Page last updated: 2024-08-17

carbachol and arecoline

carbachol has been researched along with arecoline in 90 studies

Research

Studies (90)

TimeframeStudies, this research(%)All Research%
pre-199039 (43.33)18.7374
1990's35 (38.89)18.2507
2000's13 (14.44)29.6817
2010's2 (2.22)24.3611
2020's1 (1.11)2.80

Authors

AuthorsStudies
Bymaster, FP; Honoré, T; Mitch, CH; Nielsen, S; Olesen, PH; Pike, AJ; Sauerberg, P; Sheardown, MJ; Treppendahl, S; Ward, JS1
Amstutz, R; Boelsterli, J; Bolliger, G; Floersheim, P; Gammenthaler, H; Gmelin, G; Shapiro, G; Supavilai, P; Walkinshaw, M1
Baker, R; Book, T; Freedman, SB; Marwood, RS; Patel, S; Reeve, AJ; Saunders, J; Street, LJ; Willson, T1
Baker, R; Freedman, SB; Gibbons, TL; Kneen, CO; MacLeod, AM; Merchant, K; Patel, S; Saunders, J; Showell, GA1
Baker, R; Book, T; Freedman, SB; Herbert, RH; Kneen, CO; MacLeod, AM; Merchant, KJ; Saunders, J; Showell, GA; Street, LJ1
Baker, R; Cassidy, M; Freedman, SB; Harley, EA; Iversen, LL; Kneen, C; MacLeod, AM; Merchant, KJ; Saunders, J; Snow, RJ1
Baker, R; Freedman, SB; MacLeod, AM; Merchant, KJ; Patel, S; Roe, M; Saunders, J1
Baker, R; Freedman, SB; Harley, EA; Saunders, J; Showell, GA; Snow, RJ1
Falch, E; Krogsgaard-Larsen, P; Larsen, JJ; Sauerberg, P1
Andrews, PR; Craik, DJ; Martin, JL1
Brann, MR; Bräuner-Osborne, H; Ebert, B; Falch, E; Krogsgaard-Larsen, P1
Bøgesø, KP; Frederiksen, K; Løve Lembøl, H; Meier, E; Moltzen, EK; Pedersen, H; Sánchez, C1
Dunbar, PG; Durant, GJ; el-Assadi, AA; Huzl, JJ; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Sbeih, S; Smith, DA1
Abuh, YF; Dunbar, PG; Durant, GJ; el-Assadi, AA; Fang, Z; Hoss, WP; Messer, WS; Ngur, DO; Periyasamy, S1
Abuh, YF; Dunbar, PG; Edgar, MA; El-Assadi, AA; Fang, Z; Huzl, JJ; Liu, Y; Messer, WS; Nagy, PI; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Roknich, S; Sbeih, S; Zhang, H1
Bromidge, SM; Brown, F; Cassidy, F; Clark, MS; Dabbs, S; Hadley, MS; Hawkins, J; Loudon, JM; Naylor, CB; Orlek, BS; Riley, GJ1
Badio, B; Daly, JW; Gupta, TH; Padgett, WL; Pei, XF1
Bymaster, FP; Calligaro, DO; DeLapp, NW; Fink-Jensen, A; Jeppesen, L; Olesen, PH; Rasmussen, T; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Thomsen, C; Ward, JS; Whitesitt, CA1
Daly, JW; Gupta, TH; Padgett, WL; Pei, XF1
Bodor, ET; Harden, TK; Kim, MG; Kohn, H; Wang, C1
Bruno-Blanch, L; Gálvez, J; García-Domenech, R1
Dei, S; Marconi, C; Pedretti, A; Romanelli, MN; Scapecchi, S; Vistoli, G1
Beleslin, D; Malobabić, Z; Samardzić, R1
Maayani, S; Sokolovsky, M; Treister, G1
De Montis, GM; Olianas, MC; Scheel-Krüger, J; Serra, G; Tagliamonte, A1
Green, SE; Summerfield, A1
Campbell, MD; Gala, RR; Jaques, S1
Abood, LG; Aronstam, R; Baumgold, J1
Dudar, JD; Hadházy, P; Szerb, JC1
Houser, VP1
Samoĭlovich, IM1
Gala, RR; Subramanian, MG1
Garg, LC; Mohuczy-Dominiak, D1
Dunant, Y; Sierro, CD; Vitus, J1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Aksoy, S; Gibson, VA; McKinney, M; Miller, JH; Nickelson, L1
Bockaert, J; Manzoni, OJ; Royer, M; Schmidt, BH; Sladeczek, FA1
Lambert, DG; Nahorski, SR1
Fertel, R; Hadjiconstantinou, M; Neff, NH; Qu, ZX1
Gardner, JD; Jensen, RT; Rattan, S; Sutliff, VE1
Ghataorre, AS; Lambert, DG; Nahorski, SR1
Nahorski, SR; Rooney, TA1
Channell, SL; Iversen, SD; Lalies, MD; Salamone, JD1
Reavill, C; Spivak, CE; Stolerman, IP; Waters, JA1
Barlow, RB; Weston-Smith, P1
Barker, DL; Mpitsos, GJ; Murray, TF; Siebenaller, JF1
Konno, F; Takayanagi, I1
Snyder, SH; Yamamura, HI1
Fernando, MM; Grove, DJ1
Rossen, E1
Huang, TF; Liu, HM1
Dureng, G; Labrid, C; Streichenberger, G1
Beleslin, DB; Grabović, L; Radmanović, BZ1
Aitken, ID; Parry, SH1
Lambrecht, G; Mutschler, E1
Lój, W1
Doss, J; van Zweiten, PA1
Evans, TG; Leake, LD; Walker, RJ1
Abeln, W; Bienhold, H; Flohr, H1
Baissat, J; Chassaing, C; Duchêne-Marullaz, P; Dureng, G1
Coppi, G; Leone, L; Lumachi, B; Rossini, L; Valsecchi, B1
Dishkelov, A; Iosifov, T; Ovcharov, R; Venkov, L1
Klein, WL; Shifrin, GS1
Bennett, JL; Blair, KL; Pax, RA1
Imaizumi, Y; Kawai, T; Masuda, Y; Ryang, S; Tanaka, M; Watanabe, M; Yamahara, NS1
Classen, M; Schaffer, K; Schepp, W; Schusdziarra, V; Wegner, U; Weigert, N1
Nahorski, SR; Safrany, ST1
Barzaghi, F; Bonetti, C; Cesana, R; Fortin, M; Galliani, G; Hunt, P; Maggioni, A; Nencioni, A; Parini, C; Toja, E1
Aronstam, RS; Buccafusco, JJ; Hays, AC; Lapp, CA; Shuster, LC1
Farlow, MR; Lahiri, DK1
Elazar, Z; Ganchrow, D; Paz, M1
Huang, CL; Lee, HM; Lin, CH; Tsai, KJ; Tung, CS1
Edwardson, JM; Koenig, JA; Szekeres, PG1
Gebauer, M; Versen, B1
Jaen, JC; Mirzadegan, T; Moreland, D; Schwarz, RD; Spencer, CJ; Tecle, H; Thomas, AJ1
Ball, RG; Bräuner-Osborne, H; Bøgesø, KP; Frydenvang, K; Krogsgaard-Larsen, P; Meier, E; Pedersen, H1
Gebauer, M; Schipp, R; Versen, B1
Barras, M; Bruneval, P; Corman, B; Grandadam, F; Heudes, D; Lluel, P; Martin, DJ; Palea, S1
Malomough, A; Naumenko, N; Nikolsky, E; Urazaev, A; Vyskocil, F1
Patil, PN; Stearns, R1
Drake, MJ; Gillespie, JI; Harvey, IJ1
BURGEN, AS1
Crittenden, EL; García, DM; González, A1
Bukharaeva, EA; Magazanik, LG; Nikolsky, EE; Samigullin, D; Vyskocil, F1
Drake, MJ; Gillespie, JI; Lagou, M1
De Ridder, D; Gevaert, T; Ost, D1
Finney, SM; Gillespie, JI; Stewart, LH1
Li, J; Long, CL; Pan, ZY; Wang, H; Zhang, YY1
De Wachter, S; Eastham, J; Gillespie, J; Persyn, S; Wyndaele, JJ1
Cristofaro, I; Di Bari, M; Español, AJ; Salem, A; Sales, ME; Sanchez, Y; Tata, AM1

