carbachol has been researched along with guanylyl imidodiphosphate in 94 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 54 (57.45) | 18.7374 |
1990's | 39 (41.49) | 18.2507 |
2000's | 1 (1.06) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Gardner, JD; Robberecht, P; Uhlemann, ER | 1 |
Berrie, CP; Birdsall, NJ; Burgen, AS; Hulme, EC | 1 |
Boyd, RS; Donnelly, LE; MacDermot, J | 1 |
Bangert, M; Beyer, T; Niroomand, F; Rauch, B | 1 |
Hatta, S; Ohshika, H | 1 |
Nathanson, NM; van Koppen, CJ | 1 |
Baker, HJ; Claro, E; Fain, JN; Nair, BG; Patel, TB; Shanker, G; Wallace, MA | 1 |
Golly, F; Larocca, JN; Ledeen, RW | 1 |
Allen, RA; Colvin, RA; Oibo, JA | 1 |
Fermum, R; Kosche, D; Möritz, KU | 1 |
Milligan, G; Nair, BG; Parikh, B; Patel, TB | 1 |
Hung, WC; Wei, JW | 1 |
Bonner, TI; Brann, MR; Dörje, F; Wess, J | 1 |
Dawson, RM; Poretski, M | 1 |
Minton, AP; Sokolovsky, M | 1 |
Dwyer, TM; Farley, JM; Ho, IK; Mohan, PM; Yang, CM | 1 |
Hoffman, BB; Thomas, JM | 1 |
Cohen-Armon, M; Sokolovsky, M | 1 |
Aronstam, RS; Carrier, GO | 1 |
Cohen-Armon, M; Henis, YI; Kloog, Y; Sokolovsky, M | 1 |
Flynn, DD; Palermo, N; Suarez, A | 1 |
Allen, IS; Gaa, ST; Rogers, TB | 1 |
Hattori, Y; Kanno, M; Nakao, Y; Sakuma, I | 1 |
Jagadeesh, G; Phan, NT; Sulakhe, PV | 1 |
Merritt, JE; Putney, JW; Rubin, RP; Taylor, CW | 1 |
Barnes, PJ; Cuss, FM; Grandordy, BM; Palmer, JB; Sampson, AS | 1 |
Anthony, BL; Aronstam, RS | 2 |
Flynn, DD; Potter, LT | 1 |
Hunter, DD; Nathanson, NM | 2 |
Mei, L; Roeske, WR; Wang, JX; Yamamura, HI | 1 |
Aronstam, RS; Narayanan, TK | 1 |
Milnor, WR; Sastre, A | 1 |
Henis, YI; Moscona-Amir, E; Sokolovsky, M | 1 |
Bertrand, C; Gies, JP; Landry, Y | 1 |
Dwyer, TM; Farley, JM; Mohan, PM; Yang, CM | 1 |
Chung, FZ; Lai, J; Mei, L; Roeske, WR; Venter, JC; Yamamura, HI | 1 |
Brown, JH; Orellana, S; Solski, PA | 1 |
Aguilar, JS; De Robertis, E; Ochoa, EL | 1 |
Gies, JP; Ilien, B; Landry, Y | 1 |
Hjalmarson, A; Jacobsson, B; Ransnäs, L; Sabler, E | 1 |
Green, RD; Hosey, MM; Kwatra, MM; Leung, E; Maan, AC; McMahon, KK; Ptasienski, J | 1 |
Aguilar, JS; De Robertis, E; Fonseca, MI | 1 |
Adam, LP; Pappano, AJ; Sorota, S | 1 |
Roeske, WR; Watson, M; Yamamura, HI | 1 |
Kagiya, T; Mizushima, A; Uchida, S; Yoshida, H | 1 |
Baker, SP; Posner, P | 1 |
Barenholz, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M; Yechiel, E | 1 |
Bering, B; Müller, WE | 1 |
Bloom, JW; Halonen, M; Lawrence, LJ; Rould, E; Seaver, NA; Yamamura, HI | 1 |
Bruni, P; Hewlett, EL; Moss, J | 1 |
Baker, SP; Marchand, S; Nelson, CA; O'Neil, E; Posner, P | 1 |
Kloog, Y; Sokolovsky, M | 1 |
Koike, K; Okumura, K; Takayanagi, I | 1 |
Higuchi, H; Kagiya, T; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H; Zhou, XM | 1 |
Howlett, AC | 1 |
Burgoyne, RD | 1 |
Aronstam, RS; Greenbaum, LM | 1 |
Bergh, CH; Hjalmarson, A; Jacobsson, B; Ransnäs, L; Waldenström, A | 1 |
Halvorsen, SW; Nathanson, NM | 2 |
Nathanson, NM | 1 |
Aronstam, RS; Kirby, ML | 1 |
Higuchi, H; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H | 1 |
Higuchi, H; Matsumoto, K; Mizushima, A; Uchida, S; Yoshida, H | 1 |
Bárány, E; Berrie, CP; Birdsall, NJ; Burgen, AS; Hulme, EC | 1 |
Dziekan, LC; Galper, JB; O'Hara, DS; Smith, TW | 1 |
Leppik, R; van Giersbergen, PL | 1 |
Coy, DH; Gu, ZF; Jensen, RT; Pradhan, TK | 1 |
Andrade, R | 1 |
Hescheler, J | 1 |
Yatani, A | 1 |
Abe, H; Chihara, K; Kaji, H; Okimura, Y; Tai, S | 1 |
Honda, K; Kamiya, H; Takano, Y | 1 |
Young, JM; Young, KW | 1 |
Feng, QP; Fu, LX; Hedner, T; Hjalmarson, A; Hoebeke, J; Liang, QM; Sun, XY | 1 |
Joyner, RW; Kumar, R; Osaka, T | 1 |
Hishinuma, S; Kurokawa, M; Matsumoto, Y; Uchida, MK | 1 |
