capsaicin and sb 366791

capsaicin has been researched along with sb 366791 in 54 studies

Research

Studies (54)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's23 (42.59)29.6817
2010's28 (51.85)24.3611
2020's3 (5.56)2.80

Authors

AuthorsStudies
Davies, CH; Davis, JB; Egerton, J; Gill, CH; Gunthorpe, MJ; Howett, L; Jerman, JC; Lappin, SC; Luis Hannan, S; Nasir, S; Owen, D; Rami, HK; Randall, AD; Smart, D; Smith, GD; Soffin, EM; Thompson, M; Worby, A; Wyman, PA1
Dell, H1
Desimone, JA; Ghosh, S; Heck, GL; Lyall, V; Phan, TH; Vinnikova, AK1
DeSimone, JA; Heck, GL; Lyall, V; Malik, SA; Mummalaneni, S; Phan, TH; Vinnikova, AK2
Elekes, K; Helyes, Z; McDougall, JJ; Németh, J; Pintér, E; Szabó, A; Szolcsányi, J; Varga, A; Zhang, C1
Adler-Graschinsky, E; Briones, R; Huidobro-Toro, JP; Orliac, ML; Poblete, IM1
Cowan, A; Ding, Z; Rawls, SM2
Andrade, EL; André, E; Calixto, JB; Ferreira, J1
Boudaka, A; Kobayashi, H; Neuhuber, WL; Shiina, T; Shimizu, Y; Takewaki, T; Wörl, J1
Alexander, SP; Athanasiou, A; Bagiokou, D; Bates, TE; Guo, DA; Kendall, DA; Kumaran, NM; Layfield, R; Lobo, DN; Lophatanon, A; Muir, KA; Ray, DE; Smith, PA; Turner, AE; Vakilpour, S; Watson, SA; Westwell, AD1
Medley, D; Naniwadekar, A; Pasricha, PJ; Shenoy, M; Winston, J1
Ferrini, F; Merighi, A; Salio, C; Vergnano, AM1
Asano, M; Harada, N; Mishima, A; Nakayama, T; Nomura, N; Okajima, K; Saito, T1
Pasricha, PJ; Pendyala, S; Shenoy, M; Winston, JH; Xu, GY; Yin, H1
Andrade, EL; Calixto, JB; Ferreira, J; Luiz, AP1
Cao, J; Li, HB; Mao, RR; Xu, L; Yang, Y; Zhang, JC1
Kopczyńska, B1
Cristino, L; Di Marzo, V; Drago, F; Leggio, GM; Micale, V; Petrosino, S; Tamburella, A1
Díaz-Laviada, I; Malagarie-Cazenave, S; Olea-Herrero, N; Vara, D1
Brink, TS; Potenzieri, C; Simone, DA1
Gregg, RG; Heimel, JA; Kamermans, M; Nawy, S; Peachey, NS; Shen, Y1
Brennan, FX; Bryant, RW; Devantier, HR; Long, DJ; Palmer, RK; Salemme, FR1
Fujihara, H; Hashimoto, H; Nagatomo, T; Ohbuchi, T; Otsubo, H; Saito, T; Suzuki, H; Ueta, Y; Yokoyama, T1
Andresen, MC; Fawley, JA; McDougall, SJ; Peters, JH; Smith, SM1
Harada, N; Ishikura, H; Kitamura, T; Okajima, K; Umemura, T1
Andresen, MC; Fawley, JA; McDougall, SJ; Peters, JH; Shoudai, K1
Buzas, K; Cohen, JI; Fan, H; Howard, OM; Klinman, D; Mont, E; Oppenheim, JJ; Qi, J; Wang, K1
