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carbachol and 1h-(1,2,4)oxadiazolo(4,3-a)quinoxalin-1-one

carbachol has been researched along with 1h-(1,2,4)oxadiazolo(4,3-a)quinoxalin-1-one in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (16.67)18.2507
2000's17 (70.83)29.6817
2010's3 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Kawana, S; Miyamoto, A; Namiki, A; Ohshika, H; Yamamoto, S1
Berg, G; Dominiczak, AF; Hamilton, CA; McArthur, K; Reid, JL1
Closs, EI; Förstermann, U; Nawrath, H; Wegener, JW1
Alfonzo, MJ; González de Alfonzo, R; Guerra de González, L; Lippo de Bécemberg, I; Misle, A; Napoleón de Herrera, V; Pacheco, G1
Jiang, F; Li, CG; Rand, MJ1
Golding, S; Herring, N; Paterson, DJ1
Berggren, PO; Cooney, RV; Sjöholm, A1
Ellis, DZ; Nathanson, JA; Sweadner, KJ1
Baccari, MC; Calamai, F1
Alloatti, G; Bedendi, I; Biasin, C; Gallo, MP; Levi, RC; Malan, D1
Herring, N; Paterson, DJ1
Fujita, A; Hata, F; Morimoto, H; Sugimoto, K; Takeuch, T1
Choate, JK; Danson, EJ; Morris, JF; Paterson, DJ1
Bett, GC; Campbell, DL; Dai, S1
Bnouham, M; Fischmeister, R; Hoerter, J; Legssyer, A; Mekhfi, H; Tahri, A; Ziyyat, A1
Iida, H; Inoue, N; Ishida, H; Ishikawa, Y; Yuan, Z1
Diamond, J; Sandirasegarane, L1
Ahn, DS; Chung, SS; Lee, HG; Lee, YH; Nam, TS1
Angelini, GD; Jeremy, JY; Jones, R; Persad, R; Shukla, N1
Antunes, E; Baracat, JS; Claudino, MA; De Nucci, G; Priviero, FB; Teixeira, CE; Webb, RC1
Altun, A; Bagcivan, I; Durmus, N; Sarac, B; Sencan, M; Turan, M1
Gajdus, M; Glaza, I; Gurtowska, N; Rzepka, A; Szadujkis-Szadurski, L; Szadujkis-Szadurski, R1
Adachi, T; Fujisawa, S; Hongoh, M; Ohba, T; Ono, K; Shimbo, T1

Other Studies

24 other study(ies) available for carbachol and 1h-(1,2,4)oxadiazolo(4,3-a)quinoxalin-1-one

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Role of nitric oxide production in carbachol-induced negative chronotropy in cultured rat ventricular myocytes.
    European journal of pharmacology, 1999, Jan-29, Volume: 366, Issue:1

    Topics: Animals; Animals, Newborn; Atropine; Carbachol; Cells, Cultured; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guanylate Cyclase; Heart Ventricles; Methylene Blue; Myocardial Contraction; Myocardium; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitrites; omega-N-Methylarginine; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Signal Transduction

1999
Does potassium channel opening contribute to endothelium-dependent relaxation in human internal thoracic artery?
    Clinical science (London, England : 1979), 1999, Volume: 96, Issue:6

    Topics: Aged; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Humans; In Vitro Techniques; Ion Channel Gating; Male; Middle Aged; Nitric Oxide Synthase; Nitroprusside; Oxadiazoles; Potassium; Potassium Channels; Quinoxalines; Thoracic Arteries; Vasodilation; Vasodilator Agents

1999
Failure of 1H-[1,2,4]oxadiazolo[4,3-a]quinoxalin-1-one (ODQ) to inhibit soluble guanylyl cyclase in rat ventricular cardiomyocytes.
    British journal of pharmacology, 1999, Volume: 127, Issue:3

    Topics: Animals; Aorta, Thoracic; Carbachol; Cells, Cultured; Cyclic GMP; Enzyme Inhibitors; Female; Guanylate Cyclase; Heart Ventricles; In Vitro Techniques; Male; Myocardium; Nitric Oxide Donors; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Solubility