Consolo, S; Garcia Ruiz, AJ; La Porta, C; Ladinsky, H; Zambelli, M | 1 |
Alafuzoff, I; Nordberg, A; Warpman, U | 1 |
Jakobs, KH; Mura, R; Niroomand, F; Piacentini, L | 1 |
Baker, SP; Belardinelli, L; Ruble, J; Scammells, PJ; Shryock, JC; Srinivas, M | 1 |
Kübler, W; Mura, RA; Niroomand, F; Piacentini, L; Rauch, B; Zeifang, F | 1 |
Ballard, C; Schaffer, S | 1 |
Avissar, S; Schreiber, G | 1 |
Chien, CC; Pasternak, GW; Ryan-Moro, J; Standifer, KM | 1 |
Spindler, KD; Spindler-Barth, M; Wegener, S | 1 |
Chidiac, P; Green, MA; Wells, JW | 1 |
Avissar, S; Nechamkin, Y; Roitman, G; Schreiber, G | 1 |
Gao, Y; Kunapuli, SP; Ravindra, R; Singh, SP | 2 |
Ladner, CJ; Lee, JM | 1 |
Lee, JM; Mariyappa, R; Muma, NA; Williams, K | 1 |
94 other study(ies) available for carbachol and guanylyl imidodiphosphate
Article | Year |
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Effects of alcohols on the actions of VIP and secretin on acinar cells from guinea pig pancreas.
Topics: 1-Propanol; Adenylyl Cyclases; Alcohols; Amylases; Animals; Carbachol; Cholecystokinin; Cyclic AMP; Ethanol; Gastrointestinal Hormones; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Male; Methanol; Octanols; Pancreas; Secretin; Vasoactive Intestinal Peptide | 1979 |
Guanine nucleotides modulate muscarinic receptor binding in the heart.
Topics: Animals; Carbachol; Guanine Nucleotides; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Myocardium; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Ribonucleotides; Scopolamine Derivatives | 1979 |
Opiate-dependent changes in the sensitivity of adenylate cyclase to stimulatory agonists and 5'-guanylylimidodiphosphate are independent of G protein abundance and eukaryotic ADP-ribosyltransferase activity in NG108-15 cells.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Drug Combinations; Enkephalin, Leucine-2-Alanine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immunoblotting; Niacinamide; Poly(ADP-ribose) Polymerases; Tumor Cells, Cultured | 1992 |
Reduced adenylyl cyclase inhibition by carbachol and GTP during acute myocardial ischaemia.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Colforsin; Coronary Disease; Dogs; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Receptors, Muscarinic | 1992 |
Stable inhibition of adenylate cyclase by muscarinic agonist in rat parotid gland: effects of neomycin and pertussis toxin.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Methoxamine; Neomycin; Parotid Gland; Pertussis Toxin; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic; Virulence Factors, Bordetella | 1991 |
The cysteine residue in the carboxyl-terminal domain of the m2 muscarinic acetylcholine receptor is not required for receptor-mediated inhibition of adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; Cell Line; Cyclic AMP; Cysteine; Guanylyl Imidodiphosphate; Muscarinic Antagonists; Quinuclidinyl Benzilate; Receptors, Muscarinic; Subcellular Fractions; Tissue Distribution | 1991 |
Altered phosphoinositide-specific phospholipase C and adenylyl cyclase in brain cortical membranes of cats with GM1 and GM2 gangliosidosis.
Topics: Adenylyl Cyclases; Aluminum; Aluminum Chloride; Aluminum Compounds; Animals; Calcium; Carbachol; Cat Diseases; Cats; Cell Membrane; Cerebral Cortex; Chlorides; Colforsin; G(M1) Ganglioside; Gangliosidoses; Gangliosidosis, GM1; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Kinetics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Phosphoric Diester Hydrolases; Reference Values; Sodium Fluoride | 1991 |
Phosphoinositide breakdown in isolated myelin is stimulated by GTP analogues and calcium.
