capsaicin and piperidines

capsaicin has been researched along with piperidines in 355 studies

Research

Studies (355)

TimeframeStudies, this research(%)All Research%
pre-19908 (2.25)18.7374
1990's92 (25.92)18.2507
2000's175 (49.30)29.6817
2010's72 (20.28)24.3611
2020's8 (2.25)2.80

Authors

AuthorsStudies
Jancsó-Gábor, A; Szolcsányi, J1
Lee, LY; Lou, YP; Lundberg, JM; Satoh, H2
Maggi, CA; Meli, A; Patacchini, R1
Jin, JG; Lu, YF; Nakayama, S; Takaki, M1
Szolcsànyi, J2
Goto, K; Ishikawa, T; Miyauchi, T; Saito, A; Sugishita, Y1
Lawless, HT; Stevens, DA3
Iwai, K; Kawada, T; Sakabe, S; Watanabe, T; Yamamoto, M1
Micevych, PE; Szolcsanyi, J; Yaksh, TL1
Amann, R; Donnerer, J; Holzer, P; Schuligoi, R1
Bolser, DC; Chapman, RW; DeGennaro, FC; Hey, JA; O'Reilly, S1
Ansay, M; Delaunois, A; Garbarg, M; Gustin, P1
Hay, DW; Hubbard, WC; Undem, BJ1
Advenier, C; Hirsch, A; Martin, CA; Molimard, M; Naline, E1
Besson, G; Drazen, JM; Israel, E; Lilly, CM; Rodger, IW1
Andersson, KE; Igawa, Y; Ishizuka, O; Mattiasson, A1
Brain, SD; Newbold, P1
Giuliani, S; Lecci, A; Maggi, CA; Meini, S1
Drazen, JM; Haley, KJ; Hall, AE; Kobzik, L; Lilly, CM; Rodger, IW1
Cioncolini, F; Figini, M; Geppetti, P; Javdan, P1
Barthò, L; Holzer, P; Maggi, CA; Patacchini, R1
Amann, R; Donnerer, J; Lanz, I; Schuligoi, R1
Andersson, KE; Ishizuka, O; Mattiasson, A1
Bertrand, C; Desai, MC; Hoffman, JI; Husseini, WK; Nadel, JA; Petersson, G; Piedimonte, G; Snider, RM1
Advenier, C; Emonds-Alt, X; Qian, Y1
Bertrand, C; Desai, MC; Geppetti, P; Nadel, JA; Piedimonte, G; Snider, RM1
Desai, MC; Hoffman, JI; Husseini, WK; Nadel, JA; Piedimonte, G; Snider, RM1
DeSautel, MG; Maher, JW; Sandler, AD; Schlegel, JF1
Bertrand, C; Geppetti, P; Graf, PD; Nadel, JA1
Bryce, DK; Desai, MC; Ganong, A; Longo, KP; McLean, S; Reynolds, LS; Robinson, G; Rosen, T; Seymour, PA; Snider, RM1
Maggi, CA; Meini, S1
Bennett, KL; Clark, MG; Colquhoun, EQ; Dora, KA; Eldershaw, TP1
Bannenberg, G; Kimland, M; Lundberg, JM; Moldéus, P; Ryrfeldt, A1
Auberson, S; Lundberg, JM1
Matui, T; Yoshii, K1
Bryce, DK; Desai, MC; Heym, J; Longo, KP; McLean, S; Rosen, T; Schmidt, AW; Snider, RM1
Bertrand, C; Foresi, A; Geppetti, P; Graf, PD; Nadel, JA1
Buckner, CK; Campbell, J; Dea, D; Krell, RD; Lengel, D; Liberati, N; Miller, S; Shenvi, A; Stinson-Fisher, C1
Vanner, S1
Lou, YP; Lundberg, JM; Satoh, H1
Everaert, E; Germonpré, PR; Joos, GF; Kips, JC; Pauwels, RA1
Beattie, DT; Brain, SD; Connor, HE; Escott, KJ1
Doerfler, DL; Sailstad, DM; Selgrade, M; Veronesi, B1
Conte, B; Cutrufo, C; Manzini, S1
Chiyotani, A; Kameyama, S; Konno, K; Sakai, N; Takeda, Y; Tamaoki, J; Yamawaki, I1
Kagoshima, M; Kodaira, H; Shimada, H; Tanaka, M1
Ikeda, K; Kubota, H; Miyata, K; Orita, A; Tomioka, K; Yamada, T1
Lin, Q; Peng, YB; Willis, WD1
Advenier, C; Emonds-Alt, X; Girard, V; Yavo, JC1
Bartho, L; Holzer, P1
Hodgson, WC; Hopkins, BJ; Sutherland, SK1
Inoue, H; Koshihara, Y; Nagata, N1
Juránek, I; Lembeck, F1
Lundberg, JM; Rinder, J1
Liu, L; Simon, SA1
Arakawa, M; Goto, F; Katori, M; Majima, M; Nagai, K1
Burkholder, TP; Knippenberg, RW; Kudlacz, EM; Logan, DE1
Caldwell, RW; Chiao, H1
Ellis, JL; Sham, JS; Undem, BJ1
Boucher, RC; Costa, DL; Lehmann, JR; McCarty, D; Pickles, RJ; Piedimonte, G1
Dimitriadou, V; Garbarg, M; Luffau, G; Miller, HR; Newlands, GJ; Rouleau, A; Schwartz, JC; Trung Tuong, MD1
Green, BG1
Green, BG; Rentmeister-Bryant, H1
Chen, PS; Rees, H; Sluka, KA; Tsuruoka, M; Willis, WD2
Arguelles, JH; Baumann, TK; Martenson, ME1
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M1
MacNaughton, W; Moore, B; Vanner, S1
Ishikawa, T; Menniti, FS; Mizutani, M; Nagahisa, A; Shimada, K; Shinjo, K; Taniguchi, K1
Advenier, C; Canet, E; Félétou, M; Girard, V1
Holst, JJ; Rasmussen, TN; Schmidt, PT1
Ahrén, B; Karlsson, S; Sundler, F1
Bereiter, DA; Bereiter, DF; Maclean, DB; Tonnessen, BH1
Bullock, B; Dickerson, C; Undem, B; Winchurch, RA1
Blackshaw, LA; Lynn, PA; Smid, SD; Templeman, R1
D'Orléans-Juste, P; Piovezan, AP; Rae, GA; Tonussi, CR1
Carstens, E; Handwerker, HO; Kuenzler, N1
Criscuoli, M; Giuliani, S; Lecci, A; Lippi, A; Maggi, CA; Patacchini, R; Santicioli, P; Tramontana, M1
Dong, F; Hasegawa, S; Iijima, H; Nomura, A; Uchida, Y; Xiang, A; Zhang, MJ1
Colquhoun, EQ; Eldershaw, TP; Geraghty, DP; Griffiths, CD1
Bryce, DK; Coffman, KJ; Crawford, RT; Gohda, Y; Lowe, JA; McLean, S; Nagahisa, A; Nakane, M; Rosen, TJ; Tsuchiya, M1
Fujiwara, H; Hirata, K; Kanazawa, H; Yoshikawa, J1
Guo, JZ; Otsuka, M; Yoshioka, K1
Baluk, P; Bunnett, NW; McDonald, DM; Murphy, TJ; Thurston, G1
Calixto, JB; Miguel, OG; Santos, AR; Yunes, RA1
Bakhle, YS; Bell, C; Brogan, JD1
Ko, MC; Woods, JH1
Perfumi, MC; Piccoli, M; Romagnoli, S; Santoni, G; Spreghini, E1
Geraghty, DP; Mazzone, SB1
Aoyama, M; Arai, Y; Inaba, N; Lee, B; Onodera, S; Shibata, M; Tanaka, M; Yamaura, T1
Aoyama, M; Arai, Y; Inaba, N; Nishizawa, A; Onodera, S; Sekine, Y; Shibata, M; Suzuki, T; Tanaka, M1
Fujita, A; Nishiwaki, H; Takeuchi, K; Umeda, M1
Barbara, G; Barthó, L; De Giorgio, R; Lecci, A; Lénárd, L; Maggi, CA; Patacchini, R; Stanghellini, V1
Lee, LY; Wu, ZX1
Carter, JD; Devlin, RB; Oortgiesen, M; Simon, SA; Veronesi, B1
Kato, S; Kunikata, T; Takeuchi, K; Tanaka, A; Umeda, M1
D'Orléans-Juste, P; Piovezan, AP; Rae, GA; Souza, GE1
Barthó, L; Benkó, R; Lázár, Z; Lénárd, L; Maggi, CA; Penke, B; Szolcsányi, J; Tóth, G1
Calixto, JB; Campos, MM; Ferreira, PK1
Doi, T; Ikeura, Y; Imai, S; Kamo, I; Natsugari, H; Okanishi, S1
D'Agostino, G; Erbelding, D; Kilbinger, H1
Chuang, H; Högestätt, ED; Julius, D; Movahed, P; Zygmunt, PM1
Filer-Maerten, S; Hay, DW; Hieble, JP; Ruggieri, MR1
Antunes, E; Costa, SK; da Silva, GR; Linardi, A1
Farkas, B; Helyes, ZS; Németh, J; Oroszi, G; Pintér, E; Szolcsányi, J; Thán, M1
Andrews, PL; Hagiwara, H; Kakaimoto, S; Matsuki, N; Okada, F; Toyoda, M; Woods, AJ1
Benbow, L; Corboz, MR; Egan, RW; Fawzi, AB; Hey, JA; Matasi, J; Rivelli, MA; Smith-Torhan, A; Tulshian, D; Zhang, H1
Hazato, T; Inoue, M; Matsunaga, S; Ueda, H; Yamamoto, Y1
Kim, D; Moore, BA; Vanner, S1
Carr, MJ; Schechter, NM; Undem, BJ1
Calignano, A; Désarnaud, F; Freund, TF; Giuffrida, A; Kátona, I; La Rana, G; Mackie, K; Piomelli, D1
Dahl, JB; Jones, B; Petersen, KL; Rowbotham, MC; Segredo, V1
Amadesi, S; Ansel, JC; Armstrong, CA; Bonaccorsi, P; Bunnett, NW; Geppetti, P; Gerard, NP; Grady, EF; Klein, R; Lu, B; Luger, TA; Olerud, JE; Scholzen, TE; Steinhoff, M1
Brockie, HC; Craib, SJ; Di Marzo, V; Gibson, TM; Leslie, M; Pashmi, G; Pertwee, RG; Ross, RA1
Van de Voorde, J; Vanheel, B1
Chapman, V; Kendall, DA; Millns, PJ1
Baird, AW; Goldhill, J; Moriarty, D; Selve, N1
Capasso, F; Capasso, R; Di Carlo, G; Izzo, AA; Mascolo, N; Pinto, L1
Kendall, DA; Ralevic, V1
Desouza, IA; Franco-Penteado, CF; Hyslop, S; Ribeiro-DaSilva, G2
Manning, BP; Mawe, GM1
Gitlin, JM; Mitchell, JA; Stanford, SJ1
Baird, AW; Goldhill, J; Moriarty, D; O'Donoghue, DP; Selve, N1
Corboz, MR; Egan, RW; Fernandez, X; Hey, JA1
Hayashi, K; Ishii, A; Kaise, T; Karasawa, A; Ohmori, K; Sano, J; Sato, H1
Heitmiller, DR; Hodges, J; Johanek, LM; Nader, N; Simone, DA; Turner, M1
Yonehara, N; Yoshimura, M1
Craib, SJ; Ellington, HC; Pertwee, RG; Ross, RA1
Antunes, E; Brain, SD; Camargo, EA; Costa, SK; de Nucci, G; Esquisatto, LC; Ribela, MT1
Erbelding, D; Kilbinger, H; Mang, CF1
Antunes, E; Brain, SD; Camargo, E; Costa, SK; De Nucci, G; Esquisatto, LC; Gambero, A1
Hataishi, R; Hayashi, I; Imasaki, T; Kobayashi, H; Majima, M; Tomita, T1
Kashon, ML; Krajnak, KM; Kwong, K; Lee, LY; Wise, PM; Wu, ZX1
Bottrill, FE; Ford, WR; Hiley, CR; Ho, WS; White, R1
Boachie-Ansah, G; Grainger, J1
Fowler, CJ; Jacobsson, SO; Wallin, T1
Brain, SD; Gerard, NP; Rawlingson, A1
Horie, S; Murayama, T; Tsuchiya, S; Uchida, M; Watanabe, K; Yamamoto, H1
Hayashi, I; Kamijo, Y; Majima, M; Ohwada, T; Soma, K1
Lever, IJ; Malcangio, M1
Eltorp, CT; Hansen, AJ; Ingvardsen, BK; Jørgensen, TK; Lundbaek, JA; Olsen, UB; Thomsen, C1
Antunes, E; Brain, SD; Costa, SK; De Nucci, G; Esquisatto, LC; Juliano, L; Moreno, RA1
Ko, MC; McKnight, AT; Naughton, NN; Rice, KC; Song, MS; Traynor, JR; Woods, JH1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N; Nocerino, E; Pinto, A; Sautebin, L1
Ajioka, H; Matsuura, N; Nakano, M; Nishihara, K; Nozawa, Y1
Naidu, KA; Thippeswamy, NB1
Berrino, L; Cuomo, D; de Novellis, V; Maione, S; Marabese, I; Palazzo, E; Rossi, F1
Baker, D; Bifulco, M; Bisogno, T; Bridges, D; Brooks, JW; Brown, P; Di Marzo, V; Hankey, DJ; Jaggar, SI; Ledent, C; Pryce, G; Rice, AS1
Chapnick, BM; Howlett, AC; Mukhopadhyay, S1
Cameron, NE; Cotter, MA; Ellington, HC; Ross, RA1
Ashton, D; Fransen, JF; Hens, KA; Heylen, L; Hillen, LC; Janssens, F; Jurzak, MR; Leysen, JE; Mahieu, M; Megens, AA; Vermeire, JC; Vermote, PC1
Anthes, JC; Billah, M; Carruthers, N; Chapman, RW; Corboz, M; Crawley, Y; Cuss, FM; Eckel, S; Egan, RW; Fernandez, X; Greenfeder, S; Hey, JA; Kreutner, W; McLeod, R; Piwinski, J; Reichard, G; Richard, C; Rizzo, C; Sehring, S; Shih, NY; Ting, P1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N; Pinto, A; Russo, A; Sautebin, L1
Freund, TF; Hájos, N1
Egan, RW; Hey, JA; Jia, Y; McLeod, RL; Parra, LE; Wang, X1
Bilbao, A; Cippitelli, A; Del Arco, I; Ferrer, B; Gómez, R; Nava, F; Navarro, M; Piomelli, D; Rodríguez de Fonseca, F; Trigo, JM1
Aoi, M; Kagawa, S; Kato, S; Kohama, K; Mimaki, H; Satoshi, T; Takeuchi, K1
Helyes, Z; Jakab, B; Németh, J; Pintér, E; Szolcsányi, J; Thán, M1
Adinolfi, B; Breschi, MC; Calderone, V; Martinotti, E; Nieri, P; Testai, L1
Kurosawa, M; Terano, A; Watanobe, H; Yoneda, M1
Ahluwalia, J; Bevan, S; Nagy, I; Urban, L; Yaqoob, M1
Ates, M; Gühring, H; Hamza, M; Seidel, K1
de Miguel, R; De Petrocellis, L; Di Marzo, V; Fernández-Ruiz, J; Lastres-Becker, I; Makriyannis, A1
Kaminski, NE; Li, J; Wang, DH1
Bang, R; Kiemer, AK; Neuhuber, WL; Sass, G; Tiegs, G; Vollmar, AM1
Beirith, A; Calixto, JB; Santos, AR1
Dey, RD; Satterfield, BE; Wu, ZX1
Shea-Donohue, T; Zhao, A1
Ahluwalia, J; Bevan, S; Nagy, I; Urban, L1
Curry, R; Eisenach, JC; Hood, DD1
Horie, S; Murayama, T; Someya, A; Yamamoto, H1
Barnes, PJ; Belvisi, MG; Birrell, MA; Crispino, N; Hele, DJ; Patel, HJ; Venkatesan, P; Yacoub, MH1
Itoh, M; Joh, T; Kasugai, K; Nomura, T; Ohara, H; Oshima, T; Seno, K; Sobue, M; Suzuki, H; Yokoyama, Y1
Calixto, JB; El Sayah, M1
Kato, S; Nagahama, K; Takeuchi, K; Yamato, M1
Adler-Graschinsky, E; Celuch, SM; del Carmen García, M1
Alexandre-Moreira, MS; Barreiro, EJ; Bolzani, Vda S; Palhares de Miranda, AL; Viegas, C1
Bueno, L; Bunnett, NW; Cenac, N; Coelho, AM; Compton, SJ; Garcia-Villar, R; Grady, E; Hollenberg, MD; Nguyen, C; Steinhoff, M; Vergnolle, N; Wallace, JL1
Köfalvi, A; Ledent, C; Sperlágh, B; Vizi, ES1
Dahl, JB; Hoke, F; Maloney, A; Petersen, KL; Rowbotham, MC1
Farquhar-Smith, WP; Rice, AS1
Dougalis, A; Lees, G1
Akerman, S; Goadsby, PJ; Kaube, H1
Capparelli, A; Mulè, F; Pizzuti, R; Vergnolle, N1
Green, BG; Hayes, JE1
Evans, RM; Ross, RA; Scott, RH1
Bánvölgyi, A; Brain, SD; Ghosh, M; Helyes, ZS; Melegh, B; Pintér, E; Pozsgai, G; Szolcsányi, J1
Amantini, C; Lucciarini, R; Perfumi, M; Piccoli, M; Pompei, P; Santoni, G1
Edwards, M; Schaffler, K; Seibel, K; Thomsen, M1
Belai, A; Horie, S; Michael, GJ; Murayama, T; Priestley, JV; Uchida, M; Watanabe, K; Yamamoto, H1
Godlewski, G; Malinowska, B; Schlicker, E1
Baamonde, A; Fresno, MF; Hidalgo, A; Lastra, A; Llames, S; Meana, A; Menéndez, L1
Adler-Graschinsky, E; Becu-Villalobos, D; Celuch, SM; Huidobro-Toro, JP; Orliac, ML; Peroni, RN1
Duncan, M; Kendall, DA; Ralevic, V1
Chapman, V; Kendall, DA; Millns, PJ; Sagar, DR; Smart, D; Smith, PA1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N1
Colleoni, M; Costa, B; Franke, C; Giagnoni, G; Trovato, AE1
Ahluwalia, A; Chauhan, S; Davis, C; De Felipe, C; Hunt, S; Kabir, J; Kotsonis, P; Oh, U; Scotland, RS1
Bembry, J; Chen, Y; Golech, SA; Lenz, F; McCarron, RM; Mechoulam, R; Shohami, E; Spatz, M1
Kato, S; Okayama, M; Takeuchi, K; Tsubouchi, R1
Ajioka, H; Horie, S; Kunieda, K; Murayama, T; Someya, A1
Bianchi, R; Borsani, E; Buffoli, B; Rezzani, R; Ricci, F; Rodella, LF1
Brzozowski, T; Ceranowicz, P; Dembiński, A; Dembiński, M; Konturek, SJ; Pawlik, WW; Warzecha, Z1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1
Gunthorpe, MJ; McNamara, FN; Randall, A1
Inoue, A; Kawamoto, M; Nakata, Y; Oshita, K; Tang, HB; Yuge, O1
Kendall, DA; O'Sullivan, SE; Randall, MD1
Cadet, JL; Chen, J; Deng, X; Errico, S; Freed, WJ; Lee, CT1
Breuer, A; Fride, E; Hanus, L; Ponde, D1
Maor, Y; Mechoulam, R; Pertwee, RG; Stevenson, LA; Thomas, A1
O'Reilly, M; Patton, D; Vanner, S1
Chapman, V; Kelly, S; Kendall, DA; Millns, PJ; O'Shaughnessey, CT; Sagar, DR1
Easton, AS; Fraser, PA; Hu, DE1
Adler-Graschinsky, E; Briones, R; Huidobro-Toro, JP; Orliac, ML; Poblete, IM1
Abe, T; Arisaka, O; Morimoto, H; Ohori, M; Yamada, Y; Yoshihara, S1
Farthing, JN; Gutierrez, T; Hohmann, AG; Suplita, RL1
Kaminski, NE; Wang, DH; Wang, Y1
Brain, SD; Costa, SK; Muscará, MN; Poston, RN; Yshii, LM1
Cowan, A; Ding, Z; Rawls, SM2
Fujimoto, S; Kunimatsu, M; Mori, M; Tsushima, H1
Braida, D; Guerini-Rocco, C; Pegorini, S; Sala, M; Zani, A1
Aoi, Y; Fukushima, K; Kato, S; Takeuchi, K1
Donnerer, J; Liebmann, I1
Kuramasu, A; Mobarakeh, JI; Sakurada, S; Takahashi, K; Yanai, K1
Cichewicz, DL; Haller, VL; Welch, SP1
Chabot, JG; Jhamandas, K; Ma, W; Quirion, R; Trang, T1
Baik, SK; Dehpour, AR; Gaskari, SA; Lee, SS; Liu, H; Moezi, L1
Baron, R; Chung, JM; Chung, K; Kim, HK; Lee, I; Schattschneider, J1
Boudaka, A; Kobayashi, H; Neuhuber, WL; Shiina, T; Shimizu, Y; Takewaki, T; Wörl, J1
Budai, D; Khasabov, SG; Mantyh, PW; Simone, DA1
Harada, N; Okajima, K1
Ali, N; Chapman, V; Chimenti, M; de Lago, E; Fernandez-Ruiz, J; Kendall, DA; Millns, PJ; Ryland, E1
De Ridder, D; Gevaert, T; Hutchings, G; Nilius, B; Vandepitte, J; Vriens, J1
Avezaat, CJ; de Vries, R; Garrelds, IM; Gupta, S; Lozano-Cuenca, J; MaassenVanDenBrink, A; Saxena, PR; van Kats, JP; Villalón, CM1
Matsuda, H; Nagatomo, A; Ochi, M; Yoshikawa, M1
Affeltranger, MA; Balaban, CD; McBurney, DH1
Cristino, L; Davison, JS; Di Marzo, V; Guglielmotti, V; Oland, LD; Pittman, QJ; Sharkey, KA; Starowicz, K; Van Sickle, MD1
Bianchi, R; Borsani, E; Labanca, M; Rodella, LF1
Srinivasan, K; Suresh, D3
Agrò, AF; Bagetta, G; Bari, M; Cerulli, A; Corasaniti, MT; De Simone, C; Gasperi, V; Maccarrone, M; Morrone, LA; Nucci, C; Tartaglione, R; Terrinoni, A1
Herradón, E; López-Miranda, V; Martín, MI1
Kendall, DA; Ralevic, V; Wilkinson, JD1
Wang, DH; Wang, Y1
Hatanaka, Y; Iwatani, Y; Jin, X; Kawasaki, H; Sugiyama, T1
d'amico, A; de Filippis, D; de Man, JG; de Winter, BY; Esposito, G; Herman, AG; Iuvone, T; Pelckmans, PA; Steardo, L1
Barrett, E; Xu, F; Xu, J1
Kamei, C; Kuyama, S; Ogawa, M; Yokota, E1
Cristino, L; Di Marzo, V; Drago, F; Leggio, GM; Micale, V; Petrosino, S; Tamburella, A2
Amagase, K; Hayashi, S; Komatsu, Y; Kotani, T; Murashima, Y; Nakagiri, A; Takeuchi, K1
Chang, HM; Chen, GD; Chiu, CH; Huang, PC; Lai, CH; Lai, CY; Lee, SD; Lin, TB; Peng, HY; Tung, KC1
Brandt, MR; Calvo, RR; Cheung, WS; Flores, CM; Hutchinson, T; Player, MR; Stone, DR; Tounge, BA; Zhang, SP1
Bitencourt, RM; Pamplona, FA; Takahashi, RN1
De Felice, M; Fioravanti, B; Gardell, LR; Ibrahim, M; King, T; Lai, J; Luo, MC; Malan, TP; Medler, KA; Ossipov, MH; Porreca, F; Stucky, CL; Vanderah, TW; Yamamura, HI1
Futamura, M; Goto, S; Ito, K; Kimoto, I; Kimura, R; Miyake, M; Sakamoto, T1
Boudaka, A; Neuhuber, WL; Shiina, T; Shimizu, Y; Takewaki, T; Wörl, J1
Atorino, G; Aviello, G; Borrelli, F; Capasso, R; Pagano, E; Romano, B1
Caldwell, JP; Fawzi, A; Fernandez, X; Matasi, JJ; McLeod, RL; Tulshian, DB; Zhang, H1
Donnerer, J; Liebmann, I; Schuligoi, R1
Hatakeyama, D; Kato, K; Long, NK; Makita, H; Shibata, T; Takeda, T; Toida, M; Yamashita, T1
Fantegrossi, WE; Galuska, CM; Ko, MC; Prinssen, EP; Wichmann, J; Woods, JH1
Hayes, D; Lee, LY; Lin, RL1
Jean, A; Lebrun, B; Roux, J; Trouslard, J; Wanaverbecq, N1
Buschmann, H; Grosse Maestrup, E; Holenz, J; Schepmann, D; Vela, JM; Wiese, C; Wünsch, B1
Chichorro, JG; Motta, EM; Rae, GA1
Challapalli, SC; Smith, PJ; Zhang, F1
Naidu, KA; Raghavendra, RH1
Bien, MY; Hsu, CC; Huang, YT; Kou, YR; Lin, YS; Ruan, T1
Kondo, S; Matsumoto, M; Ueda, H; Usdin, TB1
Hamity, MV; Hammond, DL; White, SR1
Brennan, FX; Bryant, RW; Devantier, HR; Long, DJ; Palmer, RK; Salemme, FR1
Calò, G; Guerrini, R; Hu, E; Ko, MC1
Chen, W; Lao, L; Marvizón, JC; Zhang, G1
Fujihara, H; Hashimoto, H; Nagatomo, T; Ohbuchi, T; Otsubo, H; Saito, T; Suzuki, H; Ueta, Y; Yokoyama, T1
Kushmerick, C; Morini, Vde C; Naves, LA; Silveira, NA; Silveira, PE1
Prakash, UN; Srinivasan, K4
Correa, EA; Echeverri, F; Högestätt, ED; Sterner, O; Zygmunt, PM1
Guindon, J; Hohmann, AG; Spradley, JM1
Azuma, M; Kang, KS; Matsuda, K; Sakashita, A; Shioda, S; Yahashi, S1
Beattie, RE; Knopp, K; Liu, B; Sher, E; Ursu, D1
Amagase, K; Kato, S; Ochi, A; Sugihara, T; Takeuchi, K1
Alexander, SP; Randall, MD; Wheal, AJ1
Capó-Aponte, JE; Pan, Z; Reinach, PS; Wang, Z; Yang, H; Zhang, F1
Akiba, Y; Kaunitz, JD1
Karaki, S; Kuwahara, A1
Chen, C; Chen, X; Zhang, J1
Almeida, MC; Balaskó, M; Dogan, MD; Eales, J; Gavva, NR; Molchanova, AY; Oliveira, DL; Patel, S; Pétervári, E; Romanovsky, AA; Steiner, AA; Székely, M; Wanner, SP1
Goadsby, PJ; Kavantzas, N; Knight, YE; Lasalandra, M; Mitsikostas, DD1
Fujita, T; Jiang, CY; Kumamoto, E; Mizuta, K; Piao, LH; Yang, L; Yue, HY1
Hayase, T1
Aguiar, DC; Casarotto, PC; Guimarães, FS; Moreira, FA; Terzian, AL; Wotjak, CT; Zangrossi, H1
Attkins, N; Bateman, L; Bictash, M; Doyle, R; Ivarsson, M; Neal-Morgan, S; Pullen, N; Ramsey, S; Russell, R; Turner, J; Weibley, L1
Beitz, AJ; Brink, TS; Khasabov, SG; Pacharinsak, C; Simone, DA1
Henry, PJ; Mann, TS; Taylor, SJ1
Jin, H; Kawasaki, H; Kitamura, Y; Koyama, T; Sun, P; Takatori, S; Tangsucharit, P; Zamami, Y1
Baranowska-Kuczko, M; Kozłowska, H; MacLean, MR; Malinowska, B1
Aguiar, DC; Fogaça, MV; Guimarães, FS; Moreira, FA1
Castellaneta, E; Cava, E; Ceccarelli, P; Claudia, S; Donini, LM; Edda, C; Emanuela, C; Faliva, M; Fioravanti, M; Klersy, C; Luciano, S; Maddalena, P; Opizzi, A; Paola, C; Paolini, M; Perna, S; Rondanelli, M; Savina, C; Scavone, L; Solerte, SB1
Claudia, S; Donini, LM; Edda, C; Emanuela, C; Faliva, M; Fioravanti, M; Klersy, C; Luciano, S; Maddalena, P; Opizzi, A; Paola, C; Perna, S; Rondanelli, M; Solerte, SB1
Srinivasan, K1
Fischer, MJ; Kageneck, C; Messlinger, K; Nixdorf-Bergweiler, BE1
Abílio, VC; Almeida, V; Calzavara, MB; Crippa, JA; Hallak, JE; Levin, R; Peres, FF; Suiama, MA; Zuardi, AW1
Alvarez-Berdugo, D; Clavé, P; Jiménez, M; Rofes, L1
Andresen, MC; Fawley, JA; Hofmann, ME1
Lee, M1
Dale, CS; Ferro, ES; Fogaça, MV; Gozzo, FC; Guimarães, FS; Rioli, V; Sonego, AB1
Binkowski, M; Czaja, M; Di Marzo, V; Kolosowska, N; Makuch, W; Malek, N; Morera, E; Mrugala, M; Przewlocka, B; Starowicz, K1
Calzetta, L; Capuano, A; Cazzola, M; Facciolo, F; Luongo, L; Maione, S; Matera, MG; Page, C; Rinaldi, B; Rogliani, P1
Camargo, LL; Costa, SK; Denadai-Souza, A; Fernandes, E; Grant, A; Lima, C; Mesquita, FP; Muscará, MN; Schenka, A; Soares, AG; Yshii, LM1
Cho, YM; Kiriyama, Y; Nishikawa, A; Ogawa, K; Shi, L; Takasu, S; Tatematsu, M; Toyoda, T; Tsukamoto, T1
Bartho, L; Bencsik, T; Sandor, Z1
Decorps, J; Fromy, B; Gohin, S; Sigaudo-Roussel, D1
Khan, M; Ma, T; Maryam, A; Mehmood, T; Zhang, Y1
Hott, SC; Lisboa, SF; Resstel, LB; Uliana, DL1
Hayes, JE; McGeary, JE; Nolden, AA1
He, Q; Jian, T; Lan, L; Shi, H; Tang, M; Tang, Z; Wang, C; Wang, Z; Wu, G; Yang, N; Yang, Y; Yu, G; Yuan, X; Zhu, C1
Hu, SS1
Adams, MJ; Geraghty, DP; Kunde, DA; Omari, SA1
Bradshaw, H; Carey, LM; Cornett, B; Hohmann, AG; Leishman, E; Mackie, K; Slivicki, RA1
Li, HB; Li, S; Li, Y; Xu, DP; Zheng, J; Zhou, Y1
Hinz, B; Ivanov, I; Scholl, A1
Lim, LY; Shamsi, S; Tan, RS; Tan, ZJ; Tran, H1
Coderre, TJ; Ding, S; Gyawali, S; Laferrière, A; Mahboubi, H; Mickeviciute, A; Nasir, H; Ragavendran, JV; Stochaj, U1
Gao, G; Heng, L; Jia, D; Qu, L; Song, J; Wang, X; Wang, Y; Zhang, H1
Giesler, GJ; Khasabov, SG; Malecha, P; Noack, J; Simone, DA; Tabakov, J1
Bae, IH; Burns, A; Choi, G; Choi, JK; Fagg, R; Gatfield, KM; Lee, CS; Naidoo, AA; Park, M; Park, YH; Powell, AJ; Vidgeon-Hart, M1
Fatahi, Z; Haghparast, A; Khani, A; Rainer, G; Reisi, Z1
Kim, TH; Shin, BS; Shin, S; Yoo, SD1
Krstin, S; Li, H; Wang, S; Wink, M1
Carneiro de Freitas, JC; Macedo Rondon, FC; Maia de Morais, S; Pereira Mendes, FN; Pinto Vieira, ÍG; Vieira-Araújo, FM1
Fernandes, PD; Giorno, TBS; Moreira, IGDS; Rezende, CM1
Aso, H; Suemaru, K; Watanabe, M; Yoshikawa, M1
Aboud, M; Comai, S; De Gregorio, D; Enns, J; Gobbi, G; Lopez-Canul, M; Maione, S; McLaughlin, RJ; Ochoa-Sanchez, R; Posa, L1
Ahmad, I; Baig, MH; Imran, M; Kausar, MA; Saeed, M; Shahid, S1
Dong, Y; Tian, Y; Vu, S; Yang, F; Yarov-Yarovoy, V; Yin, Y; Zheng, J1
Gerber, W; Hamman, J; Kotzé, A; Steyn, D; Svitina, H; Weldon, C1
Bortolanza, M; Crivelaro do Nascimento, G; Del Bel, EA; Ferrari, DP; Ferreira-Junior, NC; Guimaraes, FS1
Gaafar, AY; Istiqomah, I; Kawato, Y; Nakai, T; Ninomiya, K; Yamashita, H; Younes, A1
Buitimea-Cantúa, GV; Buitimea-Cantúa, NE; Hernández-Morales, A; Magaña-Barajas, E; Molina-Torres, J; Rocha-Pizaña, MDR1
Chung, YC; Jin, BK; Wi, R1
Hara, K; Haranishi, Y; Terada, T1
Almeida, PM; Dias, MS; Junior, EPV; Martins, FA; Peron, AP; Santos, BCD1
Ambedkar, R; Baskaran, V; Hanumanthappa, M; Lakshminarayana, R; Perumal, MK; Shilpa, S; Shwetha, HJ1
Alvarez-Berdugo, D; Clavé, P; Ortega, O; Rofes, L; Tomsen, N1

