JW1
Flynn, DD; Potter, LT1
Barker, DL; Mpitsos, GJ; Murray, TF; Siebenaller, JF1
Kloog, Y; Sokolovsky, M1
Konno, F; Takayanagi, I1
Gurwitz, D; Sokolovsky, M1
Ehlert, FJ1
Eriksson, H; Häggblad, J; Heilbronn, E1
Higuchi, H; Kagiya, T; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H; Zhou, XM1
Bianchi, C; Tomasi, L1
Snyder, SH; Yamamura, HI1
Blanton, RJ; Komiskey, HL; Rudy, TA1
Bhargava, AK; Bhargava, KP; Tangri, KK1
György, L; Phan, DV; Szelényi, Z; Varga, B1
Johnson, KG; Smith, CA1
Fozard, JR; Muscholl, E1
Birdsall, NJ; Burgen, A; Hulme, EC1
Abeln, W; Bienhold, H; Flohr, H1
Kanje, M; Lazarewicz, JW1
Peterfreund, RA; Vale, WW1
Kerkerian, L; Nieoullon, A1
Kuwata, K; Nagai, K; Okamoto, E; Toyosaka, A; Uchida, S; Ueki, S; Yoshida, H1
Jenden, DJ; Ringdahl, B1
Brown, BL; Dobson, PR; Wojcikiewicz, RJ1
Cortés, R; Palacios, JM; Pazos, A1
Barhanin, J; Cavey, D; Fosset, M; Lazdunski, M; Renaud, JF1
Blandina, P; Fantozzi, R; Mannaioni, PF; Masini, E1
Brown, JH; Rietow, M1
Harden, TK; Meeker, RB1
Brown, JH; Brown, SL1
Dahlbom, R; Ehlert, FJ; Jenden, DJ; Resul, B; Ringdahl, B1
Bergh, CH; Hjalmarson, A; Jacobsson, B; Ransnäs, L; Waldenström, A1
Barr, PJ; Clemens, LG; Dohanich, GP; Witcher, JA1
Hauser, G; Parks, JM1
Asselin, J; Christophe, J; de Neef, P; Robberecht, P; Waelbroeck, M1
Birdsall, NJ; Burgen, AS; Hulme, EC; Wong, EH1
Cheong, DK; Misgeld, U; Weiler, MH1
Halvorsen, SW; Holttum, J; Hunter, DD; Nathanson, NM1
North, RA; Tokimasa, T1
Klein, WL; Siman, RG1
Leung, E; Mitchelson, F1
Dial, E; Ecknauer, R; Johnson, LR; Rosenfeld, GC; Thompson, WJ1
Coppi, G; Leone, L; Lumachi, B; Rossini, L; Valsecchi, B1
Kwok, YH; Mitchelson, F1
Gainer, MW; Meyer, MR; Nathanson, NM1
Westermann, KH1
Bhargava, VK; Pushpavati, CP1
Bartfai, T; Hedlund, B; Järv, J1
Klein, WL; Shifrin, GS1
Ellis, J; Hoss, W1
Miller, DA; Pendleton, RG; Ridley, PT1
Ehlert, FJ; Fairhurst, AS; Kokka, N1
Bauer, MB; Gebhart, GF; Murphy, S1
Birmingham, AT; Harriss, DR; Hill, SJ; Marsh, KA1
Ogren, SO; Pramanik, A1
Gabelt, BT; Kaufman, PL; Poyer, JF1
Dorsey, WC; Ford, BD; Townsel, JG1
Ferrari-DiLeo, G; Flynn, DD; Mash, DC1
Denisova, NA; Erat, S; Joseph, JA; Kelly, JF; Mason, RP; Roth, GS1
Honda, K; Kamiya, H; Takano, Y1
Haass, M; Haunstetter, A; Krüger, C; Kübler, W; Yi, X1
Hadjiconstantinou, M; Hubble, JP; Neff, NH; Wemlinger, TA1
Nahorski, SR; Safrany, ST1
Martin, DL; Waniewski, RA1
Dalton, TK; Harris, A; Joseph, JA; Kandasamy, S; Rabin, BM; Villalobos-Molina, R1
Bowen, WD; de Costa, BR; Kirschner, BN; Rice, KC; Tolentino, PJ; Varghese, P1
Clement, JG1
Belton, CM; Fatherazi, S; Herrington, J; Izutsu, KT; Oda, D; Wellner, RB1
Allaoua, H; Alonso, R; Boksa, P; Chaudieu, I; Quirion, R1
Castoldi, AF; Costa, LG; Tang, C1
Antonsson, BM; Ek, B1
Habecker, BA; Nathanson, NM; Wang, H1
Eglen, RM; Sharif, NA; To, ZP1
Consolo, S; Garcia Ruiz, AJ; La Porta, C; Ladinsky, H; Zambelli, M1
Tonnaer, JA; van Huizen, F1
Contrera, JG; Holopainen, I; Mcleskey, SW; Wojcik, WJ; Xu, J1
Abood, LG; Hashmi, M; Lerner-Marmarosh, N; Saraswati, M1
Jones, SB; King, LB1
Barg, J; Fisher, A; Heldman, E; Kushnir, M; Levy, R; Pittel, Z; Vogel, Z; Zimlichman, R1
Cheng, E; Cline, RT; Fraser, CM; Geoghagen, NS; Lee, NH1
De Neef, P; Domenach, V; Vandermeers, A; Vandermeers-Piret, MC; Waelbroeck, M1
Drijfhout, WJ; Grol, CJ; Westerink, BH1
Mills, J; Reiner, PB1
Christopoulos, A; Lanzafame, A; Mitchelson, F1
Spindler, KD; Spindler-Barth, M; Wegener, S1
Ebihara, T; Saffen, D1
Murayama, T; Nomura, Y; Yamada, T1
Matthews, MR; Zaidi, ZF1
Schimerlik, MI; Sheehan, DM; Vogel, WK1
Edwardson, JM; Koenig, JA; Szekeres, PG1
Gebauer, M; Versen, B1
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M1
Beaucher, J; Harnois, C; Psarropoulou, C1
Koizumi, S; Moriyama, Y; Ogura, A; Yamada, H; Yamaguchi, A1
Andrade, R; Haj-Dahmane, S1
Colecraft, HM; Egamino, JP; Sharma, VK; Sheu, SS1
Jaen, JC; Mirzadegan, T; Moreland, D; Schwarz, RD; Spencer, CJ; Tecle, H; Thomas, AJ1
Brown, AM; Hunter, AJ; Middlemiss, DN; Watson, JM1
Akbulut, H; Akici, A; Karaalp, A; Oktay, S; Ulusoy, NB1
Jiang, B; Pappano, AJ; Shen, JB1
Ladner, CJ; Lee, JM1
Gebauer, M; Schipp, R; Versen, B1
Arellano, RO; Garay, E; Miledi, R1
Azpiazu, I; Cruzblanca, H; Gautam, N; Li, P; Linder, M; Zhuo, M1
Akk, G; Auerbach, A1
Malomough, A; Naumenko, N; Nikolsky, E; Urazaev, A; Vyskocil, F1
Hamilton, C; Höglund, AU; Lindblom, L1
Shapovalova, KB1
Fowler, CE; Gunn-Moore, F; Henderson, G; Samways, DS; Yeo, A1
Bymaster, FP; Carter, PA; Cohen, ML; Falcone, JF; Felder, CC; Gomeza, J; Shannon, HE; Stengel, PW; Wess, J; Zhang, L1
Choppin, A; Eglen, RM1
Park, PS; Sum, CS; Wells, JW1
de Araujo, EG; dos Santos, AA; Medina, SV; Sholl-Franco, A1
Goodhead, LH; Mitchell, SN; Moss, S; Sharott, A1
Kawamura, H; Kobayashi, M; Puro, DG; Sakagami, K; Wu, DM1
Hosoi, T; Nomura, J; Nomura, Y; Okuma, Y1
Borowitz, JL; Gunasekar, PG; Isom, GE; Li, L; Prabhakaran, K; Zhang, L1
Bukharaeva, EA; Magazanik, LG; Nikolsky, EE; Samigullin, D; Vyskocil, F1
Dong, SJ; Liu, H; Liu, KL; Ruan, JX; Wang, LY; Wang, Y; Zheng, JQ; Zhong, BH1
Fernández-López, A; Mostany, R; Paniagua, MA; Pérez, CC; Pilar-Cuéllar, F1
Liu, LL; Ruan, JX; Wang, LY; Wang, Y; Zheng, JQ; Zhong, BH1
Gamper, N; Hilgemann, DW; Li, Y; Shapiro, MS1
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S1
Kebig, A; Kostenis, E; Mohr, K; Mohr-Andrä, M1
Hancock, J; Hobson, SA; Kelly, E; Marrion, NV; Mason, A; Oldfield, S; Randall, AD; Wynick, D1
Christopoulos, A; Kenakin, T; Muniz-Medina, V; Novick, S; Watson, C1
Bao, HF; Eaton, AF; Eaton, DC; Helms, MN; Jain, L; Ramosevac, S; Self, J; Takemura, Y1
Carlin, J; Jacklin, DL; Mitchnick, KA; O'Hara, M; Stiver, ML; Vicic, N; Winters, BD1
Dolejší, E; Doležal, V; El-Fakahany, EE; Jakubík, J; Randáková, A; Rudajev, V; Zimčík, P1
Gillet, C; Kuenzel, T; Kurth, S1

Reviews

3 review(s) available for carbachol and oxotremorine

ArticleYear
Pharmacology and second messenger interactions of cloned muscarinic receptors.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Animals; Atropine; Carbachol; Cell Line; Humans; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic; Recombinant Proteins; Second Messenger Systems; Transfection

1991
Cardioselective muscarinic antagonists.
    Federation proceedings, 1987, Volume: 46, Issue:8

    Topics: Animals; Carbachol; Cardiotonic Agents; Carrier Proteins; Cyclic AMP; Cyclic AMP Receptor Protein; Dose-Response Relationship, Drug; Heart; N-Methylscopolamine; Oxotremorine; Phorbol Esters; Pirenzepine; Receptors, Adrenergic; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives

1987
The therapeutic use of cholinergic drugs acting on the vegetative nervous system. I - Direct, indirect and mixed agonists.
    Il Farmaco; edizione scientifica, 1981, Volume: 36, Issue:10

    Topics: Animals; Arecoline; Bethanechol Compounds; Carbachol; Chemical Phenomena; Chemistry; Dimethylphenylpiperazinium Iodide; Ganglia; Kinetics; Lobeline; Neuroeffector Junction; Nicotine; Oxotremorine; Parasympathomimetics; Pilocarpine; Stereoisomerism

1981

Other Studies

275 other study(ies) available for carbachol and oxotremorine

ArticleYear
Synthesis and cholinergic properties of N-aryl-2-[[[5-[(dimethylamino)methyl]-2-furanyl]methyl]thio]ethylamino analogs of ranitidine.
    Journal of medicinal chemistry, 1992, Aug-21, Volume: 35, Issue:17

    Topics: Acetylcholine; Animals; Brain; Butyrylcholinesterase; Cholinesterase Inhibitors; Drug Synergism; Erythrocytes; Humans; Ileum; Male; Mice; Muscle Contraction; Ranitidine; Rats; Receptors, Muscarinic

1992
Urea and 2-imidazolidone derivatives of the muscarinic agents oxotremorine and N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide.
    Journal of medicinal chemistry, 1992, Aug-21, Volume: 35, Issue:17

    Topics: Animals; Cerebral Cortex; Guinea Pigs; Ileum; Imidazoles; Molecular Structure; Muscarinic Antagonists; Muscle Contraction; Oxotremorine; Parasympathomimetics; Pyrrolidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Urea

1992
Synthesis and cholinergic properties of bis[[(dimethylamino)methyl]furanyl] analogues of ranitidine.
    Journal of medicinal chemistry, 1992, Mar-20, Volume: 35, Issue:6

    Topics: Animals; Cholinesterase Inhibitors; Furans; Humans; Male; Mice; Parasympathomimetics; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Structure-Activity Relationship

1992
Muscarinic activity of the thiolactone, lactam, lactol, and thiolactol analogues of pilocarpine and a hypothetical model for the binding of agonists to the m1 receptor.
    Journal of medicinal chemistry, 1992, Volume: 35, Issue:1

    Topics: Animals; Binding, Competitive; Crystallography; Guinea Pigs; Lactams; Male; Mice; Models, Biological; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Sulfhydryl Compounds

1992
Muscarinic receptor binding and activation of second messengers by substituted N-methyl-N-[4-(1-azacycloalkyl)-2-butynyl]acetamides.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:3

    Topics: Acetamides; Alkynes; Animals; Binding, Competitive; Cell Line; Cell Membrane; Cerebral Cortex; Chemical Phenomena; Chemistry; Female; Fibroblasts; Heterocyclic Compounds; Male; Molecular Structure; Parasympathomimetics; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Second Messenger Systems; Transfection

1991
Chemical and biochemical studies of 2-propynylpyrrolidine derivatives. Restricted-rotation analogues of N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide (BM-5).
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Chemical Phenomena; Chemistry; Dioxolanes; Guanylyl Imidodiphosphate; Magnetic Resonance Spectroscopy; Male; Molecular Conformation; Molecular Structure; Myocardium; Parasympathomimetics; Pirenzepine; Pyrrolidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship

1990
Tertiary 3- and 4-haloalkylamine analogues of oxotremorine as prodrugs of potent muscarinic agonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:1

    Topics: Analgesia; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Indicators and Reagents; Kinetics; Magnetic Resonance Spectroscopy; Mice; Muscle Contraction; Oxotremorine; Parasympathomimetics; Pharmaceutical Preparations; Prodrugs; Pyrrolidinones; Saliva; Structure-Activity Relationship; Tremor

1988
5-Methyl-2-pyrrolidone analogues of oxotremorine as selective muscarinic agonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Analgesia; Animals; Body Temperature; Carbachol; Guinea Pigs; In Vitro Techniques; Mice; Muscle, Smooth; Oxotremorine; Parasympathomimetics; Pyrrolidinones; Salivation; Urinary Bladder

1988
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors.
    Journal of medicinal chemistry, 1995, Jun-09, Volume: 38, Issue:12

    Topics: 3T3 Cells; Animals; Arecoline; Cerebral Cortex; Heterocyclic Compounds; Humans; In Vitro Techniques; Mice; Muscarinic Agonists; Protein Binding; Rats; Receptors, Muscarinic; Recombinant Proteins

1995
The synthesis and biochemical pharmacology of enantiomerically pure methylated oxotremorine derivatives.
    Journal of medicinal chemistry, 1993, Nov-12, Volume: 36, Issue:23

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Guanylyl Imidodiphosphate; Male; Methylation; N-Methylscopolamine; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Scopolamine Derivatives; Stereoisomerism