Reviews

1 review(s) available for carbachol and arecoline

ArticleYear
The therapeutic use of cholinergic drugs acting on the vegetative nervous system. I - Direct, indirect and mixed agonists.
    Il Farmaco; edizione scientifica, 1981, Volume: 36, Issue:10

    Topics: Animals; Arecoline; Bethanechol Compounds; Carbachol; Chemical Phenomena; Chemistry; Dimethylphenylpiperazinium Iodide; Ganglia; Kinetics; Lobeline; Neuroeffector Junction; Nicotine; Oxotremorine; Parasympathomimetics; Pilocarpine; Stereoisomerism

1981

Other Studies

89 other study(ies) available for carbachol and arecoline

ArticleYear
Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3-(1,2,5-thiadiazolyl)-1,2,5,6-tetrahydro-1-methylpyridines .
    Journal of medicinal chemistry, 1992, Jun-12, Volume: 35, Issue:12

    Topics: Animals; Atrial Function; Brain; Guinea Pigs; Heart Atria; Male; Molecular Structure; Myocardial Contraction; Parasympathomimetics; Pyridines; Rabbits; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Thiadiazoles

1992
Muscarinic activity of the thiolactone, lactam, lactol, and thiolactol analogues of pilocarpine and a hypothetical model for the binding of agonists to the m1 receptor.
    Journal of medicinal chemistry, 1992, Volume: 35, Issue:1

    Topics: Animals; Binding, Competitive; Crystallography; Guinea Pigs; Lactams; Male; Mice; Models, Biological; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Sulfhydryl Compounds

1992
Synthesis and muscarinic activity of quinuclidinyl- and (1-azanorbornyl)pyrazine derivatives.
    Journal of medicinal chemistry, 1992, Jan-24, Volume: 35, Issue:2

    Topics: Animals; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Norbornanes; Parasympathomimetics; Pyrazines; Quinuclidines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1992
Tetrahydropyridyloxadiazoles: semirigid muscarinic ligands.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:3

    Topics: Animals; Binding Sites; Chemical Phenomena; Chemistry; Crystallization; Hydrogen Bonding; Male; Molecular Conformation; Molecular Structure; Oxadiazoles; Parasympathomimetics; Pyridines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Structure-Activity Relationship; Thermodynamics; X-Ray Diffraction

1991
Synthesis and biological activity of 1,2,4-oxadiazole derivatives: highly potent and efficacious agonists for cortical muscarinic receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:10

    Topics: Animals; Cerebral Cortex; In Vitro Techniques; Ligands; Oxadiazoles; Parasympathomimetics; Rats; Receptors, Muscarinic; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

1990
Novel quinuclidine-based ligands for the muscarinic cholinergic receptor.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:4

    Topics: Animals; Binding Sites; Cerebral Cortex; Computer Simulation; Kinetics; Models, Chemical; Oxadiazoles; Quinuclidines; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1990
Synthesis and muscarinic activities of 1,2,4-thiadiazoles.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:7

