capsaicin has been researched along with sb 366791 in 54 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 23 (42.59) | 29.6817 |
2010's | 28 (51.85) | 24.3611 |
2020's | 3 (5.56) | 2.80 |
Authors | Studies |
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Davies, CH; Davis, JB; Egerton, J; Gill, CH; Gunthorpe, MJ; Howett, L; Jerman, JC; Lappin, SC; Luis Hannan, S; Nasir, S; Owen, D; Rami, HK; Randall, AD; Smart, D; Smith, GD; Soffin, EM; Thompson, M; Worby, A; Wyman, PA | 1 |
Dell, H | 1 |
Desimone, JA; Ghosh, S; Heck, GL; Lyall, V; Phan, TH; Vinnikova, AK | 1 |
DeSimone, JA; Heck, GL; Lyall, V; Malik, SA; Mummalaneni, S; Phan, TH; Vinnikova, AK | 2 |
Elekes, K; Helyes, Z; McDougall, JJ; Németh, J; Pintér, E; Szabó, A; Szolcsányi, J; Varga, A; Zhang, C | 1 |
Adler-Graschinsky, E; Briones, R; Huidobro-Toro, JP; Orliac, ML; Poblete, IM | 1 |
Cowan, A; Ding, Z; Rawls, SM | 2 |
Andrade, EL; André, E; Calixto, JB; Ferreira, J | 1 |
Boudaka, A; Kobayashi, H; Neuhuber, WL; Shiina, T; Shimizu, Y; Takewaki, T; Wörl, J | 1 |
Alexander, SP; Athanasiou, A; Bagiokou, D; Bates, TE; Guo, DA; Kendall, DA; Kumaran, NM; Layfield, R; Lobo, DN; Lophatanon, A; Muir, KA; Ray, DE; Smith, PA; Turner, AE; Vakilpour, S; Watson, SA; Westwell, AD | 1 |
Medley, D; Naniwadekar, A; Pasricha, PJ; Shenoy, M; Winston, J | 1 |
Ferrini, F; Merighi, A; Salio, C; Vergnano, AM | 1 |
Asano, M; Harada, N; Mishima, A; Nakayama, T; Nomura, N; Okajima, K; Saito, T | 1 |
Pasricha, PJ; Pendyala, S; Shenoy, M; Winston, JH; Xu, GY; Yin, H | 1 |
Andrade, EL; Calixto, JB; Ferreira, J; Luiz, AP | 1 |
Cao, J; Li, HB; Mao, RR; Xu, L; Yang, Y; Zhang, JC | 1 |
Kopczyńska, B | 1 |
Cristino, L; Di Marzo, V; Drago, F; Leggio, GM; Micale, V; Petrosino, S; Tamburella, A | 1 |
Díaz-Laviada, I; Malagarie-Cazenave, S; Olea-Herrero, N; Vara, D | 1 |
Brink, TS; Potenzieri, C; Simone, DA | 1 |
Gregg, RG; Heimel, JA; Kamermans, M; Nawy, S; Peachey, NS; Shen, Y | 1 |
Brennan, FX; Bryant, RW; Devantier, HR; Long, DJ; Palmer, RK; Salemme, FR | 1 |
Fujihara, H; Hashimoto, H; Nagatomo, T; Ohbuchi, T; Otsubo, H; Saito, T; Suzuki, H; Ueta, Y; Yokoyama, T | 1 |
Andresen, MC; Fawley, JA; McDougall, SJ; Peters, JH; Smith, SM | 1 |
Harada, N; Ishikura, H; Kitamura, T; Okajima, K; Umemura, T | 1 |
Andresen, MC; Fawley, JA; McDougall, SJ; Peters, JH; Shoudai, K | 1 |
Buzas, K; Cohen, JI; Fan, H; Howard, OM; Klinman, D; Mont, E; Oppenheim, JJ; Qi, J; Wang, K | 1 |
Andrade, EL; Calixto, JB; Rogerio, AP | 1 |
de Oliveira, SM; Ferreira, J; Gomez, MV; Hoffmeister, C; Rossato, MF; Trevisan, G | 1 |
Chen, Y; Wang, ZJ; Yang, C | 1 |
Aguiar, DC; Casarotto, PC; Guimarães, FS; Moreira, FA; Terzian, AL; Wotjak, CT; Zangrossi, H | 1 |
Bogo, MR; Campos, MM; Couture, R; Dias, JP; Gaudreau, P; Lahjouji, K; Talbot, S | 1 |
Hitomi, S; Iwata, K; Shinoda, M; Suzuki, I | 1 |