Topics: Animals; Calcium; Carbachol; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Inositol Phosphates; Myelin Proteins; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Second Messenger Systems | 1990 |
Calcium inhibition of cardiac adenylyl cyclase. Evidence for two distinct sites of inhibition.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Calmodulin; Carbachol; Colforsin; Dogs; Enzyme Activation; Guanylyl Imidodiphosphate; Magnesium; Myocardium; Pertussis Toxin; Sarcolemma; Virulence Factors, Bordetella | 1991 |
Membrane-associated signal transduction modulates contractile responses to Ca2+ in saponin-skinned coronary smooth muscle.
Topics: Aluminum; Animals; Calcium; Carbachol; Cattle; Coronary Vessels; Female; Fluorides; Guanylyl Imidodiphosphate; Histamine; In Vitro Techniques; Male; Membranes; Permeability; Phorbol 12,13-Dibutyrate; Saponins; Signal Transduction; Swine; Vasoconstriction | 1991 |
Gs alpha mediates epidermal growth factor-elicited stimulation of rat cardiac adenylate cyclase.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antibodies; Carbachol; Colforsin; Epidermal Growth Factor; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immune Sera; Isoproterenol; Kinetics; Male; Membrane Proteins; Molecular Sequence Data; Molecular Weight; Myocardium; Oligopeptides; Phenylisopropyladenosine; Rats; Rats, Inbred Strains | 1990 |
Guanine nucleotides have a direct inhibitory effect on polyphosphoinositide turnover in rat cortical synaptosomes.
Topics: Animals; Carbachol; Cerebral Cortex; GTP-Binding Proteins; Guanine Nucleotides; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Phosphates; Phosphatidic Acids; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Phosphatidylinositols; Rats; Rats, Inbred Strains; Synaptosomes | 1990 |
Delineation of muscarinic receptor domains conferring selectivity of coupling to guanine nucleotide-binding proteins and second messengers.
Topics: Adenylate Cyclase Toxin; Animals; Carbachol; Cyclic AMP; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Mice; N-Methylscopolamine; Pertussis Toxin; Phosphatidylinositols; Receptors, Muscarinic; Scopolamine Derivatives; Second Messenger Systems; Virulence Factors, Bordetella | 1990 |
Opposing effects of N-ethylmaleimide on the affinity of carbachol for muscarinic cholinoceptors of guinea-pig atrium.
Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; Guinea Pigs; Heart Atria; Premedication; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Temperature | 1990 |
A model for the interaction of muscarinic receptors, agonists, and two distinct effector substances.
Topics: Aging; Animals; Batrachotoxins; Carbachol; Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Models, Biological; Myocardium; Pertussis Toxin; Rats; Receptors, Muscarinic; Virulence Factors, Bordetella | 1990 |
Down-regulation of muscarinic receptors in the striatum of organophosphate-treated swine.
Topics: Acetylcholinesterase; Animals; Binding Sites; Binding, Competitive; Carbachol; Corpus Striatum; Down-Regulation; Guanylyl Imidodiphosphate; Isoflurophate; Magnesium; Male; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Regression Analysis; Swine | 1990 |
Agonist-induced down-regulation of muscarinic cholinergic and alpha 2-adrenergic receptors after inactivation of Ni by pertussis toxin.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Alprostadil; Animals; ATPase Inhibitory Protein; Carbachol; Cell Line; Cyclic AMP; Electrophoresis, Polyacrylamide Gel; Epinephrine; Glioma; Guanylyl Imidodiphosphate; Molecular Weight; NAD; Neuroblastoma; Pertussis Toxin; Proteins; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Virulence Factors, Bordetella; Yohimbine | 1986 |
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine | 1986 |
Insulin prevention of altered muscarinic receptor-G protein coupling in diabetic rat atria.
Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Carbachol; Diabetes Mellitus, Experimental; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Insulin; Kinetics; Male; Myocardium; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Reference Values | 1989 |
Batrachotoxin changes the properties of the muscarinic receptor in rat brain and heart: possible interaction(s) between muscarinic receptors and sodium channels.
Topics: Aconitine; Animals; Batrachotoxins; Benzilates; Binding, Competitive; Brain; Carbachol; Guanylyl Imidodiphosphate; Ion Channels; Kinetics; Macromolecular Substances; Male; Myocardium; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine | 1985 |
Agonist binding to M1 muscarinic receptors is sensitive to guanine nucleotides.
Topics: Animals; Carbachol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Indicators and Reagents; Kinetics; Male; Methacholine Compounds; Oxotremorine; Pilocarpine; Pirenzepine; Rabbits; Receptors, Muscarinic; Second Messenger Systems | 1989 |
Changes in expression of a functional Gi protein in cultured rat heart cells.
Topics: Angiotensin II; Animals; Carbachol; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Myocardium; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1988 |
Pharmacological analysis of the cardiac actions of xamoterol, a beta adrenoceptor antagonist with partial agonistic activity, in guinea pig heart: evidence for involvement of adenylate cyclase system in its cardiac stimulant actions.