1993
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
    Journal of medicinal chemistry, 1997, Apr-11, Volume: 40, Issue:8

    Topics: Animals; Arecoline; Brain; Carbachol; Cell Line; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship

1997
Design of [R-(Z)]-(+)-alpha-(methoxyimino)-1-azabicyclo[2.2.2]octane-3-acetonitri le (SB 202026), a functionally selective azabicyclic muscarinic M1 agonist incorporating the N-methoxy imidoyl nitrile group as a novel ester bioisostere.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Alzheimer Disease; Animals; Binding Sites; Blood Pressure; Brain; CHO Cells; Cricetinae; Electroencephalography; Heart Rate; Humans; Imines; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Structure; Muscarinic Agonists; Protein Binding; Quinuclidines; Rats; Rats, Inbred Strains; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Proteins; Stereoisomerism; Tremor

1997
6beta-Acyloxy(nor)tropanes: affinities for antagonist/agonist binding sites on transfected and native muscarinic receptors.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding Sites; Cerebral Cortex; CHO Cells; Cricetinae; Humans; In Vitro Techniques; Muscarinic Agonists; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Receptors, Muscarinic; Transfection; Tropanes

2000
Discovering selective agonists of endothelial target for acetylcholine (ETA) via diversity-guided pharmacophore simplification and simulation.
    Bioorganic & medicinal chemistry letters, 2004, Jun-21, Volume: 14, Issue:12

    Topics: Acetylcholine; Animals; Aorta; Endothelium, Vascular; Guinea Pigs; Muscarinic Agonists; Rabbits; Rats; Vasodilation

2004
Docking analyses on human muscarinic receptors: unveiling the subtypes peculiarities in agonists binding.
    Bioorganic & medicinal chemistry, 2008, Mar-15, Volume: 16, Issue:6

    Topics: Binding Sites; Computer Simulation; Humans; Ligands; Muscarinic Agonists; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M5; Receptors, Muscarinic

2008
The effect of miotics on the intraocular pressure of conscious owl monkeys.
    Investigative ophthalmology, 1976, Volume: 15, Issue:10

    Topics: Anesthesia, Local; Animals; Aotus trivirgatus; Carbachol; Dose-Response Relationship, Drug; Haplorhini; Intraocular Pressure; Male; Miotics; Oxotremorine; Parasympathomimetics; Pilocarpine; Quinuclidines; Spiro Compounds; Succinimides; Tonometry, Ocular

1976
Muscarinic cholinergic binding sites in the developing avian heart.
    Developmental biology, 1977, Volume: 55, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Benzyl Compounds; Carbachol; Chick Embryo; Heart; Methacholine Compounds; Microsomes; Myocardium; Nicotine; Oxotremorine; Physostigmine; Quaternary Ammonium Compounds; Quinuclidines; Receptors, Cholinergic; Scopolamine; Snake Venoms; Tubocurarine

1977
Occupancy of muscarinic acetylcholine receptors stimulates a guanylate cyclase in neuroblastoma cells.
    Biochemical Society transactions, 1977, Volume: 5, Issue:1

    Topics: Acetylcholine; Atropine; Carbachol; Cell Line; Cell Membrane; Enzyme Activation; Guanylate Cyclase; Kinetics; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1977
The effects of cholinomimetic drugs and atropine on ACTH release.
    Neuroendocrinology, 1976, Volume: 21, Issue:1

    Topics: Acetylcholine; Adrenocorticotropic Hormone; Animals; Atropine; Carbachol; Corticosterone; Drug Implants; Electric Stimulation; Female; Fluoresceins; Hypothalamo-Hypophyseal System; Hypothalamus; Hypothalamus, Anterior; Injections, Intraventricular; Male; Median Eminence; Oxotremorine; Parasympathomimetics; Rats; Stress, Physiological

1976
Drugs affecting the cholinergic system in the intact mammalian eye. I. Evaluation of the miotic activity of acetylcholine-like drugs in the mouse eye.
    Investigative ophthalmology, 1975, Volume: 14, Issue:3

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Guinea Pigs; Hydrogen-Ion Concentration; Miotics; Oxotremorine; Phencyclidine; Pupil; Quinuclidines

1975
Pharmacological properties of n1-piperonyl-n4-3,7,11-trimethyl-2,6,10-dodecatrienyl-piperazine, a new non-anticholinergic gastric antisecretory agent.
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:4

    Topics: Animals; Carbachol; Central Nervous System; Depression, Chemical; Dogs; Feeding Behavior; Female; Gastric Juice; Gastric Mucosa; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Hemodynamics; Histamine H1 Antagonists; Hydrogen-Ion Concentration; Male; Methacholine Compounds; Mice; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pentagastrin; Peptic Ulcer; Piperazines; Polyenes; Rabbits; Rats; Respiration

1975
Pharmacological study of a cholinergic mechanism within the rat posterior hypothalamic nucleus which mediates a hypertensive response.
    Brain research, 1979, Apr-13, Volume: 165, Issue:2

    Topics: Acetylcholine; Adrenalectomy; Animals; Atropine; Blood Pressure; Carbachol; Cholinergic Fibers; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Heart Rate; Hemicholinium 3; Hypophysectomy; Hypothalamus; Hypothalamus, Posterior; Male; Mecamylamine; Oxotremorine; Phentolamine; Premedication; Rats

1979
GTP-dependent inhibition of cardiac adenylate cyclase by muscarinic cholinergic agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 310, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Guanine Nucleotides; Guanosine Triphosphate; In Vitro Techniques; Myocardium; Oxotremorine; Parasympathetic Nervous System; Parasympathomimetics; Rabbits; Time Factors

1979
Effect of cholinergic drugs on the brainstem auditory evoked responses (far-field) in rats.
    Neuroscience, 1978, Volume: 3, Issue:9

    Topics: Animals; Auditory Pathways; Auditory Perception; Brain Stem; Carbachol; Cholinergic Fibers; Dose-Response Relationship, Drug; Evoked Potentials; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Rats

1978
Effects of cholinergic drugs on auditory evoked responses (CER) of rat cortex.
    Neuropharmacology, 1978, Volume: 17, Issue:12

    Topics: Acoustic Stimulation; Animals; Carbachol; Cerebral Cortex; Drug Interactions; Evoked Potentials; Hearing; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Rats; Scopolamine

1978
The effect of cholinergic drugs on [3H]acetylcholine release from slices of rat hippocampus, striatum and cortex.
    Brain research, 1977, Mar-11, Volume: 123, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cerebral Cortex; Corpus Striatum; Drug Interactions; Electric Stimulation; Hippocampus; In Vitro Techniques; Oxotremorine; Parasympathomimetics; Physostigmine; Potassium; Rats; Time Factors

1977
Release of [3H]acetylcholine from rat hippocampal slices: effect of septal lesion and of graded concentrations of muscarnic agonists and antagonists.
    Brain research, 1977, Jun-10, Volume: 128, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Carbachol; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Mecamylamine; Oxotremorine; Pilocarpine; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Septum Pellucidum

1977
Decrease in (3H)-quinuclidinyl bezilate binding to the muscarinic cholinergic receptor in the longitudinal muscle of the rat ileum following chronic administration of diisopropylfuorophosphate.
    Proceedings of the Western Pharmacology Society, 1977, Volume: 20

    Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cholinesterases; Depression, Chemical; Ileum; In Vitro Techniques; Isoflurophate; Male; Muscle, Smooth; Myocardium; Oxotremorine; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Time Factors

1977
[Nigrostiatally induced motor reactions in the rat. II. Cholinergic effect on rotational behavior and posture asymetry].
    Acta biologica et medica Germanica, 1976, Volume: 35, Issue:6

    Topics: Apomorphine; Carbachol; Caudate Nucleus; Hydroxydopamines; Movement Disorders; Oxotremorine; Posture; Receptors, Cholinergic; Receptors, Dopamine

1976
Thermoregulatory changes induced by cholinomimetic substances introduced into the cerebral ventricles of sheep.
    British journal of pharmacology, 1975, Volume: 53, Issue:4

    Topics: Animals; Atropine; Body Temperature Regulation; Carbachol; Castration; Cerebral Ventricles; Cold Temperature; Hot Temperature; Injections; Male; Nicotine; Oxotremorine; Parasympathomimetics; Pempidine; Physostigmine; Sheep; Shivering; Skin Temperature; Stimulation, Chemical

1975
[Cholinergic effect on the dopamine turnover in the rat corpus striatum].
    Acta biologica et medica Germanica, 1975, Volume: 34, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Carbachol; Corpus Striatum; Dopamine; Homovanillic Acid; Methyltyrosines; Oxotremorine; Rats

1975
Growth factor-like effects mediated by muscarinic receptors in PC12M1 cells.
    Journal of neurochemistry, 1992, Volume: 59, Issue:6

    Topics: Adenylyl Cyclases; Animals; Calcium; Carbachol; Cell Movement; Cyclic AMP; Cycloheximide; Dactinomycin; DNA; Enzyme Activation; Gene Expression Regulation; Growth Substances; Neurites; Oxotremorine; PC12 Cells; Phosphatidylinositols; Protein Kinase C; Rats; Receptors, Muscarinic; RNA, Messenger

1992
Characterization of muscarinic receptors that mediate contraction of guinea-pig isolated trachea to choline esters: effect of removing epithelium.
    British journal of pharmacology, 1992, Volume: 106, Issue:3

    Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Carbachol; Dose-Response Relationship, Drug; Epithelium; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Muscle Contraction; Oxotremorine; Receptors, Muscarinic; Trachea

1992
Enhancement of DNA synthesis in rat thymocytes by stimulating their muscarinic acetylcholine receptors.
    Cellular and molecular biology (Noisy-le-Grand, France), 1992, Volume: 38, Issue:8

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cells, Cultured; DNA; Hexamethonium; Hexamethonium Compounds; Isoflurophate; Kinetics; Male; Nicotine; Oxotremorine; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Nicotinic; Succinylcholine; T-Lymphocytes; Thymidine; Tritium; Tubocurarine

1992
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation

1992
Decrement of muscarinic receptor-stimulated low-KM GTPase in striatum and hippocampus from the aged rat.
    Brain research, 1992, Apr-03, Volume: 576, Issue:2

    Topics: Aging; Animals; Blotting, Western; Carbachol; Cell Membrane; Corpus Striatum; GTP Phosphohydrolases; GTP-Binding Proteins; Hippocampus; Kinetics; Macromolecular Substances; Male; Molecular Weight; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1992
[Biochemical studies of oxiracetam (CT-848) on cholinergic neurons].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1992, Volume: 99, Issue:1

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Carbachol; Cerebral Cortex; Choline O-Acetyltransferase; Hippocampus; Male; Oxotremorine; Pyrrolidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cholinergic

1992
Ganglionic nicotinic receptor agonists exhibit anti-muscarinic effects in guinea-pig olfactory cortical brain slices.
    European journal of pharmacology, 1992, Mar-03, Volume: 212, Issue:2-3

    Topics: Alkaloids; Animals; Azocines; Carbachol; Choline; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Ganglionic Stimulants; Guinea Pigs; In Vitro Techniques; Lobeline; Olfactory Bulb; Oxotremorine; Parasympatholytics; Quaternary Ammonium Compounds; Quinolizines

1992
Neuraminidase reduces the number of super-high-affinity [3H]oxotremorine-M binding sites in lung.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: Animals; Carbachol; Clostridium perfringens; Guinea Pigs; In Vitro Techniques; Kinetics; Lung; Male; Membranes; Muscle Contraction; Neuraminidase; Oxotremorine; Receptors, Muscarinic

1992
Effects of muscarinic agonists and depolarizing agents on inositol monophosphate accumulation in the rabbit vagus nerve.
    Journal of neurochemistry, 1992, Volume: 59, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Cadmium; Calcimycin; Calcium; Carbachol; Dose-Response Relationship, Drug; Hydrolysis; Inositol Phosphates; Lithium; Ouabain; Oxotremorine; Parasympathomimetics; Pirenzepine; Potassium; Rabbits; Receptors, Muscarinic; Time Factors; Vagus Nerve

1992
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Effects of dopamine agonists on dopamine secretion from PC12 cells: lack of functional autoreceptor activity.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 72, Issue:2

    Topics: Animals; Apomorphine; Carbachol; Dopamine; Dopamine Agents; Haloperidol; Oxotremorine; Phenalenes; Polycyclic Compounds; Potassium; Receptors, Dopamine; Tumor Cells, Cultured

1991
Sialic acid residues as catalysts for M2-muscarinic agonist-receptor interactions.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Carbachol; Cell Membrane; Kinetics; Male; Myocardium; Neuraminidase; Oxotremorine; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine; Sialic Acids

1990
Pre- and postjunctional muscarinic receptors in canine bronchi.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bethanechol Compounds; Bronchi; Carbachol; Dogs; Electric Stimulation; In Vitro Techniques; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Beta-adrenoceptor induced inhibition of muscarinic receptor-stimulated phosphoinositide metabolism is agonist specific in bovine tracheal smooth muscle.
    European journal of pharmacology, 1991, Jul-12, Volume: 207, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Carbachol; Cattle; Inositol Phosphates; Isoproterenol; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Propranolol; Receptors, Adrenergic, beta; Receptors, Muscarinic; Trachea

1991
D1 dopamine receptors of NS20Y neuroblastoma cells are functionally similar to rat striatal D1 receptors.
    Journal of neurochemistry, 1991, Volume: 57, Issue:5

    Topics: Benzazepines; Butaclamol; Carbachol; Cell Line; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Agents; Flupenthixol; Kinetics; Neuroblastoma; Oxotremorine; Phenanthridines; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride; Tubocurarine

1991
Interactions of agonists with M2 and M4 muscarinic receptor subtypes mediating cyclic AMP inhibition.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Cells, Cultured; CHO Cells; Corpus Striatum; Cricetinae; Cyclic AMP; Kinetics; Male; Muscarine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
M3 cholinoceptors and P2y purinoceptors mediating relaxation of arteries in spontaneously hypertensive rats at prehypertensive stages.
    European journal of pharmacology, 1991, Sep-04, Volume: 202, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Arteries; Carbachol; Cholinergic Antagonists; Endothelium, Vascular; Femoral Artery; Hypertension; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Oxotremorine; Parasympatholytics; Purinergic Antagonists; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Cholinergic; Receptors, Purinergic

1991
Inhibitory actions of muscarinic cholinergic receptor agonists on serotonin N-acetyltransferase in bovine pineal explants in culture.
    Neurochemical research, 1991, Volume: 16, Issue:8

    Topics: Animals; Arylamine N-Acetyltransferase; Carbachol; Cattle; Kinetics; Methacholine Chloride; Organ Culture Techniques; Oxotremorine; Parasympathomimetics; Pilocarpine; Pineal Gland; Receptors, Muscarinic

1991
Selective cross-activation/inhibition of second messenger systems and the reduction of age-related deficits in the muscarinic control of dopamine release from perifused rat striata.
    Brain research, 1990, Dec-24, Volume: 537, Issue:1-2