Bratz, IN; Damron, DS; DelloStritto, DJ; Guarini, G; Kmetz, JG; Meszaros, JG; Ohanyan, VA; Thodeti, CK; Thoppil, RJ | 1 |
Coderre, EM; Hermes, ML; Kolaj, M; Renaud, LP | 1 |
DeSimone, JA; Grider, JR; Lyall, V; Mummalaneni, S; Murthy, KS; Phan, TH; Ren, Z; Rhyu, MR | 1 |
Adamek, P; Kalynovska, N; Mrozkova, P; Palecek, J; Spicarova, D | 1 |
Matsuda, Y; Murakami, S; Nakajima, T; Tabeta, K; Takahashi, N; Yamada, H; Yamazaki, K | 1 |
Abramson, L; Aoki-Nonaka, Y; Bertin, S; Corr, M; de Jong, PR; Dong, H; Franco, A; Fu, G; González-Navajas, JM; Gwack, Y; Han, T; Herdman, S; Jefferies, WA; Lee, J; Li, X; Nohara, LL; Raz, E; Srikanth, S; Stanwood, SR; To, K; Touma, R; Xu, H; Yu, T | 1 |
Burrell, BD; Holec, S; Summers, T | 1 |
Furukawa, A; Honda, K; Iwata, K; Kita, K; Noma, N; Shinoda, M | 1 |
Dale, CS; Ferro, ES; Fogaça, MV; Gozzo, FC; Guimarães, FS; Rioli, V; Sonego, AB | 1 |
Chen, HY; Chiang, AN; Guo, BC; Lee, TS; Shyue, SK; Su, KH; Wei, J; Zhao, JF | 1 |
Binkowski, M; Czaja, M; Di Marzo, V; Kolosowska, N; Makuch, W; Malek, N; Morera, E; Mrugala, M; Przewlocka, B; Starowicz, K | 1 |
Calzetta, L; Capuano, A; Cazzola, M; Facciolo, F; Luongo, L; Maione, S; Matera, MG; Page, C; Rinaldi, B; Rogliani, P | 1 |
Chen, X; Cui, W; Han, W; Jin, X; Long, C; Pan, Z; Wang, H; Zhang, Y | 1 |
Ide, S; Kojima, S; Nakanishi, Y; Nishino, K; Tanamachi, K; Tanuma, S; Tsukimoto, M | 1 |
Burrell, BD; Wang, Y | 1 |
Borges, MH; Castro-Junior, CJ; Ferreira, J; Gomez, MV; Palhares, MR; Rezende, MJS; Santos, DC; Silva, JF; Silva-Junior, CA | 1 |
Binda, NS; Borges, MH; Carobin, NV; Castro Junior, CJ; Ferreira, J; Gomez, MV; Kushmerick, C; Pinto Nagem, RA; Ribeiro, FM; Rita Pereira, EM; Santos, DC; Silva Júnior, CA; Silva, JF; Souza, JM | 1 |
Inoue, M; Magara, J; Nagoya, K; Shiraishi, N; Suzuki, T; Terunuma, M; Tsujimura, T; Yoshihara, M | 1 |
Arkhipov, AY; Fedorov, NS; Khabibrakhmanov, AN; Malomouzh, AI; Mukhamedyarov, MA; Nurullin, LF; Samigullin, DV | 1 |
54 other study(ies) available for capsaicin and sb 366791
Article | Year |
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Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acids; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Anilides; Aniline Compounds; Animals; Calcium; Capsaicin; Carrier Proteins; Cell Line; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Hot Temperature; Humans; Intracellular Signaling Peptides and Proteins; Kidney; Membrane Potentials; N-Methylaspartate; Neuropeptides; Norepinephrine; Orexins; Patch-Clamp Techniques; Protein Binding; Radioligand Assay; Rats; Receptors, Drug; Serotonin Receptor Agonists; Xanthenes | 2004 |
New compound fires up pain research.
Topics: Anilides; Animals; Capsaicin; Cinnamates; Humans; Nociceptors; Pain; Rats; Receptors, Drug | 2003 |
A novel vanilloid receptor-1 (VR-1) variant mammalian salt taste receptor.
