Page last updated: 2024-08-17

carbachol and guanylyl imidodiphosphate

carbachol has been researched along with guanylyl imidodiphosphate in 94 studies

Research

Studies (94)

TimeframeStudies, this research(%)All Research%
pre-199054 (57.45)18.7374
1990's39 (41.49)18.2507
2000's1 (1.06)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gardner, JD; Robberecht, P; Uhlemann, ER1
Berrie, CP; Birdsall, NJ; Burgen, AS; Hulme, EC1
Boyd, RS; Donnelly, LE; MacDermot, J1
Bangert, M; Beyer, T; Niroomand, F; Rauch, B1
Hatta, S; Ohshika, H1
Nathanson, NM; van Koppen, CJ1
Baker, HJ; Claro, E; Fain, JN; Nair, BG; Patel, TB; Shanker, G; Wallace, MA1
Golly, F; Larocca, JN; Ledeen, RW1
Allen, RA; Colvin, RA; Oibo, JA1
Fermum, R; Kosche, D; Möritz, KU1
Milligan, G; Nair, BG; Parikh, B; Patel, TB1
Hung, WC; Wei, JW1
Bonner, TI; Brann, MR; Dörje, F; Wess, J1
Dawson, RM; Poretski, M1
Minton, AP; Sokolovsky, M1
Dwyer, TM; Farley, JM; Ho, IK; Mohan, PM; Yang, CM1
Hoffman, BB; Thomas, JM1
Cohen-Armon, M; Sokolovsky, M1
Aronstam, RS; Carrier, GO1
Cohen-Armon, M; Henis, YI; Kloog, Y; Sokolovsky, M1
Flynn, DD; Palermo, N; Suarez, A1
Allen, IS; Gaa, ST; Rogers, TB1
Hattori, Y; Kanno, M; Nakao, Y; Sakuma, I1
Jagadeesh, G; Phan, NT; Sulakhe, PV1
Merritt, JE; Putney, JW; Rubin, RP; Taylor, CW1
Barnes, PJ; Cuss, FM; Grandordy, BM; Palmer, JB; Sampson, AS1
Anthony, BL; Aronstam, RS2
Flynn, DD; Potter, LT1
Hunter, DD; Nathanson, NM2
Mei, L; Roeske, WR; Wang, JX; Yamamura, HI1
Aronstam, RS; Narayanan, TK1
Milnor, WR; Sastre, A1
Henis, YI; Moscona-Amir, E; Sokolovsky, M1
Bertrand, C; Gies, JP; Landry, Y1
Dwyer, TM; Farley, JM; Mohan, PM; Yang, CM1
Chung, FZ; Lai, J; Mei, L; Roeske, WR; Venter, JC; Yamamura, HI1
Brown, JH; Orellana, S; Solski, PA1
Aguilar, JS; De Robertis, E; Ochoa, EL1
Gies, JP; Ilien, B; Landry, Y1
Hjalmarson, A; Jacobsson, B; Ransnäs, L; Sabler, E1
Green, RD; Hosey, MM; Kwatra, MM; Leung, E; Maan, AC; McMahon, KK; Ptasienski, J1
Aguilar, JS; De Robertis, E; Fonseca, MI1
Adam, LP; Pappano, AJ; Sorota, S1
Roeske, WR; Watson, M; Yamamura, HI1
Kagiya, T; Mizushima, A; Uchida, S; Yoshida, H1
Baker, SP; Posner, P1
Barenholz, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M; Yechiel, E1
Bering, B; Müller, WE1
Bloom, JW; Halonen, M; Lawrence, LJ; Rould, E; Seaver, NA; Yamamura, HI1
Bruni, P; Hewlett, EL; Moss, J1
Baker, SP; Marchand, S; Nelson, CA; O'Neil, E; Posner, P1
Kloog, Y; Sokolovsky, M1
Koike, K; Okumura, K; Takayanagi, I1
Higuchi, H; Kagiya, T; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H; Zhou, XM1
Howlett, AC1
Burgoyne, RD1
Aronstam, RS; Greenbaum, LM1
Bergh, CH; Hjalmarson, A; Jacobsson, B; Ransnäs, L; Waldenström, A1
Halvorsen, SW; Nathanson, NM2
Nathanson, NM1
Aronstam, RS; Kirby, ML1
Higuchi, H; Matsumoto, K; Mizushima, A; Osugi, T; Uchida, S; Yoshida, H1
Higuchi, H; Matsumoto, K; Mizushima, A; Uchida, S; Yoshida, H1
Bárány, E; Berrie, CP; Birdsall, NJ; Burgen, AS; Hulme, EC1
Dziekan, LC; Galper, JB; O'Hara, DS; Smith, TW1
Leppik, R; van Giersbergen, PL1
Coy, DH; Gu, ZF; Jensen, RT; Pradhan, TK1
Andrade, R1
Hescheler, J1
Yatani, A1
Abe, H; Chihara, K; Kaji, H; Okimura, Y; Tai, S1
Honda, K; Kamiya, H; Takano, Y1
Young, JM; Young, KW1
Feng, QP; Fu, LX; Hedner, T; Hjalmarson, A; Hoebeke, J; Liang, QM; Sun, XY1
Joyner, RW; Kumar, R; Osaka, T1
Hishinuma, S; Kurokawa, M; Matsumoto, Y; Uchida, MK1
Consolo, S; Garcia Ruiz, AJ; La Porta, C; Ladinsky, H; Zambelli, M1
Alafuzoff, I; Nordberg, A; Warpman, U1
Jakobs, KH; Mura, R; Niroomand, F; Piacentini, L1
Baker, SP; Belardinelli, L; Ruble, J; Scammells, PJ; Shryock, JC; Srinivas, M1
Kübler, W; Mura, RA; Niroomand, F; Piacentini, L; Rauch, B; Zeifang, F1
Ballard, C; Schaffer, S1
Avissar, S; Schreiber, G1
Chien, CC; Pasternak, GW; Ryan-Moro, J; Standifer, KM1
Spindler, KD; Spindler-Barth, M; Wegener, S1
Chidiac, P; Green, MA; Wells, JW1
Avissar, S; Nechamkin, Y; Roitman, G; Schreiber, G1
Gao, Y; Kunapuli, SP; Ravindra, R; Singh, SP2
Ladner, CJ; Lee, JM1
Lee, JM; Mariyappa, R; Muma, NA; Williams, K1