1999
Effects of 1H-[1,2,4]oxadiazolo[4,3-a]quinoxalin-1-one (ODQ) and Nomega(6)-nitro-L-arginine methyl ester (NAME) on cyclic GMP levels during muscarinic activation of tracheal smooth muscle.
    Biochemical pharmacology, 1999, Aug-15, Volume: 58, Issue:4

    Topics: Animals; Carbachol; Cattle; Cyclic GMP; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Muscarinic Agonists; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Oxadiazoles; Quinoxalines; Receptors, Muscarinic; Trachea

1999
Mechanisms of nitric oxide-independent relaxations induced by carbachol and acetylcholine in rat isolated renal arteries.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: Acetylcholine; Animals; Carbachol; Charybdotoxin; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Indomethacin; Male; Miconazole; NG-Nitroarginine Methyl Ester; Nitric Oxide; Ouabain; Oxadiazoles; Peptides; Phenylephrine; Potassium; Potassium Channel Blockers; Quinoxalines; Rats; Rats, Sprague-Dawley; Renal Artery; Tetraethylammonium; Vasoconstriction; Vasoconstrictor Agents; Vasodilation

2000
Pre-synaptic NO-cGMP pathway modulates vagal control of heart rate in isolated adult guinea pig atria.
    Journal of molecular and cellular cardiology, 2000, Volume: 32, Issue:10

    Topics: Age Factors; Animals; Aortic Bodies; Arginine; Blotting, Western; Carbachol; Cardiotonic Agents; Cyclic GMP; Digestive System; Enzyme Inhibitors; Female; Guanylate Cyclase; Guinea Pigs; Heart Atria; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Ornithine; Oxadiazoles; Prosencephalon; Quinoxalines; Receptors, Atrial Natriuretic Factor; Time Factors

2000
gamma-tocopherol partially protects insulin-secreting cells against functional inhibition by nitric oxide.
    Biochemical and biophysical research communications, 2000, Oct-22, Volume: 277, Issue:2

    Topics: Adenylyl Cyclases; Animals; Calcium; Calcium Channels; Carbachol; Cell Division; Cell Line; Cell Survival; Cholinergic Agonists; Colforsin; Cyclic GMP; Enzyme Inhibitors; Insulin; Insulin Secretion; Insulinoma; Interleukin-1; Islets of Langerhans; Models, Chemical; Nitric Oxide; Nitrogen Oxides; Oxadiazoles; Phorbol Esters; Protein Kinase C; Quinoxalines; Rats; Spermine; Type C Phospholipases; Vitamin E

2000
Carbachol inhibits Na(+)-K(+)-ATPase activity in choroid plexus via stimulation of the NO/cGMP pathway.
    American journal of physiology. Cell physiology, 2000, Volume: 279, Issue:6

    Topics: Adenosine Triphosphate; Animals; Carbachol; Cattle; Cholinergic Agonists; Choroid Plexus; Cyclic GMP; Enzyme Inhibitors; Hydrolysis; In Vitro Techniques; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Ouabain; Oxadiazoles; Phosphorylation; Quinoxalines; Sodium-Potassium-Exchanging ATPase; Solubility; Thionucleotides; Triazenes; Vasodilator Agents

2000
Modulation of nitrergic relaxant responses by peptides in the mouse gastric fundus.
    Regulatory peptides, 2001, Apr-02, Volume: 98, Issue:1-2

    Topics: Animals; Apamin; Carbachol; Cholinergic Agonists; Chymotrypsin; Electric Stimulation; Enzyme Inhibitors; Gastric Fundus; Guanylate Cyclase; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Neuropeptides; Neurotransmitter Agents; Nitroarginine; Oxadiazoles; Peptide Fragments; Pituitary Adenylate Cyclase-Activating Polypeptide; Quinoxalines; Vasoactive Intestinal Peptide

2001
Regulation of cardiac calcium current by NO and cGMP-modulating agents.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 441, Issue:5

