Page last updated: 2024-08-17

carbachol and cromakalim

carbachol has been researched along with cromakalim in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.13)18.7374
1990's26 (81.25)18.2507
2000's5 (15.63)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arch, JR; Challiss, RA; Patel, N1
Alibhai, KN; Huizinga, JD; Richardson, D1
Arch, JR; Bond, J; Buckle, DR; Shaw, DJ; Taylor, JF; Taylor, SG; Ward, JS1
Albus, U; Englert, HC; Fürst, U; Gehring, D; Rosenkranz, B; Schölkens, BA; Scholz, W; Wirth, K1
Bang, L; Nielsen-Kudsk, JE1
Charette, L; Garcia, ML; Jones, TR; Kaczorowski, GJ1
Satoh, E; Taira, N; Yanagisawa, T1
MacLeod, KM; Ray, A1
Andersson, KE; Andersson, PO; Fovaeus, M; Malmgren, A; Sjögren, C1
Cook, NS; Quast, U; Scholtysik, G; Weir, SW1
Ishimura, Y; Katoh, I; Masuda, Y; Oka, M; Yoshizumi, M1
Allescher, HD; Franck, H; Puschmann, A; Schusdziarra, V1
Broadley, KJ; Ford, WR; Urquhart, RA1
Imagawa, J; Kamei, K; Kuriyama, H; Nabata, H; Yoshida, S1
Croxton, TL; Fernandes, LB; Hirshman, CA; Lindeman, KS1
Aubier, M; Brione, E; De Vernejoul, D; Pavlovic, D1
Bonev, AD; Nelson, MT1
Kamei, K; Kuriyama, H; Nabata, H1
Alouan, LA; Armour, CL; Black, JL; Johnson, PR; Marthan, R; McKay, KO; Savineau, JP; Tunon de Lara, JM; Villanove, X1
Barth, HL; Hempelmann, RG; Mehdorn, HM; Pradel, RH; Ziegler, A1
Chapple, CR; Chess-Williams, R; Korstanje, C; Martin, SW; Radley, SC1
Bianchi, L; Boselli, C; Grana, E1
Chang, M; Cheng, C; Lee, Y; Lin, C; Sheu, J; Yen, M1
March, JE; Randall, MD1
Hiley, CR; White, R2
Berg, G; Dominiczak, AF; Hamilton, CA; McArthur, K; Reid, JL1
De Los Angeles, J; Jagadeesh, JM; Jing, L; Miller, DD; Patil, PN1
Ahmed, R; Bird, NC; Chess-Williams, R; Johnson, AG1
Brading, AF; Hashitani, H; Suzuki, H1
Brune, ME; Buckner, SA; Coghlan, M; Daza, A; Fey, TA; Gopalakrishnan, M; Milicic, I1
Badawi, JK; Bross, S; Ding, A1

Other Studies

32 other study(ies) available for carbachol and cromakalim

ArticleYear
Comparative effects of BRL 38227, nitrendipine and isoprenaline on carbachol- and histamine-stimulated phosphoinositide metabolism in airway smooth muscle.
    British journal of pharmacology, 1992, Volume: 105, Issue:4

    Topics: Animals; Benzopyrans; Carbachol; Cattle; Cromakalim; Histamine; In Vitro Techniques; Isoproterenol; Muscle, Smooth; Nitrendipine; Parasympatholytics; Phosphatidylinositols; Pyrroles; Trachea

1992
On the pharmacological and physiological role of glibenclamide-sensitive potassium channels in colonic smooth muscle.
    Pharmacology & toxicology, 1992, Volume: 71, Issue:5

    Topics: Animals; Benzopyrans; Carbachol; Colforsin; Colon; Cromakalim; Dogs; Drug Interactions; Electric Stimulation; Female; Gallopamil; Glyburide; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Stereoisomerism

1992
The inhibitory effects of cromakalim and its active enantiomer BRL 38227 against various agonists in guinea pig and human airways: comparison with pinacidil and verapamil.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:2

    Topics: Animals; Benzopyrans; Bronchi; Bronchial Spasm; Bronchodilator Agents; Carbachol; Cromakalim; Drug Interactions; Female; Guanidines; Guinea Pigs; Humans; Male; Muscle Contraction; Pinacidil; Potassium Channels; Pyrroles; Stereoisomerism; Trachea; Vasodilator Agents; Verapamil

