capsaicin and capsazepine

capsaicin has been researched along with capsazepine in 721 studies

Research

Studies (721)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's80 (11.10)18.2507
2000's352 (48.82)29.6817
2010's266 (36.89)24.3611
2020's23 (3.19)2.80

Authors

AuthorsStudies
Bevan, S; Boelsterli, JJ; Bovermann, G; Breckenridge, R; Davies, JW; Hughes, GA; James, I; Oberer, L; Walpole, CS; Winter, J1
Annunziata, R; Appendino, G; Cravotto, G; Palmisano, G; Szallasi, A1
Blumberg, PM; Choi, HK; Ha, HJ; Kang, M; Kang, SU; Kim, HD; Kim, JM; Kim, YH; Lee, J; Lim, JO; Lundberg, DJ; Oh, U; Park, HG; Park, YH; Pearce, LV; Shin, M; Suh, YG; Toth, A; Tran, R; Wang, Y1
Cho, H; Choi, JY; Choi, SH; Jew, SS; Kang, SU; Kim, HD; Kyu Choi, J; Lee, J; Oh, U; Park, HG; Park, MK; Park, YH; Su Jeong, Y; Suh, YG1
Bogenstaetter, M; Breitenbucher, JG; Carruthers, NI; Chang, L; Chaplan, SR; Codd, EE; Dax, SL; Dubin, AE; Gonzales, L; Hoey, K; Jetter, M; Lee, DH; Liu, C; Lord, B; Mazur, C; Nasser, N; Rizzolio, M; Shah, C; Swanson, DM; Zhang, SP1
Bianchi, BR; El Kouhen, R; Faltynek, CR; Gomtsyan, A; Jarvis, MF; Lee, CH; McDonald, HA; Moreland, RB; Neelands, TR; Puttfarcken, PS; Raja, SN; Surber, B; Surowy, CS; Vaidyanathan, SN1
Correa, EA; Echeverri, F; Högestätt, ED; Sterner, O; Zygmunt, PM1
Horie, S; Takayama, H; Terada, Y; Tominaga, M; Uchida, K; Watanabe, T1
Lou, YP; Lundberg, JM1
Dray, A2
Lee, LY; Lou, YP; Lundberg, JM; Satoh, H1
Barnes, PJ; Belvisi, MG; Miura, M; Stretton, D1
Campbell, EA; Perkins, MN1
Bevan, S; Hothi, S; Hughes, G; James, IF; Rang, HP; Shah, K; Walpole, CS; Yeats, JC1
Franco-Cereceda, A; Lundberg, JM1
Dickenson, AH1
Dray, A; Urban, L1
Dickenson, AH; Dray, A1
Håkanson, R; Wang, ZY1
Kuraishi, Y; Satoh, M; Sugimoto, K; Ueda, M1
Goso, C; Manzini, S; Szallasi, A1
Barnes, PJ; Dray, A; Fox, AJ; Urban, L1
Baker, J; Bertrand, C; Geppetti, P; Nadel, JA; Piedimonte, G; Yamawaki, I1
Bevan, S; Giuliani, S; Maggi, CA; Rang, HP; Walpole, CS1
Bevan, S; Burgess, GM; Cholewinski, A1
Goso, C; Szallasi, A1
Acs, G; Blumberg, PM; Palkovits, M2
Lee, LY; Lundberg, JM1
Kuraishi, Y; Satoh, M; Ueda, M1
Franco-Cereceda, A; Källner, G; Lundberg, JM2
Delay-Goyet, P; Lundberg, JM; Satoh, H1
Bevan, S; Del Bianco, E; Figini, M; Maggi, CA; Santicioli, P1
Blumberg, PM; Goso, C; Manzini, S; Szallasi, A1
Blumberg, PM; Evangelista, S; Goso, C; Manzini, S; Szallasi, A; Tramontana, M1
Ellis, JL; Undem, BJ1
Dray, A; Seno, N1
Lou, YP; Lundberg, JM; Satoh, H1
Barnes, PJ; Belvisi, MG; Chung, KF; Fox, AJ; Lalloo, UG1
Colquhoun, EQ; Eldershaw, TP; Geraghty, DP; Griffiths, CD; Hall, JL1
Furey, G; Sanger, GJ; Wardle, KA1
Hwang, SW; Kim, D; Oh, U1
Szallasi, A1
Hua, XY; Jinno, S; Wong, S; Yaksh, TL1
Blumberg, PM; Hökfelt, T; Lundberg, JM; Nilsson, S; Szallasi, A1
Dale, N; Kuenzi, FM1
Ellis, JL; Sham, JS; Undem, BJ1
Belmonte, C; Chen, X; Rang, HP1
Ohkubo, T; Shibata, M1
Chen, I; Liu, L; Lo, Y; Simon, SA1
Czachurski, J; Seller, H; Zanzinger, J1
Liu, L; Simon, SA2
Chen, P; Hua, XY; Hwang, J; Yaksh, TL1
Arguelles, JH; Baumann, TK; Martenson, ME1
Docherty, RJ; Piper, AS; Yeats, JC1
Kitamura, K; Ohkubo, T1
Calixto, JB; Santos, AR1
Flores, CM; Harding-Rose, C; Hargreaves, KM; Kilo, S1
Knotková-Urbancová, H; Kress, M; Reeh, PW; Vitásková, Z; Vlachová, V; Vyklický, L1
Bowen, WP; Grattan, TJ; Morice, AH; Wright, CE1
Liu, L; Simon, SA; Szallasi, A1
Acs, P; Bíró, T; Blumberg, PM; Brodie, C; Lewin, NE; Modarres, S1
Bast, A; den Hartog, GJ; van Bree, L; van Hoof, HJ; Voss, HP1
Lopshire, JC; Nicol, GD1
Schultz, HD; Ustinova, EE1
Iwata, F; Lam, K; Leung, FW; Leung, JW; Seno, K1
Cho, TS; Jung, YS; Moon, CH; Shin, HS1
Hwang, SW; Jung, JY; Kwak, JY; Lee, WT; Oh, U1
Harrison, S; Page, CP; Reddy, S; Spina, D1
Beltramo, M; Piomelli, D1
Fushiki, T; Inoue, K; Ishihara, K; Kawada, T; Kim, KM1
Fisher, JT; Nault, MA; Vincent, SG1
Lee, SS; Park, YH; Surh, YJ1
Cho, TS; Jung, YS; Lee, B; Lee, SM; Moon, CH; Shin, HS1
Bíró, T; Blumberg, PM; Klusch, A; Krause, JE; Modarres, S; Petersen, M; Sterner, O; Szabó, T; Szallasi, A1
Furue, H; Kumamoto, E; Li, YQ; Yang, K; Yoshimura, M1
Geraghty, DP; Mazzone, SB1
Averbeck, B; Bove, GM; Reeh, PW; Sauer, SK1
Andersson, DA; Chuang, H; Di Marzo, V; Högestätt, ED; Julius, D; Petersson, J; Sørgård, M; Zygmunt, PM1
Akiba, Y; Engel, E; Guth, PH; Kaunitz, JD; Nastaskin, I1
Annicelli, LL; Blumberg, PM; Cortright, DN; Krause, JE; Szallasi, A1
Nagy, I; Rang, HP1
Büsselberg, D; Greffrath, W; Kirschstein, T; Treede, RD1
Mustafa, S; Oriowo, MA1
Clothier, RH; Downing, AT; Fry, JR; Garle, MJ; Jassi, KL; Knight, A1
Auberson, S; Lacroix, JS; Lundberg, JM1
Jerman, JC; Smart, D1
Distler, C; Habelt, C; Kessler, F; Kress, M; Reeh, PW1
Carratú, MR; Cochereau, C; Creppy, EE; Cuomo, V; Ennamany, R; Richeux, F; Saboureau, D1
Cho, H; Cho, S; Hwang, SW; Jung, J; Kang, CJ; Kim, D; Kwak, J; Lee, SY; Min, KH; Oh, U; Suh, YG1
Davis, JB; Gunthorpe, MJ; Harries, MH; Prinjha, RK; Randall, A1
Averbeck, B; Izydorczyk, I; Kress, M1
Brough, SJ; Davis, JB; Harries, MH; Jerman, JC; Prinjha, R; Smart, D1
Antunes, E; Costa, SK; da Silva, GR; Linardi, A1
Klusch, A; Marín-Burgin, A; Petersen, M; Reppenhagen, S; Wendland, JR1
Kim, JA; Lee, YS; Nam, DH1
Colquhoun, EQ; Geraghty, DP; Griffiths, CD; Szallasi, A; Vincent, MA1
Buchheit, KH; Campbell, EA; Chaudhry, N; James, IF; Kane, S; Panesar, M; Patel, S; Sandells, B; Urban, L1
Bielefeldt, K1
Bowles, WR; Engeland, WC; Guo, A; Harding-Rose, CA; Ulrich-Lai, YM1
Chessell, IP; Gauldie, SD; McQueen, DS; Pertwee, R1
Brockie, HC; Craib, SJ; Di Marzo, V; Gibson, TM; Leslie, M; Pashmi, G; Pertwee, RG; Ross, RA1
Amadesi, S; Bianchi, A; Carreras, M; Creminon, C; Geppetti, P; Harrison, S; Matera, M; Tognetto, M; Trevisani, M1
Van de Voorde, J; Vanheel, B1
Akiba, Y; Engel, E; Furukawa, O; Guth, PH; Kaunitz, JD; Nastaskin, I1
Bevan, S; Chambers, A; Clarke, M; James, IF; McIntyre, P; McLatchie, LM; Peacock, M; Phillips, E; Rang, HP; Savidge, J; Shah, K; Toms, C; Webb, M; Weerasakera, N; Winter, J1
