Page last updated: 2024-08-17

carbachol and kn 62

carbachol has been researched along with kn 62 in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (66.67)18.2507
2000's3 (20.00)29.6817
2010's2 (13.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fox, LM; Funasaka, M; Goldenring, JR; Hidaka, H; Modlin, IM; Tsunoda, Y1
Easom, RA; Hidaka, H; Landt, M; Walters, SM; Wenham, RM1
Hinds, TR; Storm, DR; Wayman, GA1
Sanderson, MJ; Schweitzer, ES; Wasterlain, CG1
Itoh, M; Joh, T; Kato, T; Miyamoto, T; Moriyama, A; Okayama, N; Suzuki, T; Takeuchi, T1
Fukunaga, K; Izumi, F; Kuroiwa, A; Minami, K; Miyamoto, E; Nakashima, Y; Tsutsui, M; Yanagihara, N1
Benz, D; Möller, K; Perrin, D; Söling, HD1
Aronstam, RS; Puhl, HL; Raman, PS; Williams, CL1
Diener, M; Heinke, B; Ribeiro, R1
Jope, RS; Pacheco, MA1
Mikoshiba, K; Muto, Y; Nagao, T; Urushidani, T; Yamada, M1
Fährmann, M; Heinzmann, A; Seidler, U1
Dehaye, JP; Garcia-Marcos, M; Marino, A; Otto, A; Pochet, S; Seil, M1
Al-Qudah, M; Anderson, CD; Grider, JR; Kendig, DM; Mahavadi, S; Murthy, KS1
Carbonetto, S; Tremblay, M; Vezina-Audette, R1

Other Studies

15 other study(ies) available for carbachol and kn 62

ArticleYear
An inhibitor of Ca2+/calmodulin-dependent protein kinase II, KN-62, inhibits cholinergic-stimulated parietal cell secretion.
    The American journal of physiology, 1992, Volume: 262, Issue:1 Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Separation; Colforsin; Gastric Acid; Isoquinolines; Parasympathomimetics; Parietal Cells, Gastric; Piperazines; Protein Kinase Inhibitors; Protein Kinases

1992
Inhibition of insulin secretion by KN-62, a specific inhibitor of the multifunctional Ca2+/calmodulin-dependent protein kinase II.
    Biochemical and biophysical research communications, 1992, Nov-30, Volume: 189, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Line; Dose-Response Relationship, Drug; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Kinetics; Myosin-Light-Chain Kinase; Phosphorylation; Piperazines; Potassium; Protein Kinase C; Protein Kinase Inhibitors; Rats

1992
Hormone stimulation of type III adenylyl cyclase induces Ca2+ oscillations in HEK-293 cells.
    The Journal of biological chemistry, 1995, Oct-13, Volume: 270, Issue:41

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Calcium; Calcium Channels; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Line; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Glucagon; Humans; Inositol 1,4,5-Trisphosphate Receptors; Isoproterenol; Isoquinolines; Kidney; Kinetics; Models, Biological; Oscillometry; Phosphatidylinositols; Piperazines; Receptors, Cytoplasmic and Nuclear; Receptors, Glucagon; Signal Transduction; Time Factors

1995
Inhibition of regulated catecholamine secretion from PC12 cells by the Ca2+/calmodulin kinase II inhibitor KN-62.
    Journal of cell science, 1995, Volume: 108 ( Pt 7)

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Isoquinolines; Kinetics; Membrane Potentials; Norepinephrine; PC12 Cells; Piperazines; Protein Kinase C; Rats; Trifluoperazine

1995
Mediation of pepsinogen secretion from guinea pig chief cells by Ca2+/calmodulin-dependent protein kinase II.
    Biochimica et biophysica acta, 1995, Aug-31, Volume: 1268, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cells, Cultured; Gastric Mucosa; Guinea Pigs; Immunohistochemistry; Ionomycin; Isoquinolines; Male; Pepsinogens; Phosphorylation; Piperazines

1995
Ca(2+)/calmodulin-dependent protein kinase II inhibitor KN-62 inhibits adrenal medullary chromaffin cell functions independent of its action on the kinase.
    Journal of neurochemistry, 1996, Volume: 66, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adolescent; Adrenal Medulla; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Catecholamines; Cattle; Chromaffin System; Enzyme Inhibitors; Humans; Ion Channels; Isoquinolines; Nicotinic Agonists; Piperazines; Sodium; Tyrosine 3-Monooxygenase

1996
The role of protein kinase C in carbachol-induced and of cAMP-dependent protein kinase in isoproterenol-induced secretion in primary cultured guinea pig parotid acinar cells.
    The Biochemical journal, 1996, Feb-15, Volume: 314 ( Pt 1)