Reviews

3 review(s) available for capsaicin and piperidines

ArticleYear
Antioxidant potential of spices and their active constituents.
    Critical reviews in food science and nutrition, 2014, Volume: 54, Issue:3

    Topics: Alkaloids; Anti-Inflammatory Agents; Antimutagenic Agents; Antioxidants; Benzodioxoles; Capsaicin; Cardiotonic Agents; Catechols; Curcumin; Eugenol; Fatty Alcohols; Garlic; Humans; Neoplasms; Onions; Oxidative Stress; Phenols; Piperidines; Polyunsaturated Alkamides; Spices; Trigonella

2014
Enhancing Activity of Anticancer Drugs in Multidrug Resistant Tumors by Modulating P-Glycoprotein through Dietary Nutraceuticals.
    Asian Pacific journal of cancer prevention : APJCP, 2015, Volume: 16, Issue:16

    Topics: Abietanes; Alkaloids; Allyl Compounds; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Benzodioxoles; beta Carotene; Biflavonoids; Capsaicin; Catechin; Catechols; Curcumin; Dietary Supplements; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Fatty Alcohols; Furocoumarins; Humans; Indoles; Limonins; Neoplasms; Phytotherapy; Piperidines; Polyunsaturated Alkamides; Proanthocyanidins; Quercetin; Resveratrol; Stilbenes; Sulfides; Tea; Triterpenes; Xanthophylls

2015
Spices for Prevention and Treatment of Cancers.
    Nutrients, 2016, Aug-12, Volume: 8, Issue:8

    Topics: Alkaloids; Antineoplastic Agents, Phytogenic; Apoptosis; Benzodioxoles; Benzoquinones; Capsaicin; Capsicum; Cell Proliferation; Crocus; Curcuma; Curcumin; Garlic; Humans; Neoplasms; Nigella sativa; Phytotherapy; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Spices; Zingiber officinale

2016

Trials

8 trial(s) available for capsaicin and piperidines

ArticleYear
Rapid recovery from capsaicin desensitization during recurrent stimulation.
    Pain, 1996, Volume: 68, Issue:2-3

    Topics: Administration, Oral; Adult; Alkaloids; Analysis of Variance; Benzodioxoles; Capsaicin; Citric Acid; Depression, Chemical; Dose-Response Relationship, Drug; Female; Guaiacol; Humans; Irritants; Logistic Models; Male; Piperidines; Polyunsaturated Alkamides; Reference Values; Stimulation, Chemical; Time Factors; Tongue

1996
Effect of remifentanil on pain and secondary hyperalgesia associated with the heat--capsaicin sensitization model in healthy volunteers.
    Anesthesiology, 2001, Volume: 94, Issue:1

    Topics: Adult; Analgesics, Opioid; Capsaicin; Female; Hot Temperature; Humans; Hyperalgesia; Male; Middle Aged; Pain Measurement; Piperidines; Remifentanil

2001
Intravenous remifentanil produces withdrawal hyperalgesia in volunteers with capsaicin-induced hyperalgesia.
    Anesthesia and analgesia, 2003, Volume: 97, Issue:3

    Topics: Adult; Analgesics, Opioid; Capsaicin; Female; Humans; Hyperalgesia; Male; Nausea; Oxyhemoglobins; Pain Measurement; Piperidines; Remifentanil

2003
A randomized study of the effect of oral lamotrigine and hydromorphone on pain and hyperalgesia following heat/capsaicin sensitization.
    The journal of pain, 2003, Volume: 4, Issue:7

    Topics: Adult; Analgesics, Opioid; Anticonvulsants; Capsaicin; Double-Blind Method; Drug Therapy, Combination; Excitatory Amino Acid Antagonists; Hot Temperature; Humans; Hydromorphone; Hyperalgesia; Lamotrigine; Pain; Pain Measurement; Piperidines; Remifentanil; Triazines

2003
Effect of the new H1-antagonist ReN1869 on capsaicin-induced hyperalgesia in human skin/Human phase-I trial using somatosensory evoked potentials induced by a CO2 laser.
    Arzneimittel-Forschung, 2004, Volume: 54, Issue:3

    Topics: Adult; Arousal; Capsaicin; Cross-Over Studies; Double-Blind Method; Electroencephalography; Evoked Potentials, Somatosensory; Histamine H1 Antagonists; Humans; Hyperalgesia; Lasers; Male; Pain Measurement; Piperidines; Skin

2004
Palliative effect of lafutidine on oral burning sensation.
    Journal of oral pathology & medicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology, 2009, Volume: 38, Issue:3

    Topics: Acetamides; Aged; Burning Mouth Syndrome; Capsaicin; Female; Histamine H2 Antagonists; Humans; Male; Neurons, Afferent; Pain Measurement; Palliative Care; Piperidines; Pyridines; Sensory System Agents; Treatment Outcome

2009
Improvement in insulin resistance and favourable changes in plasma inflammatory adipokines after weight loss associated with two months' consumption of a combination of bioactive food ingredients in overweight subjects.
    Endocrine, 2013, Volume: 44, Issue:2

    Topics: Adipokines; Adult; Alkaloids; Benzodioxoles; Capsaicin; Carnitine; Catechin; Diet, Reducing; Dietary Supplements; Double-Blind Method; Female; Humans; Inflammation Mediators; Insulin Resistance; Male; Middle Aged; Overweight; Piperidines; Polyunsaturated Alkamides; Time Factors; Weight Loss; Young Adult

2013
Acute effect on satiety, resting energy expenditure, respiratory quotient, glucagon-like peptide-1, free fatty acids, and glycerol following consumption of a combination of bioactive food ingredients in overweight subjects.
    Journal of the American College of Nutrition, 2013, Volume: 32, Issue:1

    Topics: Adult; Alkaloids; Area Under Curve; Basal Metabolism; Benzodioxoles; Capsaicin; Carnitine; Catechin; Dietary Supplements; Double-Blind Method; Fatty Acids, Nonesterified; Female; Glucagon-Like Peptide 1; Glycerol; Humans; Male; Middle Aged; Obesity; Phytotherapy; Piperidines; Plant Extracts; Polyunsaturated Alkamides; Satiation; Satiety Response

2013

Other Studies

344 other study(ies) available for capsaicin and piperidines

ArticleYear
Sensory effects of capsaicin congeners I. Relationship between chemical structure and pain-producing potency of pungent agents.
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:12

    Topics: Animals; Butanones; Capsaicin; Condiments; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Homovanillic Acid; Pain; Piperidines; Rats; Sensory Receptor Cells; Structure-Activity Relationship

1975
Inhibitory effects of capsazepine and the NK2 antagonist SR 48968 on bronchoconstriction evoked by sensory nerve stimulation in guinea-pigs.
    Acta physiologica Scandinavica, 1992, Volume: 146, Issue:4

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Electric Stimulation; Female; Guinea Pigs; Male; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter

1992
Capsaicin-like activity of some natural pungent substances on peripheral endings of visceral primary afferents.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:1

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Curcumin; Eugenol; In Vitro Techniques; Isothiocyanates; Male; Muscle Contraction; Mustard Plant; Nerve Endings; Neurons, Afferent; Piperidines; Plant Extracts; Plant Oils; Polyunsaturated Alkamides; Rats; Rats, Inbred Strains; Ruthenium Red; Tetrodotoxin; Thiocyanates

1990
Effects of piperine on the motility of the isolated guinea-pig ileum: comparison with capsaicin.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Alkaloids; Animals; Anticonvulsants; Atropine; Benzodioxoles; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nerve Endings; Neurons, Afferent; Piperidines; Polyunsaturated Alkamides; Ruthenium Red; Substance P; Tachyphylaxis; Tetrodotoxin

1990
Effect of capsaicin, resiniferatoxin and piperine on ethanol-induced gastric ulcer of the rat.
    Acta physiologica Hungarica, 1990, Volume: 75 Suppl

    Topics: Alkaloids; Animals; Anti-Ulcer Agents; Benzodioxoles; Capsaicin; Diterpenes; Ethanol; Female; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Inbred Strains; Stomach Ulcer

1990
Involvement of calcitonin gene-related peptide in the positive chronotropic and inotropic effects of piperine and development of cross-tachyphylaxis between piperine and capsaicin in the isolated rat atria.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: Alkaloids; Animals; Benzodioxoles; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Neuropeptides; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Inbred Strains; Stimulation, Chemical; Tachyphylaxis

1989
Responses by humans to oral chemical irritants as a function of locus of stimulation.
    Perception & psychophysics, 1988, Volume: 43, Issue:1

    Topics: Adolescent; Adult; Alkaloids; Benzodioxoles; Capsaicin; Female; Humans; Male; Mouth; Piperidines; Polyunsaturated Alkamides; Sensation; Time Factors; Tongue

1988
Some pungent principles of spices cause the adrenal medulla to secrete catecholamine in anesthetized rats.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1988, Volume: 188, Issue:2

    Topics: Adrenal Medulla; Alkaloids; Animals; Benzodioxoles; Capsaicin; Catecholamines; Condiments; Epinephrine; Guaiacol; Intestinal Absorption; Kinetics; Male; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Inbred Strains

1988
Enhancement of responses to sequential presentation of oral chemical irritants.
    Physiology & behavior, 1987, Volume: 39, Issue:1

    Topics: Alkaloids; Benzodioxoles; Capsaicin; Drug Administration Schedule; Drug Synergism; Humans; Irritants; Mouth; Piperidines; Polyunsaturated Alkamides

1987
Putting out the fire: effects of tastants on oral chemical irritation.
    Perception & psychophysics, 1986, Volume: 39, Issue:5

    Topics: Adult; Alkaloids; Benzodioxoles; Capsaicin; Citrates; Citric Acid; Humans; Piperidines; Polyunsaturated Alkamides; Quinine; Sodium Chloride; Sucrose; Taste; Water

1986
Effect of intrathecal capsaicin analogues on the immunofluorescence of peptides and serotonin in the dorsal horn in rats.
    Neuroscience, 1983, Volume: 8, Issue:1

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Cholecystokinin; Enkephalin, Methionine; Fatty Acids, Unsaturated; Ganglia, Spinal; Kainic Acid; Male; Microscopy, Fluorescence; Nociceptors; Peptides; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Inbred Strains; Sensory Thresholds; Serotonin; Somatostatin; Substance P

1983
Tetrodotoxin-resistant non-cholinergic neurogenic contraction evoked by capsaicinoids and piperine on the guinea-pig trachea.
    Neuroscience letters, 1983, Nov-21, Volume: 42, Issue:1

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Denervation; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Muscle, Smooth; Neuromuscular Junction; Pain; Piperidines; Polyunsaturated Alkamides; Tetrodotoxin; Trachea

1983
The non-peptide NK1 receptor antagonist SR140333 produces long-lasting inhibition of neurogenic inflammation, but does not influence acute chemo- or thermonociception in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Blood Proteins; Capillary Permeability; Capsaicin; Dinoprostone; Female; Hot Temperature; Injections, Intravenous; Injections, Subcutaneous; Male; Motor Activity; Nerve Tissue; Neurokinin-1 Receptor Antagonists; Nociceptors; Pain; Pain Measurement; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley

1995
Pharmacological studies of allergic cough in the guinea pig.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Administration, Oral; Aerosols; Albuterol; Analysis of Variance; Animals; Antitussive Agents; Capsaicin; Chlorpheniramine; Cimetidine; Codeine; Cough; Drug Hypersensitivity; Guinea Pigs; Hexamethonium; Histamine Antagonists; Indomethacin; Injections, Subcutaneous; Ipratropium; Loratadine; Male; Ovalbumin; Piperidines; Receptors, Histamine H1; Receptors, Histamine H2

1995
Modulation of acetylcholine, capsaicin and substance P effects by histamine H3 receptors in isolated perfused rabbit lungs.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Acetylcholine; Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Endothelium; Female; Histamine Agonists; Histamine Antagonists; Imidazoles; In Vitro Techniques; Lung; Male; Nerve Fibers; Piperidines; Pulmonary Edema; Rabbits; Receptors, Histamine H3; Serotonin; Substance P; Thiourea

1995
Relative contributions of direct and indirect mechanisms mediating endothelin-induced contraction of guinea-pig trachea.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dicarboxylic Acids; Endothelins; Epithelium; Guinea Pigs; Histamine Release; In Vitro Techniques; Kinetics; Leukotriene Antagonists; Male; Muscle Contraction; Neurokinin A; Piperidines; Prostaglandins; Receptors, Tachykinin; SRS-A; Tetrodotoxin; Trachea

1993
Contractile effects of bradykinin on the isolated human small bronchus.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Acetylcholine; Aged; Atropine; Benzamides; Biphenyl Compounds; Bradykinin; Bronchi; Bronchoconstriction; Capsaicin; Humans; In Vitro Techniques; Indomethacin; Middle Aged; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Bradykinin; Ruthenium Red; Tetrodotoxin

1994
Capsaicin-induced airway obstruction in tracheally perfused guinea pig lungs.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Methacholine Chloride; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Perfusion; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1994
Capsaicin-induced bladder hyperactivity in normal conscious rats.
    The Journal of urology, 1994, Volume: 152, Issue:2 Pt 1

    Topics: Administration, Intravesical; Animals; Benzamides; Capsaicin; Consciousness; Dose-Response Relationship, Drug; Female; Hexamethonium; Hexamethonium Compounds; Indoles; Isoindoles; Morphine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Urinary Bladder

1994
An investigation into the mechanism of capsaicin-induced oedema in rabbit skin.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Alprostadil; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Capillary Permeability; Capsaicin; Catalase; Dexamethasone; Drug Interactions; Edema; Histamine; Indoles; Indomethacin; Injections, Intradermal; Injections, Intravenous; Isoindoles; Male; Piperidines; Rabbits; Regional Blood Flow; Ruthenium Red; Skin; Substance P; Vasodilator Agents

1995
Pharmacological analysis of the local and reflex responses to bradykinin on rat urinary bladder motility in vivo.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Bradykinin; Capsaicin; Dose-Response Relationship, Drug; Indoles; Indomethacin; Injections, Spinal; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Quinuclidines; Rats; Rats, Wistar; Reflex; Substance P; Urinary Bladder

1995
Substance P-induced histamine release in tracheally perfused guinea pig lungs.
    Journal of applied physiology (Bethesda, Md. : 1985), 1995, Volume: 78, Issue:4

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Guinea Pigs; Histamine; In Vitro Techniques; Lung; Male; Mast Cells; Perfusion; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1995
Involvement of tachykinins in plasma extravasation induced by bradykinin and low pH medium in the guinea-pig conjunctiva.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Capsaicin; Conjunctiva; Guinea Pigs; Hydrogen-Ion Concentration; Male; Neuritis; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Bradykinin; Substance P; Tachykinins

1995
Activity of SR 142801 at peripheral tachykinin receptors.
    European journal of pharmacology, 1995, May-04, Volume: 278, Issue:1

    Topics: Analysis of Variance; Animals; Binding, Competitive; Capsaicin; Cricetinae; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mesocricetus; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Portal Vein; Pulmonary Artery; Rabbits; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Trachea

1995
Histamine-induced edema in the rat paw--effect of capsaicin denervation and a CGRP receptor antagonist.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Animals; Blood Proteins; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capillary Permeability; Capsaicin; Denervation; Edema; Foot; Histamine; Male; Miotics; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley

1995
Urodynamic effects of intravesical resiniferatoxin and capsaicin in conscious rats with and without outflow obstruction.
    The Journal of urology, 1995, Volume: 154, Issue:2 Pt 1

    Topics: Administration, Intravesical; Animals; Benzamides; Capsaicin; Consciousness; Diterpenes; Female; Neurotoxins; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Urethral Obstruction; Urinary Bladder; Urodynamics

1995
Neurogenic vasodilation in the rat nasal mucosa involves neurokinin1 tachykinin receptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:1

    Topics: Animals; Capsaicin; Male; Neurons, Afferent; Olfactory Mucosa; Piperidines; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins; Vasodilation

1993
Effects of capsaicin, (+/-)-CP-96,345 and SR 48968 on the bradykinin-induced airways microvascular leakage in guinea-pigs.
    Pulmonary pharmacology, 1993, Volume: 6, Issue:1

    Topics: Animals; Autonomic Nervous System; Benzamides; Biphenyl Compounds; Bradykinin; Capillary Permeability; Capsaicin; Evans Blue; Guinea Pigs; Hypnotics and Sedatives; In Vitro Techniques; Nerve Endings; Neurokinin A; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1993
A new NK1 receptor antagonist (CP-99,994) prevents the increase in tracheal vascular permeability produced by hypertonic saline.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Edema; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Hypertonic Solutions; Neurokinin A; Neurons, Afferent; Piperidines; Platelet Activating Factor; Rats; Rats, Inbred F344; Receptors, Neurotransmitter; Receptors, Tachykinin; Sodium Chloride; Stimulation, Chemical; Substance P; Trachea; Tracheal Diseases

1993
NK1 receptors mediate neurogenic inflammatory increase in blood flow in rat airways.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 74, Issue:5

    Topics: Animals; Capsaicin; Inflammation; Male; Microspheres; Neurons, Afferent; Peptidyl-Dipeptidase A; Piperidines; Rats; Rats, Inbred F344; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Regional Blood Flow; Respiratory System; Respiratory Tract Diseases; Substance P; Tachykinins; Vasodilation

1993
Neuroregulation of a chemosensitive afferent system in the canine distal esophagus.
    The Journal of surgical research, 1993, Volume: 55, Issue:4

    Topics: Afferent Pathways; Animals; Atropine; Blood Pressure; Capsaicin; Chemoreceptor Cells; Dogs; Esophagus; Hexamethonium; Hexamethonium Compounds; Mucous Membrane; Nociceptors; Piperidines; Pressure; Pulse; Respiration; Substance P; Tetrodotoxin; Vagotomy

1993
Capsaicin increases airflow resistance in guinea pigs in vivo by activating both NK2 and NK1 tachykinin receptors.
    The American review of respiratory disease, 1993, Volume: 148, Issue:4 Pt 1

    Topics: Airway Resistance; Animals; Atropine; Benzamides; Biphenyl Compounds; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Male; Neurokinin A; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1993
Pharmacology of CP-99,994; a nonpeptide antagonist of the tachykinin neurokinin-1 receptor.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:1

    Topics: Animals; Binding, Competitive; Calcium Channels; Capillary Permeability; Capsaicin; Cells, Cultured; Cricetinae; Guinea Pigs; Humans; In Vitro Techniques; Locus Coeruleus; Male; Motor Activity; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Species Specificity; Substance P

1993
Evidence for a capsaicin-sensitive, tachykinin-mediated, component in the NANC contraction of the rat urinary bladder to nerve stimulation.
    British journal of pharmacology, 1994, Volume: 112, Issue:4

    Topics: Adenosine Triphosphate; Animals; Atropine; Capsaicin; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins; Urinary Bladder

1994
Resiniferatoxin and piperine: capsaicin-like stimulators of oxygen uptake in the perfused rat hindlimb.
    Life sciences, 1994, Volume: 55, Issue:5

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Diterpenes; Hindlimb; Male; Nitroglycerin; Oxygen Consumption; Perfusion; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar

1994
Sensory neuropeptide-mediated bronchoconstriction of the guinea pig lung by diamide; a comparison to hydrogen peroxide.
    European journal of pharmacology, 1994, Apr-04, Volume: 270, Issue:2-3

    Topics: Animals; Benzamides; Biphenyl Compounds; Bronchoconstriction; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Diamide; Guinea Pigs; Hydrogen Peroxide; In Vitro Techniques; Lung; Male; Neurokinin A; Neurons, Afferent; Neuropeptides; Piperidines; Thromboxanes

1994
Lactic acid-induced plasma protein extravasation in rat airways by stimulation of sensory nerves and NK1 receptor activation.
    Pharmacology & toxicology, 1993, Volume: 73, Issue:6

    Topics: Animals; Benzamides; Blood Proteins; Bronchi; Capsaicin; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Indoles; Isoindoles; Lactates; Lactic Acid; Male; Nasal Mucosa; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Respiratory Physiological Phenomena; Respiratory System; Trachea

1993
Taste responses of bullfrog to pungent stimuli.
    Brain research, 1994, Feb-21, Volume: 637, Issue:1-2

    Topics: Adaptation, Physiological; Alkaloids; Animals; Benzodioxoles; Capsaicin; Chemoreceptor Cells; Electrophysiology; Glossopharyngeal Nerve; In Vitro Techniques; Isothiocyanates; Neurons, Afferent; Piperidines; Polyunsaturated Alkamides; Rana catesbeiana; Regional Blood Flow; Sensory Thresholds; Stimulation, Chemical; Taste; Tongue

1994
CP-99,994, a nonpeptide antagonist of the tachykinin NK1 receptor.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Albuterol; Animals; Binding, Competitive; Calcium Channels; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; Kinetics; Lung; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Thiorphan; Verapamil

1993
Involvement of neurogenic inflammation in antigen-induced bronchoconstriction in guinea pigs.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: Aerosols; Animals; Atropine; Benzamides; Biphenyl Compounds; Bronchoconstriction; Capsaicin; Glycopeptides; Guinea Pigs; Histamine; Immunization; Inflammation; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Pulmonary Circulation; Receptors, Neurokinin-2; Vascular Resistance

1993
Differential blockade by tachykinin NK1 and NK2 receptor antagonists of bronchoconstriction induced by direct-acting agonists and the indirect-acting mimetics capsaicin, serotonin and 2-methyl-serotonin in the anesthetized guinea pig.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Amino Acid Sequence; Anesthesia; Animals; Benzamides; Biphenyl Compounds; Bronchial Spasm; Bronchoconstriction; Capsaicin; Guinea Pigs; Hypnotics and Sedatives; Injections, Intravenous; Male; Molecular Sequence Data; Neurokinin A; Piperidines; Receptors, Tachykinin; Serotonin

1993
Mechanism of action of capsaicin on submucosal arterioles in the guinea pig ileum.
    The American journal of physiology, 1993, Volume: 265, Issue:1 Pt 1

    Topics: Animals; Arterioles; Capsaicin; Guinea Pigs; Ileum; Intestinal Mucosa; Parasympatholytics; Perfusion; Piperidines; Tetrodotoxin; Vasodilation; Vasodilator Agents

1993
Postjunctional inhibitory effect of the NK2 receptor antagonist, SR 48968, on sensory NANC bronchoconstriction in the guinea-pig.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: Animals; Atropine; Autonomic Nervous System; Benzamides; Bronchoconstriction; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Lung; Male; Neurokinin A; Neurons, Afferent; Neuropeptides; Piperidines; Receptors, Neurotransmitter; Receptors, Tachykinin

1993
Inhibitory effects of capsazepine and SR 48968 on citric acid-induced bronchoconstriction in guinea-pigs.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Administration, Inhalation; Analysis of Variance; Animals; Benzamides; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Female; Guinea Pigs; Histamine; Hydrogen-Ion Concentration; Male; Neurokinin A; Neurons, Afferent; Piperidines

1993
Characterization of neurogenic inflammation in the airways of two highly inbred rat strains.
    American journal of respiratory and critical care medicine, 1995, Volume: 152, Issue:6 Pt 1

    Topics: Animals; Benzamides; Blood Pressure; Bronchi; Capillary Permeability; Capsaicin; Cimetidine; Coloring Agents; Dose-Response Relationship, Drug; Evans Blue; Histamine Antagonists; Indoles; Inflammation; Isoindoles; Methysergide; Neurokinin-1 Receptor Antagonists; Piperidines; Pyrilamine; Rats; Rats, Inbred F344; Rats, Inbred Strains; Receptors, Neurokinin-1; Serotonin; Serotonin Antagonists; Substance P; Trachea

1995
The involvement of calcitonin gene-related peptide (CGRP) and substance P in feline pial artery diameter responses evoked by capsaicin.
    Neuropeptides, 1995, Volume: 29, Issue:3

    Topics: Anesthetics; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cats; Cerebral Arteries; Female; Injections, Intravenous; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Substance P; Trigeminal Nerve; Vasomotor System

1995
Neuropeptide modulation of chemically induced skin irritation.
    Toxicology and applied pharmacology, 1995, Volume: 135, Issue:2

    Topics: Administration, Cutaneous; Animals; Benzamides; Biphenyl Compounds; Capsaicin; Dermatitis, Contact; Dinitrofluorobenzene; Disease Models, Animal; Dose-Response Relationship, Drug; Ear, External; Female; Irritants; Mice; Mice, Inbred BALB C; Neurokinin A; Neuropeptides; Piperidines; Skin; Substance P; Synaptic Transmission

1995
Electrocorticographic desynchronization after application of visceral and somatic noxious stimuli in urethane-anesthetized rats: effect of intrathecal administration of tachykinin (NK 1 or NK 2) receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:1

    Topics: Acetylcholine; Administration, Topical; Anesthesia; Animals; Benzamides; Capsaicin; Cortical Synchronization; Electric Stimulation; Indoles; Injections, Spinal; Isoindoles; Lidocaine; Male; Perineum; Physalaemin; Piperidines; Rats; Rats, Wistar; Receptors, Tachykinin; Sensitivity and Specificity; Urethane; Urinary Bladder

1996
Effect of T-kinin on microvascular permeability and its modulation by peptidases in rat airways.
    Journal of applied physiology (Bethesda, Md. : 1985), 1995, Volume: 79, Issue:4

    Topics: Amino Acid Sequence; Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Heart Rate; Male; Molecular Sequence Data; Neprilysin; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Hydrolases; Peptidyl-Dipeptidase A; Piperidines; Rats; Rats, Sprague-Dawley; Respiratory System; Tachykinins

1995
[Effect of FRG-8813, a new histamine H2-receptor antagonist, on gastric mucus production in rats].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1995, Volume: 106, Issue:6

    Topics: 16,16-Dimethylprostaglandin E2; Acetamides; Animals; Anti-Ulcer Agents; Capsaicin; Gastric Mucosa; Histamine H2 Antagonists; Mucus; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley

1995
RP67580, a neurokinin1 receptor antagonist, decreased restraint stress-induced defecation in rat.
    Neuroscience letters, 1995, Sep-29, Volume: 198, Issue:2

    Topics: Analgesics; Animals; Benzamides; Capsaicin; Defecation; Dose-Response Relationship, Drug; Indoles; Isoindoles; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Restraint, Physical; Stereoisomerism; Stress, Psychological; Substance P

1995
Possible role of protein kinase C in the sensitization of primate spinothalamic tract neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, May-01, Volume: 16, Issue:9

    Topics: Animals; Capsaicin; Female; Injections, Intradermal; Macaca fascicularis; Male; Neural Inhibition; Neurons; Periaqueductal Gray; Physical Stimulation; Piperidines; Protein Kinase C; Spinothalamic Tracts; Tetradecanoylphorbol Acetate

1996
The tachykinin NK2 receptor antagonist SR 48968 inhibits citric acid-induced airway hyperresponsiveness in guinea pigs.
    American journal of respiratory and critical care medicine, 1996, Volume: 153, Issue:5

    Topics: Acetylcholine; Aerosols; Animals; Benzamides; Bronchial Hyperreactivity; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Codeine; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Guinea Pigs; Injections, Intraperitoneal; Injections, Intravenous; Male; Narcotics; Piperidines; Protease Inhibitors; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Stereoisomerism; Tachykinins; Thiorphan

1996
The inhibitory modulation of guinea-pig intestinal peristalsis caused by capsaicin involves calcitonin gene-related peptide and nitric oxide.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 353, Issue:1

    Topics: Animals; Benzamides; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peristalsis; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Reflex

1995
Evidence for adrenergic and tachykinin activity in venom of the stonefish (Synanceja trachynis).
    Toxicon : official journal of the International Society on Toxinology, 1996, Volume: 34, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bronchoconstriction; Capsaicin; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Fish Venoms; Ganglionic Blockers; Guinea Pigs; Heart Atria; Ileum; Injections, Intravenous; Male; Mecamylamine; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Rabbits; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Neurokinin-2; Tachykinins; Tetrodotoxin; Vas Deferens

1996
Effect of the tachykinin receptor antagonists, SR 140333, FK 888, and SR 142801, on capsaicin-induced mouse ear oedema.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:6

    Topics: Animals; Binding Sites; Capsaicin; Dipeptides; Disease Models, Animal; Ear Diseases; Edema; Indoles; Injections, Intravenous; Lethal Dose 50; Male; Mice; Piperidines; Quinuclidines; Receptors, Tachykinin; Skin; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Evidence for the participation of glutamate in reflexes involving afferent, substance P-containing nerve fibres in the rat.
    British journal of pharmacology, 1996, Volume: 117, Issue:1

    Topics: Animals; Blood Pressure; Body Temperature; Capillary Permeability; Capsaicin; Colchicine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; Male; Mustard Plant; Nerve Fibers; Piperidines; Plant Extracts; Plant Oils; Quinuclidines; Rats; Rats, Wistar; Receptors, Tachykinin; Sciatic Nerve; Stereoisomerism

1996
Effects of hCGRP 8-37 and the NK1-receptor antagonist SR 140.333 on capsaicin-evoked vasodilation in the pig nasal mucosa in vivo.
    Acta physiologica Scandinavica, 1996, Volume: 156, Issue:2

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Female; Heart Rate; Male; Nasal Cavity; Nasal Mucosa; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinuclidines; Regional Blood Flow; Substance P; Swine; Vasodilation

1996
Similarities and differences in the currents activated by capsaicin, piperine, and zingerone in rat trigeminal ganglion cells.
    Journal of neurophysiology, 1996, Volume: 76, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Biotransformation; Calcium; Capsaicin; Cells, Cultured; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Guaiacol; Ion Channels; Neurons; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptors, Drug; Structure-Activity Relationship; Tachyphylaxis; Trigeminal Ganglion

1996
Role of tachykinins in enhancement of bradykinin-induced bronchoconstriction by captopril.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Benzamides; Bradykinin; Bronchoconstriction; Capsaicin; Captopril; Dose-Response Relationship, Drug; Drug Synergism; Guinea Pigs; Male; Neurokinin A; Peptides, Cyclic; Piperidines; Substance P

1996
Effect of MDL 105,212, a nonpeptide NK-1/NK-2 receptor antagonist in an allergic guinea pig model.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Release; Hypersensitivity; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Pyrrolidines; Receptors, Neurokinin-2; Respiration

1996
The role of substance P in myocardial dysfunction during ischemia and reperfusion.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:4

    Topics: Analgesics; Animals; Capsaicin; Guinea Pigs; Heart Rate; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardial Stunning; Piperidines; Substance P; Ventricular Dysfunction, Left

1996
Tachykinin-independent effects of capsaicin on smooth muscle in human isolated bronchi.
    American journal of respiratory and critical care medicine, 1997, Volume: 155, Issue:2

    Topics: Adult; Benzamides; Bronchi; Capsaicin; Cells, Cultured; Diterpenes; Drug Interactions; Female; Humans; Male; Muscle Contraction; Muscle, Smooth; Patch-Clamp Techniques; Piperidines; Tachykinins

1997
Replication-deficient adenoviral vector for gene transfer potentiates airway neurogenic inflammation.
    American journal of respiratory cell and molecular biology, 1997, Volume: 16, Issue:3

    Topics: Adenoviruses, Human; Animals; Capillary Permeability; Capsaicin; Dexamethasone; Ficusin; Gene Transfer Techniques; Genetic Vectors; Glucocorticoids; Hot Temperature; Inflammation; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Photosensitizing Agents; Piperidines; Protein Denaturation; Rats; Rats, Inbred F344; Receptors, Neurokinin-1; Respiratory System; Substance P; Ultraviolet Rays

1997
Functional relationships between sensory nerve fibers and mast cells of dura mater in normal and inflammatory conditions.
    Neuroscience, 1997, Volume: 77, Issue:3

    Topics: Animals; Animals, Newborn; Capsaicin; Cerebral Cortex; Chymases; Denervation; Dura Mater; Enzyme-Linked Immunosorbent Assay; Histamine; Histamine Antagonists; Inflammation; Male; Mast Cells; Methylhistamines; Nerve Fibers; Neurons, Afferent; Nippostrongylus; Piperidines; Rats; Rats, Wistar; Reference Values; Sensitivity and Specificity; Serine Endopeptidases; Strongylida Infections

1997
Perceived irritation during ingestion of capsaicin or piperine: comparison of trigeminal and non-trigeminal areas.
    Chemical senses, 1997, Volume: 22, Issue:3

    Topics: Adult; Alkaloids; Benzodioxoles; Capsaicin; Chemoreceptor Cells; Female; Glossopharyngeal Nerve; Humans; Irritants; Male; Mouth; Perception; Pharynx; Piperidines; Polyunsaturated Alkamides; Tongue; Trigeminal Nerve

1997
Inhibitors of G-proteins and protein kinases reduce the sensitization to mechanical stimulation and the desensitization to heat of spinothalamic tract neurons induced by intradermal injection of capsaicin in the primate.
    Experimental brain research, 1997, Volume: 115, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Diphosphate; Animals; Capsaicin; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Haplorhini; Hot Temperature; Injections, Intradermal; Isoquinolines; Microdialysis; Nerve Fibers; Neural Pathways; Physical Stimulation; Piperidines; Protein Kinase Inhibitors; Spinal Cord; Sulfonamides; Thalamus; Thionucleotides

1997
Enhancement of rat trigeminal ganglion neuron responses to piperine in a low-pH environment and block by capsazepine.
    Brain research, 1997, Jun-27, Volume: 761, Issue:1

    Topics: Alkaloids; Animals; Anticonvulsants; Benzodioxoles; Binding, Competitive; Capsaicin; Female; Hydrogen-Ion Concentration; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Protons; Rats; Rats, Sprague-Dawley; Trigeminal Ganglion

1997
MEN 11,420, a peptide tachykinin NK2 receptor antagonist, reduces motor responses induced by the intravesical administration of capsaicin in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Animals; Capsaicin; Hexamethonium; Male; Muscle Contraction; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Tachykinin; Urinary Bladder

1997
Cellular pathways mediating tachykinin-evoked secretomotor responses in guinea pig ileum.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Capsaicin; Electric Stimulation; Evoked Potentials; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Mucosa; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins

1997
Antinociceptive activity of CP-101,606, an NMDA receptor NR2B subunit antagonist.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Analgesics, Non-Narcotic; Animals; Brain; Capsaicin; Carrageenan; Excitatory Amino Acid Antagonists; Hyperalgesia; Injections, Subcutaneous; Male; Motor Activity; Pain Measurement; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Tetradecanoylphorbol Acetate

1997
Effects of tachykinins and capsaicin on the mechanical and electrical activity of the guinea-pig isolated trachea.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Animals; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Potassium Channel Blockers; Quinuclidines; Receptors, Neurokinin-2; Substance P; Tachykinins; Tetraethylammonium; Trachea

1997
Capsaicin-induced sensitization of primate spinothalamic tract cells is prevented by a protein kinase C inhibitor.
    Brain research, 1997, Oct-24, Volume: 772, Issue:1-2

    Topics: Animals; Biomechanical Phenomena; Capsaicin; Enzyme Activation; Enzyme Inhibitors; Macaca fascicularis; Nerve Fibers; Piperidines; Protein Kinase C; Spinothalamic Tracts; Temperature

1997
Tachykinins may mediate capsaicin-induced, but not vagally induced motility in porcine antrum.
    Peptides, 1997, Volume: 18, Issue:10

    Topics: Animals; Benzamides; Biphenyl Compounds; Capsaicin; Electric Stimulation; Gastrointestinal Motility; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Pyloric Antrum; Receptors, Neurokinin-2; Substance P; Swine; Tachykinins; Vagus Nerve

1997
Insulin secretion by gastrin-releasing peptide in mice: ganglionic versus direct islet effect.
    The American journal of physiology, 1998, Volume: 274, Issue:1

    Topics: Animals; Blood Glucose; Capsaicin; Cells, Cultured; Female; Ganglia, Sympathetic; Gastrin-Releasing Peptide; Glucagon; Hexamethonium; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred Strains; Muscarinic Antagonists; Pancreas; Piperidines; Receptor, Muscarinic M3; Receptors, Muscarinic

1998
Selective blockade of substance P or neurokinin A receptors reduces the expression of c-fos in trigeminal subnucleus caudalis after corneal stimulation in the rat.
    Neuroscience, 1998, Volume: 83, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Autonomic Nervous System; Capsaicin; Cornea; Hormones; Immunohistochemistry; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Trigeminal Nucleus, Spinal

1998
Neuropeptide regulation of proinflammatory cytokine responses.
    Journal of leukocyte biology, 1998, Volume: 63, Issue:5

    Topics: Animals; Capsaicin; Cytokines; Endotoxins; Female; Gene Expression Regulation; Inflammation; Lipopolysaccharides; Liver; Mice; Mice, Inbred BALB C; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Spleen; Tachykinins; Time Factors; Transcription, Genetic; Tumor Necrosis Factor-alpha

1998
Activation of non-adrenergic non-cholinergic inhibitory pathways by endogenous and exogenous tachykinins in the ferret lower oesophageal sphincter.
    Neurogastroenterology and motility, 1998, Volume: 10, Issue:2

    Topics: Animals; Capsaicin; Electric Stimulation; Esophagogastric Junction; Female; Ferrets; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nitroarginine; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Substance P; Tachykinins; Tetrodotoxin

1998
Effects of endothelin-1 on capsaicin-induced nociception in mice.
    European journal of pharmacology, 1998, Jun-12, Volume: 351, Issue:1

    Topics: Analgesia; Animals; Bosentan; Capsaicin; Dansyl Compounds; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Hindlimb; Hyperalgesia; Male; Mice; Oligopeptides; Peptide Fragments; Peptides; Peptides, Cyclic; Piperidines; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Serotonin; Sulfonamides; Viper Venoms

1998
Activation of neurons in rat trigeminal subnucleus caudalis by different irritant chemicals applied to oral or ocular mucosa.
    Journal of neurophysiology, 1998, Volume: 80, Issue:2

    Topics: Alkaloids; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzodioxoles; Capsaicin; Conjunctiva; Cornea; Dose-Response Relationship, Drug; Electrophysiology; Ethanol; Ganglionic Stimulants; Histamine; Irritants; Male; Mouth Mucosa; Mustard Plant; Neurons; Nicotine; Piperidines; Plant Extracts; Plant Oils; Polyunsaturated Alkamides; Rats; Rats, Wistar; Reaction Time; Serotonin; Sodium Chloride; Solvents; Stimulation, Chemical; Tachyphylaxis; Tongue; Trigeminal Nuclei

1998
Characterization of the antibronchoconstrictor activity of MEN 11420, a tachykinin NK2 receptor antagonist, in guinea-pigs.
    European journal of pharmacology, 1998, Jul-10, Volume: 352, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Atropine; Benzamides; Bronchi; Bronchoconstriction; Bronchodilator Agents; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Piperidines; Receptors, Neurokinin-2

1998
Effects of airway inflammation on cough response in the guinea pig.
    Journal of applied physiology (Bethesda, Md. : 1985), 1998, Volume: 85, Issue:5

    Topics: Animals; Antitussive Agents; Benzamides; Bronchoalveolar Lavage Fluid; Capsaicin; Codeine; Cough; Dipeptides; Female; Guinea Pigs; Indoles; Inflammation; Peptides, Cyclic; Piperidines; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Respiratory Hypersensitivity; Respiratory Tract Diseases

1998
Acute and chronic effects of capsaicin in perfused rat muscle: the role of tachykinins and calcitonin gene-related peptide.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:2

    Topics: Animals; Benzamides; Calcitonin Gene-Related Peptide; Capsaicin; Male; Muscle, Skeletal; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Substance P

1998
Synthesis and structure-activity relationships of CP-122,721, a second-generation NK-1 receptor antagonist.
    Bioorganic & medicinal chemistry letters, 1998, Feb-03, Volume: 8, Issue:3