Topics: Adenosine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cyclic AMP; Dose-Response Relationship, Drug; Female; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Rate; Iodocyanopindolol; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Xamoterol | 1987 |
Comparison of cholinergic inhibition and beta-adrenergic stimulation of adenylate cyclase from rat and guinea-pig hearts: effects of guanine nucleotides and monovalent cations.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Cations, Monovalent; Chlorides; Colforsin; Cytosol; Enzyme Activation; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Lithium; Lithium Chloride; Male; Myocardium; Rats; Rats, Inbred Strains; Sodium; Sodium Chloride; Sodium Fluoride; Tissue Distribution | 1985 |
A guanine nucleotide-dependent regulatory protein couples substance P receptors to phospholipase C in rat parotid gland.
Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Epinephrine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Monophosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Inositol Phosphates; Male; Parotid Gland; Propranolol; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Sodium Fluoride; Thionucleotides; Type C Phospholipases | 1986 |
Phosphatidylinositol response to cholinergic agonists in airway smooth muscle: relationship to contraction and muscarinic receptor occupancy.
Topics: Acetylcholine; Animals; Atropine; Benzodiazepinones; Carbachol; Cattle; Chlorides; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Lithium; Lithium Chloride; Membrane Lipids; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Respiratory System; Trachea | 1986 |
Effect of pH on muscarinic acetylcholine receptors from rat brainstem.
Topics: Animals; Brain Stem; Carbachol; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Male; Mathematics; N-Methylscopolamine; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Scopolamine Derivatives; Temperature; Time Factors | 1986 |
Effect of solubilization on the distinct binding properties of muscarine receptors from rabbit hippocampus and brainstem.
Topics: Animals; Brain Stem; Carbachol; Edetic Acid; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; In Vitro Techniques; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Solubility | 1986 |
Biochemical and physical analyses of newly synthesized muscarinic acetylcholine receptors in cultured embryonic chicken cardiac cells.
Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Cell Membrane Permeability; Chick Embryo; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart; Isoelectric Point; Kinetics; Molecular Weight; Myocardium; Potassium; Receptors, Muscarinic | 1986 |
Solubilization with digitonin alters the kinetics of pirenzepine binding to muscarinic receptors from rat forebrain and heart.
Topics: Animals; Brain; Carbachol; Digitonin; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Myocardium; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Solubility | 1987 |
Temperature effect on the detection of muscarinic receptor-G protein interactions in ligand binding assays.
Topics: Animals; Brain Stem; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Myocardium; Oxotremorine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Temperature | 1988 |
Cholinergic receptors and contraction of smooth muscle in canine portal vein.
Topics: Algorithms; Animals; Calcimycin; Carbachol; Dogs; Guanylyl Imidodiphosphate; Kinetics; Muscle Contraction; Muscle, Smooth; Norepinephrine; Portal Vein; Quinuclidinyl Benzilate; Receptors, Cholinergic | 1988 |
Guanosine 5'-triphosphate binding protein (Gi) and two additional pertussis toxin substrates associated with muscarinic receptors in rat heart myocytes: characterization and age dependency.
Topics: Adenosine Diphosphate Ribose; Aging; Animals; Carbachol; Cells, Cultured; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Liposomes; Molecular Weight; Myocardium; Pertussis Toxin; Rats; Receptors, Muscarinic; Virulence Factors, Bordetella | 1988 |
Membrane phospholipid polar heads influence the coupling of M2 muscarinic receptors to G proteins.
Topics: Animals; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Membrane Proteins; Myocardium; Oxotremorine; Phospholipids; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Type C Phospholipases | 1988 |
Changes in affinity states during down-regulation of muscarinic receptors in tracheal smooth muscle of organophosphate-treated swine.
Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoflurophate; Magnesium; Male; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine; Trachea | 1988 |
The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells.
Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Line; Cell Membrane; DNA, Recombinant; Fibroblasts; Guanylyl Imidodiphosphate; Hydrolysis; Mice; Muscarine; Nucleic Acid Hybridization; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Recombinant Proteins; Sequence Homology, Nucleic Acid; Transfection | 1988 |
Guanosine 5'-O-(thiotriphosphate)-dependent inositol trisphosphate formation in membranes is inhibited by phorbol ester and protein kinase C.
Topics: Bradykinin; Carbachol; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Histamine; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Kinetics; Membranes; Phorbol Esters; Protein Kinase C; Quinuclidinyl Benzilate; Receptors, Muscarinic; Sugar Phosphates; Tetradecanoylphorbol Acetate; Thionucleotides | 1987 |
Reconstitution of solubilized atrial cholinergic muscarinic receptors in liposomes.