Andrade, EL; Calixto, JB; Rogerio, AP1
de Oliveira, SM; Ferreira, J; Gomez, MV; Hoffmeister, C; Rossato, MF; Trevisan, G1
Chen, Y; Wang, ZJ; Yang, C1
Aguiar, DC; Casarotto, PC; Guimarães, FS; Moreira, FA; Terzian, AL; Wotjak, CT; Zangrossi, H1
Bogo, MR; Campos, MM; Couture, R; Dias, JP; Gaudreau, P; Lahjouji, K; Talbot, S1
Hitomi, S; Iwata, K; Shinoda, M; Suzuki, I1
Bratz, IN; Damron, DS; DelloStritto, DJ; Guarini, G; Kmetz, JG; Meszaros, JG; Ohanyan, VA; Thodeti, CK; Thoppil, RJ1
Coderre, EM; Hermes, ML; Kolaj, M; Renaud, LP1
DeSimone, JA; Grider, JR; Lyall, V; Mummalaneni, S; Murthy, KS; Phan, TH; Ren, Z; Rhyu, MR1
Adamek, P; Kalynovska, N; Mrozkova, P; Palecek, J; Spicarova, D1
Matsuda, Y; Murakami, S; Nakajima, T; Tabeta, K; Takahashi, N; Yamada, H; Yamazaki, K1
Abramson, L; Aoki-Nonaka, Y; Bertin, S; Corr, M; de Jong, PR; Dong, H; Franco, A; Fu, G; González-Navajas, JM; Gwack, Y; Han, T; Herdman, S; Jefferies, WA; Lee, J; Li, X; Nohara, LL; Raz, E; Srikanth, S; Stanwood, SR; To, K; Touma, R; Xu, H; Yu, T1
Burrell, BD; Holec, S; Summers, T1
Furukawa, A; Honda, K; Iwata, K; Kita, K; Noma, N; Shinoda, M1
Dale, CS; Ferro, ES; Fogaça, MV; Gozzo, FC; Guimarães, FS; Rioli, V; Sonego, AB1
Chen, HY; Chiang, AN; Guo, BC; Lee, TS; Shyue, SK; Su, KH; Wei, J; Zhao, JF1
Binkowski, M; Czaja, M; Di Marzo, V; Kolosowska, N; Makuch, W; Malek, N; Morera, E; Mrugala, M; Przewlocka, B; Starowicz, K1
Calzetta, L; Capuano, A; Cazzola, M; Facciolo, F; Luongo, L; Maione, S; Matera, MG; Page, C; Rinaldi, B; Rogliani, P1
Chen, X; Cui, W; Han, W; Jin, X; Long, C; Pan, Z; Wang, H; Zhang, Y1
Ide, S; Kojima, S; Nakanishi, Y; Nishino, K; Tanamachi, K; Tanuma, S; Tsukimoto, M1
Burrell, BD; Wang, Y1
Borges, MH; Castro-Junior, CJ; Ferreira, J; Gomez, MV; Palhares, MR; Rezende, MJS; Santos, DC; Silva, JF; Silva-Junior, CA1
Binda, NS; Borges, MH; Carobin, NV; Castro Junior, CJ; Ferreira, J; Gomez, MV; Kushmerick, C; Pinto Nagem, RA; Ribeiro, FM; Rita Pereira, EM; Santos, DC; Silva Júnior, CA; Silva, JF; Souza, JM1
Inoue, M; Magara, J; Nagoya, K; Shiraishi, N; Suzuki, T; Terunuma, M; Tsujimura, T; Yoshihara, M1
Arkhipov, AY; Fedorov, NS; Khabibrakhmanov, AN; Malomouzh, AI; Mukhamedyarov, MA; Nurullin, LF; Samigullin, DV1