    Topics: Adenine; Animals; Arginine; Biological Transport; Calcium Channels, L-Type; Carbachol; Cholinergic Agonists; Cyclic GMP; Cyclic N-Oxides; Enzyme Inhibitors; Exonucleases; Free Radical Scavengers; Guinea Pigs; Imidazoles; In Vitro Techniques; Myocardium; Nitric Oxide; omega-N-Methylarginine; Orchiectomy; Oxadiazoles; Quinoxalines; Receptors, Muscarinic

2001
Nitric oxide-cGMP pathway facilitates acetylcholine release and bradycardia during vagal nerve stimulation in the guinea-pig in vitro.
    The Journal of physiology, 2001, Sep-01, Volume: 535, Issue:Pt 2

    Topics: Acetylcholine; Alkaloids; Animals; Bradycardia; Calcium Channel Blockers; Calcium Channels; Carbachol; Carbazoles; Cardiotonic Agents; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Electric Stimulation; Enzyme Inhibitors; Female; Guanylate Cyclase; Guinea Pigs; Heart Rate; In Vitro Techniques; Indoles; Isoquinolines; Milrinone; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; omega-Conotoxin GVIA; Oxadiazoles; Phosphorylation; Presynaptic Terminals; Quinoxalines; Sinoatrial Node; Sulfonamides; Synaptic Transmission; Tritium; Vagus Nerve

2001
Mechanism of a nitric oxide donor NOR 1-induced relaxation in longitudinal muscle of rat proximal colon.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:4

    Topics: Animals; Calcium; Carbachol; Colon; Culture Techniques; Cyclic GMP; DNA-Binding Proteins; Dose-Response Relationship, Drug; Male; Models, Biological; Muscle Contraction; Muscle Relaxation; Muscle, Skeletal; Nerve Tissue Proteins; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Thapsigargin; Thionucleotides

2001
Peripheral vagal control of heart rate is impaired in neuronal NOS knockout mice.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 281, Issue:6

    Topics: Animals; Anti-Arrhythmia Agents; Atropine; Carbachol; Cardiotonic Agents; Cesium; Electric Stimulation; Enzyme Inhibitors; Guanylate Cyclase; Heart Atria; Heart Rate; Hypothalamus; Imidazoles; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Ornithine; Oxadiazoles; Parasympathetic Nervous System; Parasympatholytics; Propranolol; Quinoxalines; Sinoatrial Node; Stimulation, Chemical; Vagus Nerve

2001
Cholinergic modulation of the basal L-type calcium current in ferret right ventricular myocytes.
    The Journal of physiology, 2002, Jul-01, Volume: 542, Issue:Pt 1

    Topics: Animals; Calcium Channels, L-Type; Carbachol; Cholinergic Agents; Electric Stimulation; Electrophysiology; Ferrets; Guanylate Cyclase; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Kinetics; Membrane Potentials; Muscarinic Agonists; Myocardium; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Oxadiazoles; Patch-Clamp Techniques; Quinoxalines

2002
Arbutus unedo induces endothelium-dependent relaxation of the isolated rat aorta.
    Phytotherapy research : PTR, 2002, Volume: 16, Issue:6

    Topics: Animals; Aorta, Thoracic; Atropine; Carbachol; Dogs; Drug Interactions; Endothelium, Vascular; Ericaceae; In Vitro Techniques; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Norepinephrine; Oxadiazoles; Plant Extracts; Plant Roots; Quinoxalines; Rats; Rats, Wistar; Vasoconstriction; Vasodilation

2002
Effect of SNI-2011 on amylase secretion from parotid tissue in rats and in neuronal nitric oxide synthase knockout mice.
    European journal of pharmacology, 2003, Mar-19, Volume: 464, Issue:2-3