Topics: Amiloride; Anilides; Animals; Capsaicin; Cinnamates; Diterpenes; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Salts; Sodium Channel Blockers; Sodium Chloride; Taste; Taste Buds; TRPV Cation Channels | 2005 |
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. I. Effect on TRC volume and Na+ flux.
Topics: Amiloride; Anilides; Animals; Capsaicin; Cell Size; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Cytosol; Diuretics; Ethanol; Female; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Taste; Temperature; Tongue | 2005 |
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. II. Effect on chorda tympani salt responses.
Topics: Algorithms; Amiloride; Anilides; Animals; Capsaicin; Cell Membrane; Cell Polarity; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Diterpenes; Diuretics; Ethanol; Female; In Vitro Techniques; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Stimulation, Chemical; Taste; Taste Threshold; Temperature; Tongue | 2005 |
Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat.
Topics: Analgesics; Anilides; Animals; Capsaicin; Cells, Cultured; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Hypothermia; Ion Channels; Male; Mice; Mice, Inbred BALB C; Neurons, Afferent; Nociceptors; Pain; Peripheral Nervous System; Rats; Rats, Wistar; Sensory Receptor Cells; Substance P; Trigeminal Ganglion; TRPV Cation Channels | 2005 |
Anandamide elicits an acute release of nitric oxide through endothelial TRPV1 receptor activation in the rat arterial mesenteric bed.
Topics: Anilides; Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Capsaicin; Cinnamates; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Artery, Superior; Nitric Oxide; Nitroarginine; Perfusion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; RNA, Messenger; TRPV Cation Channels; Vasodilation | 2005 |
Capsaicin evokes hypothermia independent of cannabinoid CB1 and CB2 receptors.
Topics: Anilides; Animals; Benzoxazines; Body Temperature; Calcium Channel Blockers; Camphanes; Capsaicin; Cinnamates; Hypothermia; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; TRPV Cation Channels | 2005 |
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
Topics: Amidohydrolases; Anilides; Animals; Arachidonic Acids; Body Temperature; Capsaicin; Cinnamates; Endocannabinoids; Hypothermia; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels | 2006 |
Contractile mechanisms coupled to TRPA1 receptor activation in rat urinary bladder.
Topics: Acrolein; Anilides; Animals; Ankyrins; Binding Sites; Calcium Channels; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Drug Antagonism; In Vitro Techniques; Isothiocyanates; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Wistar; Ruthenium Red; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels; Urinary Bladder | 2006 |
Involvement of TRPV1-dependent and -independent components in the regulation of vagally induced contractions in the mouse esophagus.
Topics: Alkaloids; Anilides; Animals; Benzodioxoles; Capsaicin; Cinnamates; Cricetinae; Enzyme Inhibitors; Esophagus; Female; Male; Mesocricetus; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Tachykinin; Species Specificity; TRPV Cation Channels; Tryptophan; Vagus Nerve | 2007 |
Vanilloid receptor agonists and antagonists are mitochondrial inhibitors: how vanilloids cause non-vanilloid receptor mediated cell death.
Topics: Anilides; Animals; Apoptosis; Capsaicin; Carcinoma, Non-Small-Cell Lung; Cells, Cultured; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Humans; Hydrogen Peroxide; Lung Neoplasms; Membrane Potentials; Mitochondria, Heart; Oxygen Consumption; Rats; TRPV Cation Channels | 2007 |
The vanilloid receptor initiates and maintains colonic hypersensitivity induced by neonatal colon irritation in rats.
Topics: Acetic Acid; Age Factors; Anilides; Animals; Animals, Newborn; Capsaicin; Catheterization; Cinnamates; Colon; Disease Models, Animal; Diterpenes; Electromyography; Ganglia, Spinal; Hyperalgesia; Irritable Bowel Syndrome; Male; Pain; Rats; Rats, Sprague-Dawley; Reflex, Abdominal; TRPV Cation Channels; Visceral Afferents | 2007 |
Vanilloid receptor-1 (TRPV1)-dependent activation of inhibitory neurotransmission in spinal substantia gelatinosa neurons of mouse.
Topics: Anilides; Animals; Animals, Newborn; Bicuculline; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Immunohistochemistry; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Mice; Neural Inhibition; Neurons; Patch-Clamp Techniques; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin; TRPV Cation Channels; Tryptophan | 2007 |
Atrial natriuretic peptide reduces ischemia/reperfusion-induced spinal cord injury in rats by enhancing sensory neuron activation.