    Topics: Animals; Capsaicin; Cell Line; Guinea Pigs; Humans; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Structure-Activity Relationship

1998
Subthreshold concentration of endothelin-1-enhanced, capsaicin-induced bronchoconstriction in anaesthetized guinea-pigs.
    The European respiratory journal, 1998, Volume: 12, Issue:6

    Topics: Aerosols; Airway Resistance; Anesthesia; Animals; Asthma; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelin-1; Guinea Pigs; Male; Neurokinin A; Oligopeptides; Peptides, Cyclic; Piperidines; Substance P

1998
Effects of a tachykinin NK3 receptor antagonist, SR 142801, studied in isolated neonatal rat spinal cord.
    Neuropeptides, 1998, Volume: 32, Issue:6

    Topics: Animals; Animals, Newborn; Capsaicin; Electrophysiology; Female; In Vitro Techniques; Male; Membrane Potentials; Neurokinin B; Neurons, Afferent; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Spinal Cord; Spinal Nerve Roots; Substance P

1998
Neurogenic plasma leakage in mouse airways.
    British journal of pharmacology, 1999, Volume: 126, Issue:2

    Topics: Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Benzamides; Blood Vessels; Bradykinin; Bradykinin Receptor Antagonists; Capillary Permeability; Capsaicin; Captopril; Dose-Response Relationship, Drug; Evans Blue; Glycopeptides; Lung; Male; Mice; Mice, Inbred C57BL; Neurokinin-1 Receptor Antagonists; Piperidines; Protease Inhibitors; Quinuclidines; Receptors, Neurokinin-2; Skin; Specific Pathogen-Free Organisms; Substance P; Trachea; Urinary Bladder

1999
Antinociceptive properties of the new alkaloid, cis-8, 10-di-N-propyllobelidiol hydrochloride dihydrate isolated from Siphocampylus verticillatus: evidence for the mechanism of action.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: Abdominal Muscles; Acetic Acid; Alkaloids; Analgesics; Analgesics, Opioid; Animals; Capsaicin; Female; Formaldehyde; Gastrointestinal Transit; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Morphine; Muscle Contraction; Muscle, Smooth; Pain Measurement; Piperidines; Plants, Medicinal; Postural Balance; Reaction Time; Vas Deferens

1999
Decreased vascular permeability response to substance P in airways of genetically hypertensive rats.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Animals; Blood Pressure; Capillary Permeability; Capsaicin; Hypertension; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Substance P

1999
Local administration of delta9-tetrahydrocannabinol attenuates capsaicin-induced thermal nociception in rhesus monkeys: a peripheral cannabinoid action.
    Psychopharmacology, 1999, Volume: 143, Issue:3

    Topics: Analgesics, Non-Narcotic; Animals; Cannabinoids; Capsaicin; Dronabinol; Female; Macaca mulatta; Male; Pain Measurement; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1999
Neurokinin type-1 receptor antagonist inhibits enhancement of T cell functions by substance P in normal and neuromanipulated capsaicin-treated rats.
    Journal of neuroimmunology, 1999, Jan-01, Volume: 93, Issue:1-2

    Topics: Animals; Capsaicin; CD4-Positive T-Lymphocytes; CD5 Antigens; Cell Division; Concanavalin A; Female; Interleukin-2; Lymphocyte Activation; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Specific Pathogen-Free Organisms; Spleen; Substance P

1999
Respiratory action of capsaicin microinjected into the nucleus of the solitary tract: involvement of vanilloid and tachykinin receptors.
    British journal of pharmacology, 1999, Volume: 127, Issue:2

    Topics: Anesthesia; Animals; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Indoles; Isoindoles; Male; Microinjections; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mechanics; Solitary Nucleus; Tidal Volume

1999
Gastroprotective mechanism of lafutidine, a novel anti-ulcer drug with histamine H2-receptor antagonistic activity.
    Arzneimittel-Forschung, 1999, Volume: 49, Issue:6

    Topics: 16,16-Dimethylprostaglandin E2; Acetamides; Ammonia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Capsaicin; Central Nervous System Depressants; Ethanol; Gastric Mucosa; Histamine H2 Antagonists; Indomethacin; Male; Membrane Potentials; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Stomach Ulcer

1999
Antiulcer effect of lafutidine on indomethacin-induced gastric antral ulcers in refed rats.
    Japanese journal of pharmacology, 1999, Volume: 80, Issue:3

    Topics: 16,16-Dimethylprostaglandin E2; Acetamides; Administration, Oral; Animals; Anti-Ulcer Agents; Capsaicin; Cimetidine; Denervation; Dose-Response Relationship, Drug; Enzyme Inhibitors; Famotidine; Food; Indomethacin; Male; Nitroarginine; Piperidines; Pyloric Antrum; Pyridines; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Wound Healing

1999
Effect of lafutidine, a novel histamine H2-receptor antagonist, on monochloramine-induced gastric lesions in rats: role of capsaicin-sensitive sensory neurons.
    Journal of gastroenterology and hepatology, 1999, Volume: 14, Issue:9

    Topics: Acetamides; Animals; Anti-Ulcer Agents; Capsaicin; Chloramines; Cimetidine; Gastric Mucosa; Histamine H2 Antagonists; Ischemia; Membrane Potentials; Neurons, Afferent; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Stomach; Stomach Ulcer

1999
Involvement of endogenous tachykinins and CGRP in the motor responses produced by capsaicin in the guinea-pig common bile duct.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:3

    Topics: Animals; Atropine; Calcitonin Gene-Related Peptide; Capsaicin; Common Bile Duct; Electric Stimulation; Guinea Pigs; Humans; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Peptides, Cyclic; Physalaemin; Piperidines; Potassium Chloride; Pyridoxal Phosphate; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Tachykinins; Tetrodotoxin

1999
Airway hyperresponsiveness induced by chronic exposure to cigarette smoke in guinea pigs: role of tachykinins.
    Journal of applied physiology (Bethesda, Md. : 1985), 1999, Volume: 87, Issue:5

    Topics: Acetylcholine; Air Pressure; Animals; Benzamides; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Capsaicin; Cell Count; Dose-Response Relationship, Drug; Guinea Pigs; Male; Neurokinin A; Neuropeptides; Nicotiana; Piperidines; Plants, Toxic; Receptors, Neurokinin-2; Smoke; Tachykinins; Vagotomy

1999
Neuropeptides and capsaicin stimulate the release of inflammatory cytokines in a human bronchial epithelial cell line.
    Neuropeptides, 1999, Volume: 33, Issue:6

    Topics: Bronchi; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cell Line, Transformed; Cytokines; Epithelial Cells; Gene Expression; Humans; Interleukin-6; Interleukin-8; Peptide Fragments; Piperidines; Protease Inhibitors; RNA, Messenger; Substance P; Thiorphan; Tumor Necrosis Factor-alpha

1999
Protective effect of lafutidine against indomethacin-induced intestinal ulceration in rats: relation to capsaicin-sensitive sensory neurons.
    Digestion, 2000, Volume: 61, Issue:1

    Topics: 16,16-Dimethylprostaglandin E2; Acetamides; Ampicillin; Animals; Capsaicin; Dose-Response Relationship, Drug; Duodenal Ulcer; Histamine H2 Antagonists; Indomethacin; Intestinal Mucosa; Male; Neurons, Afferent; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Peroxidase; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley

2000
Endothelin-1-induced ET(A) receptor-mediated nociception, hyperalgesia and oedema in the mouse hind-paw: modulation by simultaneous ET(B) receptor activation.
    British journal of pharmacology, 2000, Volume: 129, Issue:5

    Topics: Animals; Atrasentan; Capsaicin; Edema; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Hyperalgesia; Male; Mice; Nociceptors; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Piperidines; Pyrrolidines; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Viper Venoms

2000
Evidence for the involvement of ATP, but not of VIP/PACAP or nitric oxide, in the excitatory effect of capsaicin in the small intestine.
    European journal of pharmacology, 2000, Mar-31, Volume: 392, Issue:3

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Capsaicin; Enzyme Inhibitors; Guinea Pigs; Ileum; In Vitro Techniques; Intestine, Small; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Neuropeptides; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Physalaemin; Piperidines; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyridoxal Phosphate; Receptors, Neurokinin-3; Sincalide; Substance P; Vasoactive Intestinal Peptide

2000
The role of sensorial neuropeptides in the edematogenic responses mediated by B(1) agonist des-Arg(9)-BK in rats pre-treated with LPS.
    Regulatory peptides, 2000, May-10, Volume: 89, Issue:1-3

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Edema; Histamine H1 Antagonists; Lipopolysaccharides; Male; Methysergide; Mianserin; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; p-Methoxy-N-methylphenethylamine; Peptide Fragments; Piperidines; Pyrazoles; Pyridines; Pyrilamine; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Serotonin Antagonists

2000
Effects of TAK-637, a tachykinin receptor antagonist, on the micturition reflex in guinea pigs.
    European journal of pharmacology, 2000, May-03, Volume: 395, Issue:3

    Topics: Animals; Benzhydryl Compounds; Benzilates; Capsaicin; Cholinergic Antagonists; Cresols; Dilatation; Dose-Response Relationship, Drug; Guinea Pigs; Male; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxants, Central; Naphthyridines; Parasympatholytics; Phenylpropanolamine; Piperidines; Propiophenones; Receptors, Tachykinin; Reflex; Tolterodine Tartrate; Urinary Bladder; Urination

2000
Tachykinin NK(2) receptors facilitate acetylcholine release from guinea-pig isolated trachea.
    European journal of pharmacology, 2000, May-12, Volume: 396, Issue:1

    Topics: Acetylcholine; Animals; Benzamides; Capsaicin; Choline; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Trachea

2000
The anandamide transport inhibitor AM404 activates vanilloid receptors.
    European journal of pharmacology, 2000, May-12, Volume: 396, Issue:1

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Cannabinoids; Capsaicin; Endocannabinoids; Female; Hepatic Artery; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Oocytes; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Drug; Rimonabant; Vasodilation; Xenopus

2000
Role of neurokinin receptors in the behavioral effect of intravesical antigen infusion in guinea pig bladder.
    The Journal of urology, 2000, Volume: 164, Issue:1

    Topics: Administration, Intravesical; Animals; Antigens; Behavior, Animal; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Neurokinin-1 Receptor Antagonists; Ovalbumin; Pelvic Pain; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Urinary Bladder

2000
Involvement of kinins, mast cells and sensory neurons in the plasma exudation and paw oedema induced by staphylococcal enterotoxin B in the mouse.
    European journal of pharmacology, 2000, Jul-07, Volume: 399, Issue:2-3

    Topics: Animals; Benzamides; Bradykinin; Capillary Permeability; Capsaicin; Diabetes Mellitus, Experimental; Edema; Enterotoxins; Hindlimb; Kinins; Male; Mast Cells; Mice; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Pyrilamine; Quinuclidines; Receptors, Neurokinin-2

2000
Substance P radioimmunoassay for quantitative characterization of sensory neurotransmitter release.
    Neurobiology (Budapest, Hungary), 1999, Volume: 7, Issue:4

    Topics: Alkaloids; Animals; Benzodioxoles; Calibration; Capsaicin; Diterpenes; Electric Stimulation; Enzyme Inhibitors; Female; Neurons, Afferent; Piperidines; Polyunsaturated Alkamides; Radioimmunoassay; Rats; Rats, Wistar; Stimulation, Chemical; Substance P; Trachea

1999
The emetic and anti-emetic effects of the capsaicin analogue resiniferatoxin in Suncus murinus, the house musk shrew.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Abdomen; Animals; Animals, Newborn; Antiemetics; Behavior, Animal; Capsaicin; Cisplatin; Copper Sulfate; Diterpenes; Dose-Response Relationship, Drug; Female; Indoles; Injections, Intraventricular; Male; Medulla Oblongata; Morphine; Motion Sickness; Nicotine; Piperidines; Proto-Oncogene Proteins c-fos; Serotonin Receptor Agonists; Shrews; Tropisetron; Vagotomy; Vomiting

2000
Nociceptin inhibits capsaicin-induced bronchoconstriction in isolated guinea pig lung.
    European journal of pharmacology, 2000, Aug-18, Volume: 402, Issue:1-2

    Topics: Animals; Benzimidazoles; Bronchoconstriction; Capsaicin; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; In Vitro Techniques; Lung; Naloxone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Piperidines; Receptors, Opioid; Sulfur Radioisotopes

2000
Complete inhibition of purinoceptor agonist-induced nociception by spinorphin, but not by morphine.
    Peptides, 2000, Volume: 21, Issue:8

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; Analgesics, Opioid; Animals; Animals, Newborn; Bradykinin; Capsaicin; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Mice; Morphine; Neurons, Afferent; Neuroprotective Agents; Oligopeptides; Pain; Pertussis Toxin; Piperidines; Protease Inhibitors; Purinergic Agonists; Thionucleosides; Time Factors; Virulence Factors, Bordetella

2000
Neural pathways regulating Brunner's gland secretion in guinea pig duodenum in vitro.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 279, Issue:5

    Topics: Animals; Brunner Glands; Capsaicin; Carbachol; Choline O-Acetyltransferase; Cholinergic Agonists; Cholinergic Fibers; Dimethylphenylpiperazinium Iodide; Duodenum; Electric Stimulation; Female; Ganglia, Sympathetic; Guanethidine; Guinea Pigs; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Neural Pathways; Neurotransmitter Agents; Nicotinic Agonists; Nicotinic Antagonists; Piperidines; Submucous Plexus; Substance P; Sympatholytics; Tetrodotoxin; Vagotomy; Vagus Nerve

2000
Trypsin-induced, neurokinin-mediated contraction of guinea pig bronchus.
    American journal of respiratory and critical care medicine, 2000, Volume: 162, Issue:5

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Chymases; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Receptor, PAR-1; Receptor, PAR-2; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Thrombin; Serine Endopeptidases; Tachykinins; Thrombin; Trachea; Trypsin; Tryptases

2000
Bidirectional control of airway responsiveness by endogenous cannabinoids.
    Nature, 2000, Nov-02, Volume: 408, Issue:6808

    Topics: Animals; Arachidonic Acids; Axons; Bronchi; Bronchial Spasm; Bronchoconstriction; Cannabinoids; Capsaicin; Cough; Endocannabinoids; Guinea Pigs; Lung; Muscle Contraction; Muscle, Smooth; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2000
Neutral endopeptidase terminates substance P-induced inflammation in allergic contact dermatitis.
    Journal of immunology (Baltimore, Md. : 1950), 2001, Jan-15, Volume: 166, Issue:2

    Topics: Administration, Cutaneous; Animals; Anti-Inflammatory Agents, Non-Steroidal; Capillary Permeability; Capsaicin; Croton Oil; Dermatitis, Allergic Contact; Dermatitis, Irritant; Enzyme Inhibitors; Female; Glycopeptides; Injections, Intravenous; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neprilysin; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Skin; Substance P

2001
Structure-activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens.
    British journal of pharmacology, 2001, Volume: 132, Issue:3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Biological Transport; Calcium; Calcium Channel Blockers; Cannabinoids; Capsaicin; CHO Cells; Cricetinae; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Morpholines; Muscle Contraction; Naphthalenes; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Structure-Activity Relationship; Transfection; TRPV Cation Channels; Vas Deferens

2001
Regional differences in anandamide- and methanandamide-induced membrane potential changes in rat mesenteric arteries.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:2

    Topics: Animals; Arachidonic Acids; Benzoxazines; Biological Factors; Calcium Channel Blockers; Cannabinoids; Capsaicin; Electrophysiology; Endocannabinoids; Endothelium, Vascular; Membrane Potentials; Mesenteric Arteries; Morpholines; Muscle, Smooth, Vascular; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Drug; Rimonabant; Vasodilator Agents

2001
Cannabinoid inhibition of the capsaicin-induced calcium response in rat dorsal root ganglion neurones.
    British journal of pharmacology, 2001, Volume: 132, Issue:5

    Topics: Animals; Calcium; Cannabinoids; Capsaicin; Dronabinol; Ganglia, Spinal; Neurons; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2001
Potent NK1 antagonism by SR-140333 reduces rat colonic secretory response to immunocyte activation.
    American journal of physiology. Cell physiology, 2001, Volume: 280, Issue:4

    Topics: Animals; Benzamides; Capsaicin; Colon; Colonic Diseases, Functional; Electric Stimulation; Male; Mast Cells; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stress, Physiological; Substance P

2001
Effect of vanilloid drugs on gastrointestinal transit in mice.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Arachidonic Acids; Benzodioxoles; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Gastrointestinal Transit; Hexamethonium; Male; Mice; Mice, Inbred ICR; Naloxone; NG-Nitroarginine Methyl Ester; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Yohimbine

2001
Cannabinoid inhibition of capsaicin-sensitive sensory neurotransmission in the rat mesenteric arterial bed.
    European journal of pharmacology, 2001, Apr-20, Volume: 418, Issue:1-2

    Topics: Adenosine Diphosphate; Animals; Benzofurans; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoids; Capsaicin; Dose-Response Relationship, Drug; Dronabinol; Electric Stimulation; Electrophysiology; Male; Mesenteric Arteries; Neurons, Afferent; Nitroprusside; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Synaptic Transmission; Time Factors; Vasodilation; Vasodilator Agents

2001
Mouse macrophages release a neutrophil chemotactic mediator following stimulation by staphylococcal enterotoxin type A.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2001, Volume: 50, Issue:4

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Benzamides; Calcium; Capsaicin; Chemotactic Factors; Chemotaxis, Leukocyte; Cyclooxygenase Inhibitors; Dexamethasone; Drug Stability; Enterotoxins; Glucocorticoids; Glucose; Indomethacin; Macrophages, Peritoneal; Magnesium; Male; Mice; Molecular Weight; Neutrophils; Piperidines; Receptors, Neurokinin-2; Thioglycolates

2001
Tachykinins mediate slow excitatory postsynaptic transmission in guinea pig sphincter of Oddi ganglia.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 281, Issue:2

    Topics: Animals; Calcium; Capsaicin; Culture Techniques; Excitatory Postsynaptic Potentials; Female; Ganglia; Guinea Pigs; Male; Membrane Potentials; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Receptors, Tachykinin; Sphincter of Oddi; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin

2001
Identification of two distinct vasodilator pathways activated by ATP in the mesenteric bed of the rat.
    British journal of pharmacology, 2001, Volume: 133, Issue:6

    Topics: Adenine; Adenosine; Adenosine Triphosphate; Animals; Arachidonic Acids; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Histamine; In Vitro Techniques; Male; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Oxadiazoles; Piperidines; Polyunsaturated Alkamides; Potassium Chloride; Pyrazoles; Pyrilamine; Quinoxalines; Rats; Rats, Wistar; Rimonabant; Signal Transduction; Stereoisomerism; Theophylline; Vasodilation

2001
Human colonic anti-secretory activity of the potent NK(1) antagonist, SR140333: assessment of potential anti-diarrhoeal activity in food allergy and inflammatory bowel disease.
    British journal of pharmacology, 2001, Volume: 133, Issue:8

    Topics: Animals; Antidiarrheals; Capsaicin; Colitis, Ulcerative; Colon; Crohn Disease; Epithelial Cells; Food Hypersensitivity; Guinea Pigs; Humans; Immunoglobulin E; Inflammatory Bowel Diseases; Male; Mast Cells; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Receptors, Neurokinin-1; Species Specificity; Substance P; Tachykinins

2001
Inhibitory activity of nociceptin/orphanin FQ on capsaicin-induced bronchoconstriction in the guinea-pig.
    Life sciences, 2001, Jul-27, Volume: 69, Issue:10

    Topics: Animals; Benzimidazoles; Bronchoconstriction; Bronchoconstrictor Agents; Capsaicin; Drug Therapy, Combination; Guinea Pigs; Injections, Intravenous; Male; Naloxone; Neuropeptides; Nociceptin; Nociceptin Receptor; Opioid Peptides; Piperidines; Plethysmography, Whole Body; Protease Inhibitors; Receptors, Opioid; Vasodilator Agents

2001
Roles of mast cells and sensory nerves in cutaneous vascular hyperpermeability and scratching behavior induced by poly-L-arginine in rats.
    European journal of pharmacology, 2001, Aug-17, Volume: 425, Issue:3

    Topics: Animals; Behavior, Animal; Capillary Permeability; Capsaicin; Chlorpheniramine; Dose-Response Relationship, Drug; Glycopeptides; Histamine; Histamine H1 Antagonists; Indoles; Injections, Intradermal; Male; Mast Cells; Methysergide; Neurons, Afferent; Peptides; Piperidines; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Skin; Substance P

2001
Cannabinoids attenuate capsaicin-evoked hyperalgesia through spinal and peripheral mechanisms.
    Pain, 2001, Volume: 93, Issue:3

    Topics: Analgesics; Animals; Benzoxazines; Cannabinoids; Capsaicin; Hyperalgesia; Male; Morpholines; Naphthalenes; Neurons, Afferent; Pain Measurement; Peripheral Nerves; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Spinal Cord

2001
Influence of capsaicin cream in rats with peripheral neuropathy.
    Pharmacological research, 2001, Volume: 44, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics; Animals; Benzamides; Capsaicin; Carrageenan; Disease Models, Animal; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Hyperalgesia; Indoles; Isoindoles; Male; Neuroprotective Agents; Pain; Peripheral Nervous System Diseases; Piperidines; Postoperative Period; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Substance Withdrawal Syndrome; Time Factors

2001
A possible role of lipoxygenase in the activation of vanilloid receptors by anandamide in the guinea-pig bronchus.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonic Acids; Bronchi; Calcium Channel Blockers; Capsaicin; Cyclohexanols; Dose-Response Relationship, Drug; Endocannabinoids; Fatty Acids, Unsaturated; Guinea Pigs; Hydrazines; In Vitro Techniques; Indomethacin; Lipoxygenase; Muscle Contraction; Oxazepines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Thiorphan

2001
The plasma protein extravasation induced by adenosine and its analogues in the rat dorsal skin: evidence for the involvement of capsaicin sensitive primary afferent neurones and mast cells.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Proteins; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Female; Injections, Intradermal; Isotonic Solutions; Male; Mast Cells; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; p-Methoxy-N-methylphenethylamine; Peptide Fragments; Piperidines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Skin; Substance P; Theobromine

2001
Differential effects of anandamide on acetylcholine release in the guinea-pig ileum mediated via vanilloid and non-CB1 cannabinoid receptors.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: Acetylcholine; Animals; Arachidonic Acids; Camphanes; Capsaicin; Cyclohexanols; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methacholine Chloride; Muscle Contraction; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2001
Comparative effect of Phoneutria nigriventer spider venom and capsaicin on the rat paw oedema.
    Life sciences, 2001, Aug-17, Volume: 69, Issue:13

    Topics: Animals; Animals, Newborn; Calcitonin Gene-Related Peptide; Capillary Permeability; Capsaicin; Edema; Female; Foot; Histamine H1 Antagonists; Indicators and Reagents; Male; Mast Cells; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; p-Methoxy-N-methylphenethylamine; Piperidines; Quinuclidines; Rats; Rats, Wistar; Spider Venoms

2001
Nitric oxide is generated in smooth muscle layer by neurokinin A and counteracts constriction in guinea pig airway.
    Nitric oxide : biology and chemistry, 2001, Volume: 5, Issue:5

    Topics: Airway Resistance; Animals; Benzamides; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epithelial Cells; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitrates; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Nitrites; Piperidines; Receptors, Neurokinin-2; Trachea

2001
Chronic smoking enhances tachykinin synthesis and airway responsiveness in guinea pigs.
    American journal of respiratory cell and molecular biology, 2001, Volume: 25, Issue:3

    Topics: Analysis of Variance; Animals; Benzamides; Bronchi; Bronchial Hyperreactivity; Calcitonin Gene-Related Peptide; Capsaicin; Guinea Pigs; In Situ Hybridization; Male; Neurons, Afferent; Piperidines; Protein Precursors; Radioimmunoassay; Random Allocation; Receptors, Neurokinin-2; Smoking; Tachykinins

2001
Mechanisms of anandamide-induced vasorelaxation in rat isolated coronary arteries.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Amides; Animals; Arachidonic Acids; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Ethanolamines; Gap Junctions; Glycyrrhetinic Acid; In Vitro Techniques; Indoles; Indomethacin; Male; Palmitic Acids; Peptides; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Tetraethylammonium; Vasodilation

2001
Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Animals; Apamin; Arachidonic Acid; Arachidonic Acids; Barium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Coronary Vessels; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Miconazole; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptides; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Potassium; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Receptors, Drug; Rimonabant; Sheep; Tetraethylammonium; Vasoconstrictor Agents; Vasodilation