Ranasinghe, SP; Rang, HP; Savidge, JR1
Brough, SJ; Cairns, W; Davis, JB; Gunthorpe, MJ; Hayes, PD; Jerman, JC; Randall, AD; Ranson, J; Smart, D1
Chung, HT; Kim, IK; Kim, NY; Oh, GS; Pae, HO; Pyun, KH; Seo, WG; Shin, M1
Ahn, D; Kwon, S; Lee, Y; Leem, J; Nam, T; Yeon, D1
Rudd, JA; Wai, MK1
Harrison, C; Lambert, DG; Rowbotham, DJ; Smart, D; Sprague, J1
Eun, SY; Jung, SJ; Kim, J; Kim, SJ; Kwak, J; Park, YK1
Baumann, TK; Chaudhary, P; Martenson, ME1
McVey, DC; Vigna, SR1
Craib, SJ; Ellington, HC; Pertwee, RG; Ross, RA1
Erbelding, D; Kilbinger, H; Mang, CF1
Kohama, K; Nakamura, A; Shirakura, K; Sudo, M; Takagishi, K; Tomioka, A; Tsutsumi, S1
Bisogno, T; Brandi, I; Davis, JB; De Petrocellis, L; Di Marzo, V; Hanus, L; Mechoulam, R; Moriello, AS; Ponde, DE; Tchilibon, S1
Bottrill, FE; Ford, WR; Hiley, CR; Ho, WS; White, R1
Liddle, RA; McVey, DC; Nathan, JD; Patel, AA; Prpic, V; Thomas, JE; Vigna, SR1
Boachie-Ansah, G; Grainger, J1
Dussor, GO; Flores, CM; Harding-Rose, C; Hargreaves, KM; Kilo, S; Leong, AS1
Horie, S; Minowa, S; Murayama, T; Tsuchiya, S; Watanabe, K1
Bove, GM; Reeh, PW; Sauer, SK1
Fowler, CJ; Jacobsson, SO; Wallin, T1
Ikeda, Y; Naraba, H; Oh-ishi, S; Ueno, A1
Fushiki, T; Haramizu, S; Ohnluki, K; Watanabe, T; Yazawa, S1
Kobata, K; Sakurada, N; Watanabe, T1
Denda, M; Denda, S; Fuziwara, S; Inoue, K; Koizumi, S1
Biro, T; Blumberg, PM; Gonzalez, AF; Palkovits, M; Szabo, T1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N; Nocerino, E; Pinto, A; Sautebin, L1
Ahluwalia, A; Aston, D; McLean, PG; Sarkar, D1
Kim, KH1
Lee, LY; Lin, YS1
Berrino, L; Cuomo, D; de Novellis, V; Maione, S; Marabese, I; Palazzo, E; Rossi, F1
Kakehi, K; Kawabata, A; Kinoshita, M; Kuroda, R1
Amadesi, S; Barbieri, M; Bianchi, A; Brough, SJ; Campi, B; Davis, JB; Geppetti, P; Gray, J; Gunthorpe, MJ; Harrison, S; Jerman, JC; Owen, D; Randall, AD; Smart, D; Smith, GD; Tognetto, M; Trevisani, M1
Kagawa, S; Kato, S; Nakashima, M; Takeuchi, K; Tashima, K1
Andersson, DA; Bevan, S; Colley, S; Earley, TJ; Hergarden, AC; Hogenesch, JB; McIntyre, P; Moqrich, A; Patapoutian, A; Peier, AM; Reeve, AJ; Story, GM1
Harada, N; Katsuragi, T; Okajima, K; Uchiba, M1
Berger, AL; Price, MP; Welsh, MJ; Xie, J1
Chapman, V; Kelly, S2
Itoh, H; Kawabata, A; Kawao, N; Kuroda, R; Shimada, C1
Arden, WA; Chung, E; Gu, Q; Kwong, K; Lee, LY1
Adner, M; Andersson, DA; Högestätt, ED; Zygmunt, PM1
Kollarik, M; Undem, BJ1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N; Pinto, A; Russo, A; Sautebin, L1
Andresen, MC; Bailey, TW; Doyle, MW; Jin, YH1
Colley, S; Davis, C; Kotsonis, P; McIntyre, P; Phillips, E; Ranasinghe, S; Rang, H; Savidge, J; Shah, K; Winter, J1
Ishida, Y; Nishigaki, M; Shibata, Y; Shimada, S; Ueda, T; Ugawa, S1
Ahluwalia, J; Nagy, I; Rang, H1
Christie, MJ; Connor, M; Dedov, VN; Duke, CC; Mandadi, S; Roufogalis, BD; Tran, VH1
Egan, RW; Hey, JA; Jia, Y; McLeod, RL; Parra, LE; Wang, X1
Atweh, SF; Jabbur, SJ; Massaad, CA; Ochoa-Chaar, CI; Saadé, NE; Safieh-Garabedian, B1
Choi, JK; Choi, Jy; Choi, Sh; Jeong, YS; Jew, Ss; Kim, HD; Lee, J; Oh, U; Park, Hg; Park, Mk; Park, YH; Suh, Yg1
Fox, AJ; McIntyre, P; Medhurst, SJ; Panesar, M; Patel, S; Urban, L; Walker, KM1
Gharibova, LS; Li, T; Nicol, GD; Pei, Y; Southall, MD; Travers, JB1
Helyes, Z; Jakab, B; Németh, J; Pintér, E; Szolcsányi, J; Thán, M1
Adinolfi, B; Breschi, MC; Calderone, V; Martinotti, E; Nieri, P; Testai, L1
Christie, MJ; Jennings, EA; Roberts, LA; Vaughan, CW1
Chiang, HT; Lo, YK; Wu, SN1
Kaminski, NE; Li, J; Wang, DH1
Agopyan, N; Li, L; Simon, SA; Yu, S1
de la Fuente, SG; Fujino, K; Kihara, N; Mantyh, CR; Pappas, TN; Takahashi, T1
Li, GD; Zhao, ZQ; Zhou, Y1
Choi, H; Choi, JK; Jeong, YS; Kim, HD; Lee, HJ; Oh, U; Park, HG; Park, YH; Ryu, CH; Suh, YG; Yoon, J1
Cury, Y; Zanchet, EM1
Capasso, R; Mascolo, N1
Bernardi, G; Berretta, N; Di Marzo, V; Maccarrone, M; Marinelli, S; Matias, I; Mercuri, NB1
Matsumura, T; Moriyama, T; Sakurada, C; Sakurada, S; Sakurada, T; Ueno, S1
Hirota, K; Lambert, DG; Smart, D1
Deng, HW; Hu, CP; Li, NS; Li, YJ; Xiao, L1
Bowles, WR; Hargreaves, KM; Jackson, DL1
Gover, TD; Kao, JP; Weinreich, D1
Galoyan, SM; Mendell, LM; Petruska, JC1
Fischer, MJ; Reeh, PW; Sauer, SK1
Dux, M; Jancsó, G; Sántha, P1
Aihara, E; Kato, S; Kohama, K; Matsui, H; Nakamura, A; Takeuchi, K; Xin, H1
Calixto, JB; El Sayah, M1
Adler-Graschinsky, E; Celuch, SM; del Carmen García, M1
Kim, JS; Kim, YB; Lee, CH; Lee, JK; Oh, SB; Park, K; Piao, ZG; Yang, BH1
Chen, CW; Fu, WM; Ho, FM; Lee, ST; Lin, WW; Wu, WT1
Chen, ZH; Ding, ZH; Liu, JK; Liu, YD; Qing, C; Shen, ZQ; Yang, WM1
Akerman, S; Goadsby, PJ; Kaube, H1
Aoi, M; Kagawa, S; Kotani, T; Kubo, Y; Takeuchi, K1
Lao, LJ; Marvizón, JC; Song, B1
Cassar, SC; Esbenshade, T; Hancock, AA; Masters, JN; Witte, DG1
Benham, CD; Davies, CH; Davis, JB; Gill, CH; Gitterman, DP; Harries, M; Lanneau, C; Ray, AM; Roberts, JC1
Avelino, A; Charrua, A; Cruz, F; Matesz, K; Nagy, I; Santha, P; Sathianathan, V1
Köfalvi, A; Ledent, C; Sperlágh, B; Vizi, ES1
Farquhar-Smith, WP; Rice, AS1
Davies, CH; Davis, JB; Egerton, J; Gill, CH; Gunthorpe, MJ; Howett, L; Jerman, JC; Lappin, SC; Luis Hannan, S; Nasir, S; Owen, D; Rami, HK; Randall, AD; Smart, D; Smith, GD; Soffin, EM; Thompson, M; Worby, A; Wyman, PA1
Blumberg, PM; Chen, Z; Kozikowski, AP; Tóth, A1
Geracioti, TD; Kasckow, JW; Mulchahey, JJ1
Harada, N; Isobe, H; Okajima, K; Uchiba, M3
Bevan, S; McIntyre, P; Phillips, E; Reeve, A1
Akopian, AN; Flores, CM; Hargreaves, KM; Patwardhan, A; Price, TJ1
Evans, RM; Ross, RA; Scott, RH1
Moon, C1
Kyle, DJ; Tafesse, L1
Fujimoto, S; Mori, M1
Borrelli, F; Capasso, R; Izzo, AA; Pinto, A1
de Lago, E; de Miguel, R; Fernández-Ruiz, J; Lastres-Becker, I; Ramos, JA1
Ando, R; Kawamura, S; Watanabe, C; Yonezawa, A1
Baamonde, A; Hidalgo, A; Lastra, A; Menéndez, L1
Kim, BM; Lee, SH; Oh, U; Shim, WS1
Andresen, MC; Bailey, TW; Jin, YH; Li, BY; Schild, JH1
Izydorczyk, I; Pethö, G; Reeh, PW1
Godlewski, G; Malinowska, B; Schlicker, E1