Topics: 6-Ketoprostaglandin F1 alpha; Anilides; Animals; Atrial Natriuretic Factor; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Cells, Cultured; Cinnamates; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Indoles; Indomethacin; Male; Neurons, Afferent; Peroxidase; Psychomotor Performance; Pyrroles; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Spinal Cord; Spinal Cord Diseases; TRPV Cation Channels; Tumor Necrosis Factor-alpha | 2007 |
Transient receptor potential vanilloid 1 mediates hyperalgesia and is up-regulated in rats with chronic pancreatitis.
Topics: Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Disease Models, Animal; Electric Stimulation; Ganglia, Spinal; Hyperalgesia; Male; Membrane Potentials; Pain Measurement; Pain Threshold; Pancreas; Pancreatitis, Chronic; Rats; Rats, Sprague-Dawley; RNA, Messenger; Time Factors; Trinitrobenzenesulfonic Acid; TRPV Cation Channels; Up-Regulation | 2007 |
Pronociceptive response elicited by TRPA1 receptor activation in mice.
Topics: Analgesics; Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Isothiocyanates; Male; Mice; Pain; Pain Measurement; Ruthenium Red; Time Factors; Transient Receptor Potential Channels; TRPA1 Cation Channel | 2008 |
Antistress effect of TRPV1 channel on synaptic plasticity and spatial memory.
Topics: Anilides; Animals; Animals, Newborn; Behavior, Animal; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Male; Memory; Neuronal Plasticity; Neurons; Rats; Rats, Wistar; Space Perception; Synaptic Transmission; TRPV Cation Channels | 2008 |
Role of VR1 and CB1 receptors in modelling of cardio-respiratory response to arvanil, an endocannabinoid and vanilloid hybrid, in rats.
Topics: Anilides; Animals; Blood Pressure; Cannabinoid Receptor Modulators; Capsaicin; Cinnamates; Disease Models, Animal; Endocannabinoids; Hypertension; Injections, Intravenous; Male; Morpholines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Respiration; Respiration Disorders; Ruthenium Red; Tidal Volume; TRPV Cation Channels | 2008 |
Anxiolytic effects in mice of a dual blocker of fatty acid amide hydrolase and transient receptor potential vanilloid type-1 channels.
Topics: Amidohydrolases; Anilides; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cinnamates; Diazepam; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels | 2009 |
Capsaicin, a component of red peppers, induces expression of androgen receptor via PI3K and MAPK pathways in prostate LNCaP cells.
Topics: Anilides; Capsaicin; Capsicum; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cinnamates; Diterpenes; Gene Silencing; Humans; Male; Mitogen-Activated Protein Kinase Kinases; Phosphatidylinositol 3-Kinases; Prostate; Receptors, Androgen; RNA, Small Interfering; TRPV Cation Channels | 2009 |
Excitation of cutaneous C nociceptors by intraplantar administration of anandamide.
Topics: Action Potentials; Anilides; Animals; Arachidonic Acids; Calcium Channel Blockers; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Endocannabinoids; Hindlimb; Hot Temperature; Male; Nociceptors; Pain; Pain Measurement; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Skin; Tibial Nerve; TRPV Cation Channels | 2009 |
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
Topics: Amino Acids; Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Polyunsaturated Alkamides; Propionates; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; Ruthenium Red; Synaptic Transmission; Transient Receptor Potential Channels; TRPM Cation Channels; TRPV Cation Channels; Xanthenes | 2009 |
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
Topics: Acrylamides; Administration, Oral; Alkaloids; Anilides; Animals; Avoidance Learning; Benzodioxoles; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazines; Pyridines; Taste; TRPM Cation Channels; TRPV Cation Channels | 2010 |
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
Topics: Analysis of Variance; Angiotensin II; Anilides; Animals; Capsaicin; Chelating Agents; Cinnamates; Diuretics, Osmotic; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; In Vitro Techniques; Male; Mannitol; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Piperidines; Pyrazines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Supraoptic Nucleus; TRPV Cation Channels; Vasoconstrictor Agents | 2010 |
Primary afferent activation of thermosensitive TRPV1 triggers asynchronous glutamate release at central neurons.
Topics: Afferent Pathways; Anilides; Animals; Capsaicin; Cinnamates; Electric Stimulation; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sensory System Agents; Solitary Nucleus; Thermosensing; TRPV Cation Channels | 2010 |
Limaprost reduces motor disturbances by increasing the production of insulin-like growth factor I in rats subjected to spinal cord injury.