Other Studies

94 other study(ies) available for carbachol and guanylyl imidodiphosphate

ArticleYear
Effects of alcohols on the actions of VIP and secretin on acinar cells from guinea pig pancreas.
    Gastroenterology, 1979, Volume: 76, Issue:5 Pt 1

    Topics: 1-Propanol; Adenylyl Cyclases; Alcohols; Amylases; Animals; Carbachol; Cholecystokinin; Cyclic AMP; Ethanol; Gastrointestinal Hormones; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Male; Methanol; Octanols; Pancreas; Secretin; Vasoactive Intestinal Peptide

1979
Guanine nucleotides modulate muscarinic receptor binding in the heart.
    Biochemical and biophysical research communications, 1979, Apr-27, Volume: 87, Issue:4

    Topics: Animals; Carbachol; Guanine Nucleotides; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Myocardium; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Ribonucleotides; Scopolamine Derivatives

1979
Opiate-dependent changes in the sensitivity of adenylate cyclase to stimulatory agonists and 5'-guanylylimidodiphosphate are independent of G protein abundance and eukaryotic ADP-ribosyltransferase activity in NG108-15 cells.
    Journal of neurochemistry, 1992, Volume: 58, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Drug Combinations; Enkephalin, Leucine-2-Alanine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immunoblotting; Niacinamide; Poly(ADP-ribose) Polymerases; Tumor Cells, Cultured

1992
Reduced adenylyl cyclase inhibition by carbachol and GTP during acute myocardial ischaemia.
    Journal of molecular and cellular cardiology, 1992, Volume: 24, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Colforsin; Coronary Disease; Dogs; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Receptors, Muscarinic

1992
Stable inhibition of adenylate cyclase by muscarinic agonist in rat parotid gland: effects of neomycin and pertussis toxin.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 72, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Methoxamine; Neomycin; Parotid Gland; Pertussis Toxin; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic; Virulence Factors, Bordetella

1991
The cysteine residue in the carboxyl-terminal domain of the m2 muscarinic acetylcholine receptor is not required for receptor-mediated inhibition of adenylate cyclase.
    Journal of neurochemistry, 1991, Volume: 57, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; Cell Line; Cyclic AMP; Cysteine; Guanylyl Imidodiphosphate; Muscarinic Antagonists; Quinuclidinyl Benzilate; Receptors, Muscarinic; Subcellular Fractions; Tissue Distribution

1991
Altered phosphoinositide-specific phospholipase C and adenylyl cyclase in brain cortical membranes of cats with GM1 and GM2 gangliosidosis.
    Brain research. Molecular brain research, 1991, Volume: 11, Issue:3-4

    Topics: Adenylyl Cyclases; Aluminum; Aluminum Chloride; Aluminum Compounds; Animals; Calcium; Carbachol; Cat Diseases; Cats; Cell Membrane; Cerebral Cortex; Chlorides; Colforsin; G(M1) Ganglioside; Gangliosidoses; Gangliosidosis, GM1; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Kinetics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Diacylglycerol-Lyase; Phosphatidylinositols; Phosphoric Diester Hydrolases; Reference Values; Sodium Fluoride

1991
Phosphoinositide breakdown in isolated myelin is stimulated by GTP analogues and calcium.
    Journal of neuroscience research, 1990, Volume: 27, Issue:3

    Topics: Animals; Calcium; Carbachol; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Inositol Phosphates; Myelin Proteins; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Second Messenger Systems

1990
Calcium inhibition of cardiac adenylyl cyclase. Evidence for two distinct sites of inhibition.
    Cell calcium, 1991, Volume: 12, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Calmodulin; Carbachol; Colforsin; Dogs; Enzyme Activation; Guanylyl Imidodiphosphate; Magnesium; Myocardium; Pertussis Toxin; Sarcolemma; Virulence Factors, Bordetella

1991
Membrane-associated signal transduction modulates contractile responses to Ca2+ in saponin-skinned coronary smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:2

    Topics: Aluminum; Animals; Calcium; Carbachol; Cattle; Coronary Vessels; Female; Fluorides; Guanylyl Imidodiphosphate; Histamine; In Vitro Techniques; Male; Membranes; Permeability; Phorbol 12,13-Dibutyrate; Saponins; Signal Transduction; Swine; Vasoconstriction

1991
Gs alpha mediates epidermal growth factor-elicited stimulation of rat cardiac adenylate cyclase.
    The Journal of biological chemistry, 1990, Dec-05, Volume: 265, Issue:34

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antibodies; Carbachol; Colforsin; Epidermal Growth Factor; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immune Sera; Isoproterenol; Kinetics; Male; Membrane Proteins; Molecular Sequence Data; Molecular Weight; Myocardium; Oligopeptides; Phenylisopropyladenosine; Rats; Rats, Inbred Strains