    Topics: Aging; Animals; Arachidonic Acid; Arachidonic Acids; Biotransformation; Carbachol; Corpus Striatum; Dopamine; In Vitro Techniques; Inosine Triphosphate; Male; Neomycin; Oxotremorine; Perfusion; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Second Messenger Systems; Type C Phospholipases

1990
Partial agonist effects on the interaction between the atrial muscarinic receptor and the inhibitory guanine nucleotide-binding protein in a reconstituted system.
    Molecular pharmacology, 1990, Volume: 37, Issue:6

    Topics: Animals; Carbachol; GTP Phosphohydrolases; GTP-Binding Proteins; Heart Atria; Kinetics; Oxotremorine; Phosphoric Monoester Hydrolases; Pilocarpine; Receptors, Cholinergic; Structure-Activity Relationship; Swine

1990
Binding characteristics of the muscarinic receptor subtype in rabbit pancreas.
    Journal of receptor research, 1990, Volume: 10, Issue:1-2

    Topics: Animals; Binding, Competitive; Carbachol; Kinetics; Muscarine; Oxotremorine; Pancreas; Parasympathomimetics; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Time Factors; Tritium

1990
Endogenous aspartate release in the rat hippocampus is inhibited by M2 'cardiac' muscarinic receptors.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Acetylcholine; Animals; Aspartic Acid; Calcium; Carbachol; Chromatography, High Pressure Liquid; Heart; Hippocampus; In Vitro Techniques; Male; Myocardium; Neuromuscular Depolarizing Agents; Oxotremorine; Pirenzepine; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes

1990
Muscarinic suppression of the evoked N-wave by oxotremorine-M recorded in the guinea-pig olfactory cortex slice.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cerebral Cortex; Diamines; Electric Stimulation; Electroencephalography; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Olfactory Bulb; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pirenzepine; Receptors, Muscarinic

1990
Pretreatment of rats with an organophosphorus insecticide, chlorfenvinphos, protects against subsequent challenge with the same compound.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1990, Volume: 14, Issue:3

    Topics: Acetylcholinesterase; Animals; Brain; Carbachol; Chlorfenvinphos; Cholinesterases; Dichlorvos; Erythrocytes; Insecticides; Lethal Dose 50; Male; Oxotremorine; Rats; Rats, Inbred F344

1990
A M3 muscarinic receptor coupled to inositol phosphate formation in the rat cochlea?
    Biochemical pharmacology, 1990, Jun-15, Volume: 39, Issue:12

    Topics: Animals; Carbachol; Cells, Cultured; Cochlea; Inositol; Inositol Phosphates; Lithium; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium

1990
Evidence for two modes of Ca2+ entry following muscarinic stimulation of a human salivary epithelial cell line.
    The Journal of membrane biology, 1990, Volume: 115, Issue:2

    Topics: Calcium; Calcium Channel Blockers; Carbachol; Cell Line; Epithelium; Humans; Inositol 1,4,5-Trisphosphate; Membrane Potentials; Oxotremorine; Receptors, Muscarinic; Salivary Glands

1990
Signaling through the muscarinic receptor-adenylate cyclase system of the heart is buffered against GTP over a range of concentrations.
    Molecular pharmacology, 1990, Volume: 38, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Guanosine Triphosphate; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1990
Regional differences in the coupling of muscarinic receptors to inositol phospholipid hydrolysis in guinea pig brain.
    Journal of neurochemistry, 1985, Volume: 45, Issue:4

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Brain; Carbachol; Corpus Striatum; Guinea Pigs; Hydrolysis; Oxotremorine; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Time Factors; Tissue Distribution

1985
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
    The Japanese journal of physiology, 1985, Volume: 35, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains

1985
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
    The Journal of biological chemistry, 1986, Sep-25, Volume: 261, Issue:27

    Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1986
Positive inotropic effects of acetylcholine and BAY K 8644 in embryonic chick ventricle.
    The American journal of physiology, 1987, Volume: 252, Issue:4 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Action Potentials; Animals; Calcium; Carbachol; Chick Embryo; Cyclic AMP; Heart; Isoproterenol; Myocardial Contraction; Oxotremorine; Propranolol

1987
Muscarinic receptor-mediated increase in cAMP levels in SK-N-SH human neuroblastoma cells.
    Biochemical and biophysical research communications, 1988, Aug-15, Volume: 154, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Humans; Kinetics; Neuroblastoma; Oxotremorine; Pertussis Toxin; Receptors, Muscarinic; Virulence Factors, Bordetella

1988
Pharmacological characterization of muscarinic receptors mediating inhibition of adenylate cyclase activity in the rat retina.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Arecoline; Aziridines; Carbachol; Choline; Colforsin; Cyclic AMP; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Retina

1988
Regulation of histamine release and synthesis in the brain by muscarinic receptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:1

    Topics: Animals; Brain; Carbachol; Histamine Release; Male; Oxotremorine; Pirenzepine; Potassium; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1989
Aging of rat heart myocytes disrupts muscarinic receptor coupling that leads to inhibition of cAMP accumulation and alters the pathway of muscarinic-stimulated phosphoinositide hydrolysis.
    Biochemistry, 1989, Aug-22, Volume: 28, Issue:17

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Binding, Competitive; Carbachol; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Heart; Isoproterenol; Kinetics; Myocardium; Norepinephrine; Oxotremorine; Phosphatidylinositols; Rats; Receptors, Muscarinic; Time Factors

1989
Pharmacological and biochemical characterization of complexes of muscarinic acetylcholine receptor and guanine nucleotide-binding protein.
    The Journal of biological chemistry, 1989, Dec-25, Volume: 264, Issue:36

    Topics: Animals; Antibodies; Antigen-Antibody Complex; Atropine; Blotting, Western; Carbachol; Cell Membrane; Chromatography, Affinity; Electrophoresis, Polyacrylamide Gel; GTP-Binding Proteins; Kinetics; Macromolecular Substances; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Solubility

1989
Alinidine reverses the descending staircase of isolated rat atria by an antimuscarinic action.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:4

    Topics: Animals; Anti-Arrhythmia Agents; Atropine; Carbachol; Clonidine; Female; Guinea Pigs; Heart; In Vitro Techniques; Ipratropium; Isometric Contraction; Male; Oxotremorine; Papillary Muscles; Parasympatholytics; Rats; Rats, Inbred Strains

1989
Sodium-dependent membrane current induced by carbachol in single guinea-pig ventricular myocytes.
    The Journal of physiology, 1989, Volume: 415

    Topics: Acetylcholine; Action Potentials; Animals; Barium; Cadmium; Carbachol; Cesium; Guinea Pigs; Heart; Heart Ventricles; In Vitro Techniques; Isoproterenol; Membrane Potentials; Ouabain; Oxotremorine; Ryanodine; Sodium; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin

1989
Interaction acetylcholine-glutamate in rat hippocampus: involvement of two subtypes of M-2 muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes

1989
An embryonic Ca++ mobilizing muscarinic system in the chick embryo heart.
    Journal of developmental physiology, 1989, Volume: 12, Issue:2

    Topics: Animals; Benzofurans; Bethanechol; Bethanechol Compounds; Calcium; Carbachol; Chick Embryo; Chlortetracycline; Female; Fura-2; Heart; Heart Rate, Fetal; In Vitro Techniques; Methacholine Chloride; Methacholine Compounds; Oxotremorine; Parasympathomimetics; Pilocarpine; Pregnancy; Receptors, Muscarinic

1989
Pirenzepine distinguishes between muscarinic receptor-mediated phosphoinositide breakdown and inhibition of adenylate cyclase.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Atropine; Benzodiazepinones; Brain; Carbachol; In Vitro Techniques; Inositol; Inositol Phosphates; Male; Myocardium; Oxotremorine; Parotid Gland; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1985
The H-L subgroup of guinea-pig cardiac M2 receptors (M2 beta) regulates inositol phosphate formation.
    European journal of pharmacology, 1989, Sep-22, Volume: 168, Issue:3

    Topics: Acetylcholine; Adenylate Cyclase Toxin; Animals; Carbachol; Guinea Pigs; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Male; Myocardium; Oxotremorine; Pertussis Toxin; Pilocarpine; Receptors, Muscarinic; Virulence Factors, Bordetella

1989
Agonist binding to M1 muscarinic receptors is sensitive to guanine nucleotides.
    European journal of pharmacology, 1989, Oct-17, Volume: 172, Issue:4-5

    Topics: Animals; Carbachol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Indicators and Reagents; Kinetics; Male; Methacholine Compounds; Oxotremorine; Pilocarpine; Pirenzepine; Rabbits; Receptors, Muscarinic; Second Messenger Systems

1989
Muscarinic agonists and guinea-pig perfused tracheal tubes: effects of epithelial removal and route of administration. Smooth Muscle Research Group.
    British journal of pharmacology, 1989, Volume: 98 Suppl

    Topics: Animals; Carbachol; Epithelium; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Oxotremorine; Parasympathomimetics; Trachea

1989
Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Allosteric Regulation; Animals; Atropine; Binding Sites; Carbachol; Dose-Response Relationship, Drug; Gallamine Triethiodide; In Vitro Techniques; Male; Muscarine; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine; Trachea

1989
Cholinergic receptors in the extraocular rectus muscle of the rabbit.
    Ophthalmic research, 1989, Volume: 21, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Dimethylphenylpiperazinium Iodide; Female; Hexamethonium Compounds; Male; Muscle Contraction; Neuromuscular Blocking Agents; Oculomotor Muscles; Oxotremorine; Rabbits; Receptors, Cholinergic

1989
Presynaptic muscarinic receptors in guinea pig superior cervical ganglion.
    Neuroscience letters, 1989, Sep-25, Volume: 104, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Ganglia, Sympathetic; Guinea Pigs; Oxotremorine; Pirenzepine; Receptors, Muscarinic; Synapses

1989
An M2 muscarinic receptor subtype coupled to both adenylyl cyclase and phosphoinositide turnover.
    Science (New York, N.Y.), 1987, Oct-30, Volume: 238, Issue:4827

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Carbachol; Cell Line; Cricetinae; Cyclic AMP; Gene Expression Regulation; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Receptors, Muscarinic; Recombinant Proteins; Thionucleotides; Virulence Factors, Bordetella

1987
Lithium blocks a phosphoinositide-mediated cholinergic response in hippocampal slices.
    Science (New York, N.Y.), 1988, Mar-18, Volume: 239, Issue:4846

    Topics: Adenosine; Carbachol; Enzyme Activation; Hippocampus; Inositol Phosphates; Kinetics; Lithium; Oxotremorine; Phorbol Esters; Phosphatidylinositols; Protein Kinase C; Receptors, Muscarinic; Synapses; Synaptic Transmission

1988
Changes in muscarinic cholinergic-beta adrenergic interactions in isolated rat papillary muscle after 6-hydroxydopamine pretreatment: evidence for compensatory muscarinic supersensitivity.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Animals; Carbachol; Hydroxydopamines; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Oxidopamine; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic

1988
Cloned M1 muscarinic receptors mediate both adenylate cyclase inhibition and phosphoinositide turnover.
    The EMBO journal, 1988, Volume: 7, Issue:10

    Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Atropine; Carbachol; Cell Line; Cloning, Molecular; GTP-Binding Proteins; Oxotremorine; Phosphatidylinositols; Rats; Receptors, Muscarinic; Recombinant Proteins

1988
Calcium-dependent pirenzepine-sensitive muscarinic response in the rat hippocampal slice.
    Neuroscience letters, 1988, Aug-31, Volume: 91, Issue:2

    Topics: Animals; Calcium; Carbachol; Hippocampus; In Vitro Techniques; Membrane Potentials; Oxotremorine; Parasympathomimetics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Pirenzepine; Rats; Receptors, Muscarinic

1988
Muscarinic receptor coupling to inositol phospholipid metabolism in guinea-pig cerebral cortex, parotid gland and ileal smooth muscle.
    Biochemical pharmacology, 1988, Dec-01, Volume: 37, Issue:23

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Guanosine Triphosphate; Guinea Pigs; Ileum; Muscle, Smooth; N-Methylscopolamine; Oxotremorine; Parotid Gland; Phosphatidylinositols; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1988
The muscarinic receptor of chick embryo cells: correlation between ligand binding and calcium mobilization.
    The Journal of cell biology, 1985, Volume: 100, Issue:4

    Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Binding, Competitive; Calcium; Carbachol; Chick Embryo; Dose-Response Relationship, Drug; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Spectrometry, Fluorescence

1985
Desensitization of muscarinic acetylcholine receptors: possible relation to receptor heterogeneity and phosphoinositides.
    Brain research, 1986, Feb-26, Volume: 366, Issue:1-2

    Topics: Acetylcholine; Animals; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Carbachol; Hippocampus; Male; Molecular Conformation; Oxotremorine; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1986
In rat hippocampus, somatostatin 14 and muscarinic receptor ligands modulate an adenylate cyclase belonging to a common domain of the receptor.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Carbachol; Colforsin; GTP Phosphohydrolases; Hippocampus; Hydrolysis; Oxotremorine; Phosphatidylinositols; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Somatostatin

1987
Both presynaptic nicotinic-like and muscarinic-like autoreceptors regulate acetylcholine release at an identified neuro-neuronal synapse of Aplysia.
    Pflugers Archiv : European journal of physiology, 1988, Volume: 411, Issue:4

    Topics: Acetylcholine; Animals; Aplysia; Carbachol; Curare; Hexamethonium; Hexamethonium Compounds; Muscarine; Oxotremorine; Pilocarpine; Receptors, Muscarinic; Receptors, Nicotinic; Synapses

1988
Age-related decrements in the muscarinic enhancement of K+-evoked release of endogenous striatal dopamine: an indicator of altered cholinergic-dopaminergic reciprocal inhibitory control in senescence.
    Brain research, 1988, Jun-28, Volume: 454, Issue:1-2

    Topics: Aging; Animals; Bethanechol; Bethanechol Compounds; Carbachol; Cholinergic Fibers; Corpus Striatum; Dopamine; Haloperidol; In Vitro Techniques; Nicotine; Oxotremorine; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Muscarinic

1988
Muscarinic cholinergic receptor subtype on frog esophageal peptic cells: binding and secretion studies.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Carbachol; Esophagus; Imipramine; Kinetics; N-Methylscopolamine; Oxotremorine; Pepsinogens; Pirenzepine; Propranolol; Radioligand Assay; Rana catesbeiana; Receptors, Muscarinic; Scopolamine Derivatives

1988
Muscarinic agonists and phorbol esters increase tyrosine phosphorylation of a 40-kilodalton protein in hippocampal slices.
    Proceedings of the National Academy of Sciences of the United States of America, 1989, Volume: 86, Issue:7