2001
Inhibition of rat C6 glioma cell proliferation by endogenous and synthetic cannabinoids. Relative involvement of cannabinoid and vanilloid receptors.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:3

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Arachidonic Acids; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Cell Division; Glioma; Piperidines; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tumor Cells, Cultured

2001
Interactive contribution of NK(1) and kinin receptors to the acute inflammatory oedema observed in response to noxious heat stimulation: studies in NK(1) receptor knockout mice.
    British journal of pharmacology, 2001, Volume: 134, Issue:8

    Topics: Administration, Topical; Animals; Bradykinin; Bradykinin Receptor Antagonists; Burns; Capsaicin; Cell Movement; Dermatitis; Edema; Hot Temperature; Injections, Intravenous; Mice; Mice, Inbred C57BL; Mice, Knockout; Neutrophils; Piperidines; Quinuclidines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Neurokinin-1; Tachykinins; Time Factors

2001
Effects of vanilloid receptor agonists and antagonists on gastric antral ulcers in rats.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Acetamides; Animals; Anti-Ulcer Agents; Capsaicin; Cations; Ditiocarb; Famotidine; Ion Channels; Male; Piperidines; Pyloric Antrum; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Ruthenium Red; Stomach Ulcer

2001
Effect of neutral endopeptidase inhibitor on bradykinin-induced bronchoconstriction.
    Life sciences, 2001, Nov-21, Volume: 70, Issue:1

    Topics: Animals; Benzamides; Bradykinin; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Capsaicin; Dipeptides; Dose-Response Relationship, Drug; Drug Antagonism; Drug Interactions; Glycopeptides; Guinea Pigs; Indoles; Lung; Male; Metalloendopeptidases; Neurokinin A; Piperidines; Substance P

2001
CB(1) receptor antagonist SR141716A increases capsaicin-evoked release of Substance P from the adult mouse spinal cord.
    British journal of pharmacology, 2002, Volume: 135, Issue:1

    Topics: Adjuvants, Immunologic; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Mice; Nociceptors; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Receptors, Neurokinin-1; Rimonabant; Spinal Cord; Substance P

2002
ReN 1869, a novel tricyclic antihistamine, is active against neurogenic pain and inflammation.
    European journal of pharmacology, 2002, Jan-18, Volume: 435, Issue:1

    Topics: Animals; Benzoquinones; Binding Sites; Calcitonin Gene-Related Peptide; Calcium; Calcium Channels; Capsaicin; Carrageenan; Central Nervous System; CHO Cells; Cricetinae; Disease Models, Animal; Edema; Extravasation of Diagnostic and Therapeutic Materials; Gene Expression; Guinea Pigs; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Mice; Neurogenic Inflammation; Pain; Pain Measurement; Piperidines; Proto-Oncogene Proteins c-fos; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Species Specificity; Spinal Cord; Transfection; Tritium

2002
Role of kinins and sensory neurons in the rat pleural leukocyte migration induced by Phoneutria nigriventer spider venom.
    Neuroscience letters, 2002, Feb-01, Volume: 318, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aprotinin; Benzamides; Bradykinin; Bradykinin Receptor Antagonists; Capsaicin; Chemotaxis, Leukocyte; Dose-Response Relationship, Drug; Leukocytes; Male; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Pleura; Pleurisy; Quinuclidines; Rats; Rats, Wistar; Receptors, Bradykinin; Receptors, Neurokinin-1; Soybean Proteins; Spider Venoms; Trypsin Inhibitors

2002
Orphanin FQ inhibits capsaicin-induced thermal nociception in monkeys by activation of peripheral ORL1 receptors.
    British journal of pharmacology, 2002, Volume: 135, Issue:4

    Topics: Animals; Benzimidazoles; Capsaicin; Female; Heating; Macaca mulatta; Male; Nociceptin; Nociceptin Receptor; Opioid Peptides; Pain; Piperidines; Receptors, Opioid; Tail

2002
Relaxant effect of capsazepine in the isolated rat ileum.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 365, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Calcium Channels, L-Type; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Gastrointestinal Transit; Ileum; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptors, Drug

2002
Sensitizing effects of lafutidine on CGRP-containing afferent nerves in the rat stomach.
    British journal of pharmacology, 2002, Volume: 135, Issue:6

    Topics: Acetamides; Animals; Anti-Ulcer Agents; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Gastric Mucosa; Male; Neurons, Afferent; Nitric Oxide; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Stomach

2002
Inhibition of human low density lipoprotein oxidation by active principles from spices.
    Molecular and cellular biochemistry, 2002, Volume: 229, Issue:1-2

    Topics: Alkaloids; Allyl Compounds; Ascorbic Acid; Benzodioxoles; Butylated Hydroxyanisole; Capsaicin; Curcumin; Eugenol; Humans; In Vitro Techniques; Lipoproteins, LDL; Oxidation-Reduction; Piperidines; Polyunsaturated Alkamides; Quercetin; Spices; Sulfides

2002
Interaction between vanilloid and glutamate receptors in the central modulation of nociception.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Capsaicin; Chromones; Excitatory Amino Acid Antagonists; Male; Pain; Periaqueductal Gray; Phosphoserine; Piperidines; Protein Binding; Pyrazoles; Pyridines; Rats; Rats, Wistar; Receptors, Drug; Receptors, Glutamate; Riluzole; Rimonabant; Time Factors

2002
Arvanil-induced inhibition of spasticity and persistent pain: evidence for therapeutic sites of action different from the vanilloid VR1 receptor and cannabinoid CB(1)/CB(2) receptors.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Genotype; Mice; Mice, Inbred Strains; Mice, Knockout; Morpholines; Multiple Sclerosis; Muscle Spasticity; Naphthalenes; Pain; Pain Measurement; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
Anandamide-induced vasorelaxation in rabbit aortic rings has two components: G protein dependent and independent.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:6

    Topics: Animals; Aorta; Arachidonic Acids; Cannabinoids; Capsaicin; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Gap Junctions; GTP-Binding Proteins; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rabbits; Receptors, Calcitonin Gene-Related Peptide; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Virulence Factors, Bordetella

2002
The effect of cannabinoids on capsaicin-evoked calcitonin gene-related peptide (CGRP) release from the isolated paw skin of diabetic and non-diabetic rats.
    Neuropharmacology, 2002, Volume: 42, Issue:7

    Topics: Animals; Calcitonin Gene-Related Peptide; Cannabinoids; Capsaicin; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Hindlimb; In Vitro Techniques; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Reference Values; Rimonabant; Skin

2002
Pharmacological profile of (2R-trans)-4-[1-[3,5-bis(trifluoromethyl)benzoyl]-2-(phenylmethyl)-4-piperidinyl]-N-(2,6-dimethylphenyl)-1-acetamide (S)-Hydroxybutanedioate (R116301), an orally and centrally active neurokinin-1 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:2

    Topics: Administration, Oral; Allergens; Animals; Butanols; Capsaicin; Cats; Dogs; Edema; Ferrets; Gerbillinae; Guinea Pigs; Histamine; Kinetics; Malates; Mice; Motor Activity; Neurokinin-1 Receptor Antagonists; Piperidines; Platelet Activating Factor; Rabbits; Receptors, Neurokinin-1; Salivation; Substance P; Time Factors

2002
SCH 206272: a potent, orally active tachykinin NK(1), NK(2), and NK(3) receptor antagonist.
    European journal of pharmacology, 2002, Aug-23, Volume: 450, Issue:2

    Topics: Acetamides; Administration, Oral; Animals; Bronchoconstriction; Capillary Permeability; Capsaicin; CHO Cells; Cough; Cricetinae; Dogs; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Pulmonary Artery; Radioligand Assay; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Vas Deferens

2002
Effect of piperine, the active ingredient of black pepper, on intestinal secretion in mice.
    Life sciences, 2002, Sep-27, Volume: 71, Issue:19

    Topics: Alkaloids; Animals; Anti-Ulcer Agents; Benzodioxoles; Capsaicin; Castor Oil; Dose-Response Relationship, Drug; Drug Interactions; Injections, Intraperitoneal; Intestinal Secretions; Intestine, Small; Male; Mice; Mice, Inbred ICR; Organ Size; Piperidines; Polyunsaturated Alkamides

2002
Pharmacological separation of cannabinoid sensitive receptors on hippocampal excitatory and inhibitory fibers.
    Neuropharmacology, 2002, Volume: 43, Issue:4

    Topics: Animals; Axons; Benzoxazines; Capsaicin; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; Male; Morpholines; Naphthalenes; Nerve Fibers; Piperidines; Pyramidal Cells; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Reflex, Monosynaptic; Synaptic Transmission

2002
Anandamide induces cough in conscious guinea-pigs through VR1 receptors.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Aerosols; Animals; Arachidonic Acids; Calcium; Camphanes; Capsaicin; Cells, Cultured; Consciousness; Cough; Dronabinol; Endocannabinoids; Excitatory Amino Acid Antagonists; Guinea Pigs; Male; Nodose Ganglion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
A peripheral mechanism for CB1 cannabinoid receptor-dependent modulation of feeding.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Nov-01, Volume: 22, Issue:21

    Topics: Animals; Appetite Regulation; Arachidonic Acids; Behavior, Animal; Benzoxazines; Brain; Cannabinoid Receptor Modulators; Capsaicin; Denervation; Dose-Response Relationship, Drug; Drug Synergism; Eating; Endocannabinoids; Feeding Behavior; Gastric Mucosa; Hyperphagia; Injections, Intraperitoneal; Injections, Intraventricular; Intestine, Small; Male; Morpholines; Naphthalenes; Oleic Acid; Oleic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Satiety Response

2002
Evidence for the involvement of a macrophage-derived chemotactic mediator in the neutrophil recruitment induced by staphylococcal enterotoxin B in mice.
    Toxicon : official journal of the International Society on Toxinology, 2002, Volume: 40, Issue:12

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Benzeneacetamides; Capsaicin; Chemotaxis, Leukocyte; Cimetidine; Dexamethasone; Diterpenes; Enterotoxins; Enzyme Inhibitors; Ginkgolides; Hydroxamic Acids; Indomethacin; Interleukin-8; Lactones; Macrophages, Peritoneal; Male; Mice; Neutrophil Infiltration; Piperidines; Quinuclidines; Rats; Rats, Wistar

2002
Effect of lafutidine, a histamine H2-receptor antagonist, on gastric mucosal blood flow and duodenal HCO3- secretion in rats: relation to capsaicin-sensitive afferent neurons.
    Digestive diseases and sciences, 2002, Volume: 47, Issue:12

    Topics: Acetamides; Animals; Bicarbonates; Capsaicin; Cells, Cultured; Coloring Agents; Duodenum; Gastric Mucosa; Histamine H2 Antagonists; Male; Neurons, Afferent; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Regional Blood Flow; Ruthenium Red

2002
Concentration-dependent dual effect of anandamide on sensory neuropeptide release from isolated rat tracheae.
    Neuroscience letters, 2003, Jan-16, Volume: 336, Issue:2

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; In Vitro Techniques; Male; Neuropeptides; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Reference Values; Reproducibility of Results; Rimonabant; Sensitivity and Specificity; Somatostatin; Substance P; Trachea

2003
R+-methanandamide inhibits tracheal response to endogenously released acetylcholine via capsazepine-sensitive receptors.
    European journal of pharmacology, 2003, Jan-10, Volume: 459, Issue:1

    Topics: Acetylcholine; Animals; Arachidonic Acids; Atropine; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Trachea

2003
Lafutidine increases hepatic blood flow via potentiating the action of central thyrotropin-releasing hormone in rats.
    Journal of gastroenterology and hepatology, 2003, Volume: 18, Issue:2

    Topics: Acetamides; Analysis of Variance; Animals; Capsaicin; Drug Combinations; Drug Synergism; Gastric Mucosa; Histamine H2 Antagonists; Laser-Doppler Flowmetry; Liver; Liver Circulation; Male; Neurons, Afferent; Piperidines; Pyridines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Thyrotropin-Releasing Hormone

2003
Activation of capsaicin-sensitive primary sensory neurones induces anandamide production and release.
    Journal of neurochemistry, 2003, Volume: 84, Issue:3

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Endocannabinoids; Male; Neurons, Afferent; Piperidines; Polyunsaturated Alkamides; Potassium Chloride; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Flurbiprofen inhibits capsaicin induced calcitonin gene related peptide release from rat spinal cord via an endocannabinoid dependent mechanism.
    Neuroscience letters, 2003, Feb-27, Volume: 338, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcitonin Gene-Related Peptide; Cannabinoid Receptor Modulators; Capsaicin; Cyclooxygenase Inhibitors; Dinoprostone; Dronabinol; Endocannabinoids; Fatty Acids, Unsaturated; Flurbiprofen; Immunoassay; In Vitro Techniques; Phospholipases A; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Spinal Cord

2003
Compounds acting at the endocannabinoid and/or endovanilloid systems reduce hyperkinesia in a rat model of Huntington's disease.
    Journal of neurochemistry, 2003, Volume: 84, Issue:5

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids, Neutral; Animals; Arachidonic Acids; Basal Ganglia; Cannabinoid Receptor Modulators; Capsaicin; Corpus Striatum; Cyclohexanols; Disease Models, Animal; Dopamine; Endocannabinoids; gamma-Aminobutyric Acid; Huntington Disease; Hyperkinesis; Male; Motor Activity; Nitro Compounds; Palmitates; Piperidines; Propionates; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Anandamide-induced depressor effect in spontaneously hypertensive rats: role of the vanilloid receptor.
    Hypertension (Dallas, Tex. : 1979), 2003, Volume: 41, Issue:3 Pt 2

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Endocannabinoids; Hypertension; Male; Mesenteric Arteries; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Neurokinin-1 receptor antagonists CP-96,345 and L-733,060 protect mice from cytokine-mediated liver injury.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:1

    Topics: Animals; Base Sequence; Biphenyl Compounds; Capsaicin; Chemical and Drug Induced Liver Injury; Cytokines; Dose-Response Relationship, Drug; Gene Expression; Lipopolysaccharides; Liver Diseases; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; RNA, Messenger; Sequence Homology, Nucleic Acid; Time Factors; Transcriptional Activation

2003
The role of neuropeptides and capsaicin-sensitive fibres in glutamate-induced nociception and paw oedema in mice.
    Brain research, 2003, Apr-18, Volume: 969, Issue:1-2

    Topics: Animals; Benzamides; Bradykinin Receptor Antagonists; Calcitonin Gene-Related Peptide; Capsaicin; Dipeptides; Edema; Foot; Glutamic Acid; Indoles; Male; Mice; Nerve Fibers; Neurokinin-1 Receptor Antagonists; Nociceptors; Pain; Piperidines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Receptors, Neurokinin-2

2003
Substance P released from intrinsic airway neurons contributes to ozone-enhanced airway hyperresponsiveness in ferret trachea.
    Journal of applied physiology (Bethesda, Md. : 1985), 2003, Volume: 95, Issue:2

    Topics: Animals; Capsaicin; Electric Stimulation; Female; Ferrets; Ganglia; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nerve Fibers; Neurokinin-1 Receptor Antagonists; Neurons; Ozone; Piperidines; Substance P; Trachea

2003
PAR-2 agonists induce contraction of murine small intestine through neurokinin receptors.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:4

    Topics: Animals; Benzamides; Capsaicin; Female; Intestine, Small; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Receptor, PAR-2; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Thrombin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Substance P; Tetrodotoxin; Trypsin

2003
Anandamide regulates neuropeptide release from capsaicin-sensitive primary sensory neurons by activating both the cannabinoid 1 receptor and the vanilloid receptor 1 in vitro.
    The European journal of neuroscience, 2003, Volume: 17, Issue:12

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Calcium Channel Blockers; Cannabinoids; Capsaicin; Cells, Cultured; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Ganglia, Spinal; In Vitro Techniques; Male; Nerve Growth Factor; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tetradecanoylphorbol Acetate; TRPV Cation Channels

2003
Modifications of capsaicin-sensitive neurons in isolated guinea pig ileum by [6]-gingerol and lafutidine.
    Journal of pharmacological sciences, 2003, Volume: 92, Issue:4

    Topics: Acetamides; Animals; Capsaicin; Catechols; Dose-Response Relationship, Drug; Fatty Alcohols; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Neurons; Piperidines; Pyridines

2003
Inhibition of guinea-pig and human sensory nerve activity and the cough reflex in guinea-pigs by cannabinoid (CB2) receptor activation.
    British journal of pharmacology, 2003, Volume: 140, Issue:2

    Topics: Animals; Camphanes; Cannabinoids; Capsaicin; Consciousness; Cough; Cyclohexanols; Dinoprost; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Hypertonic Solutions; In Vitro Techniques; Male; Middle Aged; Neurons, Afferent; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reflex; Rimonabant; Vagus Nerve

2003
Contribution of capsaicin-sensitive afferent nerves to rapid recovery from ethanol-induced gastric epithelial damage in rats.
    Journal of gastroenterology and hepatology, 2003, Volume: 18, Issue:10

    Topics: Acetamides; Animals; Anti-Ulcer Agents; Capillary Permeability; Capsaicin; Edetic Acid; Ethanol; Gastric Mucosa; Male; Neurons, Afferent; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Ruthenium Red; Stomach Ulcer

2003
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
    Peptides, 2003, Volume: 24, Issue:7

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins

2003
Protective effect of lafutidine, a novel H2-receptor antagonist, on reflux esophagitis in rats through capsaicin-sensitive afferent neurons.
    Journal of pharmacological sciences, 2003, Volume: 93, Issue:1

    Topics: Acetamides; Animals; Capsaicin; Dose-Response Relationship, Drug; Esophagitis, Peptic; Histamine Antagonists; Male; Neurons, Afferent; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2

2003
Hypotensive effect of anandamide through the activation of CB1 and VR1 spinal receptors in urethane-anesthetized rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:4

    Topics: Anesthesia, Intravenous; Anesthetics, Intravenous; Animals; Antihypertensive Agents; Arachidonic Acids; Benzoxazines; Blood Pressure; Calcium Channel Blockers; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Ganglionic Blockers; Heart Rate; Hemodynamics; Hexamethonium; Injections, Spinal; Male; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; Spinal Cord; Urethane

2003
Antinociceptive profile of (-)-spectaline: a piperidine alkaloid from Cassia leptophylla.
    Planta medica, 2003, Volume: 69, Issue:9

    Topics: Acetic Acid; Alkaloids; Analgesics; Animals; Capsaicin; Cassia; Dipyrone; Dose-Response Relationship, Drug; Flowers; Formaldehyde; Fruit; Hot Temperature; Indomethacin; Male; Mice; Pain; Phytotherapy; Piperidines; Plant Extracts

2003
Colitis induced by proteinase-activated receptor-2 agonists is mediated by a neurogenic mechanism.
    Canadian journal of physiology and pharmacology, 2003, Volume: 81, Issue:9

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Colitis; Enteric Nervous System; Inflammation; Mice; Neurons, Afferent; Neuropeptides; Oligopeptides; Piperidines; Quinuclidines; Receptor, PAR-2; Receptors, Neurokinin-1

2003
Cannabinoids inhibit the release of [3H]glutamate from rodent hippocampal synaptosomes via a novel CB1 receptor-independent action.
    The European journal of neuroscience, 2003, Volume: 18, Issue:7

    Topics: Analgesics; Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Chromatography, High Pressure Liquid; Cyclohexanols; Dose-Response Relationship, Drug; Drug Interactions; Glutamic Acid; Hippocampus; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Radioactivity; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Synaptosomes; Tritium

2003
A novel neuroimmune mechanism in cannabinoid-mediated attenuation of nerve growth factor-induced hyperalgesia.
    Anesthesiology, 2003, Volume: 99, Issue:6

    Topics: Analgesics; Animals; Arachidonic Acids; Cannabinoids; Capsaicin; Cell Movement; Endocannabinoids; Hyperalgesia; Male; Nerve Growth Factor; Neutrophils; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rimonabant

2003
Differential effects of the sleep-inducing lipid oleamide and cannabinoids on the induction of long-term potentiation in the CA1 neurons of the rat hippocampus in vitro.
    Brain research, 2004, Jan-30, Volume: 997, Issue:1

    Topics: Amidohydrolases; Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Drug Interactions; Electric Stimulation; Electrophysiology; Endocannabinoids; Excitatory Postsynaptic Potentials; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Long-Term Potentiation; Male; Morpholines; Naphthalenes; Neurons; Oleic Acids; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rimonabant; Sleep

2004
Anandamide is able to inhibit trigeminal neurons using an in vivo model of trigeminovascular-mediated nociception.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:1

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; Endocannabinoids; Hypotension; Male; Neurons; Nitroprusside; Pain; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Trigeminal Caudal Nucleus; Vasodilation

2004
Evidence for the presence of functional protease activated receptor 4 (PAR4) in the rat colon.
    Gut, 2004, Volume: 53, Issue:2

    Topics: Animals; Atropine; Benzamides; Capsaicin; Colitis; Colon; Dose-Response Relationship, Drug; Gastrointestinal Motility; Immunohistochemistry; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Thrombin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrodotoxin

2004
Individual differences in perception of bitterness from capsaicin, piperine and zingerone.
    Chemical senses, 2004, Volume: 29, Issue:1

    Topics: Adolescent; Adult; Alkaloids; Benzodioxoles; Capsaicin; Female; Guaiacol; Humans; Male; Middle Aged; Perception; Piperidines; Polyunsaturated Alkamides; Receptors, Cell Surface; Taste; Taste Buds

2004
Multiple actions of anandamide on neonatal rat cultured sensory neurones.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Calcium Channels; Calcium Signaling; Capsaicin; Cells, Cultured; Drug Synergism; Endocannabinoids; Fura-2; Ganglia, Spinal; Neurons, Afferent; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium Chloride; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; TRPV Cation Channels

2004
Mustard oil induces a transient receptor potential vanilloid 1 receptor-independent neurogenic inflammation and a non-neurogenic cellular inflammatory component in mice.
    Neuroscience, 2004, Volume: 125, Issue:2

    Topics: Animals; Capillary Permeability; Capsaicin; Dose-Response Relationship, Drug; Ear; Edema; Inflammation; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Mustard Plant; Neurokinin-1 Receptor Antagonists; Piperidines; Plant Extracts; Plant Oils; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-1; Staining and Labeling; Time Factors; TRPV Cation Channels

2004
Neonatal capsaicin treatment affects rat thymocyte proliferation and cell death by modulating substance P and neurokinin-1 receptor expression.
    Neuroimmunomodulation, 2004, Volume: 11, Issue:3

    Topics: Adjuvants, Immunologic; Animals; Animals, Newborn; Atrophy; Autocrine Communication; Binding Sites; Capsaicin; Cell Death; Cell Division; Concanavalin A; Growth Substances; Male; Neuroimmunomodulation; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; RNA, Messenger; Substance P; T-Lymphocytes; Thymus Gland; Up-Regulation

2004
Protective role of vanilloid receptor type 1 in HCl-induced gastric mucosal lesions in rats.
    Scandinavian journal of gastroenterology, 2004, Volume: 39, Issue:4

    Topics: Acetamides; Animals; Anti-Ulcer Agents; Capsaicin; Catechols; Diterpenes; Famotidine; Fatty Alcohols; Gastric Mucosa; Hydrochloric Acid; Male; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Stomach Ulcer

2004
Presynaptic cannabinoid CB(1) receptors are involved in the inhibition of the neurogenic vasopressor response during septic shock in pithed rats.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: Animals; Autonomic Fibers, Postganglionic; Autonomic Fibers, Preganglionic; Blood Pressure; Camphanes; Capsaicin; Decerebrate State; Disease Models, Animal; Electric Stimulation; Germany; Imidazoles; Infusions, Intravenous; Lipopolysaccharides; Male; Norepinephrine; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Shock, Septic; Solvents; Thiourea; Vagotomy; Vasomotor System; Vasopressins

2004
Implantation of tumoral XC cells induces chronic, endothelin-dependent, thermal hyperalgesia in mice.
    Cellular and molecular neurobiology, 2004, Volume: 24, Issue:2

    Topics: Animals; Avian Sarcoma Viruses; Capsaicin; Cell Line, Transformed; Cell Line, Tumor; Chronic Disease; Endothelin Receptor Antagonists; Endothelins; Fibroblasts; Genetic Vectors; Hindlimb; Hyperalgesia; Inflammation; Male; Mice; Morphine; Neoplasm Regression, Spontaneous; Neoplasm Transplantation; Nociceptors; Oligopeptides; Pain Measurement; Peptides, Cyclic; Piperidines; Rats; Reaction Time; Receptors, Endothelin

2004
Sex-linked differences in the vasorelaxant effects of anandamide in vascular mesenteric beds: role of oestrogens.
    European journal of pharmacology, 2004, Jun-16, Volume: 493, Issue:1-3