1990
Guanine nucleotides have a direct inhibitory effect on polyphosphoinositide turnover in rat cortical synaptosomes.
    The International journal of biochemistry, 1990, Volume: 22, Issue:5

    Topics: Animals; Carbachol; Cerebral Cortex; GTP-Binding Proteins; Guanine Nucleotides; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Phosphates; Phosphatidic Acids; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Phosphatidylinositols; Rats; Rats, Inbred Strains; Synaptosomes

1990
Delineation of muscarinic receptor domains conferring selectivity of coupling to guanine nucleotide-binding proteins and second messengers.
    Molecular pharmacology, 1990, Volume: 38, Issue:4

    Topics: Adenylate Cyclase Toxin; Animals; Carbachol; Cyclic AMP; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Mice; N-Methylscopolamine; Pertussis Toxin; Phosphatidylinositols; Receptors, Muscarinic; Scopolamine Derivatives; Second Messenger Systems; Virulence Factors, Bordetella

1990
Opposing effects of N-ethylmaleimide on the affinity of carbachol for muscarinic cholinoceptors of guinea-pig atrium.
    General pharmacology, 1990, Volume: 21, Issue:6

    Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; Guinea Pigs; Heart Atria; Premedication; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Temperature

1990
A model for the interaction of muscarinic receptors, agonists, and two distinct effector substances.
    Biochemistry, 1990, Feb-13, Volume: 29, Issue:6

    Topics: Aging; Animals; Batrachotoxins; Carbachol; Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Models, Biological; Myocardium; Pertussis Toxin; Rats; Receptors, Muscarinic; Virulence Factors, Bordetella

1990
Down-regulation of muscarinic receptors in the striatum of organophosphate-treated swine.
    Toxicology and applied pharmacology, 1990, Volume: 104, Issue:3

    Topics: Acetylcholinesterase; Animals; Binding Sites; Binding, Competitive; Carbachol; Corpus Striatum; Down-Regulation; Guanylyl Imidodiphosphate; Isoflurophate; Magnesium; Male; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Regression Analysis; Swine

1990
Agonist-induced down-regulation of muscarinic cholinergic and alpha 2-adrenergic receptors after inactivation of Ni by pertussis toxin.
    Endocrinology, 1986, Volume: 119, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Alprostadil; Animals; ATPase Inhibitory Protein; Carbachol; Cell Line; Cyclic AMP; Electrophoresis, Polyacrylamide Gel; Epinephrine; Glioma; Guanylyl Imidodiphosphate; Molecular Weight; NAD; Neuroblastoma; Pertussis Toxin; Proteins; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Virulence Factors, Bordetella; Yohimbine

1986
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
    The Journal of biological chemistry, 1986, Sep-25, Volume: 261, Issue:27

    Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1986
Insulin prevention of altered muscarinic receptor-G protein coupling in diabetic rat atria.
    Diabetes, 1989, Volume: 38, Issue:12

    Topics: Acetylcholine; Animals; Bethanechol; Bethanechol Compounds; Carbachol; Diabetes Mellitus, Experimental; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Insulin; Kinetics; Male; Myocardium; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Reference Values

1989
Batrachotoxin changes the properties of the muscarinic receptor in rat brain and heart: possible interaction(s) between muscarinic receptors and sodium channels.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:10

    Topics: Aconitine; Animals; Batrachotoxins; Benzilates; Binding, Competitive; Brain; Carbachol; Guanylyl Imidodiphosphate; Ion Channels; Kinetics; Macromolecular Substances; Male; Myocardium; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1985
Agonist binding to M1 muscarinic receptors is sensitive to guanine nucleotides.
    European journal of pharmacology, 1989, Oct-17, Volume: 172, Issue:4-5

    Topics: Animals; Carbachol; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Indicators and Reagents; Kinetics; Male; Methacholine Compounds; Oxotremorine; Pilocarpine; Pirenzepine; Rabbits; Receptors, Muscarinic; Second Messenger Systems

1989
Changes in expression of a functional Gi protein in cultured rat heart cells.
    The American journal of physiology, 1988, Volume: 255, Issue:1 Pt 1

    Topics: Angiotensin II; Animals; Carbachol; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Isoproterenol; Myocardium; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Pharmacological analysis of the cardiac actions of xamoterol, a beta adrenoceptor antagonist with partial agonistic activity, in guinea pig heart: evidence for involvement of adenylate cyclase system in its cardiac stimulant actions.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Adenosine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cyclic AMP; Dose-Response Relationship, Drug; Female; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Rate; Iodocyanopindolol; Isoproterenol; Male; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Xamoterol

1987
Comparison of cholinergic inhibition and beta-adrenergic stimulation of adenylate cyclase from rat and guinea-pig hearts: effects of guanine nucleotides and monovalent cations.
    General pharmacology, 1985, Volume: 16, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Carbachol; Cations, Monovalent; Chlorides; Colforsin; Cytosol; Enzyme Activation; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Lithium; Lithium Chloride; Male; Myocardium; Rats; Rats, Inbred Strains; Sodium; Sodium Chloride; Sodium Fluoride; Tissue Distribution

1985
A guanine nucleotide-dependent regulatory protein couples substance P receptors to phospholipase C in rat parotid gland.
    Biochemical and biophysical research communications, 1986, Apr-14, Volume: 136, Issue:1

    Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Epinephrine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Monophosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Inositol Phosphates; Male; Parotid Gland; Propranolol; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Sodium Fluoride; Thionucleotides; Type C Phospholipases