Topics: Animals; Binding, Competitive; Carbachol; Cattle; Glycine max; Guanylyl Imidodiphosphate; Heart Atria; Kinetics; Liposomes; Myocardium; N-Methylscopolamine; Phosphatidylcholines; Receptors, Muscarinic; Scopolamine Derivatives; Solubility | 1987 |
Temperature-dependence and heterogeneity of muscarinic agonist and antagonist binding.
Topics: Animals; Atropine; Brain; Carbachol; Guanylyl Imidodiphosphate; Kinetics; Lung; Male; Myocardium; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Temperature | 1987 |
Effect of corticosteroids on muscarinic receptors on cultured myocardial cells.
Topics: Animals; Binding, Competitive; Carbachol; Cell Membrane; Cells, Cultured; Female; Guanylyl Imidodiphosphate; Hydrocortisone; In Vitro Techniques; Manganese; Myocardium; Phosphatidylinositols; Puromycin; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1987 |
Correlation of agonist-induced phosphorylation of chick heart muscarinic receptors with receptor desensitization.
Topics: Animals; Atropine; Carbachol; Chickens; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Heart; Magnesium; Myocardium; Oxotremorine; Phosphorylation; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1987 |
Pertussis vaccine reduces agonist binding to the rat heart muscarinic receptor and its guanine nucleotide modulation.
Topics: Animals; Carbachol; Cell Membrane; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Myocardium; Pertussis Vaccine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic | 1986 |
High-affinity agonist binding to rat brainstem muscarinic receptors is eliminated by low pH.
Topics: Animals; Brain Stem; Carbachol; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine | 1986 |
Comparison of muscarinic receptor properties in hatched chick heart atrium and ventricle.
Topics: Animals; Atropine; Benzodiazepinones; Carbachol; Chickens; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Pirenzepine; Potassium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium | 1986 |
[3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. I. Characterization and regulation of agonist binding to putative muscarinic subtypes.
Topics: Acetylcholine; Animals; Benzodiazepinones; Buffers; Carbachol; Cerebral Cortex; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Myocardium; Parasympathomimetics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1986 |
Alterations in muscarinic receptors of ventricular muscle in carbachol-induced short-term desensitization.
Topics: Animals; Carbachol; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Ventricles; Myocardial Contraction; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1986 |
Irreversible binding of acetylethylcholine mustard to cardiac cholinergic muscarinic receptors.
Topics: Acetylcholine; Animals; Atropine; Carbachol; Cell Membrane; Guanylyl Imidodiphosphate; Heart Rate; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives | 1986 |
Role of lipids in age-related changes in the properties of muscarinic receptors in cultured rat heart myocytes.
Topics: Acetylcholine; Animals; Animals, Newborn; Benzilates; Carbachol; Cells, Cultured; Guanylyl Imidodiphosphate; Kinetics; Liposomes; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic | 1986 |
Stereospecific 3H-QNB binding to human erythrocyte membranes associated with muscarinic cholinergic receptors.
Topics: Adult; Aging; Animals; Atropine; Brain; Carbachol; Erythrocyte Membrane; Female; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Male; Middle Aged; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism | 1987 |
Characterization of high affinity [3H]pirenzepine and (-)-[3H] quinuclidinyl benzilate binding to muscarinic cholinergic receptors in rabbit peripheral lung.
Topics: Animals; Binding, Competitive; Carbachol; Female; Guanylyl Imidodiphosphate; Kinetics; Lung; Male; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Stereoisomerism | 1987 |
Effects of pertussis toxin-catalyzed ADP-ribosylation on interactions of transducin and the inhibitory GTP-binding protein of adenylate cyclase with guanyl nucleotides.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Atropine; Bacterial Toxins; Carbachol; Cell Line; Cell Membrane; Enkephalin, Methionine; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Membrane Proteins; Naloxone; Norepinephrine; Nucleoside Diphosphate Sugars; Pertussis Toxin; Phentolamine; Transducin; Virulence Factors, Bordetella | 1985 |
Age-related changes in cardiac muscarinic receptors: decreased ability of the receptor to form a high affinity agonist binding state.
Topics: Aging; Animals; Body Weight; Carbachol; Guanylyl Imidodiphosphate; Heart; Male; Myocardium; Organ Size; Quinuclidinyl Benzilate; Rats; Rats, Inbred F344; Receptors, Cholinergic; Receptors, Muscarinic | 1985 |
Allosteric interactions between muscarinic agonist binding sites and effector sites demonstrated by the use of bisquaternary pyridinium oximes.
Topics: Animals; Brain Stem; Carbachol; Cerebral Cortex; Cobalt; Guanylyl Imidodiphosphate; In Vitro Techniques; Oximes; Oxotremorine; Parasympathomimetics; Pyridinium Compounds; Rats; Receptors, Muscarinic | 1985 |
Interaction of muscarinic drugs with their receptor.