Other Studies

54 other study(ies) available for capsaicin and sb 366791

ArticleYear
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.
    Neuropharmacology, 2004, Volume: 46, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acids; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Anilides; Aniline Compounds; Animals; Calcium; Capsaicin; Carrier Proteins; Cell Line; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Hot Temperature; Humans; Intracellular Signaling Peptides and Proteins; Kidney; Membrane Potentials; N-Methylaspartate; Neuropeptides; Norepinephrine; Orexins; Patch-Clamp Techniques; Protein Binding; Radioligand Assay; Rats; Receptors, Drug; Serotonin Receptor Agonists; Xanthenes

2004
New compound fires up pain research.
    Drug discovery today, 2003, Dec-01, Volume: 8, Issue:23

    Topics: Anilides; Animals; Capsaicin; Cinnamates; Humans; Nociceptors; Pain; Rats; Receptors, Drug

2003
A novel vanilloid receptor-1 (VR-1) variant mammalian salt taste receptor.
    Chemical senses, 2005, Volume: 30 Suppl 1

    Topics: Amiloride; Anilides; Animals; Capsaicin; Cinnamates; Diterpenes; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Salts; Sodium Channel Blockers; Sodium Chloride; Taste; Taste Buds; TRPV Cation Channels

2005
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. I. Effect on TRC volume and Na+ flux.
    The Journal of general physiology, 2005, Volume: 125, Issue:6

    Topics: Amiloride; Anilides; Animals; Capsaicin; Cell Size; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Cytosol; Diuretics; Ethanol; Female; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Taste; Temperature; Tongue

2005
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. II. Effect on chorda tympani salt responses.
    The Journal of general physiology, 2005, Volume: 125, Issue:6

    Topics: Algorithms; Amiloride; Anilides; Animals; Capsaicin; Cell Membrane; Cell Polarity; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Diterpenes; Diuretics; Ethanol; Female; In Vitro Techniques; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Stimulation, Chemical; Taste; Taste Threshold; Temperature; Tongue

2005
Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat.
    Neuroscience letters, 2005, Sep-09, Volume: 385, Issue:2

    Topics: Analgesics; Anilides; Animals; Capsaicin; Cells, Cultured; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Hypothermia; Ion Channels; Male; Mice; Mice, Inbred BALB C; Neurons, Afferent; Nociceptors; Pain; Peripheral Nervous System; Rats; Rats, Wistar; Sensory Receptor Cells; Substance P; Trigeminal Ganglion; TRPV Cation Channels

2005
Anandamide elicits an acute release of nitric oxide through endothelial TRPV1 receptor activation in the rat arterial mesenteric bed.
    The Journal of physiology, 2005, Oct-15, Volume: 568, Issue:Pt 2

    Topics: Anilides; Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Capsaicin; Cinnamates; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Artery, Superior; Nitric Oxide; Nitroarginine; Perfusion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; RNA, Messenger; TRPV Cation Channels; Vasodilation

2005
Capsaicin evokes hypothermia independent of cannabinoid CB1 and CB2 receptors.
    Brain research, 2005, Dec-14, Volume: 1065, Issue:1-2

    Topics: Anilides; Animals; Benzoxazines; Body Temperature; Calcium Channel Blockers; Camphanes; Capsaicin; Cinnamates; Hypothermia; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; TRPV Cation Channels

2005
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:4

    Topics: Amidohydrolases; Anilides; Animals; Arachidonic Acids; Body Temperature; Capsaicin; Cinnamates; Endocannabinoids; Hypothermia; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels

2006
Contractile mechanisms coupled to TRPA1 receptor activation in rat urinary bladder.
    Biochemical pharmacology, 2006, Jun-28, Volume: 72, Issue:1

    Topics: Acrolein; Anilides; Animals; Ankyrins; Binding Sites; Calcium Channels; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Drug Antagonism; In Vitro Techniques; Isothiocyanates; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Wistar; Ruthenium Red; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels; Urinary Bladder

2006
Involvement of TRPV1-dependent and -independent components in the regulation of vagally induced contractions in the mouse esophagus.
    European journal of pharmacology, 2007, Feb-05, Volume: 556, Issue:1-3

    Topics: Alkaloids; Anilides; Animals; Benzodioxoles; Capsaicin; Cinnamates; Cricetinae; Enzyme Inhibitors; Esophagus; Female; Male; Mesocricetus; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Tachykinin; Species Specificity; TRPV Cation Channels; Tryptophan; Vagus Nerve

2007
Vanilloid receptor agonists and antagonists are mitochondrial inhibitors: how vanilloids cause non-vanilloid receptor mediated cell death.
    Biochemical and biophysical research communications, 2007, Mar-02, Volume: 354, Issue:1

    Topics: Anilides; Animals; Apoptosis; Capsaicin; Carcinoma, Non-Small-Cell Lung; Cells, Cultured; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Humans; Hydrogen Peroxide; Lung Neoplasms; Membrane Potentials; Mitochondria, Heart; Oxygen Consumption; Rats; TRPV Cation Channels

2007
The vanilloid receptor initiates and maintains colonic hypersensitivity induced by neonatal colon irritation in rats.
    Gastroenterology, 2007, Volume: 132, Issue:2