1986
Phosphatidylinositol response to cholinergic agonists in airway smooth muscle: relationship to contraction and muscarinic receptor occupancy.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Benzodiazepinones; Carbachol; Cattle; Chlorides; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Lithium; Lithium Chloride; Membrane Lipids; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Respiratory System; Trachea

1986
Effect of pH on muscarinic acetylcholine receptors from rat brainstem.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Animals; Brain Stem; Carbachol; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Male; Mathematics; N-Methylscopolamine; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Scopolamine Derivatives; Temperature; Time Factors

1986
Effect of solubilization on the distinct binding properties of muscarine receptors from rabbit hippocampus and brainstem.
    Molecular pharmacology, 1986, Volume: 30, Issue:3

    Topics: Animals; Brain Stem; Carbachol; Edetic Acid; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; In Vitro Techniques; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Solubility

1986
Biochemical and physical analyses of newly synthesized muscarinic acetylcholine receptors in cultured embryonic chicken cardiac cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:12

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Cell Membrane Permeability; Chick Embryo; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart; Isoelectric Point; Kinetics; Molecular Weight; Myocardium; Potassium; Receptors, Muscarinic

1986
Solubilization with digitonin alters the kinetics of pirenzepine binding to muscarinic receptors from rat forebrain and heart.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Animals; Brain; Carbachol; Digitonin; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Myocardium; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Solubility

1987
Temperature effect on the detection of muscarinic receptor-G protein interactions in ligand binding assays.
    Biochemical pharmacology, 1988, Mar-15, Volume: 37, Issue:6

    Topics: Animals; Brain Stem; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Myocardium; Oxotremorine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Temperature

1988
Cholinergic receptors and contraction of smooth muscle in canine portal vein.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Algorithms; Animals; Calcimycin; Carbachol; Dogs; Guanylyl Imidodiphosphate; Kinetics; Muscle Contraction; Muscle, Smooth; Norepinephrine; Portal Vein; Quinuclidinyl Benzilate; Receptors, Cholinergic

1988
Guanosine 5'-triphosphate binding protein (Gi) and two additional pertussis toxin substrates associated with muscarinic receptors in rat heart myocytes: characterization and age dependency.
    Biochemistry, 1988, Jul-12, Volume: 27, Issue:14

    Topics: Adenosine Diphosphate Ribose; Aging; Animals; Carbachol; Cells, Cultured; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Liposomes; Molecular Weight; Myocardium; Pertussis Toxin; Rats; Receptors, Muscarinic; Virulence Factors, Bordetella

1988
Membrane phospholipid polar heads influence the coupling of M2 muscarinic receptors to G proteins.
    Neurochemical research, 1988, Volume: 13, Issue:8

    Topics: Animals; Carbachol; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Membrane Proteins; Myocardium; Oxotremorine; Phospholipids; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Type C Phospholipases

1988
Changes in affinity states during down-regulation of muscarinic receptors in tracheal smooth muscle of organophosphate-treated swine.
    Journal of autonomic pharmacology, 1988, Volume: 8, Issue:2

    Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoflurophate; Magnesium; Male; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine; Trachea

1988
The cloned murine M1 muscarinic receptor is associated with the hydrolysis of phosphatidylinositols in transfected murine B82 cells.
    Life sciences, 1988, Volume: 42, Issue:24

    Topics: Animals; Atropine; Binding, Competitive; Carbachol; Cell Line; Cell Membrane; DNA, Recombinant; Fibroblasts; Guanylyl Imidodiphosphate; Hydrolysis; Mice; Muscarine; Nucleic Acid Hybridization; Phosphatidylinositols; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Recombinant Proteins; Sequence Homology, Nucleic Acid; Transfection

1988
Guanosine 5'-O-(thiotriphosphate)-dependent inositol trisphosphate formation in membranes is inhibited by phorbol ester and protein kinase C.
    The Journal of biological chemistry, 1987, Feb-05, Volume: 262, Issue:4

    Topics: Bradykinin; Carbachol; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Histamine; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Kinetics; Membranes; Phorbol Esters; Protein Kinase C; Quinuclidinyl Benzilate; Receptors, Muscarinic; Sugar Phosphates; Tetradecanoylphorbol Acetate; Thionucleotides

1987
Reconstitution of solubilized atrial cholinergic muscarinic receptors in liposomes.
    Neurochemical research, 1987, Volume: 12, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Cattle; Glycine max; Guanylyl Imidodiphosphate; Heart Atria; Kinetics; Liposomes; Myocardium; N-Methylscopolamine; Phosphatidylcholines; Receptors, Muscarinic; Scopolamine Derivatives; Solubility

1987
Temperature-dependence and heterogeneity of muscarinic agonist and antagonist binding.
    Biochemical pharmacology, 1987, Aug-15, Volume: 36, Issue:16

    Topics: Animals; Atropine; Brain; Carbachol; Guanylyl Imidodiphosphate; Kinetics; Lung; Male; Myocardium; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Temperature

1987
Effect of corticosteroids on muscarinic receptors on cultured myocardial cells.
    Pharmacology & toxicology, 1987, Volume: 61, Issue:2

    Topics: Animals; Binding, Competitive; Carbachol; Cell Membrane; Cells, Cultured; Female; Guanylyl Imidodiphosphate; Hydrocortisone; In Vitro Techniques; Manganese; Myocardium; Phosphatidylinositols; Puromycin; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1987
Correlation of agonist-induced phosphorylation of chick heart muscarinic receptors with receptor desensitization.
    The Journal of biological chemistry, 1987, Dec-05, Volume: 262, Issue:34