    Topics: Animals; Carbachol; Hippocampus; In Vitro Techniques; Kinetics; Male; Nerve Tissue Proteins; Oxotremorine; Phorbol Esters; Phosphorylation; Protein-Tyrosine Kinases; Rats; Rats, Inbred Strains; Tyrosine

1989
Stereoselectivity of muscarinic receptors in vivo and in vitro for oxotremorine analogues. N-[4-(tertiary amino)-2-butynyl]-5-methyl-2-pyrrolidones.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:12

    Topics: Abdominal Muscles; Animals; Atropine; Carbachol; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; Lethal Dose 50; Male; Mice; Muscle Contraction; Oxotremorine; Pyrrolidinones; Rana pipiens; Receptors, Muscarinic; Stereoisomerism; Tremor

1985
Mechanisms of release of atrial natriuretic factor. I. Effect of several agonists and steroids on its release by atrial minces.
    Biochemical and biophysical research communications, 1986, Mar-28, Volume: 135, Issue:3

    Topics: Animals; Arginine Vasopressin; Atrial Natriuretic Factor; Carbachol; Enkephalin, Methionine; Epinephrine; Glucocorticoids; Heart Atria; Isoproterenol; Male; Mineralocorticoids; Oxotremorine; Phenylephrine; Rats; Secretory Rate

1986
Carbachol induces desensitization of cardiac beta-adrenergic receptors through muscarinic M1 receptors.
    Biochemical and biophysical research communications, 1985, Apr-30, Volume: 128, Issue:2

    Topics: Animals; Carbachol; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Gallamine Triethiodide; Heart; Myocardium; Oxotremorine; Propanolamines; Protein Kinase C; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic; Time Factors; Tissue Distribution

1985
Inhibition of ACTH secretion in mouse pituitary tumor cells by activation of muscarinic cholinergic receptors.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:6

    Topics: Adenylyl Cyclases; Adrenocorticotropic Hormone; Animals; Carbachol; Cells, Cultured; Cyclic AMP; Isoproterenol; Mice; Oxotremorine; Parasympatholytics; Pertussis Toxin; Pituitary Neoplasms; Receptors, Muscarinic; Scopolamine; Time Factors; Virulence Factors, Bordetella

1985
Potassium ion facilitation of phosphoinositide turnover activation by muscarinic receptor agonists in rat brain.
    Journal of neurochemistry, 1986, Volume: 46, Issue:5

    Topics: Animals; Benzodiazepinones; Carbachol; Dioxolanes; Hippocampus; Histamine; Male; Norepinephrine; Oxotremorine; Phosphatidylinositols; Pirenzepine; Potassium; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1986
Muscarinic receptors in mammalian myocardium: effects of atrial and ventricular receptors on phosphatidylinositol metabolism and adenylate cyclase.
    Journal of molecular and cellular cardiology, 1986, Volume: 18, Issue:8

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Atrial Function; Carbachol; Cats; Cyclic AMP; Heart; Inositol; Kinetics; Myocardium; Oxotremorine; Phosphatidylinositols; Quinuclidinyl Benzilate; Receptors, Muscarinic; Ventricular Function

1986
Receptor reserve in the calcium-dependent cyclic AMP response of astrocytoma cells to muscarinic receptor stimulation: demonstration by agonist-induced desensitization, receptor inactivation, and phorbol ester treatment.
    Molecular pharmacology, 1986, Volume: 30, Issue:3

    Topics: Astrocytoma; Calcium; Carbachol; Cells, Cultured; Cyclic AMP; Inositol Phosphates; Isoproterenol; Oxotremorine; Phorbols; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Tetradecanoylphorbol Acetate

1986
Muscarinic acetylcholine receptor-mediated phosphoinositide turnover in cultured cerebellar granule cells: desensitization by receptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Cerebellum; Kinetics; Male; N-Methylscopolamine; Oxotremorine; Phorbol Esters; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Virulence Factors, Bordetella

1987
Cholinergic stimulation of arachidonic acid and phosphatidic acid metabolism in C62B glioma cells.
    The Journal of biological chemistry, 1986, Mar-05, Volume: 261, Issue:7

    Topics: Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Atropine; Calcimycin; Carbachol; Cell Line; Glioma; Oxotremorine; Parasympathomimetics; Phosphatidic Acids; Pilocarpine; Rats; Time Factors; Tubocurarine

1986
Behavioural and pharmacological characterization of the mouth movements induced by muscarinic agonists in the rat.
    Psychopharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Arecoline; Brain; Carbachol; Male; Motor Activity; Mouth; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Scopolamine

1986
Cholinergic phosphatidylinositol modulation of inhibitory, G protein-linked neurotransmitter actions: electrophysiological studies in rat hippocampus.
    Proceedings of the National Academy of Sciences of the United States of America, 1987, Volume: 84, Issue:10

    Topics: Acetylcholine; Adenosine; Animals; Carbachol; GTP-Binding Proteins; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Models, Neurological; Oxotremorine; Physostigmine; Rats; Rats, Inbred F344; Rats, Inbred Strains; Tetradecanoylphorbol Acetate

1987
Pertussis toxin treatment results in tolerance to the depressant effects of opioid, monoaminergic, and muscarinic agonists on dorsal-horn network responses in mouse spinal cord-ganglion cultures.
    NIDA research monograph, 1986, Volume: 75

    Topics: Adenylate Cyclase Toxin; Animals; Carbachol; Drug Tolerance; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Fetus; Ganglia, Spinal; Mice; Morphine; Norepinephrine; Organ Culture Techniques; Oxotremorine; Pertussis Toxin; Serotonin; Spinal Cord; Virulence Factors, Bordetella

1986
Temperature effect on the detection of muscarinic receptor-G protein interactions in ligand binding assays.
    Biochemical pharmacology, 1988, Mar-15, Volume: 37, Issue:6

    Topics: Animals; Brain Stem; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Myocardium; Oxotremorine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Temperature

1988
Membrane phospholipid polar heads influence the coupling of M2 muscarinic receptors to G proteins.
    Neurochemical research, 1988, Volume: 13, Issue:8

    Topics: Animals; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Membrane Proteins; Myocardium; Oxotremorine; Phospholipids; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Type C Phospholipases

1988
Diethyl ether effects on muscarinic acetylcholine receptor complexes in rat brainstem.
    Biochemical pharmacology, 1988, Nov-01, Volume: 37, Issue:21

    Topics: Animals; Brain Stem; Carbachol; Ether; Ethyl Ethers; GTP-Binding Proteins; Guanosine Triphosphate; Halothane; In Vitro Techniques; Male; Oxotremorine; Rats; Receptors, Muscarinic; Scopolamine Derivatives

1988
Release of N-[3H]methylscopolamine from isolated guinea pig atria is controlled by diffusion and rebinding.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2

    Topics: Animals; Carbachol; Diffusion; Female; Guinea Pigs; Heart Atria; Male; Membranes; Myocardium; N-Methylscopolamine; Oxotremorine; Receptors, Muscarinic; Scopolamine Derivatives; Time Factors

1988
Carboxyl residue(s) at the ligand-binding site of rat muscarinic receptors.
    Biochemical and biophysical research communications, 1988, Nov-15, Volume: 156, Issue:3

    Topics: Affinity Labels; Animals; Atropine; Binding Sites; Brain Stem; Carbachol; Cerebral Cortex; Heart Atria; In Vitro Techniques; Male; Methylation; Onium Compounds; Oxotremorine; Rats; Receptors, Muscarinic

1988
Central muscarinic cholinergic influences on ethanol sensitivity in long-sleep and short-sleep mice.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Body Temperature; Brain; Calcium; Carbachol; Dose-Response Relationship, Drug; Ethanol; Male; Mice; Neurotensin; Oxotremorine; Phosphatidylinositols; Receptors, Muscarinic; Sleep; Species Specificity

1988
Antimuscarinic oxotremorine analogs distinguish high and low affinity agonist states of muscarinic receptors.
    Proceedings of the Western Pharmacology Society, 1988, Volume: 31

    Topics: Animals; Binding, Competitive; Carbachol; Cerebral Cortex; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Myocardium; Oxotremorine; Parasympatholytics; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Structure-Activity Relationship

1988
Characterization of muscarinic receptors in human pancreatic membranes.
    Pancreas, 1988, Volume: 3, Issue:6

    Topics: Carbachol; Cell Membrane; Humans; Oxotremorine; Pancreas; Pilocarpine; Pirenzepine; Receptors, Muscarinic

1988
Brain localization of cholinergic influence on male sex behavior in rats: agonists.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:1

    Topics: Animals; Brain; Carbachol; Copulation; Ejaculation; Injections, Intraventricular; Male; Oxotremorine; Parasympathomimetics; Preoptic Area; Rats; Sexual Behavior, Animal

1988
Impaired cardiac muscarinic receptor function in dogs with heart failure.
    The Journal of clinical investigation, 1988, Volume: 81, Issue:6

    Topics: Adenylyl Cyclases; Animals; Atropine; Carbachol; Dogs; Female; Guanosine Triphosphate; Heart Failure; Heart Ventricles; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Myocardium; Oxotremorine; Receptors, Muscarinic; Sarcolemma

1988
Characterization of cholinergic muscarinic receptors in the rabbit iris.
    Biochemical pharmacology, 1988, Jul-01, Volume: 37, Issue:13

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Ileum; Iris; Kinetics; Methacholine Chloride; Methacholine Compounds; Microsomes; N-Methylscopolamine; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives

1988
Electrophysiologic responses and adenylate cyclase activities of mouse spinal cord-dorsal root ganglion explants rendered tolerant by chronic exposure to morphine or pertussis toxin.
    Advances in experimental medicine and biology, 1987, Volume: 221

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Carbachol; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Evoked Potentials; Ganglia, Spinal; Mice; Morphine; Norepinephrine; Organ Culture Techniques; Oxotremorine; Pertussis Toxin; Serotonin; Spinal Cord; Virulence Factors, Bordetella

1987
Sialic acid is selectively involved in the interaction of agonists with M2 muscarinic acetylcholine receptors.
    Biochemical and biophysical research communications, 1988, Jan-29, Volume: 150, Issue:2

    Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Male; Myocardium; Neuraminidase; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sialic Acids

1988
Chemical modification of rat cerebral cortex M1 muscarinic receptors: role of histidyl residues in antagonist and agonist binding.
    Biochemical and biophysical research communications, 1988, Mar-30, Volume: 151, Issue:3

    Topics: Animals; Atropine; Benzilates; Binding Sites; Carbachol; Cerebral Cortex; Diethyl Pyrocarbonate; Histidine; Hydrogen-Ion Concentration; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Synaptosomes

1988
Stimulation of phosphatidylinositol (PI) turnover may mediate the muscarinic suppression of the M-current in hippocampal pyramidal cells.
    Neuroscience letters, 1988, Feb-15, Volume: 85, Issue:1

    Topics: Animals; Carbachol; Hippocampus; In Vitro Techniques; Inositol Phosphates; Membrane Potentials; Oxotremorine; Phosphatidylinositols; Potassium; Protein Kinase C; Rats; Receptors, Muscarinic

1988
Characterization of agonist and antagonist binding to muscarinic cholinergic receptors solubilized from rat cerebral cortex.
    Journal of neural transmission, 1988, Volume: 72, Issue:1

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Quantitative effects of some muscarinic agonists on evoked surface-negative field potentials recorded from the guinea-pig olfactory cortex slice.
    British journal of pharmacology, 1988, Volume: 93, Issue:4

    Topics: Acetylcholine; Animals; Bethanechol Compounds; Carbachol; Cerebral Cortex; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Methacholine Compounds; Oxotremorine; Parasympathomimetics; Temperature

1988
A quantitative study of the effects of some muscarinic antagonists on the guinea-pig olfactory cortex slice.
    British journal of pharmacology, 1988, Volume: 93, Issue:4

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Drug Interactions; Evoked Potentials; Gallamine Triethiodide; Guinea Pigs; In Vitro Techniques; Oxotremorine; Parasympathomimetics; Pirenzepine

1988
The action of pertussis toxin on heart adenylate cyclase and lipolysis in the parametrial adipose tissue of the rat.
    Biomedica biochimica acta, 1987, Volume: 46, Issue:8-9

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adipose Tissue; Animals; Carbachol; Female; Heart; Isoproterenol; Lipolysis; Myocardium; Oxotremorine; Pertussis Toxin; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Virulence Factors, Bordetella

1987
Oxygen consumption mediated by M2 muscarinic receptors in rat salivary glands.
    Journal of dental research, 1987, Volume: 66, Issue:9

    Topics: Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Female; Male; Nifedipine; Oxotremorine; Oxygen Consumption; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Salivary Glands; Trihexyphenidyl

1987
Physiological effects of muscarinic vs nicotinic ACh antagonists upon ganglion cell activity in the frog retina.
    Vision research, 1987, Volume: 27, Issue:12

    Topics: Acetylcholine; Action Potentials; Animals; Atropine; Bungarotoxins; Carbachol; Electroretinography; Neuromuscular Blocking Agents; Oxotremorine; Physostigmine; Rana esculenta; Receptors, Muscarinic; Receptors, Nicotinic; Retina; Retinal Ganglion Cells; Scopolamine

1987
Dissociation of contraction and muscarinic receptor binding to isolated smooth muscle cells.
    The American journal of physiology, 1986, Volume: 251, Issue:4 Pt 1

    Topics: Animals; Atropine; Binding, Competitive; Carbachol; Dogs; Kinetics; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Stomach; Temperature

1986
Pertussis toxin blocks depressant effects of opioid, monoaminergic and muscarinic agonists on dorsal-horn network responses in spinal cord-ganglion cultures.
    Brain research, 1987, Jan-01, Volume: 400, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Carbachol; Electrophysiology; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ganglia, Spinal; Mice; Morphine; Norepinephrine; Organ Culture Techniques; Oxotremorine; Pertussis Toxin; Serotonin; Spinal Cord; Virulence Factors, Bordetella

1987
Muscarinic and antimuscarinic activity of acetamides related to oxotremorine in the guinea pig urinary bladder.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:3

    Topics: Acetamides; Animals; Carbachol; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Oxotremorine; Receptors, Muscarinic; Urinary Bladder

1987
Selectivity of partial agonists related to oxotremorine based on differences in muscarinic receptor reserve between the guinea pig ileum and urinary bladder.
    Molecular pharmacology, 1987, Volume: 31, Issue:4

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Kinetics; Male; Mathematics; Oxotremorine; Pirenzepine; Pyrrolidines; Receptors, Muscarinic; Spasm; Structure-Activity Relationship; Urinary Bladder

1987
Muscarinic receptor heterogeneity in rat central nervous system. II. Brain receptors labeled by [3H]oxotremorine-M correspond to heterogeneous M2 receptors with very high affinity for agonists.
    Molecular pharmacology, 1987, Volume: 32, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Carbachol; Cerebral Cortex; Kinetics; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1987
Determination of thermodynamic constants for agonist binding to muscarinic receptors from rat cerebral cortex.
    Acta chemica Scandinavica. Series B: Organic chemistry and biochemistry, 1987, Volume: 41, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Cerebral Cortex; Kinetics; Male; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thermodynamics

