capsaicin and oxadiazoles

capsaicin has been researched along with oxadiazoles in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.14)18.7374
1990's2 (14.29)18.2507
2000's8 (57.14)29.6817
2010's1 (7.14)24.3611
2020's2 (14.29)2.80

Authors

AuthorsStudies
Agrawal, SG; Evans, RH1
Arányi, P; Korbonits, D; Mikus, EG; Minker, E; Pascal, M; Révész, J; Saano, V1
Ayata, G; Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ1
Huh, IH; Lee, YW; Park, JI; Shin, CY; Sohn, UD1
Kilbinger, H; Mang, CF1
de Groat, WC; Seki, S; Yoshimura, N1
Gitlin, JM; Mitchell, JA; Stanford, SJ1
Adler-Graschinsky, E; Mendizábal, VE; Orliac, ML1
Ceyhan, BB; Karakurt, S1
Barahona, MV; Benedito, S; García-Sacristán, A; Hernández, M; Martínez, AC; Orensanz, LM; Prieto, D; Recio, P; Rivera, L1
Capra, NF; Lee, J; Ro, JY; Zhang, Y1
Altamirano-Espinoza, AH; González-Hernández, A; MaassenVanDenBrink, A; Manrique-Maldonado, G; Marichal-Cancino, BA; Ruiz-Salinas, II; Villalón, CM1
Pei, FN; Tang, J; Wang, ZC; Wei, B; Yang, CG; Yang, F; Yang, S; Yang, T; Yu, LF1
Ahmad Lone, B; Ahmad, F; Ahmad, N; Ali Khan, I; Ali, I; Grover, A; Khan, A; Kumari, A; Naaz, F; Rajput, VS; Shafi, S1

Trials

1 trial(s) available for capsaicin and oxadiazoles

ArticleYear
Effect of oxolamine on cough sensitivity in COPD patients.
    Respiratory medicine, 2002, Volume: 96, Issue:1

    Topics: Aged; Antitussive Agents; Capsaicin; Cough; Cross-Over Studies; Female; Humans; Male; Middle Aged; Oxadiazoles; Pilot Projects; Pulmonary Disease, Chronic Obstructive; Respiratory Function Tests; Single-Blind Method

2002

Other Studies

13 other study(ies) available for capsaicin and oxadiazoles

ArticleYear
The primary afferent depolarizing action of kainate in the rat.
    British journal of pharmacology, 1986, Volume: 87, Issue:2

    Topics: Action Potentials; Afferent Pathways; Animals; Aspartic Acid; Capsaicin; Evoked Potentials; gamma-Aminobutyric Acid; Glutamates; In Vitro Techniques; Kainic Acid; Membrane Potentials; N-Methylaspartate; Nerve Fibers; Oxadiazoles; Quisqualic Acid; Rats; Spinal Nerve Roots

1986
Experimental studies on the antitussive properties of the new xanthine derivative 1H-purine-2,6-dione, 3,7-dihydro-3-methyl-7[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]. 1st communication: in vivo demonstration of the effects on animal models of cough and of
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:4

    Topics: Animals; Antitussive Agents; Capsaicin; Citric Acid; Cough; Female; Guinea Pigs; In Vitro Techniques; Male; Mucociliary Clearance; Oxadiazoles; Physical Stimulation; Purines; Rabbits

1997
Effects of PNU-109,291, a selective 5-HT1D receptor agonist, on electrically induced dural plasma extravasation and capsaicin-evoked c-fos immunoreactivity within trigeminal nucleus caudalis.
    Neuropharmacology, 1999, Volume: 38, Issue:7

    Topics: Animals; Benzopyrans; Binding, Competitive; Blood Pressure; Blood Proteins; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; Male; Oxadiazoles; Piperazines; Proto-Oncogene Proteins c-fos; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Trigeminal Nuclei

1999
Endothelium-dependent sensory non-adrenergic non-cholinergic vasodilatation in rat thoracic aorta: involvement of ATP and a role for NO.
    The Journal of pharmacy and pharmacology, 2000, Volume: 52, Issue:4

    Topics: Adenosine Triphosphate; Animals; Aorta, Thoracic; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Endothelium, Vascular; Evans Blue; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxadiazoles; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Serotonin; Tetrodotoxin; Theophylline; Triazines; Vasodilation

2000
Modulation of acetylcholine release in the guinea-pig trachea by the nitric oxide donor, S-nitroso-N-acetyl-DL-penicillamine (SNAP).
    British journal of pharmacology, 2000, Volume: 131, Issue:1

    Topics: Acetylcholine; Animals; Capsaicin; Guinea Pigs; In Vitro Techniques; Male; Nitric Oxide; Nitric Oxide Donors; Nitroarginine; Oxadiazoles; Penicillamine; Quinoxalines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Trachea