    Topics: Acetylcholine; Animals; Arachidonic Acids; Argentina; Capsaicin; Chile; Cycloheximide; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Estradiol; Estrogens; Female; Male; Mesentery; Muscle, Smooth, Vascular; Nitroprusside; Norepinephrine; Ovariectomy; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Sex Characteristics; Time Factors; Vasodilation

2004
Characterization of cannabinoid modulation of sensory neurotransmission in the rat isolated mesenteric arterial bed.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 311, Issue:1

    Topics: Animals; Benzofurans; Benzoxazines; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoids; Capsaicin; Cyclohexanols; Dronabinol; Electric Stimulation; Indoles; Male; Mesenteric Arteries; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Rimonabant; Vasodilation

2004
TRPV1 and CB(1) receptor-mediated effects of the endovanilloid/endocannabinoid N-arachidonoyl-dopamine on primary afferent fibre and spinal cord neuronal responses in the rat.
    The European journal of neuroscience, 2004, Volume: 20, Issue:1

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Calcium; Capsaicin; Cells, Cultured; Dopamine; Drug Interactions; Electrophysiology; Male; Membrane Potentials; Nerve Fibers; Pain Measurement; Physical Stimulation; Piperidines; Posterior Horn Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; Sensory Thresholds; Spinal Cord

2004
Inhibitory effect of the antidepressant St. John's wort (hypericum perforatum) on rat bladder contractility in vitro.
    Urology, 2004, Volume: 64, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Anthracenes; Antidepressive Agents; Atropine; Bridged Bicyclo Compounds; Capsaicin; Depression; Electric Stimulation; Female; Haloperidol; Hypericum; Kaempferols; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Naloxone; Perylene; Phentolamine; Phloroglucinol; Piperidines; Plant Extracts; Propranolol; Pyrazoles; Quercetin; Rats; Rats, Wistar; Rimonabant; Rutin; Terpenes; Tetrodotoxin; Urinary Bladder; Urinary Incontinence; Verapamil

2004
Vanilloid TRPV1 receptor mediates the antihyperalgesic effect of the nonpsychoactive cannabinoid, cannabidiol, in a rat model of acute inflammation.
    British journal of pharmacology, 2004, Volume: 143, Issue:2

    Topics: Administration, Oral; Animals; Camphanes; Cannabidiol; Capsaicin; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Therapy, Combination; Hyperalgesia; Inflammation; Italy; Male; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Drug; Rimonabant; Time Factors

2004
Vanilloid receptor TRPV1, sensory C-fibers, and vascular autoregulation: a novel mechanism involved in myogenic constriction.
    Circulation research, 2004, Nov-12, Volume: 95, Issue:10

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Capsaicin; Cation Transport Proteins; CHO Cells; Cricetinae; Endothelium, Vascular; Gadolinium; Ganglia, Sympathetic; Guanethidine; Hydroxyeicosatetraenoic Acids; Ion Channels; Male; Mesenteric Arteries; Mice; Mice, Knockout; Models, Cardiovascular; Models, Neurological; Nerve Fibers, Unmyelinated; Nociceptors; Peptides, Cyclic; Piperidines; Pressure; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Ruthenium Red; Sodium Channel Blockers; Splanchnic Circulation; Stress, Mechanical; Sympathectomy, Chemical; Tetrodotoxin; TRPV Cation Channels; Vascular Resistance; Vasoconstriction

2004
Human brain endothelium: coexpression and function of vanilloid and endocannabinoid receptors.
    Brain research. Molecular brain research, 2004, Dec-06, Volume: 132, Issue:1

    Topics: Arachidonic Acids; Blood-Brain Barrier; Brain; Camphanes; Cannabinoid Receptor Agonists; Cannabinoid Receptor Modulators; Capsaicin; Cell Adhesion Molecules; Cells, Cultured; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Endothelium, Vascular; Glycerides; Humans; Ion Channels; Microcirculation; Microfilament Proteins; Phosphoproteins; Phosphorylation; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; RNA, Messenger; TRPV Cation Channels

2004
Protective effect of lafutidine, a novel histamine H2-receptor antagonist, on dextran sulfate sodium-induced colonic inflammation through capsaicin-sensitive afferent neurons in rats.
    Digestive diseases and sciences, 2004, Volume: 49, Issue:10

    Topics: Acetamides; Animals; Capsaicin; Colitis, Ulcerative; Dextran Sulfate; Histamine H2 Antagonists; Intestinal Mucosa; Male; Neurons, Afferent; Peroxidase; Piperidines; Pyridines; Rats; Rats, Wistar

2004
Lafutidine-induced increase in intracellular ca(2+) concentrations in PC12 and endothelial cells.
    Journal of pharmacological sciences, 2005, Volume: 97, Issue:1

    Topics: Acetamides; Animals; Calcium; Calcium Chloride; Capsaicin; Dose-Response Relationship, Drug; Endothelial Cells; Humans; Imidazoles; Immunoblotting; Intracellular Fluid; PC12 Cells; Piperidines; Pyridines; Rats; Thapsigargin; Time Factors

2005
AM404, an inhibitor of anandamide reuptake decreases Fos-immunoreactivity in the spinal cord of neuropathic rats after non-noxious stimulation.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Dose-Response Relationship, Drug; Endocannabinoids; Immunohistochemistry; Indoles; Male; Physical Stimulation; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Spinal Cord

2005
Role of capsaicin-sensitive nerves and histamine H1, H2, and H3 receptors in the gastroprotective effect of histamine against stress ulcers in rats.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Capsaicin; DNA; Gastric Mucosa; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Immersion; Interleukin-1; Male; Neurons, Afferent; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Regional Blood Flow; Restraint, Physical; Stomach Ulcer; Stress, Physiological

2005
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005
Effects of piperine, the pungent component of black pepper, at the human vanilloid receptor (TRPV1).
    British journal of pharmacology, 2005, Volume: 144, Issue:6

    Topics: Alkaloids; Benzodioxoles; Capsaicin; Cell Line; Humans; Hydrogen-Ion Concentration; Patch-Clamp Techniques; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Receptors, Drug; Ruthenium Red; Structure-Activity Relationship

2005
CB(1) cannabinoid receptor stimulation modulates transient receptor potential vanilloid receptor 1 activities in calcium influx and substance P Release in cultured rat dorsal root ganglion cells.
    Journal of pharmacological sciences, 2005, Volume: 97, Issue:3

    Topics: Animals; Bradykinin; Calcium; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Capsaicin; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Cyclooxygenase 2; Dose-Response Relationship, Drug; Dronabinol; Enzyme Induction; Enzyme Inhibitors; Ganglia, Spinal; Isoquinolines; Male; Piperidines; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; RNA, Messenger; Substance P; Sulfonamides; Time Factors

2005
The effects of Delta9-tetrahydrocannabinol in rat mesenteric vasculature, and its interactions with the endocannabinoid anandamide.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Apamin; Arachidonic Acids; Azepines; Barium Compounds; Biological Factors; Calcium; Cannabinoid Receptor Modulators; Capsaicin; Charybdotoxin; Chlorides; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Endocannabinoids; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Vasodilation; Verapamil

2005
Protective effects of Delta(9)-tetrahydrocannabinol against N-methyl-d-aspartate-induced AF5 cell death.
    Brain research. Molecular brain research, 2005, Apr-04, Volume: 134, Issue:2

    Topics: alpha-Tocopherol; Animals; Benzimidazoles; Benzoxazines; Blotting, Northern; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Capsaicin; Cell Count; Cell Death; Cell Lineage; Dizocilpine Maleate; DNA, Single-Stranded; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Excitatory Amino Acid Agonists; Immunohistochemistry; In Situ Nick-End Labeling; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Neuroprotective Agents; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Ruthenium; Tetrazolium Salts; Thiazoles; TRPC Cation Channels

2005
Peripheral, but not central effects of cannabidiol derivatives: mediation by CB(1) and unidentified receptors.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Body Temperature; Camphanes; Cannabidiol; Capsaicin; Drug Interactions; Ear, External; Gastrointestinal Motility; Inflammation; Mice; Mice, Inbred ICR; Mice, Inbred Strains; Motor Activity; Pain Measurement; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant

2005
Evidence that (-)-7-hydroxy-4'-dimethylheptyl-cannabidiol activates a non-CB(1), non-CB(2), non-TRPV1 target in the mouse vas deferens.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzoxazines; Cannabidiol; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Capsaicin; In Vitro Techniques; Isometric Contraction; Male; Mice; Morpholines; Naloxone; Naphthalenes; Phenylephrine; Piperidines; Pyrazoles; Rimonabant; Ruthenium Red; TRPV Cation Channels; Vas Deferens; Yohimbine

2005
Sensory peptide neurotransmitters mediating mucosal and distension evoked neural vasodilator reflexes in guinea pig ileum.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 289, Issue:5

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Guinea Pigs; Hexamethonium; Ileum; Intestinal Mucosa; Neurons; Neurotransmitter Agents; Nifedipine; Piperidines; Signal Transduction; Tachykinins; Vasodilation

2005
Inhibitory effects of CB1 and CB2 receptor agonists on responses of DRG neurons and dorsal horn neurons in neuropathic rats.
    The European journal of neuroscience, 2005, Volume: 22, Issue:2

    Topics: Action Potentials; Animals; Arachidonic Acids; Behavior, Animal; Calcium; Camphanes; Cannabinoids; Capsaicin; Cells, Cultured; Diagnostic Imaging; Dose-Response Relationship, Drug; Drug Interactions; Evoked Potentials; Ganglia, Spinal; Hyperalgesia; Ligation; Male; Neural Inhibition; Neurons; Pain Measurement; Piperidines; Posterior Horn Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Spinal Cord Diseases; Touch

2005
TRPV1 activation results in disruption of the blood-brain barrier in the rat.
    British journal of pharmacology, 2005, Volume: 146, Issue:4

    Topics: Animals; Blood-Brain Barrier; Brain Ischemia; Capillaries; Capillary Permeability; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Male; Microspheres; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Starch; Substance P; Tetrazoles; Time Factors; TRPV Cation Channels

2005
Anandamide elicits an acute release of nitric oxide through endothelial TRPV1 receptor activation in the rat arterial mesenteric bed.
    The Journal of physiology, 2005, Oct-15, Volume: 568, Issue:Pt 2

    Topics: Anilides; Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Capsaicin; Cinnamates; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Artery, Superior; Nitric Oxide; Nitroarginine; Perfusion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; RNA, Messenger; TRPV Cation Channels; Vasodilation

2005
Endogenous cannabinoid receptor agonists inhibit neurogenic inflammations in guinea pig airways.
    International archives of allergy and immunology, 2005, Volume: 138, Issue:1

    Topics: Amides; Animals; Arachidonic Acids; Bronchi; Bronchoconstriction; Calcium Channel Blockers; Camphanes; Cannabinoid Receptor Agonists; Capsaicin; Electric Stimulation; Endocannabinoids; Ethanolamines; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Unmyelinated; Neurogenic Inflammation; Organ Culture Techniques; Palmitic Acids; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Pyrazoles; Receptors, Cannabinoid; Rimonabant; Substance P

2005
Inhibition of fatty-acid amide hydrolase enhances cannabinoid stress-induced analgesia: sites of action in the dorsolateral periaqueductal gray and rostral ventromedial medulla.
    Neuropharmacology, 2005, Volume: 49, Issue:8

    Topics: Amidohydrolases; Analgesia; Animals; Arachidonic Acids; Cannabinoids; Capsaicin; Carrier Proteins; Cytosol; Endocannabinoids; Male; Medulla Oblongata; Mice; Microinjections; Pain Measurement; Periaqueductal Gray; Phospholipases A; Phospholipases A2; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Stress, Psychological; TRPV Cation Channels

2005
VR1-mediated depressor effects during high-salt intake: role of anandamide.
    Hypertension (Dallas, Tex. : 1979), 2005, Volume: 46, Issue:4

    Topics: Animals; Arachidonic Acids; Blood Pressure; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Dose-Response Relationship, Drug; Drug Combinations; Endocannabinoids; Male; Mesenteric Arteries; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Sodium, Dietary; Time Factors; TRPV Cation Channels

2005
Pivotal role of endogenous tachykinins and the NK1 receptor in mediating leukocyte accumulation, in the absence of oedema formation, in response to TNFalpha in the cutaneous microvasculature.
    Journal of neuroimmunology, 2006, Volume: 171, Issue:1-2

    Topics: Albumins; Analysis of Variance; Animals; Capsaicin; Dose-Response Relationship, Drug; Female; Glycoproteins; Immunohistochemistry; Inflammation; Injections, Intradermal; Iodine Isotopes; Leukocytes; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neutrophils; Peroxidase; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Skin; Substance P; Tachykinins; Time Factors; Tumor Necrosis Factor-alpha

2006
Capsaicin evokes hypothermia independent of cannabinoid CB1 and CB2 receptors.
    Brain research, 2005, Dec-14, Volume: 1065, Issue:1-2

    Topics: Anilides; Animals; Benzoxazines; Body Temperature; Calcium Channel Blockers; Camphanes; Capsaicin; Cinnamates; Hypothermia; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; TRPV Cation Channels

2005
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Apamin; Barium; Benzopyrans; Caffeine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Charybdotoxin; Diclofenac; Dimethyl Sulfoxide; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanethidine; Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nitroarginine; Papaverine; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Protein Serine-Threonine Kinases; Pyrazoles; Receptor, Cannabinoid, CB1; rho-Associated Kinases; Tetraethylammonium; Vasodilator Agents

2006
Vanilloid VR1 receptor is involved in rimonabant-induced neuroprotection.
    British journal of pharmacology, 2006, Volume: 147, Issue:5

    Topics: Animals; Avoidance Learning; Brain Ischemia; Cannabinoid Receptor Antagonists; Capsaicin; Electroencephalography; Gerbillinae; Male; Motor Activity; Neuroprotective Agents; Piperidines; Pyrazoles; Rimonabant; TRPV Cation Channels

2006
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:4

    Topics: Amidohydrolases; Anilides; Animals; Arachidonic Acids; Body Temperature; Capsaicin; Cinnamates; Endocannabinoids; Hypothermia; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels

2006
Gastro-protective action of lafutidine mediated by capsaicin-sensitive afferent neurons without interaction with TRPV1 and involvement of endogenous prostaglandins.
    World journal of gastroenterology, 2006, May-21, Volume: 12, Issue:19

    Topics: 6-Ketoprostaglandin F1 alpha; Acetamides; Animals; Calcium; Capsaicin; Dinoprostone; Dose-Response Relationship, Drug; Gastric Mucosa; Histamine H2 Antagonists; Humans; Indomethacin; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; NG-Nitroarginine Methyl Ester; Piperidines; Prostaglandins; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Epoprostenol; Stomach; Stomach Diseases; TRPV Cation Channels

2006
The NK1 receptor antagonist SR140333 inhibits capsaicin-induced ERK phosphorylation in sensory neurons.
    Pharmacology, 2006, Volume: 77, Issue:3

    Topics: Animals; Capsaicin; Extracellular Signal-Regulated MAP Kinases; Ganglia, Spinal; Gene Expression Regulation; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Phosphorylation; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sciatic Nerve; STAT3 Transcription Factor; TRPV Cation Channels

2006
Enhanced antinociceptive effects of morphine in histamine H2 receptor gene knockout mice.
    Neuropharmacology, 2006, Volume: 51, Issue:3

    Topics: Analysis of Variance; Animals; Benzothiazoles; Brain; Capsaicin; Drug Synergism; Ganglia, Spinal; Histamine H2 Antagonists; Hot Temperature; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Narcotics; Pain Measurement; Phenoxypropanolamines; Piperidines; Reaction Time; Receptors, Histamine H2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Touch

2006
Non-cannabinoid CB1, non-cannabinoid CB2 antinociceptive effects of several novel compounds in the PPQ stretch test in mice.
    European journal of pharmacology, 2006, Sep-28, Volume: 546, Issue:1-3

    Topics: Acetaminophen; Amides; Analgesics; Animals; Arachidonic Acids; Benzamides; Benzoquinones; Camphanes; Capsaicin; Carbamates; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Ethanolamines; Hyperalgesia; Male; Mesencephalon; Mice; Mice, Inbred ICR; Narcotic Antagonists; Pain; Palmitic Acids; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid; Rimonabant; Spinal Cord; TRPV Cation Channels

2006
Spinal modulation of calcitonin gene-related peptide by endocannabinoids in the development of opioid physical dependence.
    Pain, 2006, Dec-15, Volume: 126, Issue:1-3

    Topics: Animals; Calcitonin Gene-Related Peptide; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Drug Administration Schedule; Endocannabinoids; Ganglia, Spinal; Hot Temperature; Immunologic Techniques; Male; Morphine; Naloxone; Narcotic Antagonists; Neurons; Nociceptors; Opioid-Related Disorders; Piperidines; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; RNA, Messenger; Spinal Cord; Substance Withdrawal Syndrome

2006
Anandamide mediates hyperdynamic circulation in cirrhotic rats via CB(1) and VR(1) receptors.
    British journal of pharmacology, 2006, Volume: 149, Issue:7

    Topics: Animals; Arachidonic Acids; Bile Ducts; Blood Flow Velocity; Blood Pressure; Blotting, Western; Capsaicin; Cardiac Output; Disease Models, Animal; Endocannabinoids; Hyperemia; Indoles; Liver Circulation; Liver Cirrhosis, Biliary; Male; Mesenteric Artery, Superior; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Splanchnic Circulation; Time Factors; TRPV Cation Channels; Vascular Resistance; Vasodilation; Vasodilator Agents

2006
Prolonged maintenance of capsaicin-induced hyperalgesia by brief daily vibration stimuli.
    Pain, 2007, Volume: 129, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Behavior, Animal; Capsaicin; Drug Interactions; Excitatory Amino Acid Antagonists; Hyperalgesia; Male; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Rats; Rats, Sprague-Dawley; Spinal Cord Injuries; Time Factors; Vibration

2007
Involvement of TRPV1-dependent and -independent components in the regulation of vagally induced contractions in the mouse esophagus.
    European journal of pharmacology, 2007, Feb-05, Volume: 556, Issue:1-3

    Topics: Alkaloids; Anilides; Animals; Benzodioxoles; Capsaicin; Cinnamates; Cricetinae; Enzyme Inhibitors; Esophagus; Female; Male; Mesocricetus; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Tachykinin; Species Specificity; TRPV Cation Channels; Tryptophan; Vagus Nerve

2007
NK-1 receptors modulate the excitability of ON cells in the rostral ventromedial medulla.
    Journal of neurophysiology, 2007, Volume: 97, Issue:2

    Topics: Animals; Capsaicin; Electrophysiology; Excitatory Amino Acid Agonists; Extracellular Space; Immunohistochemistry; Iontophoresis; Male; Medulla Oblongata; Microscopy, Confocal; N-Methylaspartate; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P

2007
Inhibition of neutrophil activation by lafutidine, an H2-receptor antagonist, through enhancement of sensory neuron activation contributes to the reduction of stress-induced gastric mucosal injury in rats.
    Digestive diseases and sciences, 2007, Volume: 52, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Acetamides; Animals; Anti-Ulcer Agents; Arachidonic Acids; Calcitonin Gene-Related Peptide; Capsaicin; Cells, Cultured; Cyclooxygenase Inhibitors; Disease Models, Animal; Endocannabinoids; Famotidine; Ganglia, Spinal; Gastric Acid; Gastric Mucosa; Histamine H2 Antagonists; Indomethacin; Male; Neurons, Afferent; Neutrophil Activation; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyridines; Rats; Rats, Wistar; Restraint, Physical; Stomach Ulcer; Stress, Psychological

2007
Effects of inhibition of fatty acid amide hydrolase vs. the anandamide membrane transporter on TRPV1-mediated calcium responses in adult DRG neurons; the role of CB receptors.
    The European journal of neuroscience, 2006, Volume: 24, Issue:12

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Calcium; Capsaicin; Carbamates; Cells, Cultured; Dopamine; Drug Interactions; Endocannabinoids; Fura-2; Furans; Ganglia, Spinal; Male; Membrane Potentials; Membrane Transport Proteins; Neurons; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2006
TRPV1 is involved in stretch-evoked contractile changes in the rat autonomous bladder model: a study with piperine, a new TRPV1 agonist.
    Neurourology and urodynamics, 2007, Volume: 26, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Indicators and Reagents; Mechanotransduction, Cellular; Muscle Contraction; Piperidines; Polyunsaturated Alkamides; Pressure; Rats; Rats, Wistar; Ruthenium Red; Stress, Mechanical; TRPV Cation Channels; Urinary Bladder

2007
Pharmacological characterisation of capsaicin-induced relaxations in human and porcine isolated arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adolescent; Adult; Aged; Analgesics, Non-Narcotic; Animals; Arteries; Calcitonin Gene-Related Peptide; Capsaicin; Coronary Vessels; Cyclic AMP; Dipeptides; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Middle Aged; NG-Nitroarginine Methyl Ester; Piperazines; Piperidines; Potassium Channel Blockers; Potassium Chloride; Protein Kinase Inhibitors; Quinazolines; Swine; Vasodilation

2007
Effects of allyl isothiocyanate from horseradish on several experimental gastric lesions in rats.
    European journal of pharmacology, 2007, Apr-30, Volume: 561, Issue:1-3

    Topics: Alkaloids; Ammonia; Animals; Armoracia; Aspirin; Benzodioxoles; Capsaicin; Dose-Response Relationship, Drug; Ethanol; Food Preservatives; Gastric Mucosa; Hydrochloric Acid; Indomethacin; Isothiocyanates; Male; NG-Nitroarginine Methyl Ester; Omeprazole; Piperidines; Polyunsaturated Alkamides; Prostaglandins; Rats; Rats, Sprague-Dawley; Ruthenium Red; Structure-Activity Relationship

2007
Temporal interactions between oral irritants: piperine, zingerone, and capsaicin.
    Chemical senses, 2007, Volume: 32, Issue:5

    Topics: Administration, Oral; Alkaloids; Benzodioxoles; Capsaicin; Guaiacol; Humans; Irritants; Piperidines; Polyunsaturated Alkamides

2007
Arvanil, anandamide and N-arachidonoyl-dopamine (NADA) inhibit emesis through cannabinoid CB1 and vanilloid TRPV1 receptors in the ferret.
    The European journal of neuroscience, 2007, Volume: 25, Issue:9

    Topics: Acrylamides; Animals; Antiemetics; Arachidonic Acids; Area Postrema; Autonomic Pathways; Brain Stem; Bridged Bicyclo Compounds, Heterocyclic; Cannabinoids; Capsaicin; Dopamine; Emetics; Endocannabinoids; Ferrets; Male; Mice; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Solitary Nucleus; TRPV Cation Channels; Vagus Nerve; Vomiting

2007
AM404 decreases Fos-immunoreactivity in the spinal cord in a model of inflammatory pain.
    Brain research, 2007, Jun-04, Volume: 1152

    Topics: Animals; Arachidonic Acids; Capsaicin; Endocannabinoids; Immunohistochemistry; Indoles; Inflammation; Male; Pain; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Spinal Cord; TRPV Cation Channels

2007
Influence of curcumin, capsaicin, and piperine on the rat liver drug-metabolizing enzyme system in vivo and in vitro.
    Canadian journal of physiology and pharmacology, 2006, Volume: 84, Issue:12

    Topics: Alkaloids; Animals; Aryl Hydrocarbon Hydroxylases; Benzodioxoles; Capsaicin; Carrier Proteins; Curcumin; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Glucuronosyltransferase; Heme-Binding Proteins; Hemeproteins; In Vitro Techniques; Liver; Male; Microsomes, Liver; NADPH-Ferrihemoprotein Reductase; Oxidoreductases, N-Demethylating; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar

2006
Studies on the in vitro absorption of spice principles--curcumin, capsaicin and piperine in rat intestines.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 2007, Volume: 45, Issue:8

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Curcumin; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Male; Micelles; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Spices

2007
Involvement of the endocannabinoid system in retinal damage after high intraocular pressure-induced ischemia in rats.
    Investigative ophthalmology & visual science, 2007, Volume: 48, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cell Count; Chromatography, High Pressure Liquid; Endocannabinoids; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Hydrolysis; Intraocular Pressure; Male; Ocular Hypertension; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reperfusion Injury; Retinal Diseases; Retinal Ganglion Cells; Retinal Vessels; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Thy-1 Antigens; TRPV Cation Channels

2007
Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Aorta, Abdominal; Apamin; Arachidonic Acids; Benzamides; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Charybdotoxin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Isoindoles; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sulfonamides; Vasodilation