1987
Genetic influences on tolerance development with chronic oxotremorine infusion.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:4

    Topics: Animals; Behavior, Animal; Carbachol; Dose-Response Relationship, Drug; Drug Tolerance; Genotype; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Inbred Strains; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tissue Distribution

1987
Correlation of agonist-induced phosphorylation of chick heart muscarinic receptors with receptor desensitization.
    The Journal of biological chemistry, 1987, Dec-05, Volume: 262, Issue:34

    Topics: Animals; Atropine; Carbachol; Chickens; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Heart; Magnesium; Myocardium; Oxotremorine; Phosphorylation; Quinuclidinyl Benzilate; Receptors, Muscarinic

1987
Choline increases endogenous GABA release in rat hippocampus by a mechanism sensitive to hemicholinium-3.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Choline; gamma-Aminobutyric Acid; Hemicholinium 3; Hippocampus; In Vitro Techniques; Male; Mecamylamine; Oxotremorine; Rats; Rats, Inbred Strains; Synaptosomes

1987
Evidence for involvement of midbrain central gray in cholinergic mediation of female sexual receptivity in rats.
    Behavioral neuroscience, 1986, Volume: 100, Issue:3

    Topics: Animals; Brain Mapping; Carbachol; Cholinergic Fibers; Estradiol; Female; Oxotremorine; Periaqueductal Gray; Posture; Progesterone; Rats; Sexual Behavior, Animal

1986
High-affinity agonist binding to rat brainstem muscarinic receptors is eliminated by low pH.
    Neuroscience letters, 1986, Aug-15, Volume: 69, Issue:1

    Topics: Animals; Brain Stem; Carbachol; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1986
Effects of N-ethylmaleimide on muscarinic acetylcholine receptor subtype autoradiography and inositide response in rat brain.
    Life sciences, 1986, Sep-29, Volume: 39, Issue:13

    Topics: Animals; Autoradiography; Benzodiazepinones; Brain; Carbachol; Ethylmaleimide; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Cholinergic

1986
Muscarinic receptor coupling to intracellular calcium release in rat pancreatic acinar carcinoma.
    Cancer research, 1986, Volume: 46, Issue:11

    Topics: Animals; Binding, Competitive; Calcium; Carbachol; Carcinoma; N-Methylscopolamine; Oxotremorine; Pancreatic Neoplasms; Proteins; Rats; Rats, Inbred F344; Receptors, Muscarinic; Scopolamine Derivatives

1986
Irreversible binding of acetylethylcholine mustard to cardiac cholinergic muscarinic receptors.
    Molecular pharmacology, 1986, Volume: 30, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cell Membrane; Guanylyl Imidodiphosphate; Heart Rate; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1986
Stimulation of phosphatidylinositol metabolism in atrial and ventricular myocytes.
    Life sciences, 1986, Dec-08, Volume: 39, Issue:23

    Topics: Acetylcholine; Adenosine; Angiotensin II; Animals; Carbachol; Guinea Pigs; Heart Atria; Heart Ventricles; Inositol Phosphates; Lithium; Muscle, Smooth, Vascular; Oxotremorine; Phosphatidylinositols; Time Factors; Vasopressins

1986
Role of lipids in age-related changes in the properties of muscarinic receptors in cultured rat heart myocytes.
    Biochemistry, 1986, Dec-02, Volume: 25, Issue:24

    Topics: Acetylcholine; Animals; Animals, Newborn; Benzilates; Carbachol; Cells, Cultured; Guanylyl Imidodiphosphate; Kinetics; Liposomes; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic

1986
Stereospecific 3H-QNB binding to human erythrocyte membranes associated with muscarinic cholinergic receptors.
    Journal of neural transmission, 1987, Volume: 68, Issue:1-2

    Topics: Adult; Aging; Animals; Atropine; Brain; Carbachol; Erythrocyte Membrane; Female; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Male; Middle Aged; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism

1987
Pharmacologic characterization and functional role of muscarinic autoreceptors in the rabbit striatum.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Corpus Striatum; Dose-Response Relationship, Drug; Drug Synergism; Haloperidol; Oxotremorine; Physostigmine; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Scopolamine; Time Factors

1987
Characterization of [3H]pirenzepine binding to muscarinic cholinergic receptors solubilized from rat brain.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Carbachol; Detergents; In Vitro Techniques; Kinetics; Male; Oxotremorine; Parasympatholytics; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Solubility; Tritium

1985
Experimental testing of Mackay's model for functional antagonism in the isolated costo-uterus of the rat.
    British journal of pharmacology, 1985, Volume: 86, Issue:1

    Topics: Animals; Carbachol; Drug Antagonism; Female; Fenoterol; In Vitro Techniques; Kinetics; Male; Models, Biological; Oxotremorine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Uterine Contraction

1985
Different effects of N-ethylmaleimide on M1 and M2 muscarine receptors in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:2

    Topics: Animals; Binding Sites; Brain; Carbachol; Ethylmaleimide; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tissue Distribution

1985
Characterization of muscarinic cholinergic receptors in the crab nervous system.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Animals; Arecoline; Binding, Competitive; Brachyura; Carbachol; Decamethonium Compounds; Kinetics; Male; Mathematics; Nervous System; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Stereoisomerism; Tissue Distribution; Tubocurarine

1986
Allosteric interactions between muscarinic agonist binding sites and effector sites demonstrated by the use of bisquaternary pyridinium oximes.
    Life sciences, 1985, Jun-03, Volume: 36, Issue:22

    Topics: Animals; Brain Stem; Carbachol; Cerebral Cortex; Cobalt; Guanylyl Imidodiphosphate; In Vitro Techniques; Oximes; Oxotremorine; Parasympathomimetics; Pyridinium Compounds; Rats; Receptors, Muscarinic

1985
Muscarinic acetylcholine receptors in the rabbit ciliary body smooth muscle: spare receptors and threshold phenomenon.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:1

    Topics: Animals; Arecoline; Atropine; Carbachol; Ciliary Body; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxotremorine; Phenoxybenzamine; Pilocarpine; Rabbits; Receptors, Muscarinic

1985
Rat brain and heart muscarinic receptors: modification with tetranitromethane.
    Biochemical and biophysical research communications, 1985, Sep-30, Volume: 131, Issue:3

    Topics: Acetylcholine; Animals; Brain; Brain Stem; Carbachol; Corpus Striatum; Heart Atria; Hippocampus; Methane; Myocardium; Nitrogen; Oxotremorine; Rats; Receptors, Muscarinic; Tetranitromethane

1985
The relationship between muscarinic receptor occupancy and adenylate cyclase inhibition in the rabbit myocardium.
    Molecular pharmacology, 1985, Volume: 28, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Guanosine Triphosphate; In Vitro Techniques; Male; Models, Structural; Myocardium; N-Methylscopolamine; Oxotremorine; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1985
Oxotremorine acts as a partial nicotinic agonist on cultured chick myotubes.
    Acta pharmacologica et toxicologica, 1985, Volume: 57, Issue:5

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Carbachol; Cells, Cultured; Chick Embryo; Microtubules; Muscles; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Nicotinic

1985
Multiple agonist binding sites of muscarinic acetylcholine receptors and their relation to the negative inotropic action of agonists in guinea-pig heart.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Binding Sites; Carbachol; Depression, Chemical; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Myocardial Contraction; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1985
Central nervous system and autonomic nervous system effects of amantadine and of some standard anti-Parkinson drugs.
    Pharmacology, 1973, Volume: 10, Issue:4

    Topics: Amantadine; Animals; Antiparkinson Agents; Atropine; Autonomic Nervous System; Body Temperature; Carbachol; Central Nervous System; Dihydroxyphenylalanine; Drug Interactions; Gastrointestinal Motility; Male; Mecamylamine; Mice; Mydriatics; Nicotine; Oxotremorine; Phenothiazines; Pupil; Rats; Trihexyphenidyl

1973
Muscarinic cholinergic binding in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1974, Volume: 71, Issue:5

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Binding Sites; Binding, Competitive; Brain; Brompheniramine; Carbachol; Chlorpheniramine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Microsomes; Mitochondria; Oxotremorine; Pilocarpine; Quaternary Ammonium Compounds; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Temperature; Time Factors; Tritium

1974
Muscarinic mediation of the biphasic temperature response to intrahypothalamic injections of carbachol in the cat.
    Experientia, 1974, May-15, Volume: 30, Issue:5

    Topics: Animals; Atropa belladonna; Body Temperature Regulation; Carbachol; Cats; Hypothalamus; Male; Mecamylamine; Nicotine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Plants, Medicinal; Plants, Toxic; Receptors, Cholinergic; Species Specificity; Synaptic Transmission

1974
Interrelation between monoaminergic and cholinergic mechanisms in the hypothalamic thermoregulatory centre of rabbits.
    Neuropharmacology, 1974, Volume: 13, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Biogenic Amines; Body Temperature Regulation; Carbachol; Cerebral Ventricles; Dopamine; Dose-Response Relationship, Drug; Epinephrine; Female; Hypothalamus; Injections; Male; Norepinephrine; Oxotremorine; Parasympathetic Nervous System; Phenoxybenzamine; Physostigmine; Pilocarpine; Propranolol; Rabbits; Receptors, Cholinergic; Serotonin; Time Factors; Tubocurarine

1974
Temperature reducing effect of oxotremorine in the rat and the mouse.
    Acta physiologica Academiae Scientiarum Hungaricae, 1973, Volume: 44, Issue:3-4

    Topics: Acetylcholine; Amyl Nitrite; Animals; Atropine; Atropine Derivatives; Blood Pressure; Body Temperature; Carbachol; Chlorpromazine; Dopamine; Dose-Response Relationship, Drug; Epinephrine; Ethanol; Female; Isoproterenol; Male; Mice; Norepinephrine; Oxotremorine; Oxygen Consumption; Temperature; Tremorine; Urethane; Vasopressins

1973
Proceedings: The nature of the thermoregulatory sensitivity to cholinomimetic drugs in the cerebral ventricles of sheep.
    The Journal of physiology, 1974, Volume: 236, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Body Temperature Regulation; Carbachol; Cerebral Ventricles; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Sheep; Shivering; Temperature

1974
Effects of several muscarinic agonists on cardiac performance and the release of noradrenaline from sympathetic nerves of the perfused rabbit heart.
    British journal of pharmacology, 1972, Volume: 45, Issue:4

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Carbamates; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Female; Heart; Heart Rate; Hexamethonium Compounds; In Vitro Techniques; Male; Methacholine Compounds; Norepinephrine; Oxotremorine; Parasympathomimetics; Perfusion; Pilocarpine; Quaternary Ammonium Compounds; Rabbits; Sympathetic Nervous System

1972
The character of the muscarinic receptors in different regions of the rat brain.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1980, Feb-13, Volume: 207, Issue:1166

    Topics: Animals; Binding Sites; Brain; Carbachol; Mathematics; Oxotremorine; Propylbenzilylcholine Mustard; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1980
Influence of cholinomimetics and cholinolytics on vestibular compensation.
    Brain research, 1981, Oct-19, Volume: 222, Issue:2

    Topics: Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Ear, Inner; Methacholine Chloride; Methacholine Compounds; Muscarine; Nicotine; Oxotremorine; Rana temporaria; Vestibule, Labyrinth

1981
Effects of neurotransmitters on calcium efflux from cultured glioma cells.
    Journal of neuroscience research, 1981, Volume: 6, Issue:3

    Topics: Astrocytoma; Atropine; Calcium; Calcium Radioisotopes; Carbachol; Cells, Cultured; Cyclic AMP; Cyclic GMP; Glutamates; Glutamic Acid; Glycine; Hexamethonium; Hexamethonium Compounds; Humans; Neoplasms, Experimental; Nicotine; Norepinephrine; Oxotremorine; Prostaglandins E; Time Factors

1981
Muscarinic cholinergic stimulation of somatostatin secretion from long term dispersed cell cultures of fetal rat hypothalamus: inhibition by gamma-aminobutyric acid and serotonin.
    Endocrinology, 1983, Volume: 112, Issue:2

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Female; gamma-Aminobutyric Acid; Hexamethonium Compounds; Hypothalamus; Oxotremorine; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic; Serotonin; Somatostatin; Tetrodotoxin

1983
Effects of acetylcholine on sodium-dependent high-affinity glutamate transport in rat striatal homogenates.
    Journal of neurochemistry, 1983, Volume: 40, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Biological Transport; Carbachol; Corpus Striatum; Glutamates; Glutamic Acid; Kinetics; Male; Nicotine; Oxotremorine; Rats; Rats, Inbred Strains; Sodium

1983
Increase in muscarinic acetylcholine receptors in mouse intestine by hexamethonium treatment.
    Life sciences, 1983, May-23, Volume: 32, Issue:21

    Topics: Animals; Brain; Carbachol; Female; Hexamethonium; Hexamethonium Compounds; Ileum; Intestinal Mucosa; Male; Mice; Muscle Contraction; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Rectum

1983
Affinity, efficacy, and stereoselectivity of oxotremorine analogues for muscarinic receptors in the isolated guinea pig ileum.
    Molecular pharmacology, 1983, Volume: 23, Issue:1

    Topics: Animals; Atropine; Carbachol; Dibenzylchlorethamine; Dose-Response Relationship, Drug; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Ileum; Isomerism; Male; Oxotremorine; Parasympatholytics; Receptors, Cholinergic; Receptors, Muscarinic; Structure-Activity Relationship

1983
Muscarinic acetylcholine receptor activation causes inhibition of cyclic AMP accumulation, prolactin and growth hormone secretion in GH3 rat anterior pituitary tumour cells.
    Biochimica et biophysica acta, 1984, Sep-14, Volume: 805, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Carbachol; Cell Line; Cyclic AMP; Growth Hormone; Kinetics; Oxotremorine; Pituitary Gland, Anterior; Pituitary Neoplasms; Prolactin; Rats; Receptors, Muscarinic; Vasoactive Intestinal Peptide

1984
A comparison of the stimulant activities of oxotremorine analogues on the frog rectus abdominis and the guinea pig ileum.
    European journal of pharmacology, 1984, Mar-23, Volume: 99, Issue:2-3

    Topics: Abdominal Muscles; Animals; Carbachol; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Oxotremorine; Rana pipiens; Receptors, Muscarinic; Receptors, Nicotinic; Structure-Activity Relationship

1984
Quantitative receptor autoradiography: application to the characterization of multiple receptor subtypes.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Autoradiography; Benzodiazepinones; Binding, Competitive; Brain; Carbachol; Hippocampus; Indoles; Oxotremorine; Pindolol; Pirenzepine; Rats; Receptors, Muscarinic; Receptors, Serotonin; Superior Colliculi; Tetrahydronaphthalenes