Adler-Graschinsky, E; Becu-Villalobos, D; Celuch, SM; Huidobro-Toro, JP; Orliac, ML; Peroni, RN1
Chapman, V; Kendall, DA; Millns, PJ; Sagar, DR; Smart, D; Smith, PA1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N1
Fujita, T; Kawasaki, Y; Kumamoto, E; Yue, HY1
Liu, M; Michael, GJ; Priestley, JV; Willmott, NJ1
Jenkins, DW; Langmead, CJ; Parsons, AA; Strijbos, PJ1
Bizik, F; Blumberg, PM; Kedei, N; Kozikowski, AP; Pearce, LV; Petukhov, PA; Szabo, T1
Nagao, M; Shimada, S; Ueda, T; Ugawa, S; Yamamura, H2
Colleoni, M; Costa, B; Franke, C; Giagnoni, G; Trovato, AE1
Bates, SA; Benham, CD; Cairns, W; Davies, CH; Gill, CH; Hill, K; Larkman, PM; Murdock, PR; Owen, D; Powell, AJ; Randall, A; Strijbos, PJ; Yusaf, SP1
Advenier, C; Chinet, T; Fagon, JY; Faisy, C; Guerot, E; Naline, E; Risse, PA; Roche, N; Rouget, C1
Akiba, Y; Hibi, T; Ishii, H; Kato, S; Katsube, K; Nakamura, M; Takeuchi, K1
Chang, HT; Chen, JS; Cheng, HH; Cheng, JS; Hsu, SS; Huang, CJ; Huang, JK; Jan, CR; Jiann, BP; Lo, YK; Teng, HP; Yeh, JH1
Han, IS; Kang, JH; Kawada, T; Kim, CS; Kim, MO; Park, JY; Park, WH; Yoo, H; Yu, R1
Amantini, C; Lucciarini, R; Morrone, S; Mosca, M; Perfumi, M; Piccoli, M; Santoni, G1
Dogan, MD; Patel, S; Romanovsky, AA; Rudaya, AY; Steiner, AA; Székely, M1
Ahluwalia, A; Chauhan, S; Davis, C; De Felipe, C; Hunt, S; Kabir, J; Kotsonis, P; Oh, U; Scotland, RS1
de la Fuente, SG; Fujino, K; Ludwig, KA; Mantyh, CR; Takami, Y1
Bembry, J; Chen, Y; Golech, SA; Lenz, F; McCarron, RM; Mechoulam, R; Shohami, E; Spatz, M1
Barritt, GJ; Zhang, L1
Kadowaki, M; Kuramoto, H; Takaki, M1
Cloutier, M; Morin, C; Proteau, S; Rousseau, E1
Sun, Q; Valenzano, KJ1
Deng, PY; Hu, CP; Li, YJ; Tan, GS; Xu, KP; Yu, J1
D'Andrea, MR; Hornby, PJ; Kimball, ES; Schneider, CR; Wallace, NH1
Avelino, A; Bevan, S; Charrua, A; Cruz, F; Dinis, P; Nagy, I; Yaqoob, M1
Deng, HW; Du, YH; Hu, CP; Li, YJ; Peng, J; Rang, WQ; Xu, KP; Ye, F1
Henderson, D; Liu, L; Lu, G; Reinhart, PH; Simon, SA1
Gu, Q; Hu, HZ; Lee, LY; Lin, RL; Zhu, MX1
Ajioka, H; Horie, S; Kunieda, K; Murayama, T; Someya, A1
Bulmer, DC; Davis, JB; Grundy, D; Hicks, GA; Jiang, W; Winchester, WJ1
Braida, D; Consalez, GG; Croci, L; Guerini-Rocco, C; Pegorini, S; Sala, M; Verzoni, C1
Bianchi, R; Borsani, E; Buffoli, B; Rezzani, R; Ricci, F; Rodella, LF1
Andrews, PL; Cheng, FH; Moreaux, B; Ngan, MP; Rudd, JA; Sam, TS; Wai, MK; Wan, C1
Gunthorpe, MJ; McNamara, FN; Randall, A1
Lam, PM; Lambert, DG; McDonald, J1
Bunnett, NW; Day, AL; Grady, EF; Hutter, MM; Jordan, TH; Kirkwood, KS; Maa, J; Mulvihill, SJ; Richmond, AC; Wick, EC; Zerega, EC1
Kendall, DA; O'Sullivan, SE; Randall, MD1
Bielefeldt, K; Dang, K; Gebhart, GF1
Cadet, JL; Chen, J; Deng, X; Errico, S; Freed, WJ; Lee, CT1
Kohama, K; Nakamura, A; Takemori, S; Tanaka, H; Xin, H; Yamaguchi, M1
Breuer, A; Fride, E; Hanus, L; Ponde, D1
Maor, Y; Mechoulam, R; Pertwee, RG; Stevenson, LA; Thomas, A1
DeSimone, JA; Heck, GL; Lyall, V; Malik, SA; Mummalaneni, S; Phan, TH; Vinnikova, AK2
Hognestad, H; Hucho, F; Illes, P; Jahnel, R; Wirkner, K1
Elekes, K; Helyes, Z; McDougall, JJ; Németh, J; Pintér, E; Szabó, A; Szolcsányi, J; Varga, A; Zhang, C1
Andersen, OS; Birn, P; Gruner, SM; Hansen, AJ; Koeppe, RE; Lundbaek, JA; Søgaard, R; Tape, SE; Toombes, GE1
Bölcskei, K; Börzsei, R; Elekes, K; Helyes, Z; Jakab, B; Keszthelyi, D; Németh, J; Petho, G; Pintér, E; Sándor, K; Szabó, A; Szolcsányi, J; Varga, A1
Ando, R; Watanabe, C1
de Vries, A; Engels, F; Nijkamp, FP; van den Worm, E1
Andersson, TL; Evilevitch, V; Högestätt, ED; Jönsson, BA; Movahed, P; Wollmer, P; Zygmunt, PM1
Asai, H; Nagamine, K; Ozaki, N; Shinoda, M; Sugiura, Y; Tohnai, I; Ueda, M1
Bryant, BP; Inoue, T1
Canning, BJ; Mazzone, SB; Mori, N1
Long, LE; Malone, DT; Taylor, DA1
Easton, AS; Fraser, PA; Hu, DE1
Adler-Graschinsky, E; Briones, R; Huidobro-Toro, JP; Orliac, ML; Poblete, IM1
Wang, DH; Wang, Y; Zhu, Y1
de la Fuente, SG; Fujino, K; Mantyh, CR; Takahashi, T; Takami, Y1
Calixto, JB; Ferreira, J; Medeiros, R; Trichês, KM1
Farthing, JN; Gutierrez, T; Hohmann, AG; Suplita, RL1
Kaminski, NE; Wang, DH; Wang, Y2
Mustafa, S; Oriowo, M1
Nagy, I; Sántha, P; Singh Tahim, A1
Bisogno, T; Di Marzo, V; Giros, B; Li, DL; Moutsimilli, L; Nomikos, GG; Phebus, LA; Tzavara, ET1
Gao, Z; Henig, O; Kehoe, V; Li, J; Sinoway, LI1
Baamonde, A; Hidalgo, A; Juarez, L; Lastra, A; Menéndez, L1
Baamonde, A; García, E; García-Suárez, O; Hidalgo, A; Juárez, L; Menéndez, L1
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Chiang, LL; Hsu, CC; Lin, YJ; Lin, YS; Su, CL; Weng, WH1
Correia Junior, CA; da Cunha, PJ; da Silva, MT; de Siqueira, RJ; dos Santos, AA; Duarte, GP; Lahlou, S; Magalhães, PJ; Maia, JG; Rodrigues, KM1
Barahona, MV; Bustamante, S; Carballido, J; Fernandes, VS; García-Sacristán, A; Hernández, M; Martínez, AC; Martínez-Sáenz, A; Orensanz, LM; Prieto, D; Recio, P; Ribeiro, AS1
Bromberg, Z; Goloubinoff, P; Saidi, Y; Weiss, YG1
Barbero, R; Cuniberti, B; Odore, R; Re, G; Vercelli, C1
Ducreux, S; Legrand, C; Lotteau, S; Romestaing, C; Van Coppenolle, F1
Ciğ, B; Nazıroğlu, M; Ozgül, C1
Chen, L; Jiang, B; Lai, K; Lomask, JM; Zhong, N1
Arote, R; Bae, JS; Choi, S; Choi, SY; Hwang, SM; Jin, M; Namkoong, E; Park, K; Shin, YH1
DeSimone, JA; Grider, JR; Lyall, V; Mummalaneni, S; Murthy, KS; Phan, TH; Ren, Z; Rhyu, MR1
Jain, S; Nair, GN; Ramachandran, S; Sharma, S1
Chen, R; Lai, K; Li, J; Li, L; Liu, X; Ma, P; Wu, Y; Yang, X; Yao, H; Ye, X; You, H; Yuan, Y1
Gomes, KS; Mascarenhas, DC; Nunes-de-Souza, RL2
Gu, JG; Ling, JX; Xu, GY; Zuo, X1
Camille, S; Caroline, F; Fabielle, A; Florian, V; Francis, C1
Battani, KA; Lindgren, CA; Morford, JJ; Newman, ZL; Ryan, SB; Su, Z1
Breit, A; Fehrentz, T; Gudermann, T; Stein, M; Trauner, D1
Ching, LC; Kou, YR; Lee, TS; Lin, SJ; Shyue, SK; Wei, J; Zhao, JF1
Imoto, H; Kikuchi, D; Miura, K; Naitoh, T; Shibata, C; Unno, M1
Horii, A; Imai, T; Inohara, H; Ishida, Y; Kamakura, T; Kitahara, T; Nakamura, Y; Okazaki, S; Shimada, S; Takimoto, Y; Uno, A; Yamada, T1
Guo, Y; Kuang, H; Ma, L; Wu, J; Zhang, X; Zhao, L1