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Indicators and Reagents; Kinetics; Ligands; Models, Molecular; Molecular Structure; N-Methylscopolamine; Oxotremorine; Parasympathomimetics; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Structure-Activity Relationship; Thiadiazoles; X-Ray Diffraction

1990
2-Methyl-1,3-dioxaazaspiro[4.5]decanes as novel muscarinic cholinergic agonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Dioxolanes; Dioxoles; In Vitro Techniques; Inositol Phosphates; Male; Molecular Conformation; N-Methylscopolamine; Oxotremorine; Parasympathomimetics; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Spiro Compounds; Structure-Activity Relationship

1988
A novel class of conformationally restricted heterocyclic muscarinic agonists.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:6

    Topics: Animals; Brain; Guinea Pigs; Ileum; In Vitro Techniques; Molecular Conformation; Parasympathomimetics; Propylbenzilylcholine Mustard; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Tritium

1986
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors.
    Journal of medicinal chemistry, 1995, Jun-09, Volume: 38, Issue:12

    Topics: 3T3 Cells; Animals; Arecoline; Cerebral Cortex; Heterocyclic Compounds; Humans; In Vitro Techniques; Mice; Muscarinic Agonists; Protein Binding; Rats; Receptors, Muscarinic; Recombinant Proteins

1995
Bioisosteres of arecoline: 1,2,3,6-tetrahydro-5-pyridyl-substituted and 3-piperidyl-substituted derivatives of tetrazoles and 1,2,3-triazoles. Synthesis and muscarinic activity.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Arecoline; Female; Guinea Pigs; Male; Mice; Rats; Rats, Wistar; Structure-Activity Relationship; Tetrazoles; Triazoles

1994
Design, synthesis, and neurochemical evaluation of 2-amino-5-(alkoxycarbonyl)-3,4,5,6-tetrahydropyridines and 2-amino-5-(alkoxycarbonyl)-1,4,5,6-tetrahydropyrimidines as M1 muscarinic receptor agonists.
    Journal of medicinal chemistry, 1994, Aug-19, Volume: 37, Issue:17

    Topics: Alzheimer Disease; Animals; Cerebral Cortex; Drug Design; Humans; In Vitro Techniques; Indicators and Reagents; Inositol; Isomerism; Kinetics; Magnetic Resonance Spectroscopy; Mass Spectrometry; Models, Molecular; Molecular Conformation; Molecular Structure; Parasympathomimetics; Phosphatidylinositols; Pyridines; Pyrimidines; Rats; Receptors, Muscarinic; Spectrophotometry, Infrared; Structure-Activity Relationship

1994
Design, synthesis, and neurochemical evaluation of 5-(3-alkyl-1,2,4- oxadiazol-5-yl)-1,4,5,6-tetrahydropyrimidines as M1 muscarinic receptor agonists.
    Journal of medicinal chemistry, 1993, Apr-02, Volume: 36, Issue:7

    Topics: Animals; Binding Sites; Brain; Oxadiazoles; Parasympathomimetics; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Structure-Activity Relationship

1993
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
    Journal of medicinal chemistry, 1997, Apr-11, Volume: 40, Issue:8

    Topics: Animals; Arecoline; Brain; Carbachol; Cell Line; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship

1997
Design of [R-(Z)]-(+)-alpha-(methoxyimino)-1-azabicyclo[2.2.2]octane-3-acetonitri le (SB 202026), a functionally selective azabicyclic muscarinic M1 agonist incorporating the N-methoxy imidoyl nitrile group as a novel ester bioisostere.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Alzheimer Disease; Animals; Binding Sites; Blood Pressure; Brain; CHO Cells; Cricetinae; Electroencephalography; Heart Rate; Humans; Imines; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Structure; Muscarinic Agonists; Protein Binding; Quinuclidines; Rats; Rats, Inbred Strains; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Proteins; Stereoisomerism; Tremor

1997
6beta-Acetoxynortropane: a potent muscarinic agonist with apparent selectivity toward M2-receptors.
    Journal of medicinal chemistry, 1998, Jun-04, Volume: 41, Issue:12

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cerebral Cortex; CHO Cells; Cricetinae; Enzyme Inhibitors; Guanosine Triphosphate; Humans; Muscarinic Agonists; Nortropanes; Phosphatidylinositols; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Receptors, Muscarinic; Receptors, Nicotinic; Structure-Activity Relationship

1998
Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic m1 receptor activation.
    Bioorganic & medicinal chemistry letters, 1998, Oct-20, Volume: 8, Issue:20

    Topics: Animals; Cells, Cultured; CHO Cells; Cricetinae; Humans; Inhibitory Concentration 50; Muscarinic Agonists; Pyridines; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Structure-Activity Relationship; Thiadiazoles; Transfection

1998
6beta-Acyloxy(nor)tropanes: affinities for antagonist/agonist binding sites on transfected and native muscarinic receptors.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding Sites; Cerebral Cortex; CHO Cells; Cricetinae; Humans; In Vitro Techniques; Muscarinic Agonists; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Receptors, Muscarinic; Transfection; Tropanes

2000
C(8) substituted 1-azabicyclo[3.3.1]non-3-enes and C(8) substituted 1-azabicyclo[3.3.1]nonan-4-ones: novel muscarinic receptor antagonists.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Crystallography, X-Ray; Humans; Inositol Phosphates; Magnetic Resonance Spectroscopy; Membranes; Muscarinic Antagonists; Radioligand Assay; Stereoisomerism; Structure-Activity Relationship

2003
Topological virtual screening: a way to find new anticonvulsant drugs from chemical diversity.
    Bioorganic & medicinal chemistry letters, 2003, Aug-18, Volume: 13, Issue:16

    Topics: Anticonvulsants; Computer Simulation; Databases, Factual; Discriminant Analysis; Drug Design; Molecular Structure; Quantitative Structure-Activity Relationship