    Topics: Acetic Acid; Age Factors; Anilides; Animals; Animals, Newborn; Capsaicin; Catheterization; Cinnamates; Colon; Disease Models, Animal; Diterpenes; Electromyography; Ganglia, Spinal; Hyperalgesia; Irritable Bowel Syndrome; Male; Pain; Rats; Rats, Sprague-Dawley; Reflex, Abdominal; TRPV Cation Channels; Visceral Afferents

2007
Vanilloid receptor-1 (TRPV1)-dependent activation of inhibitory neurotransmission in spinal substantia gelatinosa neurons of mouse.
    Pain, 2007, Volume: 129, Issue:1-2

    Topics: Anilides; Animals; Animals, Newborn; Bicuculline; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Immunohistochemistry; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Mice; Neural Inhibition; Neurons; Patch-Clamp Techniques; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin; TRPV Cation Channels; Tryptophan

2007
Atrial natriuretic peptide reduces ischemia/reperfusion-induced spinal cord injury in rats by enhancing sensory neuron activation.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Anilides; Animals; Atrial Natriuretic Factor; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Cells, Cultured; Cinnamates; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Indoles; Indomethacin; Male; Neurons, Afferent; Peroxidase; Psychomotor Performance; Pyrroles; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Spinal Cord; Spinal Cord Diseases; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2007
Transient receptor potential vanilloid 1 mediates hyperalgesia and is up-regulated in rats with chronic pancreatitis.
    Gastroenterology, 2007, Volume: 133, Issue:4

    Topics: Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Disease Models, Animal; Electric Stimulation; Ganglia, Spinal; Hyperalgesia; Male; Membrane Potentials; Pain Measurement; Pain Threshold; Pancreas; Pancreatitis, Chronic; Rats; Rats, Sprague-Dawley; RNA, Messenger; Time Factors; Trinitrobenzenesulfonic Acid; TRPV Cation Channels; Up-Regulation

2007
Pronociceptive response elicited by TRPA1 receptor activation in mice.
    Neuroscience, 2008, Mar-18, Volume: 152, Issue:2

    Topics: Analgesics; Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Isothiocyanates; Male; Mice; Pain; Pain Measurement; Ruthenium Red; Time Factors; Transient Receptor Potential Channels; TRPA1 Cation Channel

2008
Antistress effect of TRPV1 channel on synaptic plasticity and spatial memory.
    Biological psychiatry, 2008, Aug-15, Volume: 64, Issue:4

    Topics: Anilides; Animals; Animals, Newborn; Behavior, Animal; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Male; Memory; Neuronal Plasticity; Neurons; Rats; Rats, Wistar; Space Perception; Synaptic Transmission; TRPV Cation Channels

2008
Role of VR1 and CB1 receptors in modelling of cardio-respiratory response to arvanil, an endocannabinoid and vanilloid hybrid, in rats.
    Life sciences, 2008, Jul-18, Volume: 83, Issue:3-4

    Topics: Anilides; Animals; Blood Pressure; Cannabinoid Receptor Modulators; Capsaicin; Cinnamates; Disease Models, Animal; Endocannabinoids; Hypertension; Injections, Intravenous; Male; Morpholines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Respiration; Respiration Disorders; Ruthenium Red; Tidal Volume; TRPV Cation Channels

2008
Anxiolytic effects in mice of a dual blocker of fatty acid amide hydrolase and transient receptor potential vanilloid type-1 channels.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:3

    Topics: Amidohydrolases; Anilides; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cinnamates; Diazepam; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels

2009
Capsaicin, a component of red peppers, induces expression of androgen receptor via PI3K and MAPK pathways in prostate LNCaP cells.
    FEBS letters, 2009, Jan-05, Volume: 583, Issue:1

    Topics: Anilides; Capsaicin; Capsicum; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cinnamates; Diterpenes; Gene Silencing; Humans; Male; Mitogen-Activated Protein Kinase Kinases; Phosphatidylinositol 3-Kinases; Prostate; Receptors, Androgen; RNA, Small Interfering; TRPV Cation Channels

2009
Excitation of cutaneous C nociceptors by intraplantar administration of anandamide.
    Brain research, 2009, May-01, Volume: 1268