Corrêa, FM; dos Reis, DG; Guimarães, FS; Resstel, LB; Terzian, AL1
Holik, AK; Krammer, GE; Ley, JP; Pignitter, M; Rohm, B; Somoza, MM; Somoza, V; Zaunschirm, M1
Alpizar, YA; Boonen, B; Gees, M; Nilius, B; Sanchez, A; Talavera, K; Voets, T1
Chen, SL; Li, B; Li, MH; Wang, Q; Wang, ZM; Xiao, H; Zhang, JX; Zuo, GF1
Chiang, CC; Durand, DM; Gonzalez-Reyes, LE; Ladas, TP1
Chung, G; Im, ST; Jung, SJ; Kim, YH; Oh, SB; Rhyu, MR1
Islam, MS; Rebellato, P1
Cai, Q; Hu, WP; Liu, TT; Liu, YM; Qiu, CY; Qiu, F; Qu, ZW1
Abílio, VC; Almeida, V; Calzavara, MB; Crippa, JA; Hallak, JE; Levin, R; Peres, FF; Suiama, MA; Zuardi, AW1
Cai, J; Guo, J; Liu, FY; Sun, WL; Wan, Y; Xing, GG; Yang, F1
Ghazizadeh, V; Nazıroğlu, M1
Cornelius, F; Mahmmoud, YA; Pavlovic, D; Shattock, M1
Chen, CC; Chen, WN1
Andresen, MC; Fawley, JA; Hofmann, ME1
Bawankule, DU; Kalani, K; Khan, F; Luqman, S; Prakash, O; Sharma, P; Shukla, A; Singh, M; Srivastava, SK1
Cui, YY; Li, YQ; Qi, J; Shi, J; Wu, HH; Xu, H1
Nylander, O; Sjöblom, M; Sommansson, A; Wan Saudi, WS1
Baboota, RK; Bishnoi, M; Boparai, RK; Kaur, J; Kondepudi, KK; Sandhir, R; Sarma, SM; Singh, DP1
Fukushima-Miyashita, S; Goda, M; Hashikawa-Hobara, N; Hirai, K; Kawasaki, H; Ono, N; Ozaki, S; Takatori, S; Tangsucharit, P1
Gao, GD; Guo, H; Heng, LJ; Huang, B; Ma, LT; Song, J; Wang, P; Xu, GZ; Yuan, WX1
Chen, XL; Kuang, HY; Ma, LJ; Wu, JZ; Zhang, LX; Zhang, XY; Zhao, LM1
Andresen, MC; Fawley, JA; Hofmann, ME; Largent-Milnes, TM1
Battista, G; Borrelli, F; Capasso, R; Coppola, D; Di Marzo, V; Izzo, AA; Orlando, P; Pagano, E; Petrosino, S; Romano, B1
Azevedo-Santos, AP; Barboza, R; Brain, SD; Brito, CX; Costa, SK; dos Reis, AS; Fernandes, ES; Grisotto, MA; Marinho, CR; Muscará, M; Teixeira, SA1
Petrov, AM; Yakovleva, AA; Zefirov, AL1
Chen, L; Gollasch, M; Kaßmann, M; Markó, L; Wu, K; Zhu, Y1
Barragán-Iglesias, P; Granados-Soto, V; Martínez-Rojas, VA; Murbartián, J; Rocha-González, HI1
Baskaran, P; McArdle, JJ; Potian, JG; Thyagarajan, B1
Fujita, T; Jiang, CY; Kumamoto, E; Luo, QT1
Asano, A; Dayanithi, G; Forostyak, O; Hosaka, YZ; Ichimura, M; Kayano, T; Kitamura, N; Moriya, T; Shibasaki, R; Shibuya, I; Takebuchi, N; Verkhratsky, A1
Aguiar, DC; Almeida-Santos, AF; Guimarães, FS; Moreira, FA1
Chen, HY; Chiang, AN; Guo, BC; Lee, TS; Shyue, SK; Su, KH; Wei, J; Zhao, JF1
Kumamoto, N; Shibata, Y; Ueda, T; Ugawa, S; Watanabe, M1
Fazzari, J; Lin, H; Murphy, C; Singh, G; Ungard, R1
Alvarez de la Rosa, D; Armas-Capote, N; Buckley, ST; Ehrhardt, C; Fischer, H; Harvey, BJ; Huwer, H; Illek, B; Lehr, CM; Schneider-Daum, N; Schwagerus, E; Sladek, S1
Filipek, B; Sałat, K1
Nazıroğlu, M; Övey, İS1
Fujita, T; Jiang, CY; Kang, Q; Kumamoto, E1
Kikuchi, D; Miyachi, T; Nagao, M; Naitoh, T; Sasaki, H; Shibata, C; Someya, S; Tanaka, N; Unno, M1
Aizawa, F; Fujita, R; Iinuma, A; Saitou, A; Tsuchiya, Y; Wajima, N1
Chen, Q; Han, J; Sun, Z; Wang, L; Zhang, Y; Zheng, L1
Ghazizadeh, V; Nazıroğlu, M; Özdemir, ÜS; Şenol, N1
Gan, YH; Hao, T; Kou, XX; Ma, XC; Wu, YW1
Chen, X; Cui, W; Han, W; Jin, X; Long, C; Pan, Z; Wang, H; Zhang, Y1
Aoki, S; Dai, Y; Iwaoka, E; Kogure, Y; Matsuyoshi, N; Noguchi, K; Wang, S; Yamamoto, S1
Decorps, J; Fromy, B; Gohin, S; Sigaudo-Roussel, D1
Erickson, CS; Heppner, TJ; Mingin, GC; Nelson, MT; Tykocki, NR; Vizzard, MA1
Crespo, JE; Latorre-Estivalis, JM; Lazzari, CR; Lorenzo, MG; Zermoglio, PF1
Eslamizade, MJ; Hosseinmardi, N; Janahmadi, M; Meftahi, GH; Mehdizadeh, M; Mousavi, SM; Saffarzadeh, F1
Fujita, T; Jiang, CY; Kumamoto, E; Wang, C; Xu, ZH1
Ferreira-Junior, NC; Lagatta, DC; Resstel, LB1
Kaneko, S; Miyanohara, J; Nakagawa, T; Sanpei, K; Shirakawa, H1
Acharya, S; Schmidt, JJ; Vijayvergiya, V; Wilson, SP1
Dai, L; Huo, HR; Jiang, TL; Li, Q; Sui, F; Zhan, HD; Zhou, HY1
Chen, LH; Huang, Y; Li, JC; Liu, T; Peng, XY; Tian, B; Wang, XL1
Abraki, SB; Eslamizade, MJ; Gorji, A; Hadjighassem, MR; Mousavi, SM; Saffarzadeh, F1
Konno, H; Matoba, M; Miyano, K; Murakami, S; Nishimura, H; Shiraishi, S; Sudo, Y; Uezono, Y1
Ashton, JC; Milne, M1
Bo, L; Chen, X; Jin, F; Li, C; Liu, Q; Liu, W; Xu, D1
Socała, K; Wlaź, P1
Hu, SS1
Cao, X; Chai, S; Chen, Z; Dong, R; Ji, Z; Lai, K; Lv, H; Yue, J; Zhan, J; Zhang, H1
Gan, X; Hu, WP; Li, YK; Qiu, CY; Ren, C; Wu, J1
He, K; Pei, H; Su, L; Wang, Q; Wei, S; Yang, D; Yang, Y; Zhang, Y1
Baranowska-Kuczko, M; Harasim, E; Karpińska, O; Kasacka, I; Kloza, M; Kozłowska, H; Malinowska, B; Toczek, M1
Carletti, F; Ferraro, G; Gambino, G; Rizzo, V; Sardo, P1
He, L; Kumarhia, D; McCluskey, LP1
Cabral, LD; Giusti-Paiva, A1
Ide, S; Kojima, S; Nakanishi, Y; Nishino, K; Tanamachi, K; Tanuma, S; Tsukimoto, M1
Alijanpour, S; Amini-Khoei, H; Amiri, S; Ghaderi, M; Ghazi-Khansari, M; Haj-Mirzaian, A; Rahimi-Balaei, M; Rastegar, M; Tirgar, F; Zarrindast, MR1
Furube, E; Kittaka, H; Mannari, T; Miyata, S; Takayama, Y; Tominaga, M; Yoshida, A1
Deák, É; Dux, M; Jancsó, G; Sántha, P; Tassi, N1
Brzozowski, T; Czekaj, R; Magierowska, K; Magierowski, M; Majka, J; Ptak-Belowska, A; Strzalka, M; Szlachcic, A; Targosz, A1
Babes, A; Becker, C; Engel, MA; Khalil, M; Kistner, K; Neurath, MF; Reeh, PW; Selescu, T; Siklosi, N; Wirtz, S; Zimmermann, K1
Chen, X; Xiao, Y; Xu, GY; Xu, Q; Zhang, PA; Zheng, H1
da-Silva, CA; Del-Bel, E; Dos-Santos-Pereira, M; Guimarães, FS1
Demirdaş, A; Nazıroğlu, M; Övey, İS1
Ahn, KS; Baek, SH; Kim, C; Ko, JH; Lee, JH; Lee, SG; Sethi, G; Um, JY; Yang, WM1
Chen, M; Li, J; Li, M; Liu, B; Luo, L; Xin, J; Yin, W1
Hinz, B; Ivanov, I; Scholl, A1
André, E; Brusco, I; Cabrini, DA; de Oliveira, JR; Ferreira, J; Oliveira, SM; Otuki, MF1
Ding, X; Greer, JJ; Ren, J1
Joo, CK; Kwon, JY; Lee, HS1
Nanri, M; Sakakibara, F; Sasaki, E; Takahama, K1
Coutinho, HD; de Albuquerque, TR; de Lacerda Neto, LJ; de Menezes, IR; de Oliveira, LR; de Souza, SD; Dos Santos, AT; Kerntopf, MR; Quintans-Júnior, LJ; Ramos, AG; Santos Sales, V; Wanderley, AG1
Hayakawa, C; Ikeda, K; Irie, S; Kawakami, K; Kotani, S; Lin, ST; Onimaru, H; Tani, M1