2007
Delta 9-tetrahydrocannabinol inhibits electrically-evoked CGRP release and capsaicin-sensitive sensory neurogenic vasodilatation in the rat mesenteric arterial bed.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Dronabinol; Electric Stimulation; Indoles; Male; Mesenteric Arteries; Methoxamine; Neurons, Afferent; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Ruthenium Red; Time Factors; Vasodilation

2007
Increased depressor response to N-arachidonoyl-dopamine during high salt intake: role of the TRPV1 receptor.
    Journal of hypertension, 2007, Volume: 25, Issue:12

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Dopamine; Male; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Rimonabant; Sodium Chloride, Dietary; TRPV Cation Channels

2007
Lafutidine facilitates calcitonin gene-related peptide (CGRP) nerve-mediated vasodilation via vanilloid-1 receptors in rat mesenteric resistance arteries.
    Journal of pharmacological sciences, 2008, Volume: 106, Issue:3

    Topics: Acetamides; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Drug Synergism; Electric Stimulation; Male; Mesenteric Arteries; Peripheral Nervous System; Piperidines; Pyridines; Rats; Rats, Wistar; Ruthenium Red; TRPV Cation Channels; Vasodilation

2008
Effect of cannabidiol on sepsis-induced motility disturbances in mice: involvement of CB receptors and fatty acid amide hydrolase.
    Neurogastroenterology and motility, 2008, Volume: 20, Issue:8

    Topics: Amidohydrolases; Animals; Cannabidiol; Capsaicin; Gastric Emptying; Gastrointestinal Motility; Intestine, Small; Lipopolysaccharides; Male; Mice; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Sensory System Agents; Sepsis

2008
Metalloelastase in lungs and alveolar macrophages is modulated by extracellular substance P in mice.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 295, Issue:1

    Topics: Animals; Bronchoalveolar Lavage; Capsaicin; Cell Survival; Female; Gene Expression Regulation, Enzymologic; Lung; Macrophages, Alveolar; Matrix Metalloproteinase 12; Mice; Piperidines; Pulmonary Emphysema; Receptors, Neurokinin-1; RNA, Messenger; Smoking; Substance P; Up-Regulation

2008
Substance P is involved in the effect of histamine H3 receptor agonist, Sch 50971 on nasal allergic symptoms in mice.
    International immunopharmacology, 2008, Volume: 8, Issue:8

    Topics: Animals; Capsaicin; Cetirizine; Disease Models, Animal; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists, Non-Sedating; Imidazoles; Mice; Mice, Inbred BALB C; Ovalbumin; Piperidines; Pyrrolidines; Receptors, Histamine H3; Rhinitis, Allergic, Perennial; Substance P; Thiourea

2008
Anxiolytic effects in mice of a dual blocker of fatty acid amide hydrolase and transient receptor potential vanilloid type-1 channels.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:3

    Topics: Amidohydrolases; Anilides; Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Benzamides; Brain; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cinnamates; Diazepam; Exploratory Behavior; Male; Mice; Mice, Inbred C57BL; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels

2009
Impairment by 5-fluorouracil of the healing of gastric lesions in rats: effect of lafutidine, a histamine H2 receptor antagonist, mediated by capsaicin-sensitive afferent neurons.
    Digestive diseases and sciences, 2009, Volume: 54, Issue:1

    Topics: Acetamides; Animals; Antimetabolites, Antineoplastic; Capsaicin; Cell Line; Cell Movement; Cell Proliferation; Disease Models, Animal; Epithelial Cells; Fluorouracil; Gastric Mucosa; Histamine H2 Antagonists; Hydrochloric Acid; Male; Neurons, Afferent; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Sensory System Agents; Stomach Diseases; Wound Healing

2009
TRPV1 mediates the uterine capsaicin-induced NMDA NR2B-dependent cross-organ reflex sensitization in anesthetized rats.
    American journal of physiology. Renal physiology, 2008, Volume: 295, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Anesthesia; Animals; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Muscle, Smooth; Neurons, Afferent; Pelvic Pain; Phosphorylation; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reflex; Spinal Cord; TRPV Cation Channels; Uterus

2008
Discovery of piperidine carboxamide TRPV1 antagonists.
    Bioorganic & medicinal chemistry letters, 2008, Aug-15, Volume: 18, Issue:16

    Topics: Amides; Benzoxazines; Capsaicin; Carrier Proteins; Chemistry, Pharmaceutical; Drug Design; Humans; Inhibitory Concentration 50; Models, Chemical; Molecular Conformation; Piperidines; Protein Binding; Quantitative Structure-Activity Relationship; Structure-Activity Relationship; TRPV Cation Channels

2008
Facilitation of contextual fear memory extinction and anti-anxiogenic effects of AM404 and cannabidiol in conditioned rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2008, Volume: 18, Issue:12

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Arachidonic Acids; Behavior, Animal; Cannabidiol; Capsaicin; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Administration Schedule; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Injections, Intraventricular; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; TRPV Cation Channels

2008
Constitutive activity at the cannabinoid CB1 receptor is required for behavioral response to noxious chemical stimulation of TRPV1: antinociceptive actions of CB1 inverse agonists.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Nov-05, Volume: 28, Issue:45

    Topics: Analysis of Variance; Animals; Behavior, Animal; Bradykinin; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cell Line, Tumor; Dose-Response Relationship, Drug; Galanin; Gene Expression Regulation; Male; Mice; Mice, Inbred ICR; Mice, Knockout; Morphine; Narcotics; Nerve Fibers, Unmyelinated; Neuroblastoma; Pain; Pain Measurement; Pain Threshold; Piperidines; Pyrazoles; Rats; Reaction Time; Receptor, Cannabinoid, CB1; Rimonabant; Stimulation, Chemical; Sulfonamides; TRPV Cation Channels

2008
Differential effects of topically applied formalin and aromatic compounds on neurogenic-mediated microvascular leakage in rat skin.
    Toxicology, 2009, Jan-08, Volume: 255, Issue:1-2

    Topics: Administration, Topical; Animals; Antipruritics; Capillary Leak Syndrome; Capsaicin; Cell Degranulation; Disinfectants; Dose-Response Relationship, Drug; Formaldehyde; Hydrocarbons, Aromatic; Ketotifen; Male; Mast Cells; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Regional Blood Flow; Skin

2009
Galanin modulates vagally induced contractions in the mouse oesophagus.
    Neurogastroenterology and motility, 2009, Volume: 21, Issue:2

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Electric Stimulation; Enzyme Inhibitors; Esophagus; Female; Galanin; Indoles; Male; Mice; Muscle Contraction; NG-Nitroarginine Methyl Ester; Phenanthrolines; Piperidines; Polyunsaturated Alkamides; Receptors, Galanin; Sensory System Agents; Substance P; Vagus Nerve

2009
Inhibitory effect of quercetin on rat trachea contractility in vitro.
    The Journal of pharmacy and pharmacology, 2009, Volume: 61, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antioxidants; Benzamides; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phentolamine; Piperidines; Propranolol; Quercetin; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Trachea

2009
Synthesis and structure-activity relationships of N-substituted spiropiperidines as nociceptin receptor ligands: part 2.
    Bioorganic & medicinal chemistry letters, 2009, Feb-15, Volume: 19, Issue:4

    Topics: Animals; Binding Sites; Capsaicin; Combinatorial Chemistry Techniques; Cough; Disease Models, Animal; Drug Design; Guinea Pigs; Molecular Structure; Nociceptin Receptor; Piperidines; Receptors, Opioid; Spiro Compounds; Structure-Activity Relationship

2009
Capsaicin- and mustard oil-induced extracellular signal-regulated protein kinase phosphorylation in sensory neurons in vivo: effects of neurokinins 1 and 2 receptor antagonists and of a nitric oxide synthase inhibitor.
    Basic & clinical pharmacology & toxicology, 2009, Volume: 104, Issue:1

    Topics: Animals; Ankyrins; Benzamides; Calcium Channels; Capsaicin; Extracellular Signal-Regulated MAP Kinases; Ganglia, Spinal; Male; Mustard Plant; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phosphorylation; Piperidines; Plant Oils; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Sciatic Nerve; Sensory Receptor Cells; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2009
Behavioral effects of a synthetic agonist selective for nociceptin/orphanin FQ peptide receptors in monkeys.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:9

    Topics: Alfentanil; Analgesics, Opioid; Animals; Behavior, Animal; Benzimidazoles; Capsaicin; Central Nervous System Agents; Dose-Response Relationship, Drug; Female; Hot Temperature; Imidazoles; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Pain; Piperidines; Pruritus; Receptors, Opioid; Receptors, Opioid, mu; Reinforcement, Psychology; Respiratory Insufficiency; Spiro Compounds

2009
Bronchoconstriction induced by hyperventilation with humidified hot air: role of TRPV1-expressing airway afferents.
    Journal of applied physiology (Bethesda, Md. : 1985), 2009, Volume: 106, Issue:6

    Topics: Airway Resistance; Animals; Atropine; Benzamides; Bronchoconstriction; Bronchodilator Agents; Capsaicin; Disease Models, Animal; Drug Combinations; Ethanolamines; Formoterol Fumarate; Guinea Pigs; Hot Temperature; Humidity; Hyperthermia, Induced; Hyperventilation; Male; Neurons, Afferent; Piperidines; Receptors, Tachykinin; Specific Pathogen-Free Organisms; TRPV Cation Channels; Tryptophan

2009
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Capsaicin; Efferent Pathways; Endocannabinoids; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Pyridazines; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Tetrodotoxin; Vagus Nerve

2009
Pharmacological and metabolic characterisation of the potent sigma1 receptor ligand 1'-benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,4'-piperidine].
    The Journal of pharmacy and pharmacology, 2009, Volume: 61, Issue:5

    Topics: Analgesics; Animals; Capsaicin; Chromatography, High Pressure Liquid; Humans; Ligands; Mice; Microsomes, Liver; Pain; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Sigma-1 Receptor

2009
Role of ET(A) and ET(B) endothelin receptors on endothelin-1-induced potentiation of nociceptive and thermal hyperalgesic responses evoked by capsaicin in rats.
    Neuroscience letters, 2009, Jul-03, Volume: 457, Issue:3

    Topics: Analysis of Variance; Animals; Capsaicin; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Hindlimb; Hyperalgesia; Male; Oligopeptides; Pain Measurement; Peptides, Cyclic; Physical Stimulation; Piperidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Sensory System Agents; Temperature; TRPV Cation Channels

2009
Cannabinoid CB(1) receptor activation stimulates neurite outgrowth and inhibits capsaicin-induced Ca(2+) influx in an in vitro model of diabetic neuropathy.
    Neuropharmacology, 2009, Volume: 57, Issue:2

    Topics: Animals; Calcium; Capsaicin; Diabetic Neuropathies; Dose-Response Relationship, Drug; Dronabinol; Glucose; Hyperglycemia; Indoles; Nerve Growth Factor; Neurites; Neurogenesis; Neurons; Neuroprotective Agents; PC12 Cells; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; RNA, Messenger; Sensory System Agents

2009
Spice active principles as the inhibitors of human platelet aggregation and thromboxane biosynthesis.
    Prostaglandins, leukotrienes, and essential fatty acids, 2009, Volume: 81, Issue:1

    Topics: Acrolein; Adenosine Diphosphate; Alkaloids; Allyl Compounds; Arachidonic Acid; Benzodioxoles; Calcimycin; Capsaicin; Collagen Type III; Curcumin; Eugenol; Humans; Malondialdehyde; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Polyunsaturated Alkamides; Quercetin; Spices; Sulfides; Thromboxanes

2009
N-arachidonyl dopamine sensitizes rat capsaicin-sensitive lung vagal afferents via activation of TRPV1 receptors.
    Respiratory physiology & neurobiology, 2009, Jul-31, Volume: 167, Issue:3

    Topics: Adenosine; Animals; Arachidonic Acids; Capsaicin; Dopamine; Hemodynamics; Male; Nerve Fibers; Neurons, Afferent; Physical Stimulation; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Respiration, Artificial; Respiratory Mechanics; TRPV Cation Channels; Vagus Nerve

2009
Altered responses of dopamine D3 receptor null mice to excitotoxic or anxiogenic stimuli: Possible involvement of the endocannabinoid and endovanilloid systems.
    Neurobiology of disease, 2009, Volume: 36, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Anxiety; Arachidonic Acids; Brain; Cannabinoid Receptor Modulators; Capsaicin; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Epilepsy; GABA Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Picrotoxin; Piperidines; Pyrazoles; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Dopamine D3; Serotonin; TRPV Cation Channels

2009
Parathyroid hormone 2 receptor is a functional marker of nociceptive myelinated fibers responsible for neuropathic pain.
    Journal of neurochemistry, 2010, Volume: 112, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Behavior, Animal; Capsaicin; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Gene Expression Regulation; Glutamic Acid; Male; Mice; Mice, Inbred C57BL; Nerve Fibers, Myelinated; Neurons; Neuropeptides; Pain; Pain Measurement; Piperidines; Receptor, Parathyroid Hormone, Type 2; Reflex; Sciatica; Signal Transduction; Time Factors; TRPV Cation Channels

2010
Effects of neurokinin-1 receptor agonism and antagonism in the rostral ventromedial medulla of rats with acute or persistent inflammatory nociception.
    Neuroscience, 2010, Feb-03, Volume: 165, Issue:3

    Topics: Animals; Capsaicin; Central Nervous System Agents; Freund's Adjuvant; Hot Temperature; Male; Medulla Oblongata; Mustard Plant; Neurokinin-1 Receptor Antagonists; Pain; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Plant Oils; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Time Factors

2010
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: Acrylamides; Administration, Oral; Alkaloids; Anilides; Animals; Avoidance Learning; Benzodioxoles; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazines; Pyridines; Taste; TRPM Cation Channels; TRPV Cation Channels

2010
Long-lasting antinociceptive spinal effects in primates of the novel nociceptin/orphanin FQ receptor agonist UFP-112.
    Pain, 2010, Volume: 148, Issue:1

    Topics: Analgesics; Animals; Benzimidazoles; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Hyperalgesia; Injections, Spinal; Macaca mulatta; Male; Morphine; Naltrexone; Nociceptin; Opioid Peptides; Pain Measurement; Pain Threshold; Piperidines

2010
Cannabinoid CB1 receptor facilitation of substance P release in the rat spinal cord, measured as neurokinin 1 receptor internalization.
    The European journal of neuroscience, 2010, Volume: 31, Issue:2

    Topics: Animals; Capsaicin; Electric Stimulation; GABA-B Receptor Antagonists; Injections, Spinal; Male; Morpholines; Neurons; Pain; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neurokinin-1; Receptors, Opioid, mu; Sensory System Agents; Spinal Cord; Spinal Nerve Roots; Substance P; TRPV Cation Channels

2010
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: Analysis of Variance; Angiotensin II; Anilides; Animals; Capsaicin; Chelating Agents; Cinnamates; Diuretics, Osmotic; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; In Vitro Techniques; Male; Mannitol; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Piperidines; Pyrazines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Supraoptic Nucleus; TRPV Cation Channels; Vasoconstrictor Agents

2010
Opposing effects of cannabinoids and vanilloids on evoked quantal release at the frog neuromuscular junction.
    Neuroscience letters, 2010, Apr-05, Volume: 473, Issue:2

    Topics: Acetylcholine; Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Morpholines; Naphthalenes; Neuromuscular Junction; Piperidines; Pyrazoles; Rana catesbeiana; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2010
Beneficial influence of dietary spices on the ultrastructure and fluidity of the intestinal brush border in rats.
    The British journal of nutrition, 2010, Volume: 104, Issue:1

    Topics: Alkaloids; Animals; Benzodioxoles; Biological Availability; Capsaicin; Capsicum; Cell Membrane; Cholesterol; Diet; Enterocytes; Enzymes; Gastrointestinal Agents; Hydrophobic and Hydrophilic Interactions; Intestinal Absorption; Intestinal Mucosa; Intestine, Small; Lipid Metabolism; Magnoliopsida; Male; Membrane Fluidity; Microscopy, Electron, Scanning; Microvilli; Phospholipids; Piper nigrum; Piperidines; Plant Preparations; Polyunsaturated Alkamides; Protein Conformation; Rats; Rats, Wistar; Spices; Zingiber officinale

2010
In vitro TRPV1 activity of piperine derived amides.
    Bioorganic & medicinal chemistry, 2010, May-01, Volume: 18, Issue:9

    Topics: Alkaloids; Amides; Benzodioxoles; Capsaicin; Cell Line; Dose-Response Relationship, Drug; Humans; Molecular Structure; Piperidines; Polyunsaturated Alkamides; Spectrometry, Fluorescence; TRPV Cation Channels

2010
Gastrointestinal protective effect of dietary spices during ethanol-induced oxidant stress in experimental rats.
    Applied physiology, nutrition, and metabolism = Physiologie appliquee, nutrition et metabolisme, 2010, Volume: 35, Issue:2

    Topics: Alkaloids; Animals; Antioxidants; Benzodioxoles; Capsaicin; Capsicum; Catalase; Cytoprotection; Diet; Disease Models, Animal; Ethanol; Gastric Mucosa; Gastrointestinal Agents; Gastrointestinal Diseases; Glutathione Reductase; Glutathione Transferase; Glycoproteins; Intestinal Mucosa; Male; Mucus; Oxidative Stress; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Spices; Superoxide Dismutase; Zingiber officinale

2010
Inhibitors of monoacylglycerol lipase, fatty-acid amide hydrolase and endocannabinoid transport differentially suppress capsaicin-induced behavioral sensitization through peripheral endocannabinoid mechanisms.
    Pharmacological research, 2010, Volume: 62, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzodioxoles; Biological Transport; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Endocannabinoids; Male; Monoacylglycerol Lipases; Piperidines; Rats; Rats, Sprague-Dawley; Sensory System Agents

2010
Effect of intraperitoneal injection of curcumin on food intake in a goldfish model.
    Journal of molecular neuroscience : MN, 2011, Volume: 45, Issue:2

    Topics: Alkaloids; Animals; Appetite Depressants; Appetite Regulation; Benzodioxoles; Capsaicin; Corticotropin-Releasing Hormone; Curcumin; Eating; Enzyme Inhibitors; Feeding Behavior; Goldfish; Hormone Antagonists; Humans; Injections, Intraperitoneal; Molecular Structure; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Receptors, Corticotropin-Releasing Hormone; Sensory System Agents; Triterpenes; Ursolic Acid

2011
Tissue distribution & elimination of capsaicin, piperine & curcumin following oral intake in rats.
    The Indian journal of medical research, 2010, Volume: 131

    Topics: Administration, Oral; Alkaloids; Animals; Benzodioxoles; Biological Availability; Capsaicin; Chromatography, High Pressure Liquid; Curcumin; Male; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Spectrophotometry, Ultraviolet; Tissue Distribution

2010
Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicity.
    European journal of pharmacology, 2010, Sep-01, Volume: 641, Issue:2-3

    Topics: Action Potentials; Alkaloids; Animals; Benzodioxoles; Capsaicin; Diterpenes; Ganglia, Spinal; Kinetics; Lipid Metabolism; Male; Neurons, Afferent; Pain; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Sensory Receptor Cells; Solubility; TRPV Cation Channels; Urea

2010
Protective effect of lafutidine, a histamine H2 receptor antagonist, against loxoprofen-induced small intestinal lesions in rats.
    Journal of gastroenterology and hepatology, 2010, Volume: 25 Suppl 1

    Topics: 16,16-Dimethylprostaglandin E2; Acetamides; Ampicillin; Animals; Anti-Bacterial Agents; Anti-Ulcer Agents; Capsaicin; Cimetidine; Disease Models, Animal; Enterobacteriaceae; Famotidine; Histamine H2 Antagonists; Intestinal Mucosa; Intestine, Small; Male; Mucin-2; Nitric Oxide Synthase Type II; Omeprazole; Peptic Ulcer; Peroxidase; Phenylpropionates; Piperidines; Proton Pump Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sensory Receptor Cells

2010
Vasorelaxation to N-oleoylethanolamine in rat isolated arteries: mechanisms of action and modulation via cyclooxygenase activity.
    British journal of pharmacology, 2010, Volume: 160, Issue:3

    Topics: Animals; Aorta, Thoracic; Arachidonic Acids; Caffeine; Capsaicin; Chloride Channels; Endocannabinoids; Endothelium, Vascular; Ethanolamines; In Vitro Techniques; Indomethacin; Male; Mesenteric Arteries; Nitric Oxide; Oleic Acids; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Sensory Receptor Cells; Vasodilation

2010
Epidermal growth factor receptor transactivation by the cannabinoid receptor (CB1) and transient receptor potential vanilloid 1 (TRPV1) induces differential responses in corneal epithelial cells.
    Experimental eye research, 2010, Volume: 91, Issue:3

    Topics: Benzoxazines; Blotting, Western; Capsaicin; Cell Movement; Cell Proliferation; Cells, Cultured; Enzyme-Linked Immunosorbent Assay; Epithelium, Corneal; ErbB Receptors; Fluorescent Antibody Technique, Indirect; Humans; Interleukin-6; Interleukin-8; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase 8; Mitogen-Activated Protein Kinase 9; Morpholines; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Piperidines; Pyrazoles; Quinazolines; Receptor, Cannabinoid, CB1; Transcriptional Activation; TRPV Cation Channels; Tyrphostins

2010
Lafutidine, a protective H₂ receptor antagonist, enhances mucosal defense in rat esophagus.
    Digestive diseases and sciences, 2010, Volume: 55, Issue:11

    Topics: Acetamides; Animals; Capsaicin; Esophagus; Histamine H2 Antagonists; Laser-Doppler Flowmetry; Male; Mucous Membrane; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Regional Blood Flow

2010
Propionate-induced epithelial K(+) and Cl(-)/HCO3(-) secretion and free fatty acid receptor 2 (FFA2, GPR43) expression in the guinea pig distal colon.
    Pflugers Archiv : European journal of physiology, 2011, Volume: 461, Issue:1

    Topics: Animals; Atropine; Bicarbonates; Bumetanide; Capsaicin; Chlorides; Colon; Dioxanes; Enteroendocrine Cells; Fatty Acids, Nonesterified; Granisetron; Guinea Pigs; Hexamethonium; Intestinal Mucosa; Male; omega-Conotoxin GVIA; Piperidines; Potassium; Propionates; Pyridoxal Phosphate; Receptors, G-Protein-Coupled; Serous Membrane; Suramin; Tetrodotoxin

2011
Endocannabinoid 2-arachidonoylglycerol protects neurons against β-amyloid insults.
    Neuroscience, 2011, Mar-31, Volume: 178

    Topics: Amyloid beta-Peptides; Animals; Apoptosis; Arachidonic Acids; Benzodioxoles; Biphenyl Compounds; Camphanes; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Capsaicin; Cell Culture Techniques; Drug Interactions; Endocannabinoids; Glycerides; Hippocampus; Monoacylglycerol Lipases; Nerve Degeneration; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Signal Transduction

2011
The hypothermic response to bacterial lipopolysaccharide critically depends on brain CB1, but not CB2 or TRPV1, receptors.
    The Journal of physiology, 2011, May-01, Volume: 589, Issue:Pt 9

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Body Temperature Regulation; Brain; Camphanes; Capsaicin; Disease Models, Animal; Diterpenes; Endocannabinoids; Female; Hypothermia; Injections, Intraperitoneal; Injections, Intravenous; Injections, Intraventricular; Lipopolysaccharides; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Long-Evans; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Signal Transduction; Sulfonamides; Time Factors; TRPV Cation Channels

2011
Triptans attenuate capsaicin-induced CREB phosphorylation within the trigeminal nucleus caudalis: a mechanism to prevent central sensitization?
    The journal of headache and pain, 2011, Volume: 12, Issue:4

    Topics: Animals; Capsaicin; Cyclic AMP Response Element-Binding Protein; Hyperalgesia; Immunohistochemistry; Male; Pain; Phosphorylation; Piperidines; Rats; Rats, Sprague-Dawley; Sensory System Agents; Sumatriptan; Trigeminal Caudal Nucleus; Tryptamines

2011
TRPV1 agonist piperine but not olvanil enhances glutamatergic spontaneous excitatory transmission in rat spinal substantia gelatinosa neurons.
    Biochemical and biophysical research communications, 2011, Jul-15, Volume: 410, Issue:4

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Excitatory Amino Acid Agents; Glutamates; Neurons; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Rats; Substantia Gelatinosa; Synaptic Transmission; TRPV Cation Channels

2011
Differential effects of TRPV1 receptor ligands against nicotine-induced depression-like behaviors.
    BMC pharmacology, 2011, Jul-18, Volume: 11

    Topics: Animals; Antidepressive Agents; Arachidonic Acids; Capsaicin; Depression; Dopamine; Endocannabinoids; Hindlimb Suspension; Ligands; Male; Mice; Mice, Inbred ICR; Nicotine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Stress, Psychological; Swimming; TRPV Cation Channels