    Topics: Action Potentials; Anilides; Animals; Arachidonic Acids; Calcium Channel Blockers; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Endocannabinoids; Hindlimb; Hot Temperature; Male; Nociceptors; Pain; Pain Measurement; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Skin; Tibial Nerve; TRPV Cation Channels

2009
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, May-13, Volume: 29, Issue:19

    Topics: Amino Acids; Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Polyunsaturated Alkamides; Propionates; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; Ruthenium Red; Synaptic Transmission; Transient Receptor Potential Channels; TRPM Cation Channels; TRPV Cation Channels; Xanthenes

2009
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: Acrylamides; Administration, Oral; Alkaloids; Anilides; Animals; Avoidance Learning; Benzodioxoles; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazines; Pyridines; Taste; TRPM Cation Channels; TRPV Cation Channels

2010
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: Analysis of Variance; Angiotensin II; Anilides; Animals; Capsaicin; Chelating Agents; Cinnamates; Diuretics, Osmotic; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; In Vitro Techniques; Male; Mannitol; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Piperidines; Pyrazines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Supraoptic Nucleus; TRPV Cation Channels; Vasoconstrictor Agents

2010
Primary afferent activation of thermosensitive TRPV1 triggers asynchronous glutamate release at central neurons.
    Neuron, 2010, Mar-11, Volume: 65, Issue:5

    Topics: Afferent Pathways; Anilides; Animals; Capsaicin; Cinnamates; Electric Stimulation; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sensory System Agents; Solitary Nucleus; Thermosensing; TRPV Cation Channels

2010
Limaprost reduces motor disturbances by increasing the production of insulin-like growth factor I in rats subjected to spinal cord injury.
    Translational research : the journal of laboratory and clinical medicine, 2010, Volume: 156, Issue:5

    Topics: Alprostadil; Anilides; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Caspase 3; Cells, Cultured; Cinnamates; Denervation; Disease Models, Animal; Drug Therapy, Combination; Ganglia, Spinal; Gene Expression; Insulin-Like Growth Factor I; Male; Movement; Neurons; Rats; Rats, Wistar; RNA, Messenger; Sensory System Agents; Specific Pathogen-Free Organisms; Spinal Cord; Spinal Cord Injuries; Vasodilator Agents

2010
Thermally active TRPV1 tonically drives central spontaneous glutamate release.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Oct-27, Volume: 30, Issue:43

    Topics: Action Potentials; Anilides; Animals; Cadmium Compounds; Calcium; Capsaicin; Cinnamates; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Channel Blockers; Synapses; Tetrodotoxin; Thermosensing; TRPV Cation Channels

2010
Painful pathways induced by TLR stimulation of dorsal root ganglion neurons.
    Journal of immunology (Baltimore, Md. : 1950), 2011, Jun-01, Volume: 186, Issue:11

    Topics: Aminoquinolines; Anilides; Animals; Arachidonic Acids; Blotting, Western; Calcium; Capsaicin; Cells, Cultured; Cinnamates; Cytokines; Dinoprostone; Dose-Response Relationship, Drug; Endocannabinoids; Ganglia, Spinal; Humans; Imidazoles; Mice; Microscopy, Confocal; Neurons; Pain; Poly I-C; Polyunsaturated Alkamides; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Toll-Like Receptor 3; Toll-Like Receptor 7; Toll-Like Receptor 9; Toll-Like Receptors; TRPV Cation Channels

2011
C-fibers, but not the transient potential receptor vanilloid 1 (TRPV1), play a role in experimental allergic airway inflammation.
    European journal of pharmacology, 2011, Jul-15, Volume: 662, Issue:1-3

    Topics: Allergens; Anilides; Animals; Animals, Newborn; Bronchoalveolar Lavage Fluid; Capsaicin; Cell Count; Cinnamates; Cytokines; Female; Gene Expression Regulation; Hypersensitivity; Immunization; Inflammation; Leukocytes; Lung; Mice; Mice, Inbred BALB C; Nerve Fibers, Unmyelinated; NF-kappa B; Ovalbumin; P-Selectin; Respiratory System; TRPV Cation Channels