De Toni, L; Di Nisio, A; Filippi, A; Foresta, C; Garolla, A; Magagna, S; Menegazzo, M; Rocca, MS; Šabović, I; Scattolini, V1
Fujita, T; Kumamoto, E; Piao, LH; Yu, T1
Nazıroğlu, M1
Brzozowski, T; Hubalewska-Mazgaj, M; Kwiecien, S; Magierowska, K; Magierowski, M; Sliwowski, Z; Wojcik, D1
Chen, J; Choi, CH; Emala, CW; Fu, XW; Sanderson, MJ; Townsend, EA; Xu, D; Yocum, GT; Zhang, Y1
Andresen, MC; Hofmann, ME1
Acevedo-Quiroz, M; de la Rosa-Lugo, V; Déciga-Campos, M; Rios, MY1
Abe, K; Chiba, T; Kanbe, T; Oka, Y; Sashida, H; Taguchi, K; Utsunomiya, I1
Araya, EI; Chichorro, JG; Cunha, JMD; Ferreira, LEN; Kopruszinski, CM; Nones, CFM1
Akiduki, S; Goto, T; Ho, YY; Kanamoto, R; Kawada, T; Kim, M; Mizushige, T; Nakato, J; Ohinata, K; Omae, R; Takahashi, N; Tominaga, M; Uchida, K1
Bodnár, D; Boros, M; Garab, D; Hartmann, P; Jancsó, G; Járomi, P; Nyíri, S; Sántha, P; Szabó, A1
Kim, EY; Kim, JT; Kim, Y; Lee, YJ; Park, J; Rhyu, MR; Son, HJ1
Bae, IH; Burns, A; Choi, G; Choi, JK; Fagg, R; Gatfield, KM; Lee, CS; Naidoo, AA; Park, M; Park, YH; Powell, AJ; Vidgeon-Hart, M1
Brzozowski, T; Czekaj, R; Kwiecien, S; Magierowska, K; Magierowski, M; Majka, J; Pajdo, R; Ptak-Belowska, A; Sliwowski, Z; Surmiak, M1
Ismael, HN; Mustafa, S1
Irie, S; Izumizaki, M; Kotani, S; Onimaru, H1
Gross, ER; Gross, GJ; Heymann, HM; Lu, Y; Qvit, N; Wu, Y1
Brauchi, S; Cabezas-Bratesco, D; Cao, C; Chelluboina, B; Cohen, AM; Dawson, T; Demirkhanyan, L; Domene, C; Kusuda, R; Nersesyan, Y; Oakes, V; Sun, X; Veeravalli, KK; Zakharian, E; Zimmermann, K1
Chapple, C; Chess-Williams, R; Daly, DM; Grundy, D; Grundy, L1
Fatahi, Z; Haghparast, A; Khani, A; Rainer, G; Reisi, Z1
Klumpp, DJ; Miller, RJ; Rosen, JM; Schaeffer, AJ; Woida, PJ; Yaggie, RE1
Ganaes, JOF; Lopes-Pires, ME; Naime, ACA1
Bierbower, SM; Canseco-Alba, A; Gould, GG; Joshi, N; Mora, Z; Onaivi, ES; Perchuk, A; Schanz, N; Tyrell, L1
Aso, H; Suemaru, K; Watanabe, M; Yoshikawa, M1
Cheng, Y; Li, X; Wang, R; Xu, Y1
Aboud, M; Comai, S; De Gregorio, D; Enns, J; Gobbi, G; Lopez-Canul, M; Maione, S; McLaughlin, RJ; Ochoa-Sanchez, R; Posa, L1
Balbay, E; Çiğ, B; Nazıroğlu, M; Taner, AN1
Kawamata, K; Tsuchiya, Y1
Imaoka, S; Inoue, T; Kudoh, SN; Oguro, A1
Brito, BM; Gobira, PH; Joca, SRL; Sartim, AG1
Geng, Z; Jing, Y; Liu, YL; Tian, HL; Wang, ML; Xu, ZM; Yang, DX; Yuan, F1
Andrade-Talavera, Y; Balleza-Tapia, H; Chen, G; Crux, S; Dolz-Gaiton, P; Fisahn, A; Johansson, J; Papadia, D1
Baskaran, P; Krishnan, V; Thyagarajan, B1
De La Chapa, J; Gonzales, CB; Gonzales, K; Hart, M; McHardy, SF; Mitchell, W; Polusani, SR; Ruiz, F; Valdez, M1
Jankowska, M; Kletkiewicz, H; Maliszewska, J; Rogalska, J; Stankiewicz, M1
Pang, G; Song, P; Xiao, S; Xie, J; Zhang, Y1
Barragán-Iglesias, P; Flores-Murrieta, FJ; Granados-Soto, V; Huerta-Cruz, JC; Pineda-Farias, JB; Quiñonez-Bastidas, GN; Reyes-García, JG; Roa-Coria, JE; Rocha-González, HI; Zúñiga-Romero, Á1
Andreeva, YV; Khropycheva, RP; Zolotarev, VA1
Eshima, H; Hoshino, D; Ikegami, R; Ishiguro, T; Kano, Y; Mashio, T; Poole, DC1
Garg, SK; Kumar, A; Mishra, AK; Saxena, A; Singh, V; Swain, DK; Yadav, S1
Bellingham, MC; Thakre, PP1
Chang, YJ; Chueh, SH; Huang, KF; Jhap, TY; Liu, PS; Lo, LC; Ma, KH; Su, YH1
De La Chapa, JJ; Gonzales, CB; Hart, MJ; McGuff, HS; McHardy, SF; Polusani, SR; Ruiz, F; Sallaway, ML; Self, KK; Singha, PK; Valdez, MC1
Ahn, KS; Jung, SH; Sethi, G; Yang, MH1
Chen, CC; Han, DS; Lee, CH; Shieh, YD1
Adams, DJ; Finol-Urdaneta, RK; McArthur, JR1
Fujii, N; Hatta, A; Kurose, M; Meng, ID; Okamoto, K; Sullivan, C; Yamamura, K1
Ashba, AM; Bezuglov, VV; Bobrov, MY; Fedorova-Gogolina, IA; Gretskaya, NM; Melkumyan, AG; Pavlovich, SV; Yushina, MN1
Cheng, X; Dou, M; He, S; Huang, C; Ma, Z; Xiong, W; Xu, Y; Zhang, Y; Zou, G1
Hong, SI; Jang, CG; Kwon, SH; Lee, SY; Ma, SX; Nguyen, TL; You, IJ1
Chen, NH; Han, QW; Yuan, YH1
Castrejón-Téllez, V; Cervantes-Yañez, EZ; Del Valle-Mondragón, L; Flores-Chávez, P; Guarner-Lans, V; Martínez-Memije, R; Oidor-Chan, VH; Pastelín-Hernández, G; Pérez-Torres, I; Soto-Peredo, CA; Torres-Narváez, JC; Varela-López, E; Vargas-González, Á1
Bortolanza, M; Crivelaro do Nascimento, G; Del Bel, EA; Ferrari, DP; Ferreira-Junior, NC; Guimaraes, FS1
Han, Y; Hu, J; Kamau, PM; Lai, R; Luo, A; Luo, L; Tian, Y; Yao, Z; Zheng, J1
Ham, S; Han, JS; Han, S; Jung, YK; Kim, J; Lee, KW; Lee, S; Park, JHY; Shim, I1
Morita, H; Obata, K; Takaki, M1
Dong, L; Fei, X; Liu, D; Yuan, J; Zhang, C; Zhou, Y; Zhu, Y; Zhu, Z1
Bhutia, YD; Bora, NS; Chattopadhyay, P; Goyary, D; Hazarika, H; Karmakar, S; Kishor, S; Krishnatreyya, H; Mandal, S; Saha, A1
Bansal, Y; Bishnoi, M; Khare, P; Kondepudi, KK; Kuhad, A; Medhi, B; Singh, R; Sodhi, RK1
Bandeira, PN; Campos, AR; da Silva, AW; de Menezes, JESA; Dos Reis Lima, J; Dos Santos, HS; Evaristo, FFV; Ferreira, MKA; Holanda, CLA; Magalhães, FEA; Silva, FCO; Teixeira, EH1
González-Anduaga, GM; López-Ortíz, M; Navarrete, A; Palomino-Hernández, O; Quiñonez-Bastidas, GN; Regla, I; Rocha-González, HI1
Abdulla, MH; AlMarabeh, S; Cavers, J; Lucking, EF; O'Halloran, KD; O'Neill, J1
Hong, JI; Hwang, HS; Kim, HA; Kim, JR; Park, IY1
Christie, S; Zagorodnyuk, V1
Hara, K; Haranishi, Y; Terada, T1
Baudouin, C; Fakih, D; Guerrero-Moreno, A; Parsadaniantz, SM; Réaux-Le Goazigo, A1
Arenas, AP; Castrejón-Téllez, V; Del Valle-Mondragón, L; Guarner-Lans, V; Pastelín-Hernández, G; Pérez-Torres, I; Rojas, FM; Torres-Narváez, JC; Varela-López, E; Vargas-González, A1
Bäumer, W; Kietzmann, M; Mishra, SK; Rossbach, K; Stark, H; Wilzopolski, J1
Bang, SK; Cho, SJ; Choi, KH; Kang, SY; Ryu, Y; Seo, SY1
Mizogami, M; Tsuchiya, H1
Bishnoi, M; Chopra, K; Devi, K; Khan, R; Kondepudi, KK; Kumar, A; Kumar, V; Rajarammohan, S; Singh, RP1
Abdolmaleki, Z; Shahidi, S; Zarei, MM1
Benzing, T; Brinkkoetter, PT; Chen, H; Dryer, S; Hagmann, H; Khayyat, NH; Matin, M; Oezel, C; Schauss, A; Schell, C1
Çakır, M; Çiğremiş, Y; Durhan, M; Kaymak, E; Mustafa Özkut, M; Tekin, S; Yüksel, F1
Chhatwal, S; Li, A; Lucius, A; Mergler, S; Pleyer, U; Reinach, PS; Valtink, M1