2003
Docking analyses on human muscarinic receptors: unveiling the subtypes peculiarities in agonists binding.
    Bioorganic & medicinal chemistry, 2008, Mar-15, Volume: 16, Issue:6

    Topics: Binding Sites; Computer Simulation; Humans; Ligands; Muscarinic Agonists; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M5; Receptors, Muscarinic

2008
[Pharmacological analysis of the inhibition of peristalsis of the isolated guinea-pig ileum by tetramethylammonium].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1976, Volume: 170, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Female; Gastrointestinal Motility; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Neostigmine; Nicotine; Physostigmine; Pilocarpine; Quaternary Ammonium Compounds; Serotonin

1976
Drugs affecting the cholinergic system in the intact mammalian eye. I. Evaluation of the miotic activity of acetylcholine-like drugs in the mouse eye.
    Investigative ophthalmology, 1975, Volume: 14, Issue:3

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Guinea Pigs; Hydrogen-Ion Concentration; Miotics; Oxotremorine; Phencyclidine; Pupil; Quinuclidines

1975
Evidence that a nigral gabaergic--cholinergic balance controls posture.
    European journal of pharmacology, 1979, Jan-01, Volume: 53, Issue:2

    Topics: Animals; Apomorphine; Arecoline; Behavior, Animal; Carbachol; Catalepsy; Choline O-Acetyltransferase; gamma-Aminobutyric Acid; Haloperidol; Humans; Kainic Acid; Male; Posture; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Stereotyped Behavior; Substantia Nigra

1979
Central and peripheral cholinergic involvement in the habituation of investigatory head poking in rats.
    Journal of comparative and physiological psychology, 1977, Volume: 91, Issue:6

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Cholinergic Fibers; Exploratory Behavior; Habituation, Psychophysiologic; Male; Motor Activity; Nervous System Physiological Phenomena; Nicotine; Rats; Scopolamine; Scopolamine Derivatives

1977
The lack of an effect of cholinergic agonists on anterior pituitary prolactin production in vitro.
    Experientia, 1978, Nov-15, Volume: 34, Issue:11

    Topics: Animals; Arecoline; Carbachol; Dopamine; Female; In Vitro Techniques; Nicotine; Parasympathomimetics; Pituitary Gland, Anterior; Prolactin; Rats

1978
Studies on the relationship of binding affinity to psychoactive and anticholingergic potency of a group of psychotomimetic glycolates.
    Brain research, 1977, Mar-25, Volume: 124, Issue:2

    Topics: Animals; Arecoline; Atropine; Binding Sites; Binding, Competitive; Brain; Carbachol; Chemical Phenomena; Chemistry; Dose-Response Relationship, Drug; Glycolates; Hallucinogens; Kinetics; Male; Parasympatholytics; Phosphatidylserines; Quinuclidines; Rats; Receptors, Drug; Scopolamine; Stereoisomerism; Structure-Activity Relationship

1977
Release of [3H]acetylcholine from rat hippocampal slices: effect of septal lesion and of graded concentrations of muscarnic agonists and antagonists.
    Brain research, 1977, Jun-10, Volume: 128, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Carbachol; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Mecamylamine; Oxotremorine; Pilocarpine; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Septum Pellucidum

1977
Modulation of the aversive qualities of shock through a central inhibitory cholinergic system in the rat.
    Pharmacology, biochemistry, and behavior, 1976, Volume: 4, Issue:5

    Topics: Animals; Arecoline; Atropine; Avoidance Learning; Carbachol; Electroshock; Male; Neostigmine; Nicotine; Parasympathetic Nervous System; Pilocarpine; Rats; Scopolamine; Time Factors

1976
[Correlation analysis in studying the mechanism of action of smooth muscle stimulants].
    Biulleten' eksperimental'noi biologii i meditsiny, 1976, Volume: 81, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Barium; Carbachol; Magnesium; Muscle, Smooth; Parasympathomimetics; Pilocarpine; Rats; Serotonin; Stimulation, Chemical; Stomach

1976
The influence of cholinergic, adrenergic, and serotonergic drugs on the afternoon surge of plasma prolactin in ovariectomized, estrogen-treated rats.
    Endocrinology, 1976, Volume: 98, Issue:4

    Topics: Animals; Arecoline; Atropine; Carbachol; Castration; Circadian Rhythm; Estradiol; Female; Methysergide; Nicotine; Parasympathomimetics; Phenoxybenzamine; Phentolamine; Prolactin; Propranolol; Rats; Sympathomimetics; Time Factors

1976
Characterization of cholinergic receptors in Madin-Darby canine kidney cells.
    Journal of the American Society of Nephrology : JASN, 1992, Volume: 3, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Cell Line; Cyclic AMP; Dogs; Hydrolysis; Inositol Phosphates; Kidney; Proteins; Quinuclidinyl Benzilate; Receptors, Muscarinic

1992
Effects of muscarinic agonists and depolarizing agents on inositol monophosphate accumulation in the rabbit vagus nerve.
    Journal of neurochemistry, 1992, Volume: 59, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Cadmium; Calcimycin; Calcium; Carbachol; Dose-Response Relationship, Drug; Hydrolysis; Inositol Phosphates; Lithium; Ouabain; Oxotremorine; Parasympathomimetics; Pirenzepine; Potassium; Rabbits; Receptors, Muscarinic; Time Factors; Vagus Nerve

1992
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Interactions of agonists with M2 and M4 muscarinic receptor subtypes mediating cyclic AMP inhibition.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Cells, Cultured; CHO Cells; Corpus Striatum; Cricetinae; Cyclic AMP; Kinetics; Male; Muscarine; Oxotremorine; Pilocarpine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1991
Cholinergic inositol phosphate formation in striatal neurons is mediated by distinct mechanisms.
    European journal of pharmacology, 1991, Feb-25, Volume: 206, Issue:2