Topics: Alprostadil; Anilides; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Caspase 3; Cells, Cultured; Cinnamates; Denervation; Disease Models, Animal; Drug Therapy, Combination; Ganglia, Spinal; Gene Expression; Insulin-Like Growth Factor I; Male; Movement; Neurons; Rats; Rats, Wistar; RNA, Messenger; Sensory System Agents; Specific Pathogen-Free Organisms; Spinal Cord; Spinal Cord Injuries; Vasodilator Agents | 2010 |
Thermally active TRPV1 tonically drives central spontaneous glutamate release.
Topics: Action Potentials; Anilides; Animals; Cadmium Compounds; Calcium; Capsaicin; Cinnamates; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Channel Blockers; Synapses; Tetrodotoxin; Thermosensing; TRPV Cation Channels | 2010 |
Painful pathways induced by TLR stimulation of dorsal root ganglion neurons.
Topics: Aminoquinolines; Anilides; Animals; Arachidonic Acids; Blotting, Western; Calcium; Capsaicin; Cells, Cultured; Cinnamates; Cytokines; Dinoprostone; Dose-Response Relationship, Drug; Endocannabinoids; Ganglia, Spinal; Humans; Imidazoles; Mice; Microscopy, Confocal; Neurons; Pain; Poly I-C; Polyunsaturated Alkamides; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Toll-Like Receptor 3; Toll-Like Receptor 7; Toll-Like Receptor 9; Toll-Like Receptors; TRPV Cation Channels | 2011 |
C-fibers, but not the transient potential receptor vanilloid 1 (TRPV1), play a role in experimental allergic airway inflammation.
Topics: Allergens; Anilides; Animals; Animals, Newborn; Bronchoalveolar Lavage Fluid; Capsaicin; Cell Count; Cinnamates; Cytokines; Female; Gene Expression Regulation; Hypersensitivity; Immunization; Inflammation; Leukocytes; Lung; Mice; Mice, Inbred BALB C; Nerve Fibers, Unmyelinated; NF-kappa B; Ovalbumin; P-Selectin; Respiratory System; TRPV Cation Channels | 2011 |
Role of TRPV1 in nociception and edema induced by monosodium urate crystals in rats.
Topics: Acrylamides; Anilides; Animals; Anti-Allergic Agents; Anti-Asthmatic Agents; Antioxidants; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Cromolyn Sodium; Disease Models, Animal; Diterpenes; Edema; Gabexate; Histamine; Male; Mast Cells; Methysergide; Pain; Promethazine; Prostaglandin-Endoperoxide Synthases; Protein Binding; Rats; Rats, Wistar; Serine Proteinase Inhibitors; Serotonin; Serotonin Antagonists; Tritium; TRPV Cation Channels; Uric Acid | 2011 |
Proteinase-activated receptor 2 sensitizes transient receptor potential vanilloid 1, transient receptor potential vanilloid 4, and transient receptor potential ankyrin 1 in paclitaxel-induced neuropathic pain.
Topics: Analysis of Variance; Anilides; Animals; Ankyrins; Antineoplastic Agents, Phytogenic; Capsaicin; Carbazoles; Central Nervous System; Cinnamates; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Estrenes; Gene Expression Regulation; Hyperalgesia; Male; Mice; Mice, Inbred ICR; Neuralgia; Oligopeptides; Paclitaxel; Pain Measurement; Physical Stimulation; Protein Kinase C; Pyrroles; Pyrrolidinones; Receptor, PAR-2; Sulfonamides; Time Factors; TRPV Cation Channels; Tryptases; Type C Phospholipases | 2011 |
Opposing roles for cannabinoid receptor type-1 (CB₁) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats.
Topics: Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Drug Interactions; Electric Stimulation; Male; Microinjections; Panic; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels | 2012 |
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
Topics: Acetylcysteine; Analysis of Variance; Anilides; Animals; Antioxidants; Autoradiography; Bradykinin; Bradykinin B1 Receptor Antagonists; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Gene Expression Regulation; Iodine Isotopes; Male; Microglia; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; RNA, Messenger; Sensory System Agents; Spinal Cord; Superoxides; Tetrahydroisoquinolines; Time Factors; TRPV Cation Channels | 2012 |
Involvement of transient receptor potential vanilloid 1 in ectopic pain following inferior alveolar nerve transection in rats.