    Topics: Alkaloids; Amylases; Animals; Azepines; Benzoates; Benzylamines; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Chelating Agents; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Gallic Acid; Genotype; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Mice, Knockout; Molsidomine; Muscarinic Agonists; Myosin-Light-Chain Kinase; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Parotid Gland; Penicillamine; Phosphodiesterase Inhibitors; Pilocarpine; Protein Kinase Inhibitors; Pyrroles; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Wistar; Sulfonamides; Thiophenes; Type C Phospholipases

2003
Pertussis toxin-sensitive G protein but not NO/cGMP pathway mediates the negative inotropic effect of carbachol in adult rat cardiomyocytes.
    Pharmacology, 2004, Volume: 70, Issue:1

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Electric Stimulation; GTP-Binding Proteins; Injections, Intraperitoneal; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Nitric Oxide Synthase; omega-N-Methylarginine; Oxadiazoles; Pertussis Toxin; Quinoxalines; Rats; Time Factors

2004
Inhibition of carbachol-evoked oscillatory currents by the NO donor sodium nitroprusside in guinea-pig ileal myocytes.
    Experimental physiology, 2005, Volume: 90, Issue:4

    Topics: Animals; Caffeine; Carbachol; Chelating Agents; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Egtazic Acid; Guinea Pigs; Ileum; In Vitro Techniques; Membrane Potentials; Muscarinic Agonists; Muscle Contraction; Myocytes, Smooth Muscle; Nitric Oxide Donors; Nitroprusside; Oxadiazoles; Patch-Clamp Techniques; Phosphatidylinositol 3-Kinases; Phosphodiesterase Inhibitors; Quinoxalines; Type C Phospholipases

2005
Effect of sildenafil citrate and a nitric oxide donating sildenafil derivative, NCX 911, on cavernosal relaxation and superoxide formation in hypercholesterolaemic rabbits.
    European journal of pharmacology, 2005, Jul-11, Volume: 517, Issue:3

    Topics: Acetophenones; Allopurinol; Animals; Carbachol; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hypercholesterolemia; In Vitro Techniques; Male; Muscle Relaxation; NADPH Oxidases; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroprusside; Onium Compounds; Oxadiazoles; Penis; Phosphodiesterase Inhibitors; Piperazines; Purines; Quinoxalines; Rabbits; Rotenone; Sildenafil Citrate; Sulfones; Superoxides; Uncoupling Agents; Xanthine Oxidase

2005
Stimulation of soluble guanylyl cyclase by BAY 41-2272 relaxes anococcygeus muscle: interaction with nitric oxide.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: Animals; Carbachol; Carbolines; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroglycerin; Oxadiazoles; Pyrazoles; Pyridines; Quinoxalines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Tadalafil; Tetrodotoxin

2006
Investigation of relaxant effects of new agents affecting nitric oxide/cyclic guanosine monophosphate pathway on sheep oddi sphincter.
    Pancreas, 2010, Volume: 39, Issue:6

    Topics: Animals; Carbachol; Cyclic GMP; Dose-Response Relationship, Drug; Guanylate Cyclase; In Vitro Techniques; Male; Molsidomine; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Oxadiazoles; Pyrazoles; Pyridines; Quinoxalines; Sheep; Sphincter of Oddi; Triazenes

2010
Activity of guanylyl cyclase activators on the reaction of tracheal smooth muscle contraction.
    Postepy higieny i medycyny doswiadczalnej (Online), 2011, Aug-05, Volume: 65

    Topics: Animals; Carbachol; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Activators; Enzyme Inhibitors; Female; Guanylate Cyclase; Indazoles; Male; Muscle, Smooth; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Trachea

2011
In vitro effect of nicorandil on the carbachol-induced contraction of the lower esophageal sphincter of the rat.
    Journal of pharmacological sciences, 2016, Volume: 131, Issue:4

    Topics: Animals; Carbachol; Diazoxide; Dose-Response Relationship, Drug; Esophageal Sphincter, Lower; Glyburide; In Vitro Techniques; KATP Channels; Muscle Contraction; NG-Nitroarginine Methyl Ester; Nicorandil; Oxadiazoles; Peptides; Pinacidil; Potassium; Quinoxalines; Rats

2016