    Topics: Animals; Arecoline; Calcium; Carbachol; Corpus Striatum; In Vitro Techniques; Inositol Phosphates; Mice; Muscarine; Neurons; Receptors, Muscarinic; Tetrodotoxin

1991
Muscarinic-receptor-mediated changes in intracellular Ca2+ and inositol 1,4,5-trisphosphate mass in a human neuroblastoma cell line, SH-SY5Y.
    The Biochemical journal, 1990, Jan-15, Volume: 265, Issue:2

    Topics: Arecoline; Atropine; Benzofurans; Calcium; Carbachol; Cell Line; Fluorescent Dyes; Fura-2; Humans; Inositol 1,4,5-Trisphosphate; Ionomycin; Kinetics; Manganese; Muscarine; Neuroblastoma; Receptors, Muscarinic; Tumor Cells, Cultured

1990
Pharmacological characterization of muscarinic receptors mediating inhibition of adenylate cyclase activity in the rat retina.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Arecoline; Aziridines; Carbachol; Choline; Colforsin; Cyclic AMP; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Retina

1988
Characterization of cholinergic receptors mediating pepsinogen secretion from chief cells.
    The American journal of physiology, 1989, Volume: 257, Issue:2 Pt 1

    Topics: Acetylcholine; Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscarine; Pepsinogens; Propylbenzilylcholine Mustard; Receptors, Muscarinic; Scopolamine

1989
Muscarinic receptor binding characteristics of a human neuroblastoma SK-N-SH and its clones SH-SY5Y and SH-EP1.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Arecoline; Atropine; Carbachol; Cell Membrane; Humans; Neuroblastoma; Piperidines; Pirenzepine; Receptors, Muscarinic; Tumor Cells, Cultured

1989
Postnatal ontogeny of agonist and depolarization-induced phosphoinositide hydrolysis in rat cerebral cortex.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:1

    Topics: Aging; Animals; Arecoline; Calcium Channel Blockers; Carbachol; Cerebral Cortex; Hydrolysis; Male; N-Methylscopolamine; Norepinephrine; Phosphatidylinositols; Physostigmine; Potassium; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Scopolamine Derivatives

1987
Behavioural and pharmacological characterization of the mouth movements induced by muscarinic agonists in the rat.
    Psychopharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Arecoline; Brain; Carbachol; Male; Motor Activity; Mouth; Oxotremorine; Parasympathomimetics; Pilocarpine; Rats; Rats, Inbred Strains; Scopolamine

1986
Isoarecolone can inhibit nicotine binding and produce nicotine-like discriminative stimulus effects in rats.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Anura; Arecoline; Brain; Carbachol; Discrimination, Psychological; Male; Muscle Contraction; Nicotine; Rats; Rats, Inbred Strains

1987
The relative potencies of some agonists at M2 muscarinic receptors in guinea-pig ileum, atria and bronchi.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Atrial Function; Bronchi; Carbachol; Choline; Guinea Pigs; Heart Rate; Ileum; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Myocardial Contraction; Neostigmine; Receptors, Muscarinic

1985
Characterization of muscarinic cholinergic receptors in the crab nervous system.
    Journal of neurochemistry, 1986, Volume: 46, Issue:2

    Topics: Animals; Arecoline; Binding, Competitive; Brachyura; Carbachol; Decamethonium Compounds; Kinetics; Male; Mathematics; Nervous System; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Stereoisomerism; Tissue Distribution; Tubocurarine

1986
Muscarinic acetylcholine receptors in the rabbit ciliary body smooth muscle: spare receptors and threshold phenomenon.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:1

    Topics: Animals; Arecoline; Atropine; Carbachol; Ciliary Body; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxotremorine; Phenoxybenzamine; Pilocarpine; Rabbits; Receptors, Muscarinic

1985
Muscarinic cholinergic binding in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1974, Volume: 71, Issue:5

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Binding Sites; Binding, Competitive; Brain; Brompheniramine; Carbachol; Chlorpheniramine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Microsomes; Mitochondria; Oxotremorine; Pilocarpine; Quaternary Ammonium Compounds; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Temperature; Time Factors; Tritium

1974
Melanophore aggregation in the plaice (Pleuronectes platessa L) II. In vitro effects of adrenergic drugs.
    Comparative biochemistry and physiology. A, Comparative physiology, 1974, Aug-01, Volume: 48, Issue:4

    Topics: Acetylcholine; Adaptation, Physiological; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arecoline; Atropine; Calcium; Carbachol; Catecholamines; Chromatophores; Dopamine; Epinephrine; Fishes; Guanethidine; Histamine; Isoproterenol; Melanins; Norepinephrine; Phentolamine; Pilocarpine; Potassium; Reserpine; Skin; Tyramine

1974
Proceedings: Recovery of the contractility of isolated guinea-pig following removal of cholinomimetics.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:Suppl

    Topics: Animals; Arecoline; Calcium; Carbachol; Depression, Chemical; Electric Stimulation; Guinea Pigs; Heart Atria; In Vitro Techniques; Ouabain; Parasympathomimetics; Pyrrolidines; Temperature; Time Factors

1974
Algesic actions of the polypeptides and other agents.
    The Chinese journal of physiology, 1972, Dec-31, Volume: 21, Issue:2

    Topics: Angiotensin II; Animals; Arecoline; Bradykinin; Carbachol; Catecholamines; Dogs; Dopamine; Epinephrine; Injections, Intra-Arterial; Injections, Intraperitoneal; Methacholine Compounds; Norepinephrine; Oxytocin; Pain; Parasympathomimetics; Peptides; Reaction Time; Sensory Receptor Cells; Splenic Artery; Vasopressins