Topics: Anilides; Animals; Antigens, Nuclear; Behavior, Animal; Capsaicin; Cell Count; Cinnamates; Electric Stimulation; Extracellular Signal-Regulated MAP Kinases; Facial Pain; Grooming; Immunohistochemistry; Male; Mandibular Nerve; Nerve Tissue Proteins; Phosphorylation; Rats; Rats, Sprague-Dawley; Trigeminal Ganglion; TRPV Cation Channels; Vibrissae | 2012 |
Disruption of TRPV1-mediated coupling of coronary blood flow to cardiac metabolism in diabetic mice: role of nitric oxide and BK channels.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Anilides; Animals; Capsaicin; Cinnamates; Coronary Vessels; Diabetes Mellitus, Type 2; Diabetic Cardiomyopathies; Enzyme Inhibitors; Large-Conductance Calcium-Activated Potassium Channels; Male; Mice; Mice, Inbred C57BL; Microvessels; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptides; TRPV Cation Channels; Vasoconstrictor Agents; Vasodilation | 2012 |
Gastrin-releasing peptide acts via postsynaptic BB2 receptors to modulate inward rectifier K+ and TRPV1-like conductances in rat paraventricular thalamic neurons.
Topics: Anilides; Animals; Capsaicin; Cinnamates; Gastrin-Releasing Peptide; Male; Midline Thalamic Nuclei; Neurons; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Bombesin; TRPV Cation Channels | 2013 |
TRPM5-dependent amiloride- and benzamil-insensitive NaCl chorda tympani taste nerve response.
Topics: Amiloride; Anilides; Animals; Capsaicin; Chorda Tympani Nerve; Cinnamates; Diterpenes; Mice; Mice, Knockout; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Sodium Chloride; Taste; TRPM Cation Channels; TRPV Cation Channels | 2013 |
TRPV1 receptor inhibition decreases CCL2-induced hyperalgesia.
Topics: Anilides; Animals; Animals, Newborn; Capsaicin; Chemokine CCL2; Cinnamates; Disease Models, Animal; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Hyperalgesia; In Vitro Techniques; Male; MAP Kinase Kinase Kinase 3; Pain Threshold; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Rats, Wistar; Sensory System Agents; Spinal Cord; Time Factors; TRPV Cation Channels | 2014 |
Epithelial TRPV1 signaling accelerates gingival epithelial cell proliferation.
Topics: Anilides; Animals; Apoptosis; Capsaicin; Cell Line; Cell Proliferation; Cells, Cultured; Cinnamates; Epithelial Cells; Fibroblast Growth Factors; Gene Expression Profiling; Gingiva; HEK293 Cells; Humans; Male; Mice; Mice, Inbred C57BL; Nerve Growth Factors; Nociceptors; Oligonucleotide Array Sequence Analysis; Sensory System Agents; Signal Transduction; TRPV Cation Channels; Up-Regulation | 2014 |
The ion channel TRPV1 regulates the activation and proinflammatory properties of CD4⁺ T cells.
Topics: Anilides; Animals; Calcium; Calcium Channels; Calcium Signaling; Capsaicin; CD4-Positive T-Lymphocytes; Cells, Cultured; Cinnamates; Colitis; Humans; Inflammation; Interleukin-10; Intestines; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptors, Antigen, T-Cell; Sensory System Agents; TRPV Cation Channels | 2014 |
Physiological and behavioral evidence of a capsaicin-sensitive TRPV-like channel in the medicinal leech.
Topics: Anilides; Animals; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Hirudo medicinalis; Hot Temperature; Nociceptors; Sensory System Agents; TRPV Cation Channels | 2014 |
TRPA1 contributes to capsaicin-induced facial cold hyperalgesia in rats.
Topics: Acetanilides; Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Cold Temperature; Electromyography; Face; Facial Pain; Hot Temperature; Hyperalgesia; Injections, Intradermal; Male; Neural Conduction; Neurons; Physical Stimulation; Purines; Rats; Rats, Sprague-Dawley; Reflex; Sensory System Agents; Synaptic Transmission; Trigeminal Ganglion; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels | 2014 |
Anxiogenic-like effects induced by hemopressin in rats.
Topics: Anilides; Animals; Anxiety; Brain; Capsaicin; Cinnamates; Hemoglobins; Injections, Intraventricular; Male; Maze Learning; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Wistar | 2015 |
Transient receptor potential vanilloid type 1 is vital for (-)-epigallocatechin-3-gallate mediated activation of endothelial nitric oxide synthase.
Topics: AMP-Activated Protein Kinases; Anilides; Animals; Calcium; Capsaicin; Catechin; Cell Movement; Cell Proliferation; Cell Survival; Cinnamates; Endothelial Cells; HEK293 Cells; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Neovascularization, Pathologic; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphorylation; Signal Transduction; Tea; TRPV Cation Channels | 2015 |
A multi-target approach for pain treatment: dual inhibition of fatty acid amide hydrolase and TRPV1 in a rat model of osteoarthritis.
Topics: Activating Transcription Factor 3; Amidohydrolases; Anilides; Animals; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Cinnamates; Disease Models, Animal; Endocannabinoids; Ganglia, Spinal; Gene Expression; Hyperalgesia; Inflammation; Interleukin-6; Lumbar Vertebrae; Male; Osteoarthritis; Pain; Pain Management; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels | 2015 |
Contribution of sensory nerves to LPS-induced hyperresponsiveness of human isolated bronchi.
Topics: Anilides; Bronchi; Bronchial Hyperreactivity; Capsaicin; Cinnamates; Electric Stimulation; Female; Humans; Indoles; Lipopolysaccharides; Male; Middle Aged; Muscle Contraction; Neprilysin; Neurokinin A; Piperidines; Sensory Receptor Cells; TRPV Cation Channels; Up-Regulation | 2015 |
The molecular pathway of ATP-sensitive potassium channel in endothelial cells for mediating arteriole relaxation.
Topics: Allyl Compounds; Anilides; Animals; Arterioles; Calcium; Capsaicin; Cells, Cultured; Cinnamates; Down-Regulation; Endothelial Cells; KATP Channels; Mesenteric Arteries; Nitric Oxide; Propylamines; Rats; RNA, Small Interfering; TRPV Cation Channels; Vasodilation | 2015 |
Radiosensitizing Effect of TRPV1 Channel Inhibitors in Cancer Cells.
Topics: Acrylamides; Anilides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line, Tumor; Cell Survival; Cinnamates; DNA Damage; Gamma Rays; Humans; Mice; Necrosis; Neoplasms; Pyrazines; Pyridines; Radiation-Sensitizing Agents; TRPV Cation Channels | 2016 |
Differences in chloride gradients allow for three distinct types of synaptic modulation by endocannabinoids.
Topics: Anilides; Animals; Biophysics; Bumetanide; Cannabinoid Receptor Modulators; Capsaicin; Central Nervous System; Chlorides; Cinnamates; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Lactones; Leeches; Neurons; Orlistat; Patch-Clamp Techniques; Sensory System Agents; Sodium Potassium Chloride Symporter Inhibitors; Synapses | 2016 |
Synergistic antinociceptive effect of a calcium channel blocker and a TRPV1 blocker in an acute pain model in mice.
Topics: Acute Pain; Analgesics; Anilides; Animals; Body Temperature; Calcium Channel Blockers; Capsaicin; Cinnamates; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Mice; Spider Venoms; TRPV Cation Channels | 2017 |
Phoneutria toxin PnTx3-5 inhibits TRPV1 channel with antinociceptive action in an orofacial pain model.
Topics: Acrolein; Anilides; Animals; Calcium; Calcium Signaling; Capsaicin; Cinnamates; Disease Models, Animal; Facial Pain; Glutamic Acid; HEK293 Cells; Humans; Inhibitory Concentration 50; Male; Neuropeptides; Nociception; Patch-Clamp Techniques; Rats; Sensory System Agents; Transfection; Trigeminal Ganglion; TRPA1 Cation Channel; TRPV Cation Channels | 2020 |
Sustained laryngeal transient receptor potential vanilloid 1 activation inhibits mechanically induced swallowing in anesthetized rats.
Topics: Anesthesia; Anilides; Animals; Capillary Permeability; Capsaicin; Cinnamates; Deglutition; Electric Stimulation; Laryngeal Nerves; Larynx; Male; Mechanoreceptors; Physical Stimulation; Radiation; Rats; Rats, Sprague-Dawley; TRPV Cation Channels | 2020 |
Activation of TRPV1 Channels Inhibits the Release of Acetylcholine and Improves Muscle Contractility in Mice.
Topics: Acetylcholine; Animals; Capsaicin; Mice; Muscle, Skeletal; Neuromuscular Junction; TRPV Cation Channels | 2023 |