2011
Fat digestion and absorption in spice-pretreated rats.
    Journal of the science of food and agriculture, 2012, Volume: 92, Issue:3

    Topics: Adiposity; Alkaloids; Animals; Benzodioxoles; Bile; Bile Acids and Salts; Capsaicin; Curcumin; Diet, High-Fat; Dietary Fats; Digestion; Hydrolases; India; Intestinal Absorption; Lipid Metabolism; Liver; Male; Pancreas; Piperidines; Polyunsaturated Alkamides; Rats, Wistar; Rhizome; Spices; Up-Regulation; Zingiber officinale

2012
Opposing roles for cannabinoid receptor type-1 (CB₁) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:2

    Topics: Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Drug Interactions; Electric Stimulation; Male; Microinjections; Panic; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2012
In vitro and in vivo pharmacological characterisation of the potent and selective vasopressin V(1A) receptor antagonist 4-[4-(4-Chloro-phenyl)-5-[1,2,3]triazol-2-ylmethyl-4H-[1,2,4]triazol-3-yl]-piperidin-1-yl-(3,5-difluoro-phenyl) methanone (PF-00738245)
    European journal of pharmacology, 2011, Nov-30, Volume: 670, Issue:2-3

    Topics: Administration, Oral; Animals; Antidiuretic Hormone Receptor Antagonists; Aorta; Arginine Vasopressin; Blood Circulation; Capsaicin; CHO Cells; Cricetinae; Cricetulus; Dogs; Female; Humans; Male; Models, Biological; Myometrium; Piperidines; Rats; Receptors, Oxytocin; Receptors, Vasopressin; Substrate Specificity; Triazoles

2011
Differential modulation of neurons in the rostral ventromedial medulla by neurokinin-1 receptors.
    Journal of neurophysiology, 2012, Volume: 107, Issue:4

    Topics: Action Potentials; Afferent Pathways; Analysis of Variance; Animals; Capsaicin; Hyperalgesia; Male; Medulla Oblongata; Neurokinin-1 Receptor Antagonists; Neurons; Nociception; Pain Threshold; Patch-Clamp Techniques; Physical Stimulation; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Sensory System Agents

2012
Influence of influenza A infection on capsaicin-induced responses in murine airways.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:2

    Topics: Animals; Biphenyl Compounds; Bronchoalveolar Lavage Fluid; Capsaicin; Carbachol; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Indomethacin; Inflammation; Influenza A virus; Isoproterenol; Leukocytes; Male; Mice; Mice, Inbred BALB C; Models, Biological; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Orthomyxoviridae Infections; Piperidines; Prostaglandin Antagonists; Respiratory Mucosa; Specific Pathogen-Free Organisms; Substance P; Trachea; TRPV Cation Channels; Xanthones

2012
Involvement of perivascular nerves and transient receptor potential vanilloid 1 (TRPV1) in vascular responses to histamine in rat mesenteric resistance arteries.
    European journal of pharmacology, 2012, Apr-05, Volume: 680, Issue:1-3

    Topics: Acetamides; Animals; Benzoquinones; Capsaicin; Endothelium, Vascular; Heptanoic Acids; Histamine; Indomethacin; Male; Mesenteric Arteries; Methoxamine; Piperidines; Procaine; Prostaglandins; Pyridines; Rats; Rats, Wistar; Receptors, Histamine H2; Ruthenium Red; Tetrodotoxin; Thromboxane A2; TRPV Cation Channels; Vasoconstriction; Vasodilation

2012
Endothelium-dependent mechanisms of the vasodilatory effect of the endocannabinoid, anandamide, in the rat pulmonary artery.
    Pharmacological research, 2012, Volume: 66, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amidohydrolases; Animals; Anisoles; Apamin; Arachidonic Acids; Benzamides; Benzyl Compounds; Cannabinoid Receptor Antagonists; Capsaicin; Carbamates; Charybdotoxin; Cyclohexanes; Endocannabinoids; Endothelium, Vascular; Imidazoles; Indoles; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Chloride; Prostaglandin-Endoperoxide Synthases; Pulmonary Artery; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Epoprostenol; Tetraethylammonium; TRPV Cation Channels; Vasodilation

2012
The endocannabinoid and endovanilloid systems interact in the rat prelimbic medial prefrontal cortex to control anxiety-like behavior.
    Neuropharmacology, 2012, Volume: 63, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Arachidonic Acids; Behavior, Animal; Capsaicin; Endocannabinoids; Male; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2012
Enhanced intestinal uptake of iron, zinc and calcium in rats fed pungent spice principles--piperine, capsaicin and ginger (Zingiber officinale).
    Journal of trace elements in medicine and biology : organ of the Society for Minerals and Trace Elements (GMS), 2013, Volume: 27, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Calcium; Capsaicin; Intestinal Absorption; Intestinal Mucosa; Intestines; Iron; Male; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Wistar; Zinc; Zingiber officinale

2013
Release of CGRP from mouse brainstem slices indicates central inhibitory effect of triptans and kynurenate.
    The journal of headache and pain, 2014, Feb-08, Volume: 15

    Topics: Animals; Brain Stem; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Organ Culture Techniques; Piperidines; Rats, Sprague-Dawley; Tryptamines

2014
Effects of cannabinoid and vanilloid drugs on positive and negative-like symptoms on an animal model of schizophrenia: the SHR strain.
    Schizophrenia research, 2014, Volume: 153, Issue:1-3

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Interpersonal Relations; Male; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Inbred SHR; Rats, Wistar; Rimonabant; Schizophrenia; Schizophrenic Psychology; TRPV Cation Channels

2014
Pharmacodynamics of TRPV1 agonists in a bioassay using human PC-3 cells.
    TheScientificWorldJournal, 2014, Volume: 2014

    Topics: Alkaloids; Apoptosis; Benzodioxoles; Biological Assay; Capsaicin; Cell Line, Tumor; Cell Survival; Humans; Male; Metabolic Clearance Rate; Piperidines; Polyunsaturated Alkamides; Prostatic Neoplasms; TRPV Cation Channels

2014
Cannabinoid 1 and transient receptor potential vanilloid 1 receptors discretely modulate evoked glutamate separately from spontaneous glutamate transmission.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Jun-11, Volume: 34, Issue:24

    Topics: Action Potentials; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Capsaicin; Dopamine; Excitatory Postsynaptic Potentials; Glutamic Acid; Hot Temperature; In Vitro Techniques; Male; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission; TRPV Cation Channels

2014
Z944: a first in class T-type calcium channel modulator for the treatment of pain.
    Journal of the peripheral nervous system : JPNS, 2014, Volume: 19 Suppl 2

    Topics: Acetamides; Administration, Oral; Benzamides; Calcium Channel Blockers; Capsaicin; Clinical Trials, Phase I as Topic; Dose-Response Relationship, Drug; Evoked Potentials, Somatosensory; Humans; Lasers; Male; Pain; Piperidines; Time Factors

2014
Anxiogenic-like effects induced by hemopressin in rats.
    Pharmacology, biochemistry, and behavior, 2015, Volume: 129

    Topics: Anilides; Animals; Anxiety; Brain; Capsaicin; Cinnamates; Hemoglobins; Injections, Intraventricular; Male; Maze Learning; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Wistar

2015
A multi-target approach for pain treatment: dual inhibition of fatty acid amide hydrolase and TRPV1 in a rat model of osteoarthritis.
    Pain, 2015, Volume: 156, Issue:5

    Topics: Activating Transcription Factor 3; Amidohydrolases; Anilides; Animals; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Cinnamates; Disease Models, Animal; Endocannabinoids; Ganglia, Spinal; Gene Expression; Hyperalgesia; Inflammation; Interleukin-6; Lumbar Vertebrae; Male; Osteoarthritis; Pain; Pain Management; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2015
Contribution of sensory nerves to LPS-induced hyperresponsiveness of human isolated bronchi.
    Life sciences, 2015, Jun-15, Volume: 131

    Topics: Anilides; Bronchi; Bronchial Hyperreactivity; Capsaicin; Cinnamates; Electric Stimulation; Female; Humans; Indoles; Lipopolysaccharides; Male; Middle Aged; Muscle Contraction; Neprilysin; Neurokinin A; Piperidines; Sensory Receptor Cells; TRPV Cation Channels; Up-Regulation

2015
Peripheral neurokinin-1 receptors contribute to kaolin-induced acute monoarthritis in rats.
    Neuroimmunomodulation, 2015, Volume: 22, Issue:6

    Topics: Animals; Animals, Newborn; Antidiarrheals; Arthritis; Capsaicin; Cytokines; Disease Models, Animal; Edema; Enzyme Inhibitors; Hyperalgesia; Indomethacin; Kaolin; Knee Joint; Male; Pain Measurement; Peroxidase; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Synovial Fluid

2015
Anti-Inflammatory Effects of Capsaicin and Piperine on Helicobacter pylori-Induced Chronic Gastritis in Mongolian Gerbils.
    Helicobacter, 2016, Volume: 21, Issue:2

    Topics: Alkaloids; Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents; Benzodioxoles; Capsaicin; Chemoprevention; Colony Count, Microbial; Diet Therapy; Gastritis; Gerbillinae; Helicobacter Infections; Helicobacter pylori; Male; Piperidines; Polyunsaturated Alkamides; Real-Time Polymerase Chain Reaction; Sequence Analysis, DNA; Stomach

2016
High-Concentration Piperine: Capsaicin-Sensitive and -Insensitive Effects on Isolated Organs.
    Pharmacology, 2015, Volume: 96, Issue:1-2

    Topics: Acetanilides; Alkaloids; Animals; Benzodioxoles; Capsaicin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Nifedipine; Piperidines; Polyunsaturated Alkamides; Purines; Pyrazines; Pyridines; Trachea; TRPV Cation Channels; Urinary Bladder

2015
Sensory nerves contribute to cutaneous vasodilator response to cathodal stimulation in healthy rats.
    Microvascular research, 2015, Volume: 101

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Electrodes; Electrophysiology; Hydrogen-Ion Concentration; Laser-Doppler Flowmetry; Male; Microcirculation; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory Receptor Cells; Skin; Substance P; TRPV Cation Channels; Vasodilation; Vasodilator Agents

2015
Dorsolateral periaqueductal gray matter CB1 and TRPV1 receptors exert opposite modulation on expression of contextual fear conditioning.
    Neuropharmacology, 2016, Volume: 103

    Topics: Animals; Capsaicin; Conditioning, Classical; Fear; Male; Nitric Oxide; Nitric Oxide Synthase Type I; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Soluble Guanylyl Cyclase; TRPV Cation Channels

2016
Differential bitterness in capsaicin, piperine, and ethanol associates with polymorphisms in multiple bitter taste receptor genes.
    Physiology & behavior, 2016, Mar-15, Volume: 156

    Topics: Adult; Alkaloids; Benzodioxoles; Capsaicin; Ethanol; Female; Genetic Variation; Genotype; Humans; Male; Piperidines; Polymorphism, Single Nucleotide; Polyunsaturated Alkamides; Receptors, G-Protein-Coupled; Taste; Tongue

2016
TRPV1 and PLC Participate in Histamine H4 Receptor-Induced Itch.
    Neural plasticity, 2016, Volume: 2016

    Topics: Acetanilides; Acrylamides; Animals; Antipruritics; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Capsaicin; Dose-Response Relationship, Drug; Ganglia, Spinal; Histamine Agonists; Imidazoles; Mice; Neurons; Piperidines; Pruritus; Purines; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; TRPV Cation Channels; Type C Phospholipases

2016
Involvement of TRPV1 in the Olfactory Bulb in Rimonabant-Induced Olfactory Discrimination Deficit.
    The Chinese journal of physiology, 2016, 02-29, Volume: 59, Issue:1

    Topics: Animals; Capsaicin; Male; Mice; Mice, Inbred C57BL; Motor Activity; Olfactory Bulb; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Smell; TRPV Cation Channels

2016
Capsaicin-Induced Death of Human Haematological Malignant Cell Lines Is Independent of TRPV1 Activation.
    Pharmacology, 2016, Volume: 98, Issue:1-2

    Topics: Cannabinoid Receptor Antagonists; Capsaicin; Cell Death; Cell Line, Tumor; Hematologic Neoplasms; Humans; Indoles; Oxazines; Piperidines; Pyrazoles; TRPV Cation Channels; Xanthenes

2016
A pro-nociceptive phenotype unmasked in mice lacking fatty-acid amide hydrolase.
    Molecular pain, 2016, Volume: 12

    Topics: Acrylamides; Amidohydrolases; Analgesia; Animals; Arachidonic Acid; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Carrageenan; Disease Models, Animal; Ethanolamines; Formaldehyde; Genotype; Hyperalgesia; Inflammation; Injections, Intraperitoneal; Ligands; Lumbar Vertebrae; Mice, Inbred C57BL; Mice, Knockout; Nociception; Pain; Pain Threshold; Phenotype; Piperidines; Proto-Oncogene Proteins c-fos; Pyrazoles; Receptor, Cannabinoid, CB1; Skin; Spinal Cord Dorsal Horn; TRPV Cation Channels

2016
Inhibition of interleukin-1β-induced endothelial tissue factor expression by the synthetic cannabinoid WIN 55,212-2.
    Oncotarget, 2016, 09-20, Volume: 7, Issue:38

    Topics: Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cannabinoids; Capsaicin; Cells, Cultured; Ceramides; Human Umbilical Vein Endothelial Cells; Humans; Indoles; Interleukin-1beta; JNK Mitogen-Activated Protein Kinases; Monocytes; Morpholines; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Partial Thromboplastin Time; Phosphorylation; Piperidines; Pyrazoles; RNA, Messenger; Signal Transduction; Sphingomyelin Phosphodiesterase; Thromboplastin; TRPV Cation Channels

2016
Curcumin, Piperine, and Capsaicin: A Comparative Study of Spice-Mediated Inhibition of Human Cytochrome P450 Isozyme Activities.
    Drug metabolism and disposition: the biological fate of chemicals, 2017, Volume: 45, Issue:1

    Topics: Alkaloids; Benzodioxoles; Capsaicin; Curcumin; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Humans; Molecular Structure; Piperidines; Polyunsaturated Alkamides; Recombinant Proteins; Spices

2017
Consistent sex-dependent effects of PKMζ gene ablation and pharmacological inhibition on the maintenance of referred pain.
    Molecular pain, 2016, Volume: 12

    Topics: Animals; Capsaicin; Cell-Penetrating Peptides; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Freund's Adjuvant; Inflammation; Lipopeptides; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neuralgia; Pain Threshold; Piperidines; Protein Kinase C; Rats; Rats, Long-Evans; Sex Characteristics; Spinal Cord

2016
Enhanced ability of TRPV1 channels in regulating glutamatergic transmission after repeated morphine exposure in the nucleus accumbens of rat.
    Brain research, 2017, 04-01, Volume: 1660

    Topics: Animals; Capsaicin; Corpus Striatum; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Morphine; Narcotics; Neuronal Plasticity; Neurotransmitter Agents; Nucleus Accumbens; Piperidines; Presynaptic Terminals; Pyrazoles; Random Allocation; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Substance Withdrawal Syndrome; Synaptic Transmission; Tissue Culture Techniques; TRPV Cation Channels

2017
Hyperalgesia and sensitization of dorsal horn neurons following activation of NK-1 receptors in the rostral ventromedial medulla.
    Journal of neurophysiology, 2017, 11-01, Volume: 118, Issue:5

    Topics: Animals; Capsaicin; Catheters, Indwelling; Central Nervous System Sensitization; Hot Temperature; Hyperalgesia; Immunohistochemistry; Male; Medulla Oblongata; Microelectrodes; Neurokinin-1 Receptor Antagonists; Piperidines; Posterior Horn Cells; Proto-Oncogene Proteins c-fos; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Touch

2017
Do TRPV1 antagonists increase the risk for skin tumourigenesis? A collaborative in vitro and in vivo assessment.
    Cell biology and toxicology, 2018, Volume: 34, Issue:2

    Topics: Acrylamides; Animals; Anthracenes; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line; Cell Proliferation; Cell Survival; Cocarcinogenesis; Female; Humans; Keratinocytes; Mice; Mice, Hairless; Piperidines; Primary Cell Culture; Pyridines; Pyrrolidines; Risk; Skin Neoplasms; TRPV Cation Channels; Urea

2018
Cannabinoids induce apathetic and impulsive patterns of choice through CB1 receptors and TRPV1 channels.
    Neuropharmacology, 2018, 05-01, Volume: 133

    Topics: Animals; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Cerebral Cortex; Choice Behavior; Dose-Response Relationship, Drug; Impulsive Behavior; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2018
Effects of Phytochemical P-Glycoprotein Modulators on the Pharmacokinetics and Tissue Distribution of Doxorubicin in Mice.
    Molecules (Basel, Switzerland), 2018, Feb-07, Volume: 23, Issue:2

    Topics: Alkaloids; Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzodioxoles; Biological Transport; Capsaicin; Catechols; Doxorubicin; Fatty Alcohols; Mice; Phytochemicals; Piperidines; Polyunsaturated Alkamides; Tissue Distribution

2018
Capsaicin and Piperine Can Overcome Multidrug Resistance in Cancer Cells to Doxorubicin.
    Molecules (Basel, Switzerland), 2018, Mar-02, Volume: 23, Issue:3

    Topics: Alkaloids; Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzodioxoles; Biological Transport; Caco-2 Cells; Capsaicin; Capsicum; Cell Line, Tumor; Doxorubicin; Drug Combinations; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Fluoresceins; Gene Expression; HCT116 Cells; Humans; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Rhodamine 123

2018
Sinergism between alkaloids piperine and capsaicin with meglumine antimoniate against Leishmania infantum.
    Experimental parasitology, 2018, Volume: 188

    Topics: Alkaloids; Antiprotozoal Agents; Benzodioxoles; Capsaicin; Chromatography, High Pressure Liquid; Drug Synergism; Inhibitory Concentration 50; Leishmania infantum; Leishmaniasis, Visceral; Magnetic Resonance Spectroscopy; Meglumine; Meglumine Antimoniate; Organometallic Compounds; Piperidines; Polyunsaturated Alkamides; Spectrophotometry, Ultraviolet

2018
New
    Scientific reports, 2018, 07-03, Volume: 8, Issue:1

    Topics: Analgesics; Animals; Behavior, Animal; Capsaicin; Coffee; Disease Models, Animal; Female; Formaldehyde; Glutamic Acid; Hot Temperature; Hyperalgesia; Male; Mice; Naloxone; Narcotic Antagonists; Ondansetron; Pain; Pain Measurement; Piperidines; Pyrazoles; Serotonin

2018
TRPV1 mediates the anticonvulsant effects of acetaminophen in mice.
    Epilepsy research, 2018, Volume: 145

    Topics: Acetaminophen; Acetanilides; Acrylamides; Animals; Anticonvulsants; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Pentylenetetrazole; Piperidines; Purines; Pyrazoles; Seizures; Time Factors; TRPV Cation Channels

2018
Cannabidiol modulates serotonergic transmission and reverses both allodynia and anxiety-like behavior in a model of neuropathic pain.
    Pain, 2019, Volume: 160, Issue:1

    Topics: Action Potentials; Animals; Anxiety; Cannabidiol; Capsaicin; Disease Models, Animal; Exploratory Behavior; Feeding Behavior; Ganglia, Spinal; Hyperalgesia; Lysergic Acid Diethylamide; Male; Maze Learning; Neuralgia; Piperazines; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Swimming

2019
Virtual screening of natural anti-filarial compounds against glutathione-S-transferase of Brugia malayi and Wuchereria bancrofti.
    Cellular and molecular biology (Noisy-le-Grand, France), 2018, Oct-30, Volume: 64, Issue:13

    Topics: Alkaloids; Animals; Anthelmintics; Benzodioxoles; Biological Products; Brugia malayi; Capsaicin; Catalytic Domain; Curcumin; Drug Evaluation, Preclinical; Glutathione Transferase; Molecular Docking Simulation; Piperidines; Polyunsaturated Alkamides; Strychnine; Wuchereria bancrofti

2018
A distinct structural mechanism underlies TRPV1 activation by piperine.
    Biochemical and biophysical research communications, 2019, 08-20, Volume: 516, Issue:2

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Hydrogen Bonding; Ion Channel Gating; Mice; Mutation; Piperidines; Polyunsaturated Alkamides; Structure-Activity Relationship; TRPV Cation Channels

2019
Capsaicin and Piperine as Functional Excipients for Improved Drug Delivery across Nasal Epithelial Models.
    Planta medica, 2019, Volume: 85, Issue:13

    Topics: Alkaloids; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzodioxoles; Capsaicin; Drug Delivery Systems; Nasal Mucosa; Pharmaceutical Vehicles; Piperidines; Polyunsaturated Alkamides; Sheep

2019
Cannabidiol increases the nociceptive threshold in a preclinical model of Parkinson's disease.
    Neuropharmacology, 2020, Volume: 163

    Topics: Amidohydrolases; Analgesics; Animals; Benzamides; Brain; Cannabidiol; Capsaicin; Carbamates; Celecoxib; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Nociception; Oxidopamine; Pain; Parkinson Disease; Piperidines; Pyrazoles; Thienamycins

2020
Comparative immunohistological study on using capsaicin, piperine, and okadaic acid for the transepithelial passage of the inactivated viral and bacterial vaccines in fish.
    Microscopy research and technique, 2020, Volume: 83, Issue:8

    Topics: Adjuvants, Immunologic; Administration, Oral; Alkaloids; Animals; Bacterial Vaccines; Benzodioxoles; Biological Transport; Capsaicin; Fish Diseases; Okadaic Acid; Piperidines; Polyunsaturated Alkamides; Sea Bream; Viral Vaccines

2020
Inhibitory effect of
    Journal of environmental science and health. Part. B, Pesticides, food contaminants, and agricultural wastes, 2020, Volume: 55, Issue:9

    Topics: Aflatoxins; Alkaloids; Antifungal Agents; Aspergillus; Benzodioxoles; Biosynthetic Pathways; Capsaicin; Capsicum; DNA-Binding Proteins; Fruit; Fungal Proteins; Gene Expression Regulation, Fungal; Genes, Fungal; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Transcription Factors

2020
Functional Crosstalk between CB and TRPV1 Receptors Protects Nigrostriatal Dopaminergic Neurons in the MPTP Model of Parkinson's Disease.
    Journal of immunology research, 2020, Volume: 2020

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Capsaicin; Disease Models, Animal; Dopaminergic Neurons; Humans; Indoles; Mice; Mice, Inbred C57BL; Neurogenic Inflammation; Neuroglia; Neuroprotection; Parkinson Disease; Piperidines; Pyrazoles; Receptor Cross-Talk; Receptors, Cannabinoid; Substantia Nigra; TRPV Cation Channels

2020
Inhibitory effect of intrathecally administered AM404, an endocannabinoid reuptake inhibitor, on neuropathic pain in a rat chronic constriction injury model.
    Pharmacological reports : PR, 2021, Volume: 73, Issue:3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Disease Models, Animal; Endocannabinoids; Hyperalgesia; Indoles; Male; Neuralgia; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rotarod Performance Test; Spinal Cord; TRPV Cation Channels

2021
Cytogenotoxicity and protective effect of piperine and capsaicin on meristematic cells of Allium cepa L.
    Anais da Academia Brasileira de Ciencias, 2021, Volume: 93, Issue:suppl 3

    Topics: Alkaloids; Benzodioxoles; Capsaicin; DNA Damage; Onions; Piperidines; Plant Roots; Polyunsaturated Alkamides

2021
Turmeric, red pepper, and black pepper affect carotenoids solubilized micelles properties and bioaccessibility: Capsaicin/piperine improves and curcumin inhibits carotenoids uptake and transport in Caco-2 cells.
    Journal of food science, 2021, Volume: 86, Issue:11

    Topics: Alkaloids; Benzodioxoles; Biological Availability; Caco-2 Cells; Capsaicin; Capsicum; Carotenoids; Curcuma; Curcumin; Humans; Micelles; Piper nigrum; Piperidines; Polyunsaturated Alkamides

2021
A Comparative Study on the Effect of Acute Pharyngeal Stimulation with TRP Agonists on the Biomechanics and Neurophysiology of Swallow Response in Patients with Oropharyngeal Dysphagia.
    International journal of molecular sciences, 2022, Sep-15, Volume: 23, Issue:18

    Topics: Acrolein; Acyclic Monoterpenes; Alkaloids; Benzodioxoles; Biomechanical Phenomena; Capsaicin; Deglutition; Deglutition Disorders; Humans; Menthol; Piperidines; Polyunsaturated Alkamides; Retrospective Studies; Zinc

2022