1972
[Interaction of N-methyl and N-butyl scopolammonium and some parasympathomimetics on cholinergic receptors in the jejunum of the rat].
    Archives internationales de pharmacodynamie et de therapie, 1974, Volume: 210, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Jejunum; Muscle Contraction; Parasympathomimetics; Physostigmine; Quaternary Ammonium Compounds; Rats; Receptors, Cholinergic; Scopolamine; Scopolamine Derivatives

1974
The pharmacology fo gross behavioural effects of cholinomimetic substances injected into the cerebral ventricles of unanaesthetized cats: evidence for central muscarinic mediation.
    Neuropharmacology, 1974, Volume: 13, Issue:12

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Autonomic Nervous System; Behavior, Animal; Carbachol; Cats; Cerebral Ventricles; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Emotions; Female; Gallamine Triethiodide; Hexamethonium Compounds; Injections; Male; Methacholine Compounds; Motor Activity; Nicotine; Parasympathetic Nervous System; Parasympathomimetics; Pilocarpine; Quaternary Ammonium Compounds; Scopolamine; Tubocurarine

1974
Stimulation of lachrymation and salivation in the adult fowl (Gallus domesticus).
    Research in veterinary science, 1972, Volume: 13, Issue:5

    Topics: Animals; Arecoline; Atropine; Carbachol; Chickens; Female; Injections, Intramuscular; Irritants; Lacrimal Apparatus; Neostigmine; Parasympathomimetics; Physostigmine; Pilocarpine; Saliva; Secretory Rate; Spasm; Stimulation, Chemical; Tears

1972
[Structure-activity relationships of isoarecaidine esters].
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:10

    Topics: Animals; Arecoline; Atropine; Blood Pressure; Carbachol; Depression, Chemical; Dose-Response Relationship, Drug; Esters; Female; Guinea Pigs; Heart Atria; Heart Rate; Hydrogenation; Ileum; In Vitro Techniques; Isomerism; Male; Muscle Contraction; Rats; Structure-Activity Relationship; Sympathomimetics

1973
Pharmacological analysis of regulation of the intestinal blood flow in sheep. The effect of parasympathicomimetic drugs.
    Acta physiologica Polonica, 1974, Volume: 25, Issue:3

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Injections, Intra-Arterial; Intestine, Small; Parasympathomimetics; Physostigmine; Picrotoxin; Regional Blood Flow; Sheep; Vagotomy; Vagus Nerve

1974
Cholinergic receptors involved in the production of gastric acid.
    Archives internationales de pharmacodynamie et de therapie, 1972, Volume: 197, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Blood Pressure; Carbachol; Gastric Juice; Gastric Mucosa; Hydrogen-Ion Concentration; Isoflurophate; Male; Methacholine Compounds; Neostigmine; Parasympathomimetics; Pilocarpine; Rats; Receptors, Cholinergic; Receptors, Drug; Salivation; Tremorine

1972
The action of cholinergic drugs on the heart-beat of the limpet, Patella vulgata.
    Comparative and general pharmacology, 1971, Volume: 2, Issue:5

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Choline; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Heart Rate; Lobeline; Mollusca; Nicotine; Parasympatholytics; Perfusion

1971
Influence of cholinomimetics and cholinolytics on vestibular compensation.
    Brain research, 1981, Oct-19, Volume: 222, Issue:2

    Topics: Animals; Arecoline; Bethanechol; Bethanechol Compounds; Carbachol; Ear, Inner; Methacholine Chloride; Methacholine Compounds; Muscarine; Nicotine; Oxotremorine; Rana temporaria; Vestibule, Labyrinth

1981
Pharmacological evidence for cardiac muscarinic receptor subtypes.
    Life sciences, 1984, Oct-22, Volume: 35, Issue:17

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzodiazepinones; Binding Sites; Butylscopolammonium Bromide; Carbachol; Female; Guinea Pigs; Heart Rate; Male; Myocardial Contraction; Myocardium; N-Methylscopolamine; Pirenzepine; Quaternary Ammonium Compounds; Receptors, Muscarinic; Scopolamine Derivatives

1984
[Changes in the brain content of lipids and the fatty acid composition after treatment with carbachol, arecoline, and nicotine].
    Eksperimentalna meditsina i morfologiia, 1982, Volume: 21, Issue:1

    Topics: Animals; Arecoline; Brain Chemistry; Carbachol; Fatty Acids; Nicotine; Parasympathomimetics; Phospholipids; Rats; Rats, Inbred Strains

1982
Regulation of muscarinic acetylcholine receptor concentration in cloned neuroblastoma cells.
    Journal of neurochemistry, 1980, Volume: 34, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Cell Line; Clone Cells; Dose-Response Relationship, Drug; Kinetics; Mice; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic

1980
Serotonin and acetylcholine: further analysis of praziquantel-induced contraction of magnesium-paralysed Schistosoma mansoni.
    Parasitology, 1993, Volume: 107 ( Pt 4)

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Amifampridine; Animals; Arecoline; Carbachol; Colforsin; Dose-Response Relationship, Drug; In Vitro Techniques; Ions; Magnesium; Male; Muscle Contraction; Paralysis; Phorbol 12,13-Dibutyrate; Praziquantel; Schistosoma mansoni; Serotonin

1993
Characterization of muscarinic receptors mediating relaxation and contraction in the rat iris dilator muscle.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Alkaloids; Animals; Arecoline; Bethanechol; Carbachol; Diamines; Dose-Response Relationship, Drug; Furans; Ganglia, Parasympathetic; Ganglionectomy; Iris; Male; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1995
Functional characterization of a muscarinic receptor stimulating gastrin release from rabbit antral G-cells in primary culture.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Arecoline; Atropine; Benzodiazepinones; Carbachol; Cell Adhesion; Cell Separation; Cells, Cultured; Gastrins; Immunohistochemistry; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Rabbits; Receptors, Muscarinic