Reviews

7 review(s) available for capsaicin and capsazepine

ArticleYear
Mechanism of action of capsaicin-like molecules on sensory neurons.
    Life sciences, 1992, Volume: 51, Issue:23

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcium Channels; Capsaicin; Cell Membrane; Humans; Neurons, Afferent; Nociceptors; Pain; Pain Threshold; Receptors, Drug

1992
Neuropharmacological mechanisms of capsaicin and related substances.
    Biochemical pharmacology, 1992, Aug-18, Volume: 44, Issue:4

    Topics: Animals; Capsaicin; Humans; Ion Channels; Nervous System; Neuropeptides; Receptors, Drug

1992
Capsaicin: gaps in our knowledge start to be filled.
    Trends in neurosciences, 1991, Volume: 14, Issue:7

    Topics: Animals; Axonal Transport; Capsaicin; Nerve Degeneration; Nerve Endings; Nerve Fibers; Nerve Growth Factors; Neurons, Afferent; Pain; Receptors, Drug; Sciatic Nerve; Silver Nitrate; Spinal Cord; Staining and Labeling

1991
Current perspectives on the therapeutic utility of VR1 antagonists.
    Current medicinal chemistry, 2004, Volume: 11, Issue:24

    Topics: Animals; Capsaicin; Humans; Receptors, Drug

2004
Sepsis: The Involvement of Platelets and the Current Treatments.
    Current molecular pharmacology, 2018, Volume: 11, Issue:4

    Topics: Acetylcysteine; Animals; Blood Platelets; Capsaicin; Chloroquine; Disseminated Intravascular Coagulation; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Interleukin-7; Platelet Aggregation Inhibitors; Sepsis; Software; Thrombocytopenia; Toll-Like Receptor 4

2018
Pleiotropic Pharmacological Actions of Capsazepine, a Synthetic Analogue of Capsaicin, against Various Cancers and Inflammatory Diseases.
    Molecules (Basel, Switzerland), 2019, Mar-12, Volume: 24, Issue:5

    Topics: Animals; Anti-Inflammatory Agents; Antineoplastic Agents; Capsaicin; Cell Line, Tumor; Humans; Janus Kinases; NF-kappa B; Reactive Oxygen Species; Signal Transduction; TRPV Cation Channels

2019
The therapeutic role of cannabinoid receptors and its agonists or antagonists in Parkinson's disease.
    Progress in neuro-psychopharmacology & biological psychiatry, 2020, 01-10, Volume: 96

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Endocannabinoids; Humans; Parkinson Disease; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2

2020

Trials

2 trial(s) available for capsaicin and capsazepine

ArticleYear
Transient receptor potential vanilloid type-1 (TRPV-1) channels contribute to cutaneous thermal hyperaemia in humans.
    The Journal of physiology, 2010, Nov-01, Volume: 588, Issue:Pt 21

    Topics: Adult; Capsaicin; Enzyme Inhibitors; Female; Hot Temperature; Humans; Hyperemia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Regional Blood Flow; Sensory Receptor Cells; Skin; Skin Temperature; TRPV Cation Channels

2010
Transient receptor potential vanilloid type 1 channels contribute to reflex cutaneous vasodilation in humans.
    Journal of applied physiology (Bethesda, Md. : 1985), 2012, Volume: 112, Issue:12

    Topics: Adult; Blood Pressure; Body Temperature; Capsaicin; Female; Forearm; Heating; Humans; Male; Microdialysis; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Reflex; Regional Blood Flow; Skin; TRPV Cation Channels; Vasodilation; Young Adult

2012

Other Studies

712 other study(ies) available for capsaicin and capsazepine

ArticleYear
The discovery of capsazepine, the first competitive antagonist of the sensory neuron excitants capsaicin and resiniferatoxin.
    Journal of medicinal chemistry, 1994, Jun-24, Volume: 37, Issue:13

    Topics: Animals; Calcium; Capsaicin; Cells, Cultured; Crystallography, X-Ray; Diterpenes; Ganglia, Spinal; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Neurons, Afferent; Neurotoxins; Rats; Receptors, Drug; Structure-Activity Relationship

1994
Synthesis and evaluation of phorboid 20-homovanillates: discovery of a class of ligands binding to the vanilloid (capsaicin) receptor with different degrees of cooperativity.
    Journal of medicinal chemistry, 1996, Aug-02, Volume: 39, Issue:16

    Topics: Animals; Body Temperature; Diterpenes; Edema; Homovanillic Acid; Magnetic Resonance Spectroscopy; Mass Spectrometry; Membrane Proteins; Molecular Structure; Phorbol Esters; Protein Binding; Rats; Receptors, Drug; Spinal Cord

1996
N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: novel potent and high affinity antagonists and partial antagonists of the vanilloid receptor.
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Analgesics; Animals; Calcium; Capsaicin; CHO Cells; Cricetinae; Ligands; Male; Mice; Mice, Inbred ICR; Rats; Receptors, Drug; Structure-Activity Relationship; Sulfonamides; Thiourea

2003
N-4-Substituted-benzyl-N'-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity.
    Bioorganic & medicinal chemistry letters, 2004, Feb-09, Volume: 14, Issue:3

    Topics: Animals; Animals, Newborn; Calcium; Capsaicin; Cells, Cultured; Ganglia, Spinal; Ligands; Molecular Structure; Neurons; Rats; Receptors, Drug; Structure-Activity Relationship; Sulfonamides; Thiourea