2011
Role of TRPV1 in nociception and edema induced by monosodium urate crystals in rats.
    Pain, 2011, Volume: 152, Issue:8

    Topics: Acrylamides; Anilides; Animals; Anti-Allergic Agents; Anti-Asthmatic Agents; Antioxidants; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Cromolyn Sodium; Disease Models, Animal; Diterpenes; Edema; Gabexate; Histamine; Male; Mast Cells; Methysergide; Pain; Promethazine; Prostaglandin-Endoperoxide Synthases; Protein Binding; Rats; Rats, Wistar; Serine Proteinase Inhibitors; Serotonin; Serotonin Antagonists; Tritium; TRPV Cation Channels; Uric Acid

2011
Proteinase-activated receptor 2 sensitizes transient receptor potential vanilloid 1, transient receptor potential vanilloid 4, and transient receptor potential ankyrin 1 in paclitaxel-induced neuropathic pain.
    Neuroscience, 2011, Oct-13, Volume: 193

    Topics: Analysis of Variance; Anilides; Animals; Ankyrins; Antineoplastic Agents, Phytogenic; Capsaicin; Carbazoles; Central Nervous System; Cinnamates; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Estrenes; Gene Expression Regulation; Hyperalgesia; Male; Mice; Mice, Inbred ICR; Neuralgia; Oligopeptides; Paclitaxel; Pain Measurement; Physical Stimulation; Protein Kinase C; Pyrroles; Pyrrolidinones; Receptor, PAR-2; Sulfonamides; Time Factors; TRPV Cation Channels; Tryptases; Type C Phospholipases

2011
Opposing roles for cannabinoid receptor type-1 (CB₁) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:2

    Topics: Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Drug Interactions; Electric Stimulation; Male; Microinjections; Panic; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2012
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
    Journal of neuroinflammation, 2012, Jan-20, Volume: 9

    Topics: Acetylcysteine; Analysis of Variance; Anilides; Animals; Antioxidants; Autoradiography; Bradykinin; Bradykinin B1 Receptor Antagonists; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Gene Expression Regulation; Iodine Isotopes; Male; Microglia; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; RNA, Messenger; Sensory System Agents; Spinal Cord; Superoxides; Tetrahydroisoquinolines; Time Factors; TRPV Cation Channels

2012
Involvement of transient receptor potential vanilloid 1 in ectopic pain following inferior alveolar nerve transection in rats.
    Neuroscience letters, 2012, Mar-28, Volume: 513, Issue:1

    Topics: Anilides; Animals; Antigens, Nuclear; Behavior, Animal; Capsaicin; Cell Count; Cinnamates; Electric Stimulation; Extracellular Signal-Regulated MAP Kinases; Facial Pain; Grooming; Immunohistochemistry; Male; Mandibular Nerve; Nerve Tissue Proteins; Phosphorylation; Rats; Rats, Sprague-Dawley; Trigeminal Ganglion; TRPV Cation Channels; Vibrissae

2012
Disruption of TRPV1-mediated coupling of coronary blood flow to cardiac metabolism in diabetic mice: role of nitric oxide and BK channels.
    American journal of physiology. Heart and circulatory physiology, 2012, Jul-15, Volume: 303, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Anilides; Animals; Capsaicin; Cinnamates; Coronary Vessels; Diabetes Mellitus, Type 2; Diabetic Cardiomyopathies; Enzyme Inhibitors; Large-Conductance Calcium-Activated Potassium Channels; Male; Mice; Mice, Inbred C57BL; Microvessels; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptides; TRPV Cation Channels; Vasoconstrictor Agents; Vasodilation

2012
Gastrin-releasing peptide acts via postsynaptic BB2 receptors to modulate inward rectifier K+ and TRPV1-like conductances in rat paraventricular thalamic neurons.
    The Journal of physiology, 2013, Apr-01, Volume: 591, Issue:7

    Topics: Anilides; Animals; Capsaicin; Cinnamates; Gastrin-Releasing Peptide; Male; Midline Thalamic Nuclei; Neurons; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Bombesin; TRPV Cation Channels

2013
TRPM5-dependent amiloride- and benzamil-insensitive NaCl chorda tympani taste nerve response.
    American journal of physiology. Gastrointestinal and liver physiology, 2013, Jul-01, Volume: 305, Issue:1