Topics: Animals; Atropine; Carbachol; Guanylyl Imidodiphosphate; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Microsomes; Muscle, Smooth; Parasympathomimetics; Quaternary Ammonium Compounds; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1985 |
Multiple agonist binding sites of muscarinic acetylcholine receptors and their relation to the negative inotropic action of agonists in guinea-pig heart.
Topics: Animals; Binding Sites; Carbachol; Depression, Chemical; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Myocardial Contraction; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1985 |
Inhibition of neuroblastoma adenylate cyclase by cannabinoid and nantradol compounds.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclase Inhibitors; Alprostadil; Animals; Carbachol; Cell Line; Cyclic AMP; Dronabinol; Epoprostenol; Guanylyl Imidodiphosphate; Neuroblastoma; Phenanthridines; Phosphodiesterase Inhibitors; Prostaglandins E; Secretin; Sodium Fluoride | 1984 |
Regulation of the muscarinic acetylcholine receptor: effects of phosphorylating conditions on agonist and antagonist binding.
Topics: Animals; Brain; Calcium-Binding Proteins; Calmodulin; Carbachol; Cerebral Cortex; Cyclic AMP; Guanylyl Imidodiphosphate; Phosphorylation; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Synaptic Membranes | 1983 |
Guanine nucleotide sensitivity of muscarinic acetylcholine receptors from rat brainstem is eliminated by endogenous proteolytic activity.
Topics: Animals; Brain Stem; Carbachol; Endopeptidases; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Protease Inhibitors; Rats; Receptors, Muscarinic | 1984 |
Effects of acute ketotic and non-ketotic diabetes on the myocardial muscarinic receptors.
Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; Computers; Diabetes Mellitus, Experimental; Diabetic Ketoacidosis; Guanylyl Imidodiphosphate; Insulin; Male; Models, Biological; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1984 |
Ontogenesis of physiological responsiveness and guanine nucleotide sensitivity of cardiac muscarinic receptors during chick embryonic development.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atrial Function; Bacterial Toxins; Carbachol; Chick Embryo; Depression, Chemical; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart; Heart Rate; Isoproterenol; Myocardium; Pertussis Toxin; Quinuclidinyl Benzilate; Receptors, Muscarinic; Virulence Factors, Bordetella | 1984 |
Decreased physiological sensitivity mediated by newly synthesized muscarinic acetylcholine receptors in embryonic chicken heart.
Topics: Adenylyl Cyclase Inhibitors; Animals; Atropine; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Rate; Protein Processing, Post-Translational; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1984 |
Binding of agonists and antagonists to muscarinic acetylcholine receptors on intact cultured heart cells.
Topics: Animals; Binding, Competitive; Carbachol; Cells, Cultured; Chick Embryo; Guanylyl Imidodiphosphate; Kinetics; Myocardium; N-Methylscopolamine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Scopolamine Derivatives | 1983 |
Atropine-induced alterations of normal development of muscarinic receptors in the embryonic chick heart.
Topics: Animals; Atropine; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Atria; Heart Ventricles; Myocardium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Time Factors | 1983 |
Effects of guanine nucleotide and sulfhydryl reagent on subpopulations of muscarinic acetylcholine receptors in mammalian hearts: possible evidence for interconversion of super-high and low affinity agonist binding sites.
Topics: Animals; Carbachol; Dogs; Guanine Nucleotides; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Membranes; Myocardium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Sulfhydryl Reagents; Temperature | 1984 |
Effect of urea-treatment on agonist binding affinity of the muscarinic acetylcholine receptor.
Topics: Animals; Atropine; Binding, Competitive; Carbachol; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Male; Microsomes; Myocardium; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Urea | 1983 |
The binding properties of the muscarinic receptors of the cynomolgus monkey ciliary body and the response to the induction of agonist subsensitivity.
Topics: Animals; Benzodiazepinones; Carbachol; Ciliary Body; Guanylyl Imidodiphosphate; Kinetics; Macaca fascicularis; N-Methylscopolamine; Pilocarpine; Pirenzepine; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives | 1982 |
The biphasic response of muscarinic cholinergic receptors in cultured heart cells to agonists. Effects on receptor number and affinity in intact cells and homogenates.
Topics: Animals; Carbachol; Cell Membrane; Cells, Cultured; Chick Embryo; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Myocardium; N-Methylscopolamine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives | 1982 |
In vivo regulation of muscarinic acetylcholine receptor number and function in embryonic chick heart.
Topics: Animals; Binding, Competitive; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Rate; Kinetics; Mathematics; Myocardium; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic | 1981 |
Modulation of agonist binding by guanine nucleotides in CHO cells expressing muscarinic m1-m5 receptors.
Topics: Animals; Atropine; Carbachol; CHO Cells; Cricetinae; Guanine Nucleotides; Guanylyl Imidodiphosphate; Humans; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Parasympatholytics; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives | 1995 |
Smooth muscle cells from guinea pig stomach possess high-affinity galanin receptors that mediate relaxation.