1984
Comparative properties of the in ovo and in vitro differentiation of the muscarinic cholinergic receptor in embryonic heart cells.
    Developmental biology, 1980, Volume: 78, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; Cells, Cultured; Chick Embryo; Cyclic GMP; Heart; Heart Rate; Myocardial Contraction; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic

1980
Characteristics of histamine release evoked by acetylcholine in isolated rat mast cells.
    The Journal of physiology, 1980, Volume: 301

    Topics: Acetylcholine; Animals; Atropine; Bucladesine; Carbachol; Choline; Epinephrine; Histamine Release; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Mast Cells; Oxotremorine; Rats; Secretory Rate; Sodium

1980
Muscarinic-dopaminergic synergism on retinal cyclic AMP formation.
    Brain research, 1981, Jun-29, Volume: 215, Issue:1-2

    Topics: Animals; Atropine; Carbachol; Cyclic AMP; Female; Oxotremorine; Rats; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Muscarinic; Retina

1981
Muscarinic cholinergic receptor-mediated control of cyclic AMP metabolism. Agonist-induced changes in nucleotide synthesis and degradation.
    Molecular pharmacology, 1983, Volume: 23, Issue:2

    Topics: Alprostadil; Astrocytoma; Carbachol; Cell Line; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Isoproterenol; Oxotremorine; Prostaglandins E; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic

1983
Agonists differentiate muscarinic receptors that inhibit cyclic AMP formation from those that stimulate phosphoinositide metabolism.
    The Journal of biological chemistry, 1984, Mar-25, Volume: 259, Issue:6

    Topics: Animals; Carbachol; Chick Embryo; Cyclic AMP; In Vitro Techniques; Kinetics; Myocardium; Oxotremorine; Phosphatidylinositols; Quinuclidinyl Benzilate; Receptors, Muscarinic

1984
The conversion of 2-chloroalkylamine analogues of oxotremorine to aziridinium ions and their interactions with muscarinic receptors in the guinea pig ileum.
    Molecular pharmacology, 1984, Volume: 26, Issue:2

    Topics: Alkylation; Animals; Aziridines; Azirines; Binding, Competitive; Carbachol; Chlorides; Guinea Pigs; Hydrolysis; Ileum; Indicators and Reagents; Kinetics; Muscle Contraction; Oxotremorine; Pyrrolidinones; Quinuclidinyl Benzilate; Rana pipiens; Receptors, Muscarinic

1984
Effects of acute ketotic and non-ketotic diabetes on the myocardial muscarinic receptors.
    Acta pharmacologica et toxicologica, 1984, Volume: 55, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; Computers; Diabetes Mellitus, Experimental; Diabetic Ketoacidosis; Guanylyl Imidodiphosphate; Insulin; Male; Models, Biological; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1984
Pharmacological and anatomical aspects of cholinergic activation of female sexual behavior.
    Physiology & behavior, 1984, Volume: 32, Issue:6

    Topics: Animals; Atropine; Carbachol; Castration; Dose-Response Relationship, Drug; Female; Injections, Intraventricular; Oxotremorine; Preoptic Area; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus

1984
Evidence from phospholipid metabolism changes for muscarinic cholinergic receptors on rat anterior pituitary cells.
    Journal of neuroscience research, 1983, Volume: 10, Issue:3

    Topics: Animals; Carbachol; Culture Techniques; Male; Membrane Lipids; Oxotremorine; Phospholipids; Pilocarpine; Pituitary Gland, Anterior; Rats; Receptors, Muscarinic

1983
Effect of pH on binding of agonists and antagonists to rat heart muscarinic receptors.
    The Biochemical journal, 1983, Oct-15, Volume: 216, Issue:1

    Topics: Animals; Atropine; Carbachol; Cell Membrane; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Models, Biological; Myocardium; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Receptors, Muscarinic; Scopolamine; Solanaceous Alkaloids

1983
The effects of p-chloromercuribenzoate on muscarinic receptors in the cerebral cortex.
    British journal of pharmacology, 1983, Volume: 80, Issue:1

    Topics: Animals; Carbachol; Cerebral Cortex; Chloromercuribenzoates; Drug Interactions; In Vitro Techniques; Oxotremorine; p-Chloromercuribenzoic Acid; Propylbenzilylcholine Mustard; Rats; Receptors, Muscarinic; Tritium

1983
Determination of dissociation constants and relative efficacies of oxotremorine analogs at muscarinic receptors in the guinea-pig ileum by pharmacological procedures.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:1

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Kinetics; Mathematics; Oxotremorine; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Structure-Activity Relationship

1984
Presynaptic muscarinic modulation of nicotinic excitation in the rat neostriatum.
    Brain research, 1984, Mar-26, Volume: 296, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Corpus Striatum; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Muscarine; Nicotine; Oxotremorine; Potassium; Rats; Receptors, Muscarinic; Receptors, Nicotinic

1984
Partial agonist activity of oxotremorine at muscarinic acetylcholine receptors in the embryonic chick heart.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:2

    Topics: Animals; Carbachol; Chick Embryo; Heart; Heart Rate; Oxotremorine; Receptors, Muscarinic

1984
The time course of muscarinic depolarization of guinea-pig myenteric neurones.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Acetylcholine; Animals; Barium; Carbachol; Guinea Pigs; In Vitro Techniques; Methacholine Compounds; Myenteric Plexus; Neostigmine; Neurons; Oxotremorine; Receptors, Muscarinic; Scopolamine; Temperature; Time Factors

1984
Differential regulation of muscarinic and nicotinic receptors by cholinergic stimulation in cultured avian retina cells.
    Brain research, 1983, Feb-28, Volume: 262, Issue:1

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Chick Embryo; N-Methylscopolamine; Neurons; Nicotine; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Receptors, Nicotinic; Retina; Scopolamine Derivatives; Tubocurarine

1983
Modification by hexamethonium of the muscarinic receptors blocking activity of pancuronium and homatropine in isolated tissues of the guinea-pig.
    European journal of pharmacology, 1982, May-07, Volume: 80, Issue:1

    Topics: Animals; Carbachol; Female; Guinea Pigs; Heart; Hexamethonium Compounds; Ileum; Male; Mecamylamine; Oxotremorine; Pancuronium; Receptors, Cholinergic; Receptors, Muscarinic; Tropanes

1982
Isolated rat gastric parietal cells: cholinergic response and pharmacology.
    Life sciences, 1981, Feb-09, Volume: 28, Issue:6

    Topics: Acetylcholine; Aminopyrine; Animals; Atropine; Biological Transport; Carbachol; Dose-Response Relationship, Drug; Gastric Mucosa; In Vitro Techniques; Methacholine Chloride; Methacholine Compounds; Oxotremorine; Rats

1981
The effect of amitriptyline, mianserin, and viloxazine at pre- and post-junctional muscarinic receptors in guinea-pig ileal longitudinal muscle.
    Canadian journal of physiology and pharmacology, 1982, Volume: 60, Issue:2

    Topics: Acetylcholine; Amitriptyline; Animals; Antidepressive Agents; Atropine; Carbachol; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mianserin; Muscle, Smooth; Oxotremorine; Receptors, Cholinergic; Receptors, Muscarinic; Viloxazine

1982
In vivo regulation of muscarinic cholinergic receptors in embryonic chick brain.
    Molecular pharmacology, 1982, Volume: 21, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Carbachol; Chick Embryo; Kinetics; Membranes; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Time Factors

1982
Do cholinomimetics specifically antagonize rotational behavior?
    Pharmacology, biochemistry, and behavior, 1981, Volume: 15, Issue:5

    Topics: Animals; Carbachol; Caudate Nucleus; Dopamine; Female; Humans; Injections; Oxotremorine; Parasympathomimetics; Posture; Rats; Rats, Inbred Strains; Rotation; Stereotyped Behavior; Substantia Nigra

1981
Effect of some cholinergic drugs on the conditioned pole jump response in rats.
    Pharmacology, biochemistry, and behavior, 1981, Volume: 15, Issue:4

    Topics: Animals; Avoidance Learning; Carbachol; Conditioning, Psychological; Female; Male; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Rats; Time Factors

1981
Kinetic studies on muscarinic antagonist-agonist competition.
    The Journal of biological chemistry, 1980, Apr-10, Volume: 255, Issue:7

    Topics: Animals; Atropine; Benzilates; Binding, Competitive; Carbachol; Intestine, Small; Kinetics; Male; Muscle, Smooth; Oxotremorine; Parasympatholytics; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1980
Regulation of muscarinic acetylcholine receptor concentration in cloned neuroblastoma cells.
    Journal of neurochemistry, 1980, Volume: 34, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Cell Line; Clone Cells; Dose-Response Relationship, Drug; Kinetics; Mice; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic

1980
Analysis of regional variations in the affinities of muscarinic agonists in the rat brain.
    Brain research, 1980, Jul-07, Volume: 193, Issue:1

    Topics: Animals; Atropine; Binding, Competitive; Brain; Carbachol; Male; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1980
Studies on the putative anticholinergic effects of desmethylimipramine.
    Archives internationales de pharmacodynamie et de therapie, 1980, Volume: 243, Issue:1

    Topics: Animals; Atropine; Blepharoptosis; Carbachol; Defecation; Desipramine; Gastric Juice; Male; Mice; Mydriatics; Oxotremorine; Parasympatholytics; Rats; Salivation

1980
Muscarinic receptor subsensitivity in the longitudinal muscle of the rat ileum following chronic anticholinesterase treatment with diisopropylfluorophosphate.
    Biochemical pharmacology, 1980, May-15, Volume: 29, Issue:10

    Topics: Acetylcholine; Animals; Carbachol; Cholinesterases; Drug Tolerance; Ileum; In Vitro Techniques; Isoflurophate; Kinetics; Male; Muscle, Smooth; Oxotremorine; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Time Factors

1980
Muscarinic cholinergic stimulation of the nitric oxide-cyclic GMP signaling system in cultured rat sensory neurons.
    Neuroscience, 1994, Volume: 62, Issue:2

    Topics: Acetylcholine; Amino Acid Oxidoreductases; Animals; Arginine; Atropine; Capsaicin; Carbachol; Cells, Cultured; Cyclic GMP; Embryo, Mammalian; Ganglia, Spinal; Guanylate Cyclase; Methacholine Chloride; Methylene Blue; Neurons, Afferent; Nicotine; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; omega-N-Methylarginine; Oxotremorine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Signal Transduction

1994
Expression of muscarinic M3-receptors coupled to inositol phospholipid hydrolysis in human detrusor cultured smooth muscle cells.
    The Journal of urology, 1995, Volume: 154, Issue:3

    Topics: Carbachol; Cells, Cultured; Diamines; Humans; Hydrolysis; Inositol Phosphates; Methacholine Chloride; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Urinary Bladder

1995
Galanin stimulates striatal acetylcholine release via a mechanism unrelated to cholinergic receptor stimulation.
    Regulatory peptides, 1993, Jun-11, Volume: 45, Issue:3

    Topics: Acetylcholine; Animals; Bupivacaine; Carbachol; Chromatography, High Pressure Liquid; Corpus Striatum; Galanin; Injections, Intraperitoneal; Male; Neuropeptides; Oxotremorine; Peptides; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Receptors, Galanin; Receptors, Gastrointestinal Hormone; Scopolamine; Substance P

1993
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
    Experimental eye research, 1994, Volume: 59, Issue:6

    Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines

1994
Neurotransmitter and neuropeptide modulation of high affinity choline uptake in Limulus brain.
    Comparative biochemistry and physiology. Part A, Physiology, 1995, Volume: 111, Issue:1

    Topics: Animals; Atropine; Brain; Carbachol; Choline; FMRFamide; Horseshoe Crabs; Neuropeptides; Neurotransmitter Agents; Octopamine; Oligopeptides; Oxotremorine; Pirenzepine; Potassium; Serotonin; Tubocurarine

1995
Attenuation of muscarinic receptor-G-protein interaction in Alzheimer disease.
    Molecular and chemical neuropathology, 1995, Volume: 24, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Carbachol; Cerebral Cortex; Choline O-Acetyltransferase; Female; Frontal Lobe; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Humans; Male; Middle Aged; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Pirenzepine; Receptors, Muscarinic; Reference Values; Regression Analysis; Synaptic Membranes; Synaptosomes

1995
Dissociation of striatal GTPase and dopamine release responses to muscarinic cholinergic agonists in F344 rats: influence of age and dietary manipulation.
    Journal of neurochemistry, 1995, Volume: 64, Issue:6

    Topics: Aging; Animals; Carbachol; Cholesterol; Cholinergic Agents; Corpus Striatum; Diet; Dopamine; GTP Phosphohydrolases; Male; Oxotremorine; Phospholipids; Potassium Chloride; Rats; Rats, Inbred F344; Synaptosomes

1995
The mechanism of muscarinic agonist-stimulated inositol phosphate formation in permeabilized ileal smooth muscle.
    Japanese journal of pharmacology, 1994, Volume: 65, Issue:3

    Topics: Acetylcholine; Animals; Calcium; Carbachol; Dose-Response Relationship, Drug; Drug Synergism; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Substrate Specificity; Time Factors; Type C Phospholipases

1994
Muscarinic inhibition of cardiac norepinephrine and neuropeptide Y release during ischemia and reperfusion.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Atropine; Carbachol; Electric Stimulation; Guinea Pigs; Heart; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Neuropeptide Y; Norepinephrine; Oxotremorine; Parasympatholytics; Pirenzepine; Receptors, Muscarinic

1994
Enhanced MPTP neurotoxicity after treatment with isoflurophate or cholinergic agonists.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Acetylcholine; Animals; Carbachol; Corpus Striatum; Dopamine; Drug Synergism; Isoflurophate; Male; Mice; MPTP Poisoning; Nicotine; Oxotremorine; Parasympathomimetics; Receptors, Cholinergic; Tyrosine 3-Monooxygenase

1994
A comparison between muscarinic receptor occupancy, inositol 1,4,5-trisphosphate accumulation and Ca2+ mobilization in permeabilized SH-SY5Y neuroblastoma cells.
    Neuropharmacology, 1994, Volume: 33, Issue:7

    Topics: Arecoline; Brain Neoplasms; Calcium; Calcium Radioisotopes; Carbachol; Guanine Nucleotides; Humans; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Neuroblastoma; Oxotremorine; Patch-Clamp Techniques; Receptors, Muscarinic; Signal Transduction; Tumor Cells, Cultured

1994
Acetylcholine receptor agonists stimulate [3H]taurine release from rat sympathetic ganglia.
    European journal of pharmacology, 1994, Aug-01, Volume: 260, Issue:2-3

    Topics: Amino Acids; Animals; Atropine; Carbachol; Cholinergic Agonists; Chromatography, High Pressure Liquid; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Drug Interactions; Fluorometry; Hexamethonium; Male; Microscopy; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Rats; Rats, Wistar; Regression Analysis; Superior Cervical Ganglion; Taurine