    Topics: Animals; Atropine; Carbachol; Chickens; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Heart; Magnesium; Myocardium; Oxotremorine; Phosphorylation; Quinuclidinyl Benzilate; Receptors, Muscarinic

1987
Pertussis vaccine reduces agonist binding to the rat heart muscarinic receptor and its guanine nucleotide modulation.
    Neurochemical research, 1986, Volume: 11, Issue:5

    Topics: Animals; Carbachol; Cell Membrane; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Myocardium; Pertussis Vaccine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic

1986
High-affinity agonist binding to rat brainstem muscarinic receptors is eliminated by low pH.
    Neuroscience letters, 1986, Aug-15, Volume: 69, Issue:1

    Topics: Animals; Brain Stem; Carbachol; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1986
Comparison of muscarinic receptor properties in hatched chick heart atrium and ventricle.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Animals; Atropine; Benzodiazepinones; Carbachol; Chickens; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Pirenzepine; Potassium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tritium

1986
[3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. I. Characterization and regulation of agonist binding to putative muscarinic subtypes.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Acetylcholine; Animals; Benzodiazepinones; Buffers; Carbachol; Cerebral Cortex; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Myocardium; Parasympathomimetics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium

1986
Alterations in muscarinic receptors of ventricular muscle in carbachol-induced short-term desensitization.
    Japanese journal of pharmacology, 1986, Volume: 41, Issue:4

    Topics: Animals; Carbachol; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Ventricles; Myocardial Contraction; Quinuclidinyl Benzilate; Receptors, Muscarinic

1986
Irreversible binding of acetylethylcholine mustard to cardiac cholinergic muscarinic receptors.
    Molecular pharmacology, 1986, Volume: 30, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Carbachol; Cell Membrane; Guanylyl Imidodiphosphate; Heart Rate; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1986
Role of lipids in age-related changes in the properties of muscarinic receptors in cultured rat heart myocytes.
    Biochemistry, 1986, Dec-02, Volume: 25, Issue:24

    Topics: Acetylcholine; Animals; Animals, Newborn; Benzilates; Carbachol; Cells, Cultured; Guanylyl Imidodiphosphate; Kinetics; Liposomes; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic

1986
Stereospecific 3H-QNB binding to human erythrocyte membranes associated with muscarinic cholinergic receptors.
    Journal of neural transmission, 1987, Volume: 68, Issue:1-2

    Topics: Adult; Aging; Animals; Atropine; Brain; Carbachol; Erythrocyte Membrane; Female; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Male; Middle Aged; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism

1987
Characterization of high affinity [3H]pirenzepine and (-)-[3H] quinuclidinyl benzilate binding to muscarinic cholinergic receptors in rabbit peripheral lung.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Animals; Binding, Competitive; Carbachol; Female; Guanylyl Imidodiphosphate; Kinetics; Lung; Male; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Stereoisomerism

1987
Effects of pertussis toxin-catalyzed ADP-ribosylation on interactions of transducin and the inhibitory GTP-binding protein of adenylate cyclase with guanyl nucleotides.
    Biochemical and biophysical research communications, 1985, Mar-29, Volume: 127, Issue:3

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Atropine; Bacterial Toxins; Carbachol; Cell Line; Cell Membrane; Enkephalin, Methionine; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Membrane Proteins; Naloxone; Norepinephrine; Nucleoside Diphosphate Sugars; Pertussis Toxin; Phentolamine; Transducin; Virulence Factors, Bordetella

1985
Age-related changes in cardiac muscarinic receptors: decreased ability of the receptor to form a high affinity agonist binding state.
    Journal of gerontology, 1985, Volume: 40, Issue:2

    Topics: Aging; Animals; Body Weight; Carbachol; Guanylyl Imidodiphosphate; Heart; Male; Myocardium; Organ Size; Quinuclidinyl Benzilate; Rats; Rats, Inbred F344; Receptors, Cholinergic; Receptors, Muscarinic

1985
Allosteric interactions between muscarinic agonist binding sites and effector sites demonstrated by the use of bisquaternary pyridinium oximes.
    Life sciences, 1985, Jun-03, Volume: 36, Issue:22

    Topics: Animals; Brain Stem; Carbachol; Cerebral Cortex; Cobalt; Guanylyl Imidodiphosphate; In Vitro Techniques; Oximes; Oxotremorine; Parasympathomimetics; Pyridinium Compounds; Rats; Receptors, Muscarinic

1985
Interaction of muscarinic drugs with their receptor.
    General pharmacology, 1985, Volume: 16, Issue:3

    Topics: Animals; Atropine; Carbachol; Guanylyl Imidodiphosphate; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Microsomes; Muscle, Smooth; Parasympathomimetics; Quaternary Ammonium Compounds; Quinuclidinyl Benzilate; Receptors, Muscarinic

1985
Multiple agonist binding sites of muscarinic acetylcholine receptors and their relation to the negative inotropic action of agonists in guinea-pig heart.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Binding Sites; Carbachol; Depression, Chemical; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Isoproterenol; Myocardial Contraction; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1985
Inhibition of neuroblastoma adenylate cyclase by cannabinoid and nantradol compounds.
    Life sciences, 1984, Oct-22, Volume: 35, Issue:17

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclase Inhibitors; Alprostadil; Animals; Carbachol; Cell Line; Cyclic AMP; Dronabinol; Epoprostenol; Guanylyl Imidodiphosphate; Neuroblastoma; Phenanthridines; Phosphodiesterase Inhibitors; Prostaglandins E; Secretin; Sodium Fluoride