1992
Airway pharmacology of the potassium channel opener, HOE 234, in guinea pigs: in vitro and in vivo studies.
    European journal of pharmacology, 1992, Jan-07, Volume: 210, Issue:1

    Topics: Animals; Benzopyrans; Bronchoconstrictor Agents; Bronchodilator Agents; Carbachol; Chromans; Cromakalim; Dinoprostone; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Pyrroles; Pyrrolidines; Trachea

1992
Smooth muscle relaxation and inhibition of responses to pinacidil and cromakalim induced by phentolamine in guinea-pig isolated trachea.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dinoprost; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Pinacidil; Pyrroles; SRS-A; Trachea

1992
Selective inhibition of relaxation of guinea-pig trachea by charybdotoxin, a potent Ca(++)-activated K+ channel inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2

    Topics: Aminophylline; Animals; Benzopyrans; Calcium; Carbachol; Charybdotoxin; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Guanidines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nitroprusside; Pinacidil; Potassium Channels; Pyrroles; Scorpion Venoms; Serotonin; Trachea

1990
Specific antagonism by glibenclamide of negative inotropic effects of potassium channel openers in canine atrial muscle.
    Japanese journal of pharmacology, 1990, Volume: 54, Issue:2

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dogs; Female; Glyburide; Guanidines; Heart Atria; Male; Myocardial Contraction; Niacinamide; Nicorandil; Nifedipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1990
Adrenergic-cholinergic interactions in left atria: a study using K+ channel agonists, antagonist and pertussis toxin.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 4-Aminopyridine; Animals; Benzopyrans; Carbachol; Cromakalim; Cyclic AMP; Dogs; Female; Guanidines; Heart; Isoproterenol; Male; Myocardial Contraction; Parasympathetic Nervous System; Pertussis Toxin; Phenylephrine; Pinacidil; Potassium Channels; Pyrroles; Rabbits; Sympathetic Nervous System; Virulence Factors, Bordetella

1990
Effects of cromakalim (BRL 34915) and pinacidil on normal and hypertrophied rat detrusor in vitro.
    The Journal of urology, 1990, Volume: 143, Issue:4

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Electric Stimulation; Female; Guanidines; Hypertrophy; In Vitro Techniques; Muscle Contraction; Pinacidil; Potassium; Pyrroles; Rats; Rats, Inbred Strains; Urinary Bladder; Vasodilator Agents

1990
Pertussis toxin treatment does not inhibit the effects of the potassium channel opener BRL 34915 on rat isolated vascular and cardiac tissues.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:1

    Topics: Action Potentials; Animals; Benzopyrans; Carbachol; Cromakalim; Heart; Heart Rate; In Vitro Techniques; Ion Channels; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Pertussis Toxin; Potassium; Pyrroles; Rats; Rats, Inbred Strains; Virulence Factors, Bordetella

1988
Effects of the potassium channel openers cromakalim and pinacidil on catecholamine secretion and calcium mobilization in cultured bovine adrenal chromaffin cells.
    Biochemical pharmacology, 1994, May-18, Volume: 47, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Barium; Benzopyrans; Bradykinin; Calcimycin; Calcium; Carbachol; Catecholamines; Cattle; Cells, Cultured; Cromakalim; Guanidines; Histamine; Pinacidil; Potassium; Potassium Channels; Pyrroles; Rubidium Radioisotopes

1994
Functional evidence for a glibenclamide-sensitive K+ channel in rat ileal smooth muscle.
    European journal of pharmacology, 1994, Dec-27, Volume: 271, Issue:2-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Carbachol; Cromakalim; Glyburide; Ileum; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Rats; Rats, Wistar

1994
Potassium channel blockade of atrial negative inotropic responses to P1-purinoceptor and muscarinic receptor agonists and to cromakalim.
    Journal of cardiovascular pharmacology, 1993, Volume: 21, Issue:2

    Topics: 4-Aminopyridine; Adenosine; Animals; Benzopyrans; Carbachol; Cromakalim; Depression, Chemical; Glyburide; Guinea Pigs; Heart Atria; Hydrochloric Acid; In Vitro Techniques; Male; Myocardial Contraction; Parasympatholytics; Phenylisopropyladenosine; Potassium Channels; Pyrroles; Receptors, Muscarinic; Receptors, Purinergic; Rubidium Radioisotopes