Topics: Animals; Carbachol; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Galanin; Gastric Mucosa; Guanylyl Imidodiphosphate; Guinea Pigs; Kinetics; Male; Muscle Relaxation; Muscle, Smooth; Neuropeptides; Peptides; Protein Precursors; Rats; Receptors, Galanin; Receptors, Gastrointestinal Hormone; Stomach; Swine; Time Factors; Vasoactive Intestinal Peptide | 1994 |
Infusion of guanine nucleotides through recording electrodes for studies on G-protein regulation of ion currents and channels.
Topics: Animals; Baclofen; Carbachol; Electrophysiology; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hippocampus; Ion Channels; Membrane Potentials; Microelectrodes; Pyramidal Cells; Rats; Serotonin; Thionucleotides | 1994 |
Whole-cell clamp analysis for G-protein regulation of channels.
Topics: Adenosine Diphosphate Ribose; Animals; Calcium Channels; Carbachol; Cholera Toxin; Electrophysiology; Epinephrine; Glioma; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Homeostasis; Hybrid Cells; Ion Channels; Macromolecular Substances; Neuroblastoma; Oligonucleotides, Antisense; Patch-Clamp Techniques; PC12 Cells; Potassium Channels; Rats; RNA, Messenger; Virulence Factors, Bordetella | 1994 |
Reconstitution of receptor-regulated ion channels in isolated patch membrane.
Topics: Acetylcholine; Animals; Carbachol; Cell Membrane; Electrophysiology; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels; Receptors, Muscarinic; Virulence Factors, Bordetella | 1994 |
Neurokinin receptor antagonists inhibit the binding of growth hormone-releasing peptide to EP-1 human neuroblastoma cells.
Topics: Alprostadil; Animals; Atropine; Carbachol; Cell Line; Growth Hormone-Releasing Hormone; Guanylyl Imidodiphosphate; HeLa Cells; Humans; Hypothalamus; Kinetics; Neuroblastoma; Neuropeptides; Oligopeptides; Pituitary Gland; Rats; Receptors, Tachykinin; Structure-Activity Relationship; Tumor Cells, Cultured | 1995 |
The mechanism of muscarinic agonist-stimulated inositol phosphate formation in permeabilized ileal smooth muscle.
Topics: Acetylcholine; Animals; Calcium; Carbachol; Dose-Response Relationship, Drug; Drug Synergism; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Substrate Specificity; Time Factors; Type C Phospholipases | 1994 |
Potentiation by 1,4-dithiothreitol of histamine-induced inositol phosphate formation in rat cerebral cortex and human HeLa cells.
Topics: Animals; Binding, Competitive; Carbachol; Cerebral Cortex; Chromatography, Ion Exchange; Culture Techniques; Dithiothreitol; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; HeLa Cells; Histamine; Humans; Inositol Phosphates; Male; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1 | 1994 |
Hypersensitivity of Gi protein mediated muscarinic receptor adenylyl cyclase in chronic ischaemic heart failure in the rat.
Topics: Adenylyl Cyclases; Animals; Carbachol; Cell Membrane; Colforsin; Enzyme-Linked Immunosorbent Assay; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immunoblotting; Male; Myocardial Ischemia; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Sarcolemma | 1993 |
Postnatal decrease in muscarinic cholinergic influence on Ca2+ currents of rabbit ventricular cells.
Topics: Adenylate Cyclase Toxin; Aging; Animals; Animals, Newborn; Calcium; Calcium Channel Blockers; Carbachol; Colforsin; Electric Conductivity; Female; Guanylyl Imidodiphosphate; Heart Ventricles; Isoproterenol; Male; Myocardium; Pertussis Toxin; Rabbits; Receptors, Muscarinic; Virulence Factors, Bordetella | 1993 |
Novel regulation of muscarinic receptors and their coupling with G proteins in smooth muscle: transient resensitization during desensitizing process.
Topics: Animals; Carbachol; Cecum; Female; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1993 |
Differences between rat dorsal and ventral hippocampus in muscarinic receptor agonist binding and interaction with phospholipase C.
Topics: Alkaloids; Animals; Carbachol; Furans; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Mitochondria; N-Methylscopolamine; Naphthalenes; Oxotremorine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Synaptosomes; Type C Phospholipases | 1993 |
Coupling of muscarinic receptors to GTP proteins in postmortem human brain--alterations in Alzheimer's disease.
Topics: Aged; Aged, 80 and over; Alzheimer Disease; Autopsy; Binding, Competitive; Brain; Carbachol; Female; Frontal Lobe; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Kinetics; Male; Quinuclidinyl Benzilate; Receptors, Muscarinic; Reference Values; Temporal Lobe; Thalamus | 1993 |
Stable GDP analog-induced inactivation of G(i) proteins promotes cardiac adenylyl cyclase inhibition by guanosine 5'-(beta gamma-imino)triphosphate and muscarinic acetylcholine receptor.
Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Dogs; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanylyl Imidodiphosphate; Magnesium; Manganese; Myocardium; Receptors, Muscarinic; Sarcolemma; Thionucleotides | 1996 |
A novel irreversible antagonist of the A1-adenosine receptor.
Topics: Adenosine; Animals; Carbachol; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Kinetics; Membrane Potentials; Myocardium; Patch-Clamp Techniques; Potassium Channels; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptors, Purinergic P1; Theophylline; Xanthines | 1996 |
Evidence against a regulation of Na+/K(+)-ATPase by Gi proteins. Failure to detect an influence of G proteins on Na+/Ca(2+)-exchange in cardiac sarcolemmal membranes.
Topics: 4-Nitrophenylphosphatase; Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Calcium; Carbachol; Carrier Proteins; Dogs; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Muscarinic Agonists; Myocardial Contraction; Myocardium; Phenylisopropyladenosine; Potassium Channels; Receptors, Muscarinic; Receptors, Purinergic P1; Sarcolemma; Sodium; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase | 1996 |
Stimulation of the Na+/Ca2+ exchanger by phenylephrine, angiotensin II and endothelin 1.
Topics: Alkaloids; Angiotensin II; Animals; Benzophenanthridines; Calcium; Carbachol; Carrier Proteins; Endothelins; Enzyme Inhibitors; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Myocardium; Phenanthridines; Phenylephrine; Protein Kinase C; Rats; Sarcolemma; Sodium-Calcium Exchanger | 1996 |
Measurement of early events in signal transduction beyond receptors involving G proteins function in mononuclear leucocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adult; Aged; Carbachol; Depressive Disorder; Dopamine; Female; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Muscarinic Agonists; Pertussis Toxin; Poly(ADP-ribose) Polymerases; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Muscarinic; Signal Transduction; Virulence Factors, Bordetella | 1996 |
Sigma binding in a human neuroblastoma cell line.
Topics: Adenylyl Cyclases; Analgesics; Analysis of Variance; Animals; Binding, Competitive; Brain; Carbachol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanylyl Imidodiphosphate; Guinea Pigs; Haloperidol; Humans; Kinetics; Morphine; Naloxone; Neuroblastoma; Pentazocine; Phosphatidylinositols; Receptors, Opioid; Receptors, sigma; Trypsin; Tumor Cells, Cultured | 1996 |
A muscarinic acetylcholine receptor, present in the epithelial cell line from Chironomus tentans.
Topics: Animals; Atropine; Binding Sites; Binding, Competitive; Blotting, Western; Carbachol; Cell Line; Chironomidae; Ecdysterone; Epithelium; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Cholinergic | 1996 |
Cardiac muscarinic receptors. Relationship between the G protein and multiple states of affinity.
Topics: Animals; Carbachol; Cell Membrane; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanylyl Imidodiphosphate; Mesocricetus; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Osmolar Concentration; Parasympatholytics; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Scopolamine Derivatives; Tritium | 1997 |
Dynamics of ECT normalization of low G protein function and immunoreactivity in mononuclear leukocytes of patients with major depression.
Topics: Biomarkers; Carbachol; Depressive Disorder; Electroconvulsive Therapy; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Isoproterenol; Leukocytes, Mononuclear | 1998 |
Glucose uptake by C6 glioma cells is mediated by G(q alpha).
Topics: Animals; Carbachol; Deoxyglucose; Glioma; Glucose; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Pertussis Toxin; Rats; Stimulation, Chemical; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1998 |
Ethanol inhibits G-protein-mediated glucose uptake by C6 glioma cells.
Topics: Animals; Carbachol; Cell Count; Cell Survival; Culture Media; Deoxyglucose; Ethanol; Glioma; Glucose; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Insulin; Muscarinic Agonists; Rats; Tumor Cells, Cultured | 1999 |
Reduced high-affinity agonist binding at the M(1) muscarinic receptor in Alzheimer's disease brain: differential sensitivity to agonists and divalent cations.
Topics: Acetylcholine; Aged; Alzheimer Disease; Brain; Carbachol; Cations, Divalent; Chlorides; Edetic Acid; Female; Guanylyl Imidodiphosphate; Humans; Kinetics; Magnesium Chloride; Male; Manganese Compounds; Muscarinic Agonists; Oxotremorine; Pirenzepine; Receptor, Muscarinic M1; Receptors, Muscarinic; Reference Values | 1999 |
Differences in regional and subcellular localization of G(q/11) and RGS4 protein levels in Alzheimer's disease: correlation with muscarinic M1 receptor binding parameters.
Topics: Aged; Aged, 80 and over; Alzheimer Disease; Autopsy; Brain; Brain Chemistry; Carbachol; Case-Control Studies; Cell Membrane; Cerebellum; Cholinergic Agonists; Cytosol; Frontal Lobe; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Neurons; Parietal Lobe; Receptor, Muscarinic M1; Receptors, Muscarinic; RGS Proteins | 2003 |