1984
Regulation of the muscarinic acetylcholine receptor: effects of phosphorylating conditions on agonist and antagonist binding.
    Journal of neurochemistry, 1983, Volume: 40, Issue:2

    Topics: Animals; Brain; Calcium-Binding Proteins; Calmodulin; Carbachol; Cerebral Cortex; Cyclic AMP; Guanylyl Imidodiphosphate; Phosphorylation; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Synaptic Membranes

1983
Guanine nucleotide sensitivity of muscarinic acetylcholine receptors from rat brainstem is eliminated by endogenous proteolytic activity.
    Neuroscience letters, 1984, Jun-15, Volume: 47, Issue:2

    Topics: Animals; Brain Stem; Carbachol; Endopeptidases; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Protease Inhibitors; Rats; Receptors, Muscarinic

1984
Effects of acute ketotic and non-ketotic diabetes on the myocardial muscarinic receptors.
    Acta pharmacologica et toxicologica, 1984, Volume: 55, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Carbachol; Computers; Diabetes Mellitus, Experimental; Diabetic Ketoacidosis; Guanylyl Imidodiphosphate; Insulin; Male; Models, Biological; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1984
Ontogenesis of physiological responsiveness and guanine nucleotide sensitivity of cardiac muscarinic receptors during chick embryonic development.
    Biochemistry, 1984, Nov-20, Volume: 23, Issue:24

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atrial Function; Bacterial Toxins; Carbachol; Chick Embryo; Depression, Chemical; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Heart; Heart Rate; Isoproterenol; Myocardium; Pertussis Toxin; Quinuclidinyl Benzilate; Receptors, Muscarinic; Virulence Factors, Bordetella

1984
Decreased physiological sensitivity mediated by newly synthesized muscarinic acetylcholine receptors in embryonic chicken heart.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:11

    Topics: Adenylyl Cyclase Inhibitors; Animals; Atropine; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Rate; Protein Processing, Post-Translational; Quinuclidinyl Benzilate; Receptors, Muscarinic

1984
Binding of agonists and antagonists to muscarinic acetylcholine receptors on intact cultured heart cells.
    Journal of neurochemistry, 1983, Volume: 41, Issue:6

    Topics: Animals; Binding, Competitive; Carbachol; Cells, Cultured; Chick Embryo; Guanylyl Imidodiphosphate; Kinetics; Myocardium; N-Methylscopolamine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Scopolamine Derivatives

1983
Atropine-induced alterations of normal development of muscarinic receptors in the embryonic chick heart.
    Journal of molecular and cellular cardiology, 1983, Volume: 15, Issue:10

    Topics: Animals; Atropine; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Atria; Heart Ventricles; Myocardium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Time Factors

1983
Effects of guanine nucleotide and sulfhydryl reagent on subpopulations of muscarinic acetylcholine receptors in mammalian hearts: possible evidence for interconversion of super-high and low affinity agonist binding sites.
    European journal of pharmacology, 1984, May-04, Volume: 100, Issue:3-4

    Topics: Animals; Carbachol; Dogs; Guanine Nucleotides; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Membranes; Myocardium; Quinuclidinyl Benzilate; Receptors, Muscarinic; Sulfhydryl Reagents; Temperature

1984
Effect of urea-treatment on agonist binding affinity of the muscarinic acetylcholine receptor.
    Life sciences, 1983, Sep-05, Volume: 33, Issue:10

    Topics: Animals; Atropine; Binding, Competitive; Carbachol; Dithionitrobenzoic Acid; Guanylyl Imidodiphosphate; Guinea Pigs; Male; Microsomes; Myocardium; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Urea

1983
The binding properties of the muscarinic receptors of the cynomolgus monkey ciliary body and the response to the induction of agonist subsensitivity.
    British journal of pharmacology, 1982, Volume: 77, Issue:4

    Topics: Animals; Benzodiazepinones; Carbachol; Ciliary Body; Guanylyl Imidodiphosphate; Kinetics; Macaca fascicularis; N-Methylscopolamine; Pilocarpine; Pirenzepine; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives

1982
The biphasic response of muscarinic cholinergic receptors in cultured heart cells to agonists. Effects on receptor number and affinity in intact cells and homogenates.
    The Journal of biological chemistry, 1982, Sep-10, Volume: 257, Issue:17

    Topics: Animals; Carbachol; Cell Membrane; Cells, Cultured; Chick Embryo; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Myocardium; N-Methylscopolamine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine Derivatives

1982
In vivo regulation of muscarinic acetylcholine receptor number and function in embryonic chick heart.
    The Journal of biological chemistry, 1981, Aug-10, Volume: 256, Issue:15

    Topics: Animals; Binding, Competitive; Carbachol; Chick Embryo; Guanylyl Imidodiphosphate; Heart; Heart Rate; Kinetics; Mathematics; Myocardium; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic

1981
Modulation of agonist binding by guanine nucleotides in CHO cells expressing muscarinic m1-m5 receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: Animals; Atropine; Carbachol; CHO Cells; Cricetinae; Guanine Nucleotides; Guanylyl Imidodiphosphate; Humans; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Parasympatholytics; Radioligand Assay; Receptors, Muscarinic; Scopolamine Derivatives

1995
Smooth muscle cells from guinea pig stomach possess high-affinity galanin receptors that mediate relaxation.
    The American journal of physiology, 1994, Volume: 266, Issue:5 Pt 1