1994
Reductions of 56Fe heavy-particle irradiation-induced deficits in striatal muscarinic receptor sensitivity by selective cross-activation/inhibition of second-messenger systems.
    Radiation research, 1994, Volume: 139, Issue:1

    Topics: Analysis of Variance; Animals; Arachidonic Acid; Arginine Vasopressin; Carbachol; Corpus Striatum; Dopamine; In Vitro Techniques; Iron Radioisotopes; Male; Oxotremorine; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Second Messenger Systems; Whole-Body Irradiation

1994
Sigma receptors and signal transduction: negative modulation of signaling through phosphoinositide-linked receptor systems.
    NIDA research monograph, 1993, Volume: 133

    Topics: Animals; Carbachol; Male; Oxotremorine; Pentazocine; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, sigma; Signal Transduction

1993
Chromodacryorrhea in rats: absence following soman poisoning.
    Toxicology and applied pharmacology, 1994, Volume: 124, Issue:1

    Topics: Acetylcholinesterase; Animals; Brain; Carbachol; Carboxylesterase; Carboxylic Ester Hydrolases; Harderian Gland; Lacrimal Apparatus Diseases; Male; Nicotine; Oxotremorine; Parasympathomimetics; Physostigmine; Pilocarpine; Rats; Rats, Sprague-Dawley; Soman

1994
Characteristics and regulation of a muscarinically activated K current in HSG-PA cells.
    The American journal of physiology, 1994, Volume: 266, Issue:1 Pt 1

    Topics: Calcium; Carbachol; Cell Line; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Oxotremorine; Parasympathomimetics; Potassium; Potassium Channel Blockers; Salivary Glands; Signal Transduction; Tetraethylammonium; Tetraethylammonium Compounds

1994
Muscarinic potentiation of excitatory amino acid-evoked dopamine release in mesencephalic cells: specificity for the NMDA response and role of intracellular messengers.
    Synapse (New York, N.Y.), 1993, Volume: 15, Issue:1

    Topics: Alkaloids; Animals; Carbachol; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dopamine; Drug Synergism; Fetus; Isoquinolines; Kainic Acid; Kinetics; Mesencephalon; N-Methylaspartate; Neurons; Oxotremorine; Protein Kinase C; Quisqualic Acid; Rats; Receptors, Muscarinic; Receptors, N-Methyl-D-Aspartate; Second Messenger Systems; Staurosporine

1993
Effects of the muscarinic agonist oxotremorine on membrane fluidity in rat lymphocytes.
    Biochemistry and molecular biology international, 1993, Volume: 29, Issue:6

    Topics: Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Fluorescence Polarization; Lymphocytes; Male; Membrane Fluidity; Oxotremorine; Pilocarpine; Rats; Rats, Sprague-Dawley; Scopolamine; Spleen

1993
Studies of muscarinic receptor reserve linked to phosphoinositide hydrolysis in parotid gland and cerebral cortex.
    Acta physiologica Scandinavica, 1993, Volume: 147, Issue:3

    Topics: Animals; Carbachol; Cerebral Cortex; Choline; Guinea Pigs; Hydrolysis; In Vitro Techniques; Kinetics; N-Methylscopolamine; Oxotremorine; Parasympathomimetics; Parotid Gland; Phosphatidylinositols; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1993
Multiple second-messenger pathways mediate agonist regulation of muscarinic receptor mRNA expression.
    Biochemistry, 1993, May-18, Volume: 32, Issue:19

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Chick Embryo; Cyclic AMP; Enzyme Activation; Gene Expression Regulation; Heart; Myocardium; Oxotremorine; Pertussis Toxin; Pilocarpine; Receptors, Muscarinic; RNA, Messenger; Second Messenger Systems; Type C Phospholipases; Virulence Factors, Bordetella

1993
Muscarinic M3 receptors mediate total inositol phosphates accumulation in murine HSDM1C1 fibrosarcoma cells.
    European journal of pharmacology, 1993, Jan-04, Volume: 244, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Dioxolanes; Fibrosarcoma; Inositol Phosphates; Mice; Muscarine; Muscarinic Antagonists; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Parasympathomimetics; Pirenzepine; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives; Tumor Cells, Cultured

1993
Differences between rat dorsal and ventral hippocampus in muscarinic receptor agonist binding and interaction with phospholipase C.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: Alkaloids; Animals; Carbachol; Furans; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Mitochondria; N-Methylscopolamine; Naphthalenes; Oxotremorine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Synaptosomes; Type C Phospholipases

1993
Muscarinic receptor regulation and 2nd messenger responses in rat neocortex cultures.
    Journal of receptor research, 1993, Volume: 13, Issue:1-4

    Topics: Animals; Binding, Competitive; Carbachol; Cells, Cultured; Cerebral Cortex; Down-Regulation; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Second Messenger Systems

1993
Muscarinic m2 receptors in cerebellar granule cell cultures from rat: mechanism of short-term desensitization.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; beta-Adrenergic Receptor Kinases; Carbachol; Cells, Cultured; Cerebellum; Cyclic AMP-Dependent Protein Kinases; Muscarine; Neurons; Oxotremorine; Protein Kinases; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1993
Affinity ligands and related agents for brain muscarinic and nicotinic cholinergic receptors.
    Biochemical pharmacology, 1993, May-25, Volume: 45, Issue:10

    Topics: Affinity Labels; Animals; Brain; Carbachol; Choline; Kinetics; Ligands; Mice; Naloxone; Nicotine; Oxotremorine; Procaine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; Seizures; Tritium

1993
Muscarinic cholinergic receptors in brain and atrial membranes of adult brook trout (Salvelinus fontinalis) measured by radioligand binding techniques.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1995, Volume: 112, Issue:1

    Topics: Animals; Atropine; Binding, Competitive; Brain Chemistry; Carbachol; Heart Atria; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Pirenzepine; Radioligand Assay; Receptors, Muscarinic; Scopolamine; Scopolamine Derivatives; Trout

1995
Pharmacological basis for functional selectivity of partial muscarinic receptor agonists.
    European journal of pharmacology, 1996, Feb-22, Volume: 297, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; CHO Cells; Cricetinae; Humans; Hydrolysis; Muscarinic Agonists; Oxotremorine; Phosphatidylinositols; Receptors, Muscarinic; Signal Transduction

1996
Alanine scanning mutagenesis of conserved arginine/lysine-arginine/lysine-X-X-arginine/lysine G protein-activating motifs on m1 muscarinic acetylcholine receptors.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Alanine; Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; CHO Cells; Conserved Sequence; Cricetinae; DNA Primers; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; N-Methylscopolamine; Oxotremorine; Protein Structure, Secondary; Quinuclidinyl Benzilate; Receptor, Muscarinic M2; Receptors, Muscarinic; Recombinant Proteins; Scopolamine Derivatives; Second Messenger Systems; Transfection

1996
Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Elapid Venoms; Furans; Gallamine Triethiodide; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Naphthalenes; Oxotremorine; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Protein Binding; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Membranes; Tubocurarine

1996
Parasympathetic inhibition of pineal indole metabolism by prejunctional modulation of noradrenaline release.
    European journal of pharmacology, 1996, Jul-18, Volume: 308, Issue:2

    Topics: Animals; Carbachol; Cholinergic Agonists; Male; Melatonin; Microdialysis; Nicotine; Norepinephrine; Oxotremorine; Pineal Gland; Rats; Serotonin; Tryptamines

1996
Phorbol esters but not the cholinergic agonists oxotremorine-M and carbachol increase release of the amyloid precursor protein in cultured rat cortical neurons.
    Journal of neurochemistry, 1996, Volume: 67, Issue:4

    Topics: Amyloid beta-Protein Precursor; Animals; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Embryo, Mammalian; Muscarinic Agonists; Neurons; Oxotremorine; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Signal Transduction; Tetradecanoylphorbol Acetate

1996
Interactions of agonists with an allosteric antagonist at muscarinic acetylcholine M2 receptors.
    European journal of pharmacology, 1996, Nov-28, Volume: 316, Issue:1

    Topics: Acetylcholine; Animals; Binding, Competitive; Bis-Trimethylammonium Compounds; Buffers; Carbachol; Dioxolanes; Drug Interactions; Female; Guinea Pigs; In Vitro Techniques; Isoindoles; Kinetics; Male; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Receptor, Muscarinic M2; Receptors, Muscarinic

1996
A muscarinic acetylcholine receptor, present in the epithelial cell line from Chironomus tentans.
    Biological chemistry, 1996, Volume: 377, Issue:12

    Topics: Animals; Atropine; Binding Sites; Binding, Competitive; Blotting, Western; Carbachol; Cell Line; Chironomidae; Ecdysterone; Epithelium; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Cholinergic

1996
Muscarinic acetylcholine receptor-mediated induction of zif268 mRNA in PC12D cells requires protein kinase C and the influx of extracellular calcium.
    Journal of neurochemistry, 1997, Volume: 68, Issue:3

    Topics: Animals; Calcium; Carbachol; DNA-Binding Proteins; Early Growth Response Protein 1; Extracellular Space; Immediate-Early Proteins; Muscarinic Agonists; Oxotremorine; PC12 Cells; Phosphatidylinositol 4,5-Diphosphate; Protein Kinase C; Rats; Receptors, Muscarinic; RNA, Messenger; Transcription Factors

1997
Muscarinic acetylcholine receptors on rat thymocytes: their possible involvement in DNA fragmentation.
    Japanese journal of pharmacology, 1997, Volume: 73, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Apoptosis; Atropine; Binding, Competitive; Carbachol; DNA Fragmentation; Electrophoresis, Agar Gel; Hydrocortisone; Injections, Subcutaneous; Isotope Labeling; Male; Muscarinic Agonists; Muscarinic Antagonists; Nucleosomes; Oxotremorine; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Thymus Gland

1997
Exocytotic release from neuronal cell bodies, dendrites and nerve terminals in sympathetic ganglia of the rat, and its differential regulation.
    Neuroscience, 1997, Volume: 80, Issue:3

    Topics: Animals; Atropine; Carbachol; Cell Membrane; Dendrites; Exocytosis; Ganglia, Sympathetic; Male; Membrane Potentials; Nerve Endings; Neurons; Nicotine; Oxotremorine; Parasympatholytics; Pirenzepine; Potassium; Rats; Rats, Wistar; Receptors, Muscarinic; Regression Analysis; Synapses

1997
Site-directed mutagenesis on the m2 muscarinic acetylcholine receptor: the significance of Tyr403 in the binding of agonists and functional coupling.
    Molecular pharmacology, 1997, Volume: 52, Issue:6

    Topics: Acetylcholine; Animals; Binding Sites; Carbachol; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Mutagenesis, Site-Directed; Mutation; Oxotremorine; Receptor, Muscarinic M2; Receptors, Muscarinic; Tyrosine

1997
The relationship between agonist intrinsic activity and the rate of endocytosis of muscarinic receptors in a human neuroblastoma cell line.
    Molecular pharmacology, 1998, Volume: 53, Issue:4

    Topics: Arecoline; Bethanechol; Carbachol; Endocytosis; Humans; Kinetics; Ligands; Methacholine Chloride; Muscarinic Agonists; Neuroblastoma; Oxotremorine; Pilocarpine; Receptor, Muscarinic M3; Receptors, Muscarinic; Tumor Cells, Cultured

1998
Cholinergic mechanisms in the neurocontrol of the branchial heart of the cephalopod Sepia officinalis L.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1998, Volume: 119, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Branchial Region; Bungarotoxins; Carbachol; Dose-Response Relationship, Drug; Heart; Hexamethonium; Mollusca; Muscarine; Nicotine; Oxotremorine; Pilocarpine; Receptors, Cholinergic; Tetraethylammonium; Tubocurarine

1998
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
    Experimental neurology, 1998, Volume: 151, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon

1998
Comparison of the effects of M1 and M2 muscarinic receptor activation in the absence of GABAergic inhibition in immature rat hippocampal CA3 area.
    Brain research. Developmental brain research, 1998, May-15, Volume: 107, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Bicuculline; Carbachol; Dose-Response Relationship, Drug; Epilepsy; Evoked Potentials; GABA Antagonists; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Muscarinic Agonists; Oxotremorine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1998
Acetylcholine triggers L-glutamate exocytosis via nicotinic receptors and inhibits melatonin synthesis in rat pinealocytes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jul-01, Volume: 18, Issue:13

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Arylamine N-Acetyltransferase; Atropine; Bungarotoxins; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Carbachol; Cells, Cultured; Diltiazem; Exocytosis; Glutamic Acid; Melatonin; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Nifedipine; Nitrendipine; Oxotremorine; Parasympathetic Nervous System; Pineal Gland; Rats; Rats, Wistar; Receptors, Nicotinic; Scopolamine; Synaptic Vesicles; Tubocurarine

1998
Ionic mechanism of the slow afterdepolarization induced by muscarinic receptor activation in rat prefrontal cortex.
    Journal of neurophysiology, 1998, Volume: 80, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cesium; Chelating Agents; Egtazic Acid; Male; Membrane Potentials; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Patch-Clamp Techniques; Potassium; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Sodium; Vasodilator Agents

1998
Signaling mechanisms underlying muscarinic receptor-mediated increase in contraction rate in cultured heart cells.
    The Journal of biological chemistry, 1998, Nov-27, Volume: 273, Issue:48

    Topics: Animals; Animals, Newborn; Atropine; Base Sequence; Carbachol; Cells, Cultured; Estrenes; GTP-Binding Proteins; Heart; Heart Ventricles; Isoproterenol; Muscarinic Agonists; Myocardial Contraction; Myocardium; Oligodeoxyribonucleotides, Antisense; Oxotremorine; Phosphatidylinositols; Polymerase Chain Reaction; Propranolol; Protein Isoforms; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; RNA, Messenger; Transcription, Genetic

1998
Mutations of aspartate 103 in the Hm2 receptor and alterations in receptor binding properties of muscarinic agonists.
    Life sciences, 1995, Volume: 56, Issue:11-12

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Alanine; Amino Acid Substitution; Animals; Arecoline; Asparagine; Aspartic Acid; Carbachol; COS Cells; Muscarinic Agonists; Mutagenesis, Site-Directed; Oxotremorine; Pilocarpine; Receptor, Muscarinic M2; Receptors, Muscarinic; Transfection

1995
In vitro characterisation of the muscarinic receptor partial agonist, sabcomeline, in rat cortical and heart membranes.
    European journal of pharmacology, 1999, Apr-01, Volume: 370, Issue:1

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cell Membrane; Cells, Cultured; Cerebral Cortex; Drug Interactions; Heart; Imines; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth, Vascular; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Sprague-Dawley

1999
Distinct functional muscarinic receptors in guinea-pig gallbladder, ileum and atria.
    Pharmacological research, 1999, Volume: 39, Issue:5