    Topics: Amiloride; Anilides; Animals; Capsaicin; Chorda Tympani Nerve; Cinnamates; Diterpenes; Mice; Mice, Knockout; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Sodium Chloride; Taste; TRPM Cation Channels; TRPV Cation Channels

2013
TRPV1 receptor inhibition decreases CCL2-induced hyperalgesia.
    Neuropharmacology, 2014, Volume: 81

    Topics: Anilides; Animals; Animals, Newborn; Capsaicin; Chemokine CCL2; Cinnamates; Disease Models, Animal; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Hyperalgesia; In Vitro Techniques; Male; MAP Kinase Kinase Kinase 3; Pain Threshold; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Rats, Wistar; Sensory System Agents; Spinal Cord; Time Factors; TRPV Cation Channels

2014
Epithelial TRPV1 signaling accelerates gingival epithelial cell proliferation.
    Journal of dental research, 2014, Volume: 93, Issue:11

    Topics: Anilides; Animals; Apoptosis; Capsaicin; Cell Line; Cell Proliferation; Cells, Cultured; Cinnamates; Epithelial Cells; Fibroblast Growth Factors; Gene Expression Profiling; Gingiva; HEK293 Cells; Humans; Male; Mice; Mice, Inbred C57BL; Nerve Growth Factors; Nociceptors; Oligonucleotide Array Sequence Analysis; Sensory System Agents; Signal Transduction; TRPV Cation Channels; Up-Regulation

2014
The ion channel TRPV1 regulates the activation and proinflammatory properties of CD4⁺ T cells.
    Nature immunology, 2014, Volume: 15, Issue:11

    Topics: Anilides; Animals; Calcium; Calcium Channels; Calcium Signaling; Capsaicin; CD4-Positive T-Lymphocytes; Cells, Cultured; Cinnamates; Colitis; Humans; Inflammation; Interleukin-10; Intestines; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptors, Antigen, T-Cell; Sensory System Agents; TRPV Cation Channels

2014
Physiological and behavioral evidence of a capsaicin-sensitive TRPV-like channel in the medicinal leech.
    The Journal of experimental biology, 2014, Dec-01, Volume: 217, Issue:Pt 23

    Topics: Anilides; Animals; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Hirudo medicinalis; Hot Temperature; Nociceptors; Sensory System Agents; TRPV Cation Channels

2014
TRPA1 contributes to capsaicin-induced facial cold hyperalgesia in rats.
    European journal of oral sciences, 2014, Volume: 122, Issue:6

    Topics: Acetanilides; Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Cold Temperature; Electromyography; Face; Facial Pain; Hot Temperature; Hyperalgesia; Injections, Intradermal; Male; Neural Conduction; Neurons; Physical Stimulation; Purines; Rats; Rats, Sprague-Dawley; Reflex; Sensory System Agents; Synaptic Transmission; Trigeminal Ganglion; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2014
Anxiogenic-like effects induced by hemopressin in rats.
    Pharmacology, biochemistry, and behavior, 2015, Volume: 129

    Topics: Anilides; Animals; Anxiety; Brain; Capsaicin; Cinnamates; Hemoglobins; Injections, Intraventricular; Male; Maze Learning; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Wistar

2015
Transient receptor potential vanilloid type 1 is vital for (-)-epigallocatechin-3-gallate mediated activation of endothelial nitric oxide synthase.
    Molecular nutrition & food research, 2015, Volume: 59, Issue:4

    Topics: AMP-Activated Protein Kinases; Anilides; Animals; Calcium; Capsaicin; Catechin; Cell Movement; Cell Proliferation; Cell Survival; Cinnamates; Endothelial Cells; HEK293 Cells; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Neovascularization, Pathologic; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphorylation; Signal Transduction; Tea; TRPV Cation Channels

2015
A multi-target approach for pain treatment: dual inhibition of fatty acid amide hydrolase and TRPV1 in a rat model of osteoarthritis.
    Pain, 2015, Volume: 156, Issue:5