    Topics: Animals; Carbachol; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Galanin; Gastric Mucosa; Guanylyl Imidodiphosphate; Guinea Pigs; Kinetics; Male; Muscle Relaxation; Muscle, Smooth; Neuropeptides; Peptides; Protein Precursors; Rats; Receptors, Galanin; Receptors, Gastrointestinal Hormone; Stomach; Swine; Time Factors; Vasoactive Intestinal Peptide

1994
Infusion of guanine nucleotides through recording electrodes for studies on G-protein regulation of ion currents and channels.
    Methods in enzymology, 1994, Volume: 238

    Topics: Animals; Baclofen; Carbachol; Electrophysiology; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hippocampus; Ion Channels; Membrane Potentials; Microelectrodes; Pyramidal Cells; Rats; Serotonin; Thionucleotides

1994
Whole-cell clamp analysis for G-protein regulation of channels.
    Methods in enzymology, 1994, Volume: 238

    Topics: Adenosine Diphosphate Ribose; Animals; Calcium Channels; Carbachol; Cholera Toxin; Electrophysiology; Epinephrine; Glioma; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Homeostasis; Hybrid Cells; Ion Channels; Macromolecular Substances; Neuroblastoma; Oligonucleotides, Antisense; Patch-Clamp Techniques; PC12 Cells; Potassium Channels; Rats; RNA, Messenger; Virulence Factors, Bordetella

1994
Reconstitution of receptor-regulated ion channels in isolated patch membrane.
    Methods in enzymology, 1994, Volume: 238

    Topics: Acetylcholine; Animals; Carbachol; Cell Membrane; Electrophysiology; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels; Receptors, Muscarinic; Virulence Factors, Bordetella

1994
Neurokinin receptor antagonists inhibit the binding of growth hormone-releasing peptide to EP-1 human neuroblastoma cells.
    Biochemical and biophysical research communications, 1995, Sep-14, Volume: 214, Issue:2

    Topics: Alprostadil; Animals; Atropine; Carbachol; Cell Line; Growth Hormone-Releasing Hormone; Guanylyl Imidodiphosphate; HeLa Cells; Humans; Hypothalamus; Kinetics; Neuroblastoma; Neuropeptides; Oligopeptides; Pituitary Gland; Rats; Receptors, Tachykinin; Structure-Activity Relationship; Tumor Cells, Cultured

1995
The mechanism of muscarinic agonist-stimulated inositol phosphate formation in permeabilized ileal smooth muscle.
    Japanese journal of pharmacology, 1994, Volume: 65, Issue:3

    Topics: Acetylcholine; Animals; Calcium; Carbachol; Dose-Response Relationship, Drug; Drug Synergism; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Pilocarpine; Substrate Specificity; Time Factors; Type C Phospholipases

1994
Potentiation by 1,4-dithiothreitol of histamine-induced inositol phosphate formation in rat cerebral cortex and human HeLa cells.
    European journal of pharmacology, 1994, Nov-15, Volume: 269, Issue:3

    Topics: Animals; Binding, Competitive; Carbachol; Cerebral Cortex; Chromatography, Ion Exchange; Culture Techniques; Dithiothreitol; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; HeLa Cells; Histamine; Humans; Inositol Phosphates; Male; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1

1994
Hypersensitivity of Gi protein mediated muscarinic receptor adenylyl cyclase in chronic ischaemic heart failure in the rat.
    Cardiovascular research, 1993, Volume: 27, Issue:11

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cell Membrane; Colforsin; Enzyme-Linked Immunosorbent Assay; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Immunoblotting; Male; Myocardial Ischemia; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Sarcolemma

1993
Postnatal decrease in muscarinic cholinergic influence on Ca2+ currents of rabbit ventricular cells.
    The American journal of physiology, 1993, Volume: 264, Issue:6 Pt 2

    Topics: Adenylate Cyclase Toxin; Aging; Animals; Animals, Newborn; Calcium; Calcium Channel Blockers; Carbachol; Colforsin; Electric Conductivity; Female; Guanylyl Imidodiphosphate; Heart Ventricles; Isoproterenol; Male; Myocardium; Pertussis Toxin; Rabbits; Receptors, Muscarinic; Virulence Factors, Bordetella

1993
Novel regulation of muscarinic receptors and their coupling with G proteins in smooth muscle: transient resensitization during desensitizing process.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Animals; Carbachol; Cecum; Female; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Quinuclidinyl Benzilate; Receptors, Muscarinic

1993
Differences between rat dorsal and ventral hippocampus in muscarinic receptor agonist binding and interaction with phospholipase C.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: Alkaloids; Animals; Carbachol; Furans; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Mitochondria; N-Methylscopolamine; Naphthalenes; Oxotremorine; Parasympatholytics; Parasympathomimetics; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Synaptosomes; Type C Phospholipases

1993
Coupling of muscarinic receptors to GTP proteins in postmortem human brain--alterations in Alzheimer's disease.
    Neuroscience letters, 1993, Feb-05, Volume: 150, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Autopsy; Binding, Competitive; Brain; Carbachol; Female; Frontal Lobe; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Kinetics; Male; Quinuclidinyl Benzilate; Receptors, Muscarinic; Reference Values; Temporal Lobe; Thalamus

1993
Stable GDP analog-induced inactivation of G(i) proteins promotes cardiac adenylyl cyclase inhibition by guanosine 5'-(beta gamma-imino)triphosphate and muscarinic acetylcholine receptor.
    Biochimica et biophysica acta, 1996, Jun-13, Volume: 1282, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Dogs; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanylyl Imidodiphosphate; Magnesium; Manganese; Myocardium; Receptors, Muscarinic; Sarcolemma; Thionucleotides