2004
Identification and biological evaluation of 4-(3-trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide, a high affinity TRPV1 (VR1) vanilloid receptor antagonist.
    Journal of medicinal chemistry, 2005, Mar-24, Volume: 48, Issue:6

    Topics: Administration, Oral; Aminopyridines; Analgesics; Animals; Biological Availability; Body Temperature; Calcium; Capsaicin; Cell Line; Humans; Hypothermia; Ion Channels; Male; Pain Measurement; Piperazines; Rats; Structure-Activity Relationship; TRPV Cation Channels

2005
[3H]A-778317 [1-((R)-5-tert-butyl-indan-1-yl)-3-isoquinolin-5-yl-urea]: a novel, stereoselective, high-affinity antagonist is a useful radioligand for the human transient receptor potential vanilloid-1 (TRPV1) receptor.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 323, Issue:1

    Topics: Animals; Binding, Competitive; Calcium Signaling; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Ganglia, Spinal; Humans; Isoquinolines; Ligands; Molecular Structure; Neurons, Afferent; Radioligand Assay; Rats; Recombinant Proteins; Stereoisomerism; Transfection; Tritium; TRPV Cation Channels; Urea

2007
In vitro TRPV1 activity of piperine derived amides.
    Bioorganic & medicinal chemistry, 2010, May-01, Volume: 18, Issue:9

    Topics: Alkaloids; Amides; Benzodioxoles; Capsaicin; Cell Line; Dose-Response Relationship, Drug; Humans; Molecular Structure; Piperidines; Polyunsaturated Alkamides; Spectrometry, Fluorescence; TRPV Cation Channels

2010
Activation and inhibition of thermosensitive TRP channels by voacangine, an alkaloid present in Voacanga africana, an African tree.
    Journal of natural products, 2014, Feb-28, Volume: 77, Issue:2

    Topics: Africa; Alkaloids; Calcium; Capsaicin; Humans; Ibogaine; Menthol; Molecular Structure; Plant Bark; Pyrimidinones; Transient Receptor Potential Channels; Trees; TRPV Cation Channels; Voacanga

2014
Inhibition of low pH evoked activation of airway sensory nerves by capsazepine, a novel capsaicin-receptor antagonist.
    Biochemical and biophysical research communications, 1992, Nov-30, Volume: 189, Issue:1

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Citrates; Citric Acid; Electric Stimulation; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Lung; Neurokinin A; Neurons, Afferent; Nicotine; Receptors, Drug; Respiratory Physiological Phenomena; Respiratory System; Ruthenium Red; Tidal Volume; Vagus Nerve

1992
Inhibitory effects of capsazepine and the NK2 antagonist SR 48968 on bronchoconstriction evoked by sensory nerve stimulation in guinea-pigs.
    Acta physiologica Scandinavica, 1992, Volume: 146, Issue:4

    Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Electric Stimulation; Female; Guinea Pigs; Male; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Neurokinin-2; Receptors, Neurotransmitter

1992
Capsazepine as a selective antagonist of capsaicin-induced activation of C-fibres in guinea-pig bronchi.
    European journal of pharmacology, 1992, May-14, Volume: 215, Issue:2-3

    Topics: Animals; Bronchi; Capsaicin; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Nerve Fibers; Ruthenium Red; Tetrodotoxin

1992
Capsazepine reversal of the antinociceptive action of capsaicin in vivo.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Capsaicin; Female; Freund's Adjuvant; Hyperalgesia; Irritants; Mice; Morphine; Naloxone; Pain Measurement; Rats; Rats, Wistar; Uric Acid

1992
Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Adenosine Triphosphate; Animals; Calcium; Capsaicin; Cells, Cultured; Diterpenes; Electrophysiology; gamma-Aminobutyric Acid; Ganglia, Spinal; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Vagus Nerve

1992
Capsazepine inhibits low pH- and lactic acid-evoked release of calcitonin gene-related peptide from sensory nerves in guinea-pig heart.
    European journal of pharmacology, 1992, Oct-06, Volume: 221, Issue:1

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Guinea Pigs; Heart; Hydrogen-Ion Concentration; In Vitro Techniques; Lactates; Lactic Acid; Nerve Fibers

1992
Capsazepine, a novel capsaicin antagonist, selectively antagonises the effects of capsaicin in the mouse spinal cord in vitro.
    Neuroscience letters, 1991, Dec-16, Volume: 134, Issue:1

    Topics: Action Potentials; Afferent Pathways; Animals; Capsaicin; Electric Stimulation; Ganglia, Spinal; Mice; Receptors, Drug; Spinal Cord; Substance P

1991
Selective antagonism of capsaicin by capsazepine: evidence for a spinal receptor site in capsaicin-induced antinociception.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: Analgesics; Animals; Bradykinin; Capsaicin; Electric Stimulation; In Vitro Techniques; Injections, Spinal; Nerve Fibers; Rats; Receptors, Drug; Spinal Cord; Spinal Nerve Roots

1991
Effects of ruthenium red and capsazepine on C-fibres in the rabbit iris.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: Animals; Bradykinin; Capsaicin; Drug Interactions; Electric Stimulation; Female; Iris; Male; Muscle Contraction; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neuromuscular Junction; Rabbits; Ruthenium Red

1993
Evidence that glutamate is released from capsaicin-sensitive primary afferent fibers in rats: study with on-line continuous monitoring of glutamate.
    Neuroscience research, 1994, Volume: 20, Issue:3

    Topics: Animals; Calcium; Capsaicin; Enzymes, Immobilized; Glutamate Dehydrogenase; Glutamic Acid; In Vitro Techniques; Male; Nerve Endings; Nerve Fibers; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Spinal Cord; Substance P

1994
Resiniferatoxin binding to vanilloid receptors in guinea pig and human airways.
    American journal of respiratory and critical care medicine, 1995, Volume: 152, Issue:1

    Topics: Adult; Animals; Binding Sites; Bronchi; Capsaicin; Diterpenes; Female; Guinea Pigs; Humans; Male; Middle Aged; Neurotoxins; Receptors, Drug; Trachea; Tritium

1995
Effects of capsazepine against capsaicin- and proton-evoked excitation of single airway C-fibres and vagus nerve from the guinea-pig.
    Neuroscience, 1995, Volume: 67, Issue:3

    Topics: Afferent Pathways; Animals; Capsaicin; Electrophysiology; Evoked Potentials; Female; Guinea Pigs; Hydrogen-Ion Concentration; Male; Nerve Fibers; Protons; Trachea; Vagus Nerve

1995
Ruthenium red, but not capsazepine reduces plasma extravasation by cigarette smoke in rat airways.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Aerosols; Animals; Capillary Permeability; Capsaicin; Evans Blue; Nerve Fibers; Rats; Rats, Inbred F344; Ruthenium Red; Smoking

1993
A comparison of capsazepine and ruthenium red as capsaicin antagonists in the rat isolated urinary bladder and vas deferens.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Rats; Rats, Wistar; Ruthenium Red; Urinary Bladder; Vas Deferens

1993
The role of calcium in capsaicin-induced desensitization in rat cultured dorsal root ganglion neurons.
    Neuroscience, 1993, Volume: 55, Issue:4

    Topics: Animals; Bradykinin; Calcium; Capsaicin; Cells, Cultured; Drug Tolerance; Ethers, Cyclic; Extracellular Space; Ganglia, Spinal; Inositol Phosphates; Ion Channels; Ionomycin; Mitochondria; Neurons, Afferent; Okadaic Acid; Potassium Chloride; Rats; Rats, Sprague-Dawley; Signal Transduction

1993
Characterization by [3H]resiniferatoxin binding of a human vanilloid (capsaicin) receptor in post-mortem spinal cord.
    Neuroscience letters, 1994, Jan-03, Volume: 165, Issue:1-2

    Topics: Animals; Binding, Competitive; Capsaicin; Diterpenes; Guinea Pigs; Humans; In Vitro Techniques; Kinetics; Membranes; Neurotoxins; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Receptors, Drug; Spinal Cord

1994
[3H]resiniferatoxin binding by the human vanilloid (capsaicin) receptor.
    Brain research. Molecular brain research, 1994, Volume: 23, Issue:3

    Topics: Animals; Binding, Competitive; Capsaicin; Diterpenes; Female; Humans; Kinetics; Medulla Oblongata; Nerve Tissue Proteins; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, Drug; Species Specificity; Spinal Cord; Trigeminal Nuclei

1994
Capsazepine abolishes pulmonary chemoreflexes induced by capsaicin in anesthetized rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 1994, Volume: 76, Issue:5

    Topics: Anesthesia; Animals; Biguanides; Capsaicin; Chemoreceptor Cells; Female; Lung; Male; Nerve Fibers; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reflex; Respiration

1994
Comparison of [3H]resiniferatoxin binding by the vanilloid (capsaicin) receptor in dorsal root ganglia, spinal cord, dorsal vagal complex, sciatic and vagal nerve and urinary bladder of the rat.
    Life sciences, 1994, Volume: 55, Issue:13

    Topics: Animals; Axons; Binding Sites; Binding, Competitive; Capsaicin; Diterpenes; Female; Ganglia, Spinal; Kinetics; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sciatic Nerve; Spinal Cord; Substrate Specificity; Tritium; Urinary Bladder; Vagus Nerve