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amylases; Animals; Calcium; Carbachol; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Inhibitors; Exocytosis; Guinea Pigs; Immunoblotting; Isoproterenol; Isoquinolines; Male; Parotid Gland; Phorbol 12,13-Dibutyrate; Piperazines; Protein Binding; Protein Kinase C; Sulfonamides; Tetradecanoylphorbol Acetate

1996
Inhibition of M3 muscarinic acetylcholine receptor-mediated Ca2+ influx and intracellular Ca2+ mobilization in neuroblastoma cells by the Ca2+/calmodulin-dependent protein kinase inhibitor 1-[N,O-bis(5-isoquinolinesulfonyl)-N-methyl-L-trosyl]-4-phenylpipe
    Biochemical pharmacology, 1997, Apr-25, Volume: 53, Issue:8

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Enzyme Inhibitors; Humans; Neuroblastoma; Piperidines; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Tumor Cells, Cultured

1997
Involvement of calmodulin and protein kinase C in the regulation of K+ transport by carbachol across the rat distal colon.
    European journal of pharmacology, 1999, Jul-14, Volume: 377, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Carbachol; Cholinergic Agonists; Colon; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Ion Transport; Potassium; Protein Kinase C; Rats; Rats, Wistar; Rubidium Radioisotopes; Staurosporine

1999
Modulation of carbachol-stimulated AP-1 DNA binding activity by therapeutic agents for bipolar disorder in human neuroblastoma SH-SY5Y cells.
    Brain research. Molecular brain research, 1999, Oct-01, Volume: 72, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Antipsychotic Agents; Bipolar Disorder; Calcium; Calcium Signaling; Carbachol; Carbamazepine; Chelating Agents; DNA; Dose-Response Relationship, Drug; Edetic Acid; Egtazic Acid; Gene Expression Regulation; Humans; Indoles; Ionomycin; Ionophores; Lithium; Muscarinic Agonists; Nerve Tissue Proteins; Neuroblastoma; Neurons; Phosphatidylinositols; Protein Binding; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Tumor Cells, Cultured; Valproic Acid

1999
A proposed mechanism for the potentiation of cAMP-mediated acid secretion by carbachol.
    American journal of physiology. Cell physiology, 2001, Volume: 280, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Aminopyrine; Animals; Bucladesine; Calcium; Calcium Channels; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbon Radioisotopes; Cyclic AMP; Cytochalasin D; Cytoskeleton; Drug Interactions; Enzyme Inhibitors; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate Receptors; Maleimides; Parietal Cells, Gastric; Protein Kinase C; Rabbits; Receptors, Cytoplasmic and Nuclear; Stomach

2001
CaMKII is activated and translocated to the secretory apical membrane during cholinergically conveyed gastric acid secretion.
    Cellular signalling, 2002, Volume: 14, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aminopyrine; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Membrane; Cell Polarity; Cells, Cultured; Cholinergic Agonists; Dose-Response Relationship, Drug; Enzyme Activation; Gastric Acid; H(+)-K(+)-Exchanging ATPase; Male; Parietal Cells, Gastric; Protein Transport; Rabbits; Rats; Rats, Wistar; Secretory Vesicles

2002
Contribution of two ionotropic purinergic receptors to ATP responses in submandibular gland ductal cells.
    Cellular signalling, 2007, Volume: 19, Issue:10

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Biological Transport; Calcium; Carbachol; Ethidium; Interleukin-1beta; Mice; Mice, Knockout; Phospholipases A2; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Receptors, Purinergic P2X7; Saliva; Submandibular Gland

2007
Role of various kinases in muscarinic M3 receptor-mediated contraction of longitudinal muscle of rat colon.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2014, Volume: 50

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Benzimidazoles; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Carbachol; Cholinergic Neurons; Colon; Enzyme Inhibitors; In Vitro Techniques; Mitogen-Activated Protein Kinase 3; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Myosin-Light-Chain Kinase; Naphthalimides; Peptide Fragments; Pyridines; Rats, Sprague-Dawley; Receptor, Muscarinic M3; rho-Associated Kinases

2014
Laminin is instructive and calmodulin dependent kinase II is non-permissive for the formation of complex aggregates of acetylcholine receptors on myotubes in culture.
    Matrix biology : journal of the International Society for Matrix Biology, 2017, Volume: 57-58

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Agrin; Animals; Benzoquinones; Bungarotoxins; Calcium Channel Blockers; Calcium Channels; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Carbachol; Cell Line; Gene Expression; Lactams, Macrocyclic; Laminin; Mice; Muscle Fibers, Skeletal; Muscle Proteins; Protein Aggregates; Receptors, Cholinergic; Sodium Channel Blockers; Sodium Channels; Staining and Labeling; Tetrodotoxin; Verapamil

2017