1994
A comparison between muscarinic receptor occupancy, inositol 1,4,5-trisphosphate accumulation and Ca2+ mobilization in permeabilized SH-SY5Y neuroblastoma cells.
    Neuropharmacology, 1994, Volume: 33, Issue:7

    Topics: Arecoline; Brain Neoplasms; Calcium; Calcium Radioisotopes; Carbachol; Guanine Nucleotides; Humans; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Neuroblastoma; Oxotremorine; Patch-Clamp Techniques; Receptors, Muscarinic; Signal Transduction; Tumor Cells, Cultured

1994
New classes of antimuscarinic agents endowed with selective antispasmodic properties. 1-Arylsulfonyl pyrrolidin-2-ones and 2-thiones, 1-arylsulfonyl piperidin-2-ones and 2-thiones and 1-arylsulfonyl hexahydro-2H-azepin-2-one.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:4

    Topics: Animals; Arecoline; Atropine; Azepines; Butylscopolammonium Bromide; Carbachol; Gastric Acid; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pupil; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Scopolamine Derivatives; Sulfones

1994
Role of prostanoids in the regulation of central cholinergic receptor sensitivity.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Animals; Arecoline; Blood Pressure; Body Temperature; Brain; Carbachol; Central Nervous System; Indomethacin; Male; Meclofenamic Acid; Physostigmine; Prostaglandins; Rats; Rats, Wistar; Receptors, Cholinergic; Receptors, Muscarinic; Sensitivity and Specificity

1993
Differential effect of tacrine and physostigmine on the secretion of the beta-amyloid precursor protein in cell lines.
    Journal of molecular neuroscience : MN, 1996,Spring, Volume: 7, Issue:1

    Topics: Amyloid beta-Protein Precursor; Animals; Arecoline; Astrocytes; Atropine; Calcimycin; Carbachol; Cholinesterase Inhibitors; Enzyme Inhibitors; HeLa Cells; Humans; Ionophores; Muscarinic Agonists; Muscarinic Antagonists; Neuroblastoma; PC12 Cells; Physostigmine; Rats; Staurosporine; Tacrine

1996
Pontine reticular formation is involved in catalepsy produced by cholinergic drugs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Animals; Arecoline; Atropine; Carbachol; Catalepsy; Cholinergic Agents; Drug Interactions; Injections, Intraperitoneal; Kainic Acid; Male; Microinjections; Physostigmine; Rats; Reticular Formation; Stereotaxic Techniques; Thalamic Nuclei

1997
Arecoline desensitizes carbachol-stimulated phosphatidylinositol breakdown in rat brain cortices.
    Journal of neurochemistry, 1998, Volume: 70, Issue:3

    Topics: Animals; Arecoline; Carbachol; Cerebral Cortex; Female; GTP-Binding Proteins; Inositol Phosphates; Muscarinic Agonists; N-Methylscopolamine; Organ Culture Techniques; Parasympatholytics; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Tritium

1998
The relationship between agonist intrinsic activity and the rate of endocytosis of muscarinic receptors in a human neuroblastoma cell line.
    Molecular pharmacology, 1998, Volume: 53, Issue:4

    Topics: Arecoline; Bethanechol; Carbachol; Endocytosis; Humans; Kinetics; Ligands; Methacholine Chloride; Muscarinic Agonists; Neuroblastoma; Oxotremorine; Pilocarpine; Receptor, Muscarinic M3; Receptors, Muscarinic; Tumor Cells, Cultured

1998
Cholinergic mechanisms in the neurocontrol of the branchial heart of the cephalopod Sepia officinalis L.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1998, Volume: 119, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Branchial Region; Bungarotoxins; Carbachol; Dose-Response Relationship, Drug; Heart; Hexamethonium; Mollusca; Muscarine; Nicotine; Oxotremorine; Pilocarpine; Receptors, Cholinergic; Tetraethylammonium; Tubocurarine

1998
Mutations of aspartate 103 in the Hm2 receptor and alterations in receptor binding properties of muscarinic agonists.
    Life sciences, 1995, Volume: 56, Issue:11-12

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Alanine; Amino Acid Substitution; Animals; Arecoline; Asparagine; Aspartic Acid; Carbachol; COS Cells; Muscarinic Agonists; Mutagenesis, Site-Directed; Oxotremorine; Pilocarpine; Receptor, Muscarinic M2; Receptors, Muscarinic; Transfection

1995
Synthesis and muscarinic receptor pharmacology of a series of 4,5,6,7-tetrahydroisothiazolo[4,5-c]pyridine bioisosteres of arecoline.
    Bioorganic & medicinal chemistry, 1999, Volume: 7, Issue:5

    Topics: Animals; Arecoline; Brain; Carbachol; Crystallography, X-Ray; Dose-Response Relationship, Drug; Humans; Models, Chemical; Models, Molecular; Myocardium; Pyridines; Rats; Receptors, Muscarinic

1999
Inhibitory cholinergic effects on the autonomously contractile bulbus cordis branchialis of the cephalopod Sepia officinalis L.
    General pharmacology, 1999, Volume: 33, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Bungarotoxins; Carbachol; Cholinergic Agents; Cholinergic Agonists; Cholinergic Antagonists; Female; Heart; Male; Mollusca; Muscarine; Myocardial Contraction; Nicotine; Oxotremorine; Pilocarpine; Quinuclidinyl Benzilate

1999
Functional and morphological modifications of the urinary bladder in aging female rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 278, Issue:4

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Aging; Animals; Arecoline; Carbachol; Cholinergic Agonists; Consciousness; Female; Isoproterenol; Muscle Contraction; Muscle, Smooth; Norepinephrine; Organ Size; Phenylephrine; Potassium Chloride; Rats; Rats, Wistar; Urinary Bladder; Urodynamics