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Carbachol; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Heart; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Oxotremorine; Rats; Rats, Wistar; Receptors, Muscarinic

1999
Lack of effect of McN-A-343 on membrane current and contraction in guinea pig ventricular myocytes.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adrenergic beta-Agonists; Animals; Calcium Channels; Calcium Channels, L-Type; Carbachol; Cell Membrane; Cyclic AMP; Electrophysiology; Guinea Pigs; Heart; Heart Ventricles; In Vitro Techniques; Isoproterenol; Muscarinic Agonists; Myocardial Contraction; Oxotremorine; Patch-Clamp Techniques; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptors, Muscarinic

1999
Reduced high-affinity agonist binding at the M(1) muscarinic receptor in Alzheimer's disease brain: differential sensitivity to agonists and divalent cations.
    Experimental neurology, 1999, Volume: 158, Issue:2

    Topics: Acetylcholine; Aged; Alzheimer Disease; Brain; Carbachol; Cations, Divalent; Chlorides; Edetic Acid; Female; Guanylyl Imidodiphosphate; Humans; Kinetics; Magnesium Chloride; Male; Manganese Compounds; Muscarinic Agonists; Oxotremorine; Pirenzepine; Receptor, Muscarinic M1; Receptors, Muscarinic; Reference Values

1999
Inhibitory cholinergic effects on the autonomously contractile bulbus cordis branchialis of the cephalopod Sepia officinalis L.
    General pharmacology, 1999, Volume: 33, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Bungarotoxins; Carbachol; Cholinergic Agents; Cholinergic Agonists; Cholinergic Antagonists; Female; Heart; Male; Mollusca; Muscarine; Myocardial Contraction; Nicotine; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate

1999
Muscarinic receptor heterogeneity in follicle-enclosed Xenopus oocytes.
    The Journal of physiology, 1999, Dec-01, Volume: 521 Pt 2

    Topics: Acetylcholine; Animals; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Follicle Stimulating Hormone; Gene Expression; Membrane Potentials; Muscarinic Antagonists; Oocytes; Ovarian Follicle; Oxotremorine; Patch-Clamp Techniques; Piperidines; Pirenzepine; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Transcription, Genetic; Tropicamide; Xenopus laevis

1999
A G protein gamma subunit-specific peptide inhibits muscarinic receptor signaling.
    The Journal of biological chemistry, 1999, Dec-10, Volume: 274, Issue:50

    Topics: Amino Acid Sequence; Animals; Brain; Calcium; Calcium Channels; Carbachol; Cattle; Cells, Cultured; CHO Cells; Clonidine; Cricetinae; Cytoplasm; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; In Vitro Techniques; N-Methylscopolamine; Neurons; Oxotremorine; Peptide Fragments; Receptor, Muscarinic M4; Receptors, Adrenergic, alpha-2; Receptors, Muscarinic; Receptors, Somatostatin; Signal Transduction; Spinal Cord; Superior Cervical Ganglion; Transfection

1999
Activation of muscle nicotinic acetylcholine receptor channels by nicotinic and muscarinic agonists.
    British journal of pharmacology, 1999, Volume: 128, Issue:7

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Humans; Ion Channels; Kinetics; Mice; Muscarine; Muscarinic Agonists; Muscle, Skeletal; Neurons; Nicotine; Nicotinic Agonists; Oxotremorine; Rats; Receptors, Nicotinic; Recombinant Proteins; Structure-Activity Relationship

1999
Carbachol and acetylcholine delay the early postdenervation depolarization of muscle fibres through M1-cholinergic receptors.
    Neuroscience research, 2000, Volume: 37, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Carbachol; Culture Techniques; Diaphragm; Male; Membrane Potentials; Muscarinic Agonists; Muscarinic Antagonists; Muscle Denervation; Muscle Fibers, Skeletal; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic

2000
Effects of microdialyzed oxotremorine, carbachol, epibatidine, and scopolamine on intraspinal release of acetylcholine in the rat.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:1

    Topics: Acetylcholine; Animals; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Male; Microdialysis; Oxotremorine; Pyridines; Rats; Rats, Sprague-Dawley; Scopolamine; Spinal Cord

2000
[Muscarinic receptors in the neostriatum--participation in the operant behavior regulation in dogs].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2000, Volume: 86, Issue:11

    Topics: Animals; Carbachol; Cognition; Conditioning, Operant; Dogs; Escape Reaction; Functional Laterality; Microinjections; Motor Activity; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Oxotremorine; Posture; Reaction Time; Receptors, Muscarinic; Scopolamine

2000
Coincident signalling between the Gi/Go-coupled delta-opioid receptor and the Gq-coupled m3 muscarinic receptor at the level of intracellular free calcium in SH-SY5Y cells.
    Journal of neurochemistry, 2001, Volume: 76, Issue:6

    Topics: Animals; Calcium; Carbachol; CHO Cells; Cricetinae; Enkephalin, D-Penicillamine (2,5)-; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; Humans; Kinetics; Neuroblastoma; Oxotremorine; Receptor Cross-Talk; Receptor, Muscarinic M3; Receptors, Muscarinic; Receptors, Opioid, delta; Transfection; Tumor Cells, Cultured

2001
Investigations into the physiological role of muscarinic M2 and M4 muscarinic and M4 receptor subtypes using receptor knockout mice.
    Life sciences, 2001, Apr-27, Volume: 68, Issue:22-23

    Topics: Animals; Carbachol; Cerebral Cortex; Heart; Heart Rate; Humans; Hypothermia; Male; Mice; Mice, Knockout; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Radioligand Assay; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Salivation; Tremor

2001
Pharmacological characterization of muscarinic receptors in mouse isolated urinary bladder smooth muscle.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Acetylcholine; Animals; Carbachol; Diamines; Dioxolanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pilocarpine; Piperidines; Receptors, Muscarinic; Urinary Bladder

2001
Effects of N-ethylmaleimide on conformational equilibria in purified cardiac muscarinic receptors.
    The Journal of biological chemistry, 2002, Sep-27, Volume: 277, Issue:39

    Topics: Animals; Blotting, Western; Carbachol; Cell Line; Enzyme Inhibitors; Ethylmaleimide; Humans; Insecta; Kinetics; Ligands; Models, Chemical; Muscarinic Agonists; N-Methylscopolamine; Oxotremorine; Parasympatholytics; Precipitin Tests; Protein Binding; Protein Conformation; Quinuclidinyl Benzilate; Receptor, Muscarinic M2; Receptors, Muscarinic; Sulfhydryl Reagents; Swine; Time Factors

2002
PMA decreases the proliferation of retinal cells in vitro: the involvement of acetylcholine and BDNF.
    Neurochemistry international, 2003, Volume: 42, Issue:1

    Topics: Acetylcholine; Alkaloids; Amacrine Cells; Animals; Atropine; Benzophenanthridines; Brain-Derived Neurotrophic Factor; Calcium; Carbachol; Cell Division; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Eye Proteins; Growth Inhibitors; Isoenzymes; MAP Kinase Signaling System; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Phenanthridines; Pirenzepine; Protein Kinase C; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Retina; Signal Transduction; Tetradecanoylphorbol Acetate

2003
Role of muscarinic receptors in the activation of the ventral subiculum and the consequences for dopamine release in the nucleus accumbens.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Animals; Atropine; Bicuculline; Bridged-Ring Compounds; Carbachol; Cholinergic Agonists; Diamines; Dopamine; Hippocampus; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nucleus Accumbens; Oxotremorine; Pilocarpine; Pyridines; Rats; Receptors, Muscarinic; Spiro Compounds; Thiadiazoles; Tropanes

2003
Cholinergic regulation of pericyte-containing retinal microvessels.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:6

    Topics: Acetylcholine; Animals; Calcium; Capillaries; Carbachol; Electric Stimulation; Fluorescent Dyes; Fura-2; Gap Junctions; In Vitro Techniques; Ion Channels; Membrane Potentials; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth, Vascular; Neurotransmitter Agents; Oxotremorine; Parasympathetic Nervous System; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Retinal Vessels; Signal Transduction

2003
A beta-induced TNF-alpha expression and acetylcholine action in mouse glial cells.
    Life sciences, 2003, Mar-28, Volume: 72, Issue:18-19

    Topics: Acetylcholine; Amyloid beta-Peptides; Animals; Carbachol; Cells, Cultured; Glyceraldehyde-3-Phosphate Dehydrogenases; Inflammation; Mice; Muscarinic Agonists; Neuroglia; Nicotine; Nicotinic Agonists; Oxotremorine; Peptide Fragments; Reverse Transcriptase Polymerase Chain Reaction; Tumor Necrosis Factor-alpha

2003
Receptor mechanisms mediating cyanide generation in PC12 cells and rat brain.
    Neuroscience research, 2004, Volume: 49, Issue:1

    Topics: Analysis of Variance; Animals; Atropine; Brain; Carbachol; Cells, Cultured; Cholinergic Agonists; Cyanides; Drug Interactions; Embryo, Mammalian; Hydromorphone; Morphine; Muscarinic Agonists; Muscarinic Antagonists; Naloxone; Narcotic Antagonists; Narcotics; Oxotremorine; PC12 Cells; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface

2004
Cholinergic regulation of the evoked quantal release at frog neuromuscular junction.
    The Journal of physiology, 2004, Oct-01, Volume: 560, Issue:Pt 1

    Topics: Acetylcholine; Action Potentials; Animals; Arecoline; Carbachol; Cholinergic Agonists; Diamines; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Neural Conduction; Neuromuscular Junction; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Parasympatholytics; Pirenzepine; Rana ridibunda; Receptors, Muscarinic; Synaptic Transmission; Tubocurarine

2004
Pharmacological profiles of an anticholinergic agent, phencynonate hydrochloride, and its optical isomers.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:5

    Topics: Animals; Aza Compounds; Binding, Competitive; Carbachol; Cerebral Cortex; Cholinergic Antagonists; Female; Glycolates; Guinea Pigs; Hypnotics and Sedatives; Male; Mice; Muscle Contraction; Oxotremorine; Pentobarbital; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Muscarinic; Salivation; Sleep; Stereoisomerism

2005
Differential effects on [35S]GTPgammaS binding using muscarinic agonists and antagonists in the gerbil brain.
    Journal of chemical neuroanatomy, 2005, Volume: 30, Issue:2-3

    Topics: Acetylcholine; Animals; Binding, Competitive; Brain; Brain Chemistry; Carbachol; Dose-Response Relationship, Drug; Gerbillinae; Guanosine 5'-O-(3-Thiotriphosphate); Male; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Radioligand Assay; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, G-Protein-Coupled; Receptors, Muscarinic; Sulfur Radioisotopes; Synaptic Transmission

2005
Comparative study on pharmacological effects of DM-phencynonate hydrochloride and its optical isomers.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:10

    Topics: Animals; Aza Compounds; Binding, Competitive; Carbachol; Cerebral Cortex; Female; Glycolates; Guinea Pigs; Male; Mice; Muscle Contraction; Oxotremorine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Wistar; Salivation; Stereoisomerism

2005
Regulation of Kv7 (KCNQ) K+ channel open probability by phosphatidylinositol 4,5-bisphosphate.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Oct-26, Volume: 25, Issue:43

    Topics: Animals; Carbachol; CHO Cells; Cholinergic Agonists; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Electric Stimulation; Extracellular Space; Green Fluorescent Proteins; Humans; Ion Channel Gating; KCNQ Potassium Channels; Membrane Potentials; Muscarinic Agonists; Oncogene Protein v-akt; Oxotremorine; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phospholipase C gamma; Phosphotransferases (Alcohol Group Acceptor); Probability; src-Family Kinases; Structure-Activity Relationship; Transfection

2005
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection

2007
An optical dynamic mass redistribution assay reveals biased signaling of dualsteric GPCR activators.
    Journal of receptor and signal transduction research, 2009, Volume: 29, Issue:3-4

    Topics: Acetylcholine; Animals; Atropine; Biosensing Techniques; Carbachol; Cell Line; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Drug Evaluation, Preclinical; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Receptors, G-Protein-Coupled; Signal Transduction

2009
Receptor-mediated suppression of potassium currents requires colocalization within lipid rafts.
    Molecular pharmacology, 2009, Volume: 76, Issue:6

    Topics: Animals; Blotting, Western; Calcium; Carbachol; Cell Line; Cholinergic Agents; Ganglia, Spinal; Humans; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Membrane Microdomains; Membrane Potentials; Mice; Muscarine; Oxotremorine; Phosphatidylinositol 4,5-Diphosphate; Potassium Channel Blockers; Potassium Channels; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Receptors, Muscarinic

2009
A simple method for quantifying functional selectivity and agonist bias.
    ACS chemical neuroscience, 2012, Mar-21, Volume: 3, Issue:3

    Topics: Animals; Carbachol; CHO Cells; Cricetinae; Cricetulus; Guinea Pigs; Ileum; Organ Culture Techniques; Oxotremorine; Receptors, Cytoplasmic and Nuclear

2012
Cholinergic regulation of epithelial sodium channels in rat alveolar type 2 epithelial cells.
    American journal of physiology. Lung cellular and molecular physiology, 2013, Mar-15, Volume: 304, Issue:6

    Topics: Alveolar Epithelial Cells; Amides; Animals; Atropine; Carbachol; Cells, Cultured; Enzyme Activation; Epithelial Sodium Channel Agonists; Epithelial Sodium Channels; Membrane Potentials; Mice; Mice, Inbred C57BL; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Oxotremorine; Patch-Clamp Techniques; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; rho-Associated Kinases; rhoA GTP-Binding Protein

2013
Cholinergic manipulations bidirectionally regulate object memory destabilization.
    Learning & memory (Cold Spring Harbor, N.Y.), 2015, Volume: 22, Issue:4

    Topics: Acetylcholine; Animals; Carbachol; Cerebral Cortex; Male; Muscarinic Agonists; Muscarinic Antagonists; Neuropsychological Tests; Oxotremorine; Rats, Long-Evans; Receptors, Muscarinic; Recognition, Psychology; Scopolamine

2015
Classical and atypical agonists activate M1 muscarinic acetylcholine receptors through common mechanisms.
    Pharmacological research, 2015, Volume: 97

    Topics: Animals; Binding Sites; Calcium; Carbachol; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Inositol Phosphates; Models, Molecular; Muscarinic Agonists; Mutation; Oxotremorine; Pyridines; Receptor, Muscarinic M1; Receptors, G-Protein-Coupled; Thiadiazoles

2015
Muscarinic modulation of M and h currents in gerbil spherical bushy cells.
    PloS one, 2020, Volume: 15, Issue:1

    Topics: Animals; Carbachol; Cholinergic Fibers; Cochlear Nucleus; Gerbillinae; Membrane Potentials; Muscarinic Agonists; Oxotremorine; Patch-Clamp Techniques; Receptors, Muscarinic

2020