1994
Detection of capsaicin-evoked release of glutamate from spinal dorsal horn slices of rat with on-line monitoring system.
    Neuroscience letters, 1993, Jun-11, Volume: 155, Issue:2

    Topics: Animals; Biosensing Techniques; Capsaicin; Enzymes, Immobilized; Fluorometry; Glutamate Dehydrogenase; Glutamates; Glutamic Acid; Male; Monitoring, Physiologic; Nerve Endings; Neurons, Afferent; Online Systems; Perfusion; Potassium; Rats; Rats, Sprague-Dawley; Spinal Cord; Tetrodotoxin

1993
Cyclo-oxygenase products released by low pH have capsaicin-like actions on sensory nerves in the isolated guinea pig heart.
    Cardiovascular research, 1994, Volume: 28, Issue:3

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Diclofenac; Epoprostenol; Guinea Pigs; Heart; Hydrogen-Ion Concentration; Indomethacin; Lactates; Lactic Acid; Neurons, Afferent; Perfusion; Receptors, Drug

1994
Involvement of tachykinin and CGRP receptors in the cardio-pulmonary effects evoked by capsaicin in the guinea-pig.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Blood Proteins; Bronchoconstriction; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Female; Glycopeptides; Guinea Pigs; Heart Rate; Male; Metalloendopeptidases; Receptors, Calcitonin Gene-Related Peptide; Receptors, Tachykinin

1993
Effect of capsazepine on the release of calcitonin gene-related peptide-like immunoreactivity (CGRP-LI) induced by low pH, capsaicin and potassium in rat soleus muscle.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Muscles; Neurons, Afferent; Potassium; Rats; Rats, Wistar

1993
Competitive inhibition by capsazepine of [3H]resiniferatoxin binding to central (spinal cord and dorsal root ganglia) and peripheral (urinary bladder and airways) vanilloid (capsaicin) receptors in the rat.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Bronchi; Capsaicin; Diterpenes; Ganglia, Spinal; Kinetics; Membranes; Neurons; Rats; Receptors, Drug; Sensitivity and Specificity; Spinal Cord; Trachea; Tritium; Urinary Bladder

1993
Topical capsaicin administration protects against trinitrobenzene sulfonic acid-induced colitis in the rat.
    European journal of pharmacology, 1993, Nov-09, Volume: 249, Issue:2

    Topics: Administration, Topical; Animals; Capsaicin; Colitis; Diterpenes; In Vitro Techniques; Kinetics; Male; Membranes; Rats; Rats, Sprague-Dawley; Receptors, Drug; Trinitrobenzenesulfonic Acid

1993
Inhibition by capsazepine of resiniferatoxin- and capsaicin-induced contractions of guinea pig trachea.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:1

    Topics: Animals; Capsaicin; Diterpenes; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins; Trachea

1994
Capsaicin-induced activation of fine afferent fibres from rat skin in vitro.
    Neuroscience, 1993, Volume: 55, Issue:2

    Topics: Afferent Pathways; Animals; Capsaicin; Cold Temperature; Dose-Response Relationship, Drug; Electric Stimulation; Hot Temperature; In Vitro Techniques; Mechanoreceptors; Nerve Fibers; Rats; Rats, Sprague-Dawley; Skin

1993
Inhibitory effects of capsazepine and SR 48968 on citric acid-induced bronchoconstriction in guinea-pigs.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Administration, Inhalation; Analysis of Variance; Animals; Benzamides; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Female; Guinea Pigs; Histamine; Hydrogen-Ion Concentration; Male; Neurokinin A; Neurons, Afferent; Piperidines

1993
Capsazepine-sensitive release of calcitonin gene-related peptide from C-fibre afferents in the guinea-pig heart by low pH and lactic acid.
    European journal of pharmacology, 1993, Jul-20, Volume: 238, Issue:2-3

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Guinea Pigs; Heart; Heart Rate; Hydrogen-Ion Concentration; In Vitro Techniques; Lactates; Lactic Acid; Nerve Fibers; Neurons, Afferent; Nicotine

1993
Capsazepine inhibits cough induced by capsaicin and citric acid but not by hypertonic saline in guinea pigs.
    Journal of applied physiology (Bethesda, Md. : 1985), 1995, Volume: 79, Issue:4

    Topics: Animals; Antitussive Agents; Bronchodilator Agents; Capsaicin; Citrates; Citric Acid; Cough; Guinea Pigs; Irritants; Male; Protons; Saline Solution, Hypertonic; Terbutaline

1995
Capsaicin-induced biphasic oxygen uptake in rat muscle: antagonism by capsazepine and ruthenium red provides further evidence for peripheral vanilloid receptor subtypes (VN1/VN2).
    Life sciences, 1996, Volume: 59, Issue:2

    Topics: Animals; Capsaicin; Dose-Response Relationship, Drug; Hindlimb; Male; Muscles; Oxygen; Rats; Rats, Wistar; Receptors, Drug; Ruthenium Red

1996
Pharmacological characterization of the vanilloid receptor in the rat isolated vas deferens.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:3

    Topics: Animals; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Drug Antagonism; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Wistar; Receptors, Drug; Vas Deferens

1996
Capsaicin activates a nonselective cation channel in cultured neonatal rat dorsal root ganglion neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Mar-01, Volume: 16, Issue:5

    Topics: Acids; Animals; Animals, Newborn; Capsaicin; Cations; Cells, Cultured; Diterpenes; Ganglia, Spinal; Ion Channels; Models, Neurological; Neurons; Neurotoxins; Rats

1996
Autoradiographic visualization and pharmacological characterization of vanilloid (capsaicin) receptors in several species, including man.
    Acta physiologica Scandinavica. Supplementum, 1995, Volume: 629

    Topics: Animals; Antipsychotic Agents; Autoradiography; Binding, Competitive; Bronchi; Capsaicin; Cricetinae; Diterpenes; Female; Guinea Pigs; Humans; Male; Mesocricetus; Neurotoxins; Rats; Rats, Sprague-Dawley; Receptors, Drug; Spinal Cord; Swine

1995
Pharmacology of calcitonin gene related peptide release from sensory terminals in the rat trachea.
    Canadian journal of physiology and pharmacology, 1995, Volume: 73, Issue:7

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Indomethacin; Male; Nerve Fibers; Oxidopamine; Prostaglandins; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Trachea

1995
Binding of neuroleptic drugs (trifluoperazine and rimcazole) to vanilloid receptors in porcine dorsal horn.
    European journal of pharmacology, 1996, Mar-18, Volume: 298, Issue:3

    Topics: Adult; Animals; Antipsychotic Agents; Autoradiography; Binding Sites; Binding, Competitive; Capsaicin; Carbazoles; Diterpenes; Female; Humans; In Vitro Techniques; Membranes; Neurotoxins; Rats; Rats, Sprague-Dawley; Receptors, Drug; Spinal Cord; Trifluoperazine

1996
Effect of capsaicin and analogues on potassium and calcium currents and vanilloid receptors in Xenopus embryo spinal neurones.
    British journal of pharmacology, 1996, Volume: 119, Issue:1

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Capsaicin; Embryo, Nonmammalian; Membrane Potentials; Neurons; Potassium Channel Blockers; Potassium Channels; Receptors, Drug; Spinal Cord; Time Factors; Xenopus

1996
Tachykinin-independent effects of capsaicin on smooth muscle in human isolated bronchi.
    American journal of respiratory and critical care medicine, 1997, Volume: 155, Issue:2

    Topics: Adult; Benzamides; Bronchi; Capsaicin; Cells, Cultured; Diterpenes; Drug Interactions; Female; Humans; Male; Muscle Contraction; Muscle, Smooth; Patch-Clamp Techniques; Piperidines; Tachykinins

1997
Capsaicin and carbon dioxide act by distinct mechanisms on sensory nerve terminals in the cat cornea.
    Pain, 1997, Volume: 70, Issue:1

    Topics: Animals; Capsaicin; Carbon Dioxide; Cats; Cornea; Drug Interactions; Electrophysiology; Female; Male; Nerve Endings; Neurons, Afferent

1997
The selective capsaicin antagonist capsazepine abolishes the antinociceptive action of eugenol and guaiacol.
    Journal of dental research, 1997, Volume: 76, Issue:4

    Topics: Analgesics, Non-Narcotic; Analysis of Variance; Animals; Capsaicin; Eugenol; Guaiacol; Male; Mice; Mice, Inbred Strains; Nociceptors; Pain Threshold; Receptors, Drug; Structure-Activity Relationship

1997
The responses of rat trigeminal ganglion neurons to capsaicin and two nonpungent vanilloid receptor agonists, olvanil and glyceryl nonamide.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jun-01, Volume: 17, Issue:11

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Glycerol; Neurons; Pain; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Drug; Tachyphylaxis; Taste; Trigeminal Ganglion

1997
Activation of chemosensitive neurons in the ventrolateral medulla by capsaicin in cats.
    Neuroscience letters, 1997, May-02, Volume: 226, Issue:3

    Topics: Analysis of Variance; Animals; Autonomic Fibers, Preganglionic; Blood Pressure; Capsaicin; Cats; Drug Evaluation, Preclinical; Heart Rate; