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carbachol and 8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate

carbachol has been researched along with 8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19909 (42.86)18.7374
1990's8 (38.10)18.2507
2000's4 (19.05)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Nakagawa-Yagi, Y; Nakamura, H; Saito, Y; Takada, Y1
Morley, P; Schwartz, JL; Tsang, BK; Whitfield, JF1
Matsui, S; Matsumoto, Y; Tanimura, A; Tojyo, Y2
Melvin, JE; Zhang, GH2
Blanchard, LM; Larose, L; Morisset, J; Paquette, B1
De Pont, JJ; Van Nooij, IG; Willems, PH1
Axelrod, J; Felder, CC; Kanterman, RY; Ma, AL1
Cusolito, S; Donowitz, M; Sharp, GW1
Cosowsky, L; Raufman, JP1
Armour, C; Black, J; Johnson, P; Vincenc, K1
Dartt, DA; Donowitz, M; Joshi, VM; Rose, PE; Sharp, GW1
Fujino, M; Ikeda, M; Nagai, M; Niwa, H; Oka, H; Suzuki, H; Suzuki, S1
Kennedy, JA; Roberts, ML; Tennes, KA1
Ishii, K; Kato, R; Sasakawa, N; Yamamoto, S1
Greger, R; Leipziger, J; Nitschke, R; Rubini-Illes, P; Thomas, J1
Iida, H; Inoue, N; Ishida, H; Ishikawa, Y; Yuan, Z1
Adamczyk, A; Jesko, H; Strosznajder, RP2

Other Studies

21 other study(ies) available for carbachol and 8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Suppressive effect of carbachol on forskolin-stimulated neurite outgrowth in human neuroblastoma NB-OK1 cells.
    Biochemical and biophysical research communications, 1992, Jan-15, Volume: 182, Issue:1

    Topics: Atropine; Calcium; Calcium Channel Blockers; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Egtazic Acid; Gallic Acid; Humans; Inositol; Inositol Phosphates; Kinetics; Neurites; Neuroblastoma; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide

1992
The effect of muscarinic cholinergic agonists on intracellular calcium and progesterone production by chicken granulosa cells.
    Endocrinology, 1992, Volume: 130, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Calcium; Calcium Channel Blockers; Carbachol; Chickens; Cyclic AMP; Female; Gallic Acid; Gallopamil; Granulosa Cells; In Vitro Techniques; Kinetics; Lanthanum; Luteinizing Hormone; Nifedipine; Progesterone; Receptors, Muscarinic

1992
Relationship between cytosolic Ca2+ concentration and amylase release in rat parotid acinar cells following muscarinic stimulation.
    Biochimica et biophysica acta, 1992, Apr-07, Volume: 1134, Issue:3

    Topics: Alkaloids; Amylases; Animals; Calcium; Carbachol; Cytosol; Dose-Response Relationship, Drug; Egtazic Acid; Gallic Acid; Ionomycin; Male; Parotid Gland; Rats; Rats, Inbred Strains; Staurosporine; Tetradecanoylphorbol Acetate

1992
Secretagogue-induced mobilization of an intracellular Mg2+ pool in rat sublingual mucous acini.
    The Journal of biological chemistry, 1992, Oct-15, Volume: 267, Issue:29

    Topics: Animals; Calcium Channel Blockers; Carbachol; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Fluorescent Dyes; Gallic Acid; Hydroquinones; Kinetics; Magnesium; Male; Monensin; Mouth Mucosa; Ouabain; Rats; Rats, Wistar; Spectrometry, Fluorescence; Substance P

1992
Carbamylcholine and phorbol esters desensitize muscarinic receptors by different mechanisms in rat pancreatic acini.
    Pancreas, 1990, Volume: 5, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amylases; Animals; Calcimycin; Carbachol; Dose-Response Relationship, Drug; Down-Regulation; Gallic Acid; Isoquinolines; Male; Pancreas; Phorbol 12,13-Dibutyrate; Phorbol Esters; Piperazines; Protein Kinase C; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Secretory Rate; Tetradecanoylphorbol Acetate

1990
Stimulatory and inhibitory effects of TMB-8 on pancreatic enzyme secretion.
    Biochimica et biophysica acta, 1986, Oct-10, Volume: 888, Issue:3

    Topics: Amylases; Animals; Calcimycin; Calcium; Carbachol; Dose-Response Relationship, Drug; Gallic Acid; L-Lactate Dehydrogenase; Pancreas; Rabbits; Sincalide; Tetradecanoylphorbol Acetate

1986
A transfected m1 muscarinic acetylcholine receptor stimulates adenylate cyclase via phosphatidylinositol hydrolysis.
    The Journal of biological chemistry, 1989, Dec-05, Volume: 264, Issue:34

    Topics: Adenylyl Cyclases; Animals; Arachidonic Acid; Arachidonic Acids; Calcium Channel Blockers; Calmodulin; Carbachol; Cell Membrane; Cyclic AMP; Cytosol; Gallic Acid; Gene Expression; Genes; Inositol Phosphates; Kinetics; L Cells; Mice; Models, Biological; Phosphatidylinositols; Protein Kinase C; Receptors, Muscarinic; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection

1989
Effects of calcium antagonist TMB-8 on active Na and Cl transport in rabbit ileum.
    The American journal of physiology, 1986, Volume: 250, Issue:5 Pt 1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atropine; Biological Transport, Active; Calcium; Calcium Channel Blockers; Carbachol; Cell Membrane; Chlorides; Cyclic AMP; Gallic Acid; Ileum; Intestinal Absorption; Intestinal Mucosa; Male; Rabbits; Serotonin; Sodium; Verapamil

1986
Interaction between the calcium and adenylate cyclase messenger systems in dispersed chief cells from guinea pig stomach. Possible cellular mechanism for potentiation of pepsinogen secretion.
    The Journal of biological chemistry, 1987, May-05, Volume: 262, Issue:13

    Topics: Adenylyl Cyclases; Animals; Calcimycin; Calcium; Carbachol; Cholera Toxin; Gallic Acid; Gastric Mucosa; Guinea Pigs; Male; Models, Biological; Pepsinogens; Sincalide; Stomach; Time Factors; Trifluoperazine

1987
The calcium dependence of histamine, carbachol and potassium chloride-induced contraction in human airways in vitro.
    European journal of pharmacology, 1986, Jun-17, Volume: 125, Issue:2

    Topics: Bronchi; Calcium; Calcium Channel Blockers; Carbachol; Gallic Acid; Histamine; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Verapamil

1986
Role of calcium in cholinergic stimulation of lacrimal gland protein secretion.
    Current eye research, 1985, Volume: 4, Issue:4

    Topics: Animals; Calcium; Carbachol; Cell Membrane; Eye Proteins; Gallic Acid; Intracellular Membranes; Lacrimal Apparatus; Male; Ouabain; Parasympathetic Nervous System; Peroxidases; Rats; Rats, Inbred Strains; Sulfonamides; Verapamil

1985
Effect of an intracellular calcium antagonist (TMB-8) on carbamylcholine-induced amylase release from dispersed rat pancreatic acini.
    Life sciences, 1984, Feb-06, Volume: 34, Issue:6

    Topics: Amylases; Animals; Calcium; Calcium Channel Blockers; Carbachol; Diltiazem; Dose-Response Relationship, Drug; Gallic Acid; Pancreas; Rats; Verapamil

1984
Inhibition of agonist-induced hydrolysis of phosphatidylinositol and muscarinic receptor binding by the calcium antagonist 8-(N,N-diethylamino)-octyl-3,4,5-trimethoxybenzoate-HCl (TMB-8).
    Biochemical pharmacology, 1983, Jul-01, Volume: 32, Issue:13

    Topics: Animals; Calcium Channel Blockers; Carbachol; Cholecystokinin; Gallic Acid; Hydrolysis; In Vitro Techniques; Mice; Pancreas; Peptide Fragments; Phosphatidylinositols; Receptors, Cholinergic; Receptors, Muscarinic; Sincalide; Submandibular Gland

1983
Inhibition of calcium uptake and catecholamine release by 8-(N,N-diethylamino)-octyl-3,4,5-trimethoxybenzoate hydrochloride (TMB-8) in cultured bovine adrenal chromaffin cells.
    Biochemical pharmacology, 1984, Dec-15, Volume: 33, Issue:24

    Topics: Adrenal Glands; Animals; Calcium; Calcium Channel Blockers; Carbachol; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Dantrolene; Gallic Acid; Verapamil

1984
Carbachol-induced potassium release in rat parotid acini: comparison of the roles of cytosolic Ca2+ and protein kinase C.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:4

    Topics: Alkaloids; Amylases; Animals; Calcium; Calcium Channel Blockers; Carbachol; Cytosol; Egtazic Acid; Enzyme Activation; Gallic Acid; Ionomycin; Male; Parotid Gland; Potassium; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1993
Inhibitors of the intracellular Ca2+ release mechanism prevent muscarinic-induced Ca2+ influx in rat sublingual mucous acini.
    FEBS letters, 1993, Jul-19, Volume: 327, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Carbachol; Dantrolene; Fura-2; Gallic Acid; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Male; Manganese; Mucous Membrane; Rats; Rats, Wistar; Sublingual Gland; Terpenes; Thapsigargin

1993
8-(N,N-diethylamino)octyl 3,4,5-trimethoxybenzoate (TMB-8) acts as a muscarinic receptor antagonist in the epithelial cell line HT29.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: Adenosine Triphosphate; Binding, Competitive; Calcium; Calcium Channel Blockers; Carbachol; Colon; Dose-Response Relationship, Drug; Epithelial Cells; Epithelium; Fura-2; Gallic Acid; HT29 Cells; Humans; Muscarinic Antagonists; Neurotensin; Type C Phospholipases

1996
Effect of SNI-2011 on amylase secretion from parotid tissue in rats and in neuronal nitric oxide synthase knockout mice.
    European journal of pharmacology, 2003, Mar-19, Volume: 464, Issue:2-3

    Topics: Alkaloids; Amylases; Animals; Azepines; Benzoates; Benzylamines; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Chelating Agents; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Gallic Acid; Genotype; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Mice, Knockout; Molsidomine; Muscarinic Agonists; Myosin-Light-Chain Kinase; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Parotid Gland; Penicillamine; Phosphodiesterase Inhibitors; Pilocarpine; Protein Kinase Inhibitors; Pyrroles; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Wistar; Sulfonamides; Thiophenes; Type C Phospholipases

2003
Poly(ADP-ribose) polymerase-1 is a novel nuclear target for cholinergic receptor signaling in the hippocampus.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2005, Volume: 56 Suppl 4

    Topics: Animals; Calcium Signaling; Carbachol; Cholinergic Agonists; Diglycerides; Gallic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate Receptors; Male; Maleimides; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerases; Protein Kinase C; Protein Kinase Inhibitors; Rats; Rats, Wistar; Receptors, Muscarinic; Signal Transduction

2005
Alzheimer's disease related peptides affected cholinergic receptor mediated poly(ADP-ribose) polymerase activity in the hippocampus.
    Folia neuropathologica, 2005, Volume: 43, Issue:3

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Calcium Channel Blockers; Calcium Channels; Carbachol; Cholinergic Agonists; Enzyme Activation; Free Radicals; Gallic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Inositol 1,4,5-Trisphosphate Receptors; Male; Peptide Fragments; Poly(ADP-ribose) Polymerases; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Receptors, Muscarinic; Signal Transduction

2005
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