    Topics: Activating Transcription Factor 3; Amidohydrolases; Anilides; Animals; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Cinnamates; Disease Models, Animal; Endocannabinoids; Ganglia, Spinal; Gene Expression; Hyperalgesia; Inflammation; Interleukin-6; Lumbar Vertebrae; Male; Osteoarthritis; Pain; Pain Management; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2015
Contribution of sensory nerves to LPS-induced hyperresponsiveness of human isolated bronchi.
    Life sciences, 2015, Jun-15, Volume: 131

    Topics: Anilides; Bronchi; Bronchial Hyperreactivity; Capsaicin; Cinnamates; Electric Stimulation; Female; Humans; Indoles; Lipopolysaccharides; Male; Middle Aged; Muscle Contraction; Neprilysin; Neurokinin A; Piperidines; Sensory Receptor Cells; TRPV Cation Channels; Up-Regulation

2015
The molecular pathway of ATP-sensitive potassium channel in endothelial cells for mediating arteriole relaxation.
    Life sciences, 2015, Sep-15, Volume: 137

    Topics: Allyl Compounds; Anilides; Animals; Arterioles; Calcium; Capsaicin; Cells, Cultured; Cinnamates; Down-Regulation; Endothelial Cells; KATP Channels; Mesenteric Arteries; Nitric Oxide; Propylamines; Rats; RNA, Small Interfering; TRPV Cation Channels; Vasodilation

2015
Radiosensitizing Effect of TRPV1 Channel Inhibitors in Cancer Cells.
    Biological & pharmaceutical bulletin, 2016, Jul-01, Volume: 39, Issue:7

    Topics: Acrylamides; Anilides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line, Tumor; Cell Survival; Cinnamates; DNA Damage; Gamma Rays; Humans; Mice; Necrosis; Neoplasms; Pyrazines; Pyridines; Radiation-Sensitizing Agents; TRPV Cation Channels

2016
Differences in chloride gradients allow for three distinct types of synaptic modulation by endocannabinoids.
    Journal of neurophysiology, 2016, 08-01, Volume: 116, Issue:2

    Topics: Anilides; Animals; Biophysics; Bumetanide; Cannabinoid Receptor Modulators; Capsaicin; Central Nervous System; Chlorides; Cinnamates; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Lactones; Leeches; Neurons; Orlistat; Patch-Clamp Techniques; Sensory System Agents; Sodium Potassium Chloride Symporter Inhibitors; Synapses

2016
Synergistic antinociceptive effect of a calcium channel blocker and a TRPV1 blocker in an acute pain model in mice.
    Life sciences, 2017, Aug-01, Volume: 182

    Topics: Acute Pain; Analgesics; Anilides; Animals; Body Temperature; Calcium Channel Blockers; Capsaicin; Cinnamates; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Mice; Spider Venoms; TRPV Cation Channels

2017
Phoneutria toxin PnTx3-5 inhibits TRPV1 channel with antinociceptive action in an orofacial pain model.
    Neuropharmacology, 2020, 01-01, Volume: 162

    Topics: Acrolein; Anilides; Animals; Calcium; Calcium Signaling; Capsaicin; Cinnamates; Disease Models, Animal; Facial Pain; Glutamic Acid; HEK293 Cells; Humans; Inhibitory Concentration 50; Male; Neuropeptides; Nociception; Patch-Clamp Techniques; Rats; Sensory System Agents; Transfection; Trigeminal Ganglion; TRPA1 Cation Channel; TRPV Cation Channels

2020
Sustained laryngeal transient receptor potential vanilloid 1 activation inhibits mechanically induced swallowing in anesthetized rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2020, 09-01, Volume: 319, Issue:3

    Topics: Anesthesia; Anilides; Animals; Capillary Permeability; Capsaicin; Cinnamates; Deglutition; Electric Stimulation; Laryngeal Nerves; Larynx; Male; Mechanoreceptors; Physical Stimulation; Radiation; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2020
Activation of TRPV1 Channels Inhibits the Release of Acetylcholine and Improves Muscle Contractility in Mice.
    Cellular and molecular neurobiology, 2023, Volume: 43, Issue:8

    Topics: Acetylcholine; Animals; Capsaicin; Mice; Muscle, Skeletal; Neuromuscular Junction; TRPV Cation Channels

2023