1993
Regional and species differences in glyburide-sensitive K+ channels in airway smooth muscles as estimated from actions of KC 128 and levcromakalim.
    British journal of pharmacology, 1994, Volume: 113, Issue:3

    Topics: Animals; Benzopyrans; Bronchi; Carbachol; Cromakalim; Dogs; Dose-Response Relationship, Drug; Female; Glyburide; Guinea Pigs; Humans; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Pyrroles; Species Specificity; Trachea

1994
Role of potassium channels in hypoxic relaxation of porcine bronchi in vitro.
    The American journal of physiology, 1994, Volume: 266, Issue:3 Pt 1

    Topics: Animals; Benzopyrans; Bronchi; Bronchodilator Agents; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Hypoxia; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Potassium Channels; Pyrroles; Swine

1994
Partial inhibition by epithelium of tracheal smooth muscle relaxation induced by the potassium channel activator, BRL 38227.
    British journal of pharmacology, 1993, Volume: 110, Issue:1

    Topics: Aminophylline; Animals; Benzopyrans; Biotransformation; Bronchodilator Agents; Carbachol; Cromakalim; Epithelium; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Pyrroles; Rats; Rats, Sprague-Dawley; Trachea

1993
Muscarinic inhibition of ATP-sensitive K+ channels by protein kinase C in urinary bladder smooth muscle.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Carbachol; Cromakalim; Diglycerides; Glyburide; Guanosine Diphosphate; Guinea Pigs; In Vitro Techniques; Indoles; Maleimides; Membrane Potentials; Muscarinic Antagonists; Muscle, Smooth; Potassium Channels; Protein Kinase C; Pyrroles; Receptors, Muscarinic; Tetradecanoylphorbol Acetate; Thionucleotides; Urinary Bladder

1993
Effects of KC 399, a novel ATP-sensitive K+ channel opener, on electrical and mechanical responses in dog tracheal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Carbachol; Cromakalim; Cyclic AMP; Cyclic GMP; Dogs; Female; Glyburide; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Trachea

1994
Sensitization decreases relaxation in human isolated airways.
    The American review of respiratory disease, 1993, Volume: 148, Issue:1

    Topics: Asthma; Benzopyrans; Bronchi; Bucladesine; Carbachol; Colforsin; Cromakalim; Dose-Response Relationship, Drug; Humans; Immunization, Passive; Immunoglobulin E; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle Tonus; Parasympatholytics; Pyrroles; Verapamil

1993
Effects of potassium channel openers in isolated human cerebral arteries.
    Neurosurgery, 1995, Volume: 37, Issue:6

    Topics: Benzopyrans; Calcium Channel Blockers; Carbachol; Cerebral Arteries; Cromakalim; Culture Techniques; Dose-Response Relationship, Drug; Endothelium, Vascular; Guanidines; Humans; Iloprost; Nifedipine; Nimodipine; Pinacidil; Potassium Channels; Pyrroles; Vasodilator Agents

1995
Relaxant effects of potassium-channel openers on normal and hyper-reflexic detrusor muscle.
    British journal of urology, 1997, Volume: 80, Issue:3

    Topics: Benzopyrans; Benzoxazines; Carbachol; Cromakalim; Cyclic N-Oxides; Dose-Response Relationship, Drug; Electric Stimulation; Humans; Muscle Relaxation; Oxazines; Parasympatholytics; Potassium Channels; Pyrroles; Reflex, Abnormal; Urinary Bladder

1997
Effect of cromakalim on the purinergic and cholinergic transmission in the rat detrusor muscle.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: Adenosine Triphosphate; Animals; Carbachol; Cromakalim; Electric Stimulation; In Vitro Techniques; Male; Muscle, Smooth; Nifedipine; Rats; Rats, Wistar; Receptors, Cholinergic; Receptors, Purinergic; Urinary Bladder

1997
Pharmacological characteristics of MJ-451, a new benzopyran- derived ATP-sensitive potassium channel opener, in guinea pig isolated trachea.
    Pharmacology, 1998, Volume: 57, Issue:6

    Topics: Animals; Benzopyrans; Carbachol; Cromakalim; Drug Interactions; Female; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Parasympathomimetics; Potassium Channels; Potassium Chloride; Pyrrolidinones; Trachea