1996
A novel irreversible antagonist of the A1-adenosine receptor.
    Molecular pharmacology, 1996, Volume: 50, Issue:1

    Topics: Adenosine; Animals; Carbachol; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Kinetics; Membrane Potentials; Myocardium; Patch-Clamp Techniques; Potassium Channels; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptors, Purinergic P1; Theophylline; Xanthines

1996
Evidence against a regulation of Na+/K(+)-ATPase by Gi proteins. Failure to detect an influence of G proteins on Na+/Ca(2+)-exchange in cardiac sarcolemmal membranes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: 4-Nitrophenylphosphatase; Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Calcium; Carbachol; Carrier Proteins; Dogs; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Muscarinic Agonists; Myocardial Contraction; Myocardium; Phenylisopropyladenosine; Potassium Channels; Receptors, Muscarinic; Receptors, Purinergic P1; Sarcolemma; Sodium; Sodium-Calcium Exchanger; Sodium-Potassium-Exchanging ATPase

1996
Stimulation of the Na+/Ca2+ exchanger by phenylephrine, angiotensin II and endothelin 1.
    Journal of molecular and cellular cardiology, 1996, Volume: 28, Issue:1

    Topics: Alkaloids; Angiotensin II; Animals; Benzophenanthridines; Calcium; Carbachol; Carrier Proteins; Endothelins; Enzyme Inhibitors; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Myocardium; Phenanthridines; Phenylephrine; Protein Kinase C; Rats; Sarcolemma; Sodium-Calcium Exchanger

1996
Measurement of early events in signal transduction beyond receptors involving G proteins function in mononuclear leucocytes.
    Journal of neuroimmunology, 1996, Volume: 70, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adult; Aged; Carbachol; Depressive Disorder; Dopamine; Female; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Isoproterenol; Leukocytes, Mononuclear; Male; Middle Aged; Muscarinic Agonists; Pertussis Toxin; Poly(ADP-ribose) Polymerases; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Muscarinic; Signal Transduction; Virulence Factors, Bordetella

1996
Sigma binding in a human neuroblastoma cell line.
    Neurochemical research, 1996, Volume: 21, Issue:11

    Topics: Adenylyl Cyclases; Analgesics; Analysis of Variance; Animals; Binding, Competitive; Brain; Carbachol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanylyl Imidodiphosphate; Guinea Pigs; Haloperidol; Humans; Kinetics; Morphine; Naloxone; Neuroblastoma; Pentazocine; Phosphatidylinositols; Receptors, Opioid; Receptors, sigma; Trypsin; Tumor Cells, Cultured

1996
A muscarinic acetylcholine receptor, present in the epithelial cell line from Chironomus tentans.
    Biological chemistry, 1996, Volume: 377, Issue:12

    Topics: Animals; Atropine; Binding Sites; Binding, Competitive; Blotting, Western; Carbachol; Cell Line; Chironomidae; Ecdysterone; Epithelium; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Cholinergic

1996
Cardiac muscarinic receptors. Relationship between the G protein and multiple states of affinity.
    Biochemistry, 1997, Jun-17, Volume: 36, Issue:24

    Topics: Animals; Carbachol; Cell Membrane; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanylyl Imidodiphosphate; Mesocricetus; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Osmolar Concentration; Parasympatholytics; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1997
Dynamics of ECT normalization of low G protein function and immunoreactivity in mononuclear leukocytes of patients with major depression.
    The American journal of psychiatry, 1998, Volume: 155, Issue:5

    Topics: Biomarkers; Carbachol; Depressive Disorder; Electroconvulsive Therapy; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Isoproterenol; Leukocytes, Mononuclear

1998
Glucose uptake by C6 glioma cells is mediated by G(q alpha).
    Neuroreport, 1998, Jan-05, Volume: 9, Issue:1

    Topics: Animals; Carbachol; Deoxyglucose; Glioma; Glucose; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Pertussis Toxin; Rats; Stimulation, Chemical; Tumor Cells, Cultured; Virulence Factors, Bordetella

1998
Ethanol inhibits G-protein-mediated glucose uptake by C6 glioma cells.
    Neuroreport, 1999, Feb-25, Volume: 10, Issue:3

    Topics: Animals; Carbachol; Cell Count; Cell Survival; Culture Media; Deoxyglucose; Ethanol; Glioma; Glucose; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Insulin; Muscarinic Agonists; Rats; Tumor Cells, Cultured

1999
Reduced high-affinity agonist binding at the M(1) muscarinic receptor in Alzheimer's disease brain: differential sensitivity to agonists and divalent cations.
    Experimental neurology, 1999, Volume: 158, Issue:2

    Topics: Acetylcholine; Aged; Alzheimer Disease; Brain; Carbachol; Cations, Divalent; Chlorides; Edetic Acid; Female; Guanylyl Imidodiphosphate; Humans; Kinetics; Magnesium Chloride; Male; Manganese Compounds; Muscarinic Agonists; Oxotremorine; Pirenzepine; Receptor, Muscarinic M1; Receptors, Muscarinic; Reference Values

1999
Differences in regional and subcellular localization of G(q/11) and RGS4 protein levels in Alzheimer's disease: correlation with muscarinic M1 receptor binding parameters.
    Synapse (New York, N.Y.), 2003, Volume: 47, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Autopsy; Brain; Brain Chemistry; Carbachol; Case-Control Studies; Cell Membrane; Cerebellum; Cholinergic Agonists; Cytosol; Frontal Lobe; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Immunoblotting; Neurons; Parietal Lobe; Receptor, Muscarinic M1; Receptors, Muscarinic; RGS Proteins

2003