2000
Carbachol and acetylcholine delay the early postdenervation depolarization of muscle fibres through M1-cholinergic receptors.
    Neuroscience research, 2000, Volume: 37, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Carbachol; Culture Techniques; Diaphragm; Male; Membrane Potentials; Muscarinic Agonists; Muscarinic Antagonists; Muscle Denervation; Muscle Fibers, Skeletal; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic

2000
Mechanism of vascular relaxation by cholinomimetic drugs with special reference to pilocarpine and arecoline.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2002, Volume: 18, Issue:1

    Topics: Animals; Arecoline; Atropine; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; In Vitro Techniques; Latanoprost; Phenylephrine; Physostigmine; Pilocarpine; Prostaglandins F, Synthetic; Rats; Vasodilation; Vasodilator Agents

2002
Agonist- and nerve-induced phasic activity in the isolated whole bladder of the guinea pig: evidence for two types of bladder activity.
    Experimental physiology, 2003, Volume: 88, Issue:3

    Topics: Anesthetics, Local; Animals; Arecoline; Atropine; Carbachol; Cholinergic Agonists; Electric Stimulation; Female; Guinea Pigs; Hexamethonium; Lobeline; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Nicotinic Agonists; Nicotinic Antagonists; Stimulation, Chemical; Tetrodotoxin; Urinary Bladder

2003
THE COMPARATIVE ACTIVITY OF ARECOLINE AND ARECOLINE N-METHO SALT.
    The Journal of pharmacy and pharmacology, 1964, Volume: 16

    Topics: Animals; Anura; Arecoline; Carbachol; Guinea Pigs; Muscle, Smooth; Muscles; Parasympathomimetics; Pharmacology; Research

1964
Activation of muscarinic acetylcholine receptors elicits pigment granule dispersion in retinal pigment epithelium isolated from bluegill.
    BMC neuroscience, 2004, Jul-13, Volume: 5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Arecoline; Atropine; Carbachol; Colforsin; Cyclic AMP; Cytoplasmic Granules; Light; Muscarinic Agonists; Muscarinic Antagonists; Perciformes; Pigment Epithelium of Eye; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Retinal Pigments; Second Messenger Systems; Tropicamide

2004
Cholinergic regulation of the evoked quantal release at frog neuromuscular junction.
    The Journal of physiology, 2004, Oct-01, Volume: 560, Issue:Pt 1

    Topics: Acetylcholine; Action Potentials; Animals; Arecoline; Carbachol; Cholinergic Agonists; Diamines; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Neural Conduction; Neuromuscular Junction; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Parasympatholytics; Pirenzepine; Rana ridibunda; Receptors, Muscarinic; Synaptic Transmission; Tubocurarine

2004
Volume-induced effects on the isolated bladder: a possible local reflex.
    BJU international, 2004, Volume: 94, Issue:9

    Topics: Animals; Arecoline; Autonomic Nervous System; Carbachol; Electrophysiology; Female; Guinea Pigs; In Vitro Techniques; Muscarinic Agonists; Pressure; Reflex, Stretch; Tetrodotoxin; Urinary Bladder; Vesico-Ureteral Reflux

2004
Comparison study of autonomous activity in bladders from normal and paraplegic rats.
    Neurourology and urodynamics, 2006, Volume: 25, Issue:4

    Topics: Animals; Arecoline; Carbachol; Cholinergic Agonists; Female; Muscarinic Agonists; Muscle Contraction; Paraplegia; Pressure; Rats; Rats, Wistar; Urinary Bladder; Urinary Bladder, Neurogenic; Urodynamics

2006
Cholinergic activation of phasic activity in the isolated bladder: possible evidence for M3- and M2-dependent components of a motor/sensory system.
    BJU international, 2007, Volume: 100, Issue:3

    Topics: Animals; Arecoline; Benzofurans; Carbachol; Cholinergic Agonists; Female; Guinea Pigs; Muscarinic Agonists; Piperidines; Pyrrolidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder; Urination

2007
Non-neuronal muscarinic receptor activation prevents apoptosis of endothelial cells induced by homocysteine.
    Zhongguo ying yong sheng li xue za zhi = Zhongguo yingyong shenglixue zazhi = Chinese journal of applied physiology, 2013, Volume: 29, Issue:6

    Topics: Animals; Aorta; Apoptosis; Apoptosis Regulatory Proteins; Arecoline; Carbachol; Cell Cycle; Endoplasmic Reticulum; Endothelial Cells; Homocysteine; Mitochondria; Rats; Receptors, Muscarinic

2013
The actions of isoprenaline and mirabegron in the isolated whole rat and guinea pig bladder.
    Autonomic neuroscience : basic & clinical, 2016, Volume: 198

    Topics: Acetanilides; Animals; Arecoline; Carbachol; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Muscarinic Agonists; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder

2016
The metronomic combination of paclitaxel with cholinergic agonists inhibits triple negative breast tumor progression. Participation of M2 receptor subtype.
    PloS one, 2020, Volume: 15, Issue:9

    Topics: Administration, Metronomic; Animals; Antineoplastic Combined Chemotherapy Protocols; Arecoline; ATP Binding Cassette Transporter, Subfamily G, Member 2; Carbachol; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Cholinergic Agonists; Down-Regulation; ErbB Receptors; Female; Gene Expression Regulation, Neoplastic; Humans; Mice; Neoplasm Proteins; Neovascularization, Pathologic; Paclitaxel; Receptor, Muscarinic M2; RNA, Small Interfering; Triple Negative Breast Neoplasms; Vascular Endothelial Growth Factor A; Xenograft Model Antitumor Assays

2020