1998
Characterization of endothelium-dependent relaxations in mesenteries from transgenic hypertensive rats.
    European journal of pharmacology, 1998, Sep-25, Volume: 358, Issue:1

    Topics: Animals; Animals, Genetically Modified; Carbachol; Cardiotonic Agents; Cardiovascular Physiological Phenomena; Cromakalim; Endothelium, Vascular; Enzyme Inhibitors; Female; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; NG-Nitroarginine Methyl Ester; Nitroprusside; Potassium Chloride; Rats; Rats, Sprague-Dawley; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

1998
The actions of the cannabinoid receptor antagonist, SR 141716A, in the rat isolated mesenteric artery.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Animals; Benzimidazoles; Calcium; Cannabinoids; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Relaxation; Muscle, Smooth, Vascular; Penicillamine; Piperidines; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant

1998
Does potassium channel opening contribute to endothelium-dependent relaxation in human internal thoracic artery?
    Clinical science (London, England : 1979), 1999, Volume: 96, Issue:6

    Topics: Aged; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Humans; In Vitro Techniques; Ion Channel Gating; Male; Middle Aged; Nitric Oxide Synthase; Nitroprusside; Oxadiazoles; Potassium; Potassium Channels; Quinoxalines; Thoracic Arteries; Vasodilation; Vasodilator Agents

1999
Depolarization of membrane potential and the smooth muscle contraction by isothiocyanatobenzyl imidazoline in guinea-pig stomach circular muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:3

    Topics: Animals; Atropine; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Nifedipine; Oxymetazoline; Stomach; Tolazoline; Vasodilator Agents

1999
Hyperpolarisation of rat mesenteric endothelial cells by ATP-sensitive K(+) channel openers.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Adenosine Triphosphate; Animals; Apamin; Barium Compounds; Benzimidazoles; Carbachol; Charybdotoxin; Chlorides; Cromakalim; Dose-Response Relationship, Drug; Electrophysiology; Endothelium, Vascular; Glyburide; Glycyrrhetinic Acid; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Ouabain; Potassium Channels; Rats; Rats, Wistar; Vasodilator Agents

2000
Active relaxation of human gallbladder muscle is mediated by ATP-sensitive potassium channels.
    Digestion, 2002, Volume: 65, Issue:4

    Topics: Adenosine Triphosphate; Animals; Carbachol; Cromakalim; Gallbladder; Glyburide; Guinea Pigs; Humans; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Potassium Channels; Sincalide

2002
Correlation between spontaneous electrical, calcium and mechanical activity in detrusor smooth muscle of the guinea-pig bladder.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: Action Potentials; Amides; Animals; Apamin; Boron Compounds; Calcium; Calcium Signaling; Carbachol; Charybdotoxin; Colforsin; Cromakalim; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Female; Fura-2; Guinea Pigs; Isotonic Contraction; Male; Mechanotransduction, Cellular; Microelectrodes; Muscle Contraction; Muscle, Smooth; Nifedipine; Pyridines; Transducers; Urinary Bladder

2004
Pharmacological characterization of urinary bladder smooth muscle contractility following partial bladder outlet obstruction in pigs.
    European journal of pharmacology, 2006, Feb-17, Volume: 532, Issue:1-2

    Topics: Adenosine Triphosphate; Amides; Animals; Benzophenones; Carbachol; Cholinergic Agonists; Cromakalim; Cyclic S-Oxides; Diazoxide; Dose-Response Relationship, Drug; Electric Stimulation; Female; Guanidines; Histamine; Hypertrophy; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Potassium Channels; Potassium Chloride; Pyridines; Quinolones; Serotonin; Serotonin Agents; Swine; Urinary Bladder; Urinary Bladder Neck Obstruction; Vasodilator Agents

2006
Inhibitory effects of different ATP-sensitive potassium channel openers on electrically generated and carbachol-induced contractions of porcine and human detrusor muscle.
    Fundamental & clinical pharmacology, 2008, Volume: 22, Issue:1

    Topics: Aged; Amides; Animals; Benzophenones; Carbachol; Cromakalim; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Minoxidil; Muscle Contraction; Muscle, Smooth; Pinacidil; Potassium Channels; Swine; Urinary Bladder

2008
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