2000
Nitric oxide modulates Ca(2+) channels in dorsal root ganglion neurons innervating rat urinary bladder.
    Journal of neurophysiology, 2001, Volume: 86, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, N-Type; Capsaicin; Cyclic GMP; Enzyme Inhibitors; Female; Ganglia, Spinal; Nerve Fibers; Nerve Fibers, Myelinated; Neurons, Afferent; Nimodipine; Nitric Oxide; Nitric Oxide Donors; omega-Conotoxin GVIA; Oxadiazoles; Penicillamine; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Urinary Bladder

2001
Identification of two distinct vasodilator pathways activated by ATP in the mesenteric bed of the rat.
    British journal of pharmacology, 2001, Volume: 133, Issue:6

    Topics: Adenine; Adenosine; Adenosine Triphosphate; Animals; Arachidonic Acids; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Histamine; In Vitro Techniques; Male; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Oxadiazoles; Piperidines; Polyunsaturated Alkamides; Potassium Chloride; Pyrazoles; Pyrilamine; Quinoxalines; Rats; Rats, Wistar; Rimonabant; Signal Transduction; Stereoisomerism; Theophylline; Vasodilation

2001
Long-term inhibition of nitric oxide synthase potentiates effects of anandamide in the rat mesenteric bed.
    European journal of pharmacology, 2001, Sep-21, Volume: 427, Issue:3

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Capsaicin; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Norepinephrine; Oxadiazoles; Phenylmethylsulfonyl Fluoride; Polyunsaturated Alkamides; Pyrazoles; Quinoxalines; Rats; Rats, Wistar; Time Factors; Vasoconstriction; Vasoconstrictor Agents

2001
Heterogeneity of neuronal and smooth muscle receptors involved in the VIP- and PACAP-induced relaxations of the pig intravesical ureter.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Apamin; Capsaicin; Charybdotoxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Female; Guanylate Cyclase; Male; Muscle, Smooth; Neurons, Afferent; Neuropeptide Y; Neuropeptides; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; omega-Conotoxin GVIA; Oxadiazoles; Peptide Fragments; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium Channels, Calcium-Activated; Quinoxalines; Receptors, Calcitonin Gene-Related Peptide; Receptors, Peptide; Receptors, Vasoactive Intestinal Peptide; Rolipram; Sensory Receptor Cells; Swine; Tetraethylammonium; Ureter; Vasoactive Intestinal Peptide

2004
Role of soluble guanylate cyclase in the trigeminal subnucleus caudalis in capsaicin-induced muscle hypersensitivity.
    Brain research, 2007, Dec-12, Volume: 1184

    Topics: Analysis of Variance; Animals; Area Under Curve; Behavior, Animal; Capsaicin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guanylate Cyclase; Hyperalgesia; Male; Masseter Muscle; Methylene Blue; Mice; Nerve Tissue Proteins; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Sensory Thresholds; Soluble Guanylyl Cyclase; Time Factors; Trigeminal Caudal Nucleus

2007
Intrathecal dihydroergotamine inhibits capsaicin-induced vasodilatation in the canine external carotid circulation via GR127935- and rauwolscine-sensitive receptors.
    European journal of pharmacology, 2012, Oct-05, Volume: 692, Issue:1-3

    Topics: Acetylcholine; Animals; Blood Circulation; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Arteries; Dihydroergotamine; Dogs; Dose-Response Relationship, Drug; Hemodynamics; Injections, Spinal; Male; Oxadiazoles; Piperazines; Propylene Glycol; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Antagonists; Vasodilation; Vasodilator Agents; Yohimbine

2012
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus.
    European journal of medicinal chemistry, 2020, Jul-15, Volume: 198

    Topics: Anti-Bacterial Agents; Capsaicin; Cell Survival; Drug Design; Drug Resistance, Multiple; HEK293 Cells; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Oxadiazoles; Staphylococcal Infections; Structure-Activity Relationship; Thiophenes; Vancomycin

2020
1,3,4-oxadiazole conjugates of capsaicin as potent NorA efflux pump inhibitors of Staphylococcus aureus.
    Bioorganic chemistry, 2021, Volume: 113

    Topics: Anti-Bacterial Agents; Bacterial Proteins; Binding Sites; Capsaicin; Cell Line, Tumor; Cell Survival; Ciprofloxacin; Drug Resistance, Multiple, Bacterial; Humans; Kinetics; Microbial Sensitivity Tests; Molecular Docking Simulation; Multidrug Resistance-Associated Proteins; Oxadiazoles; Staphylococcus aureus; Structure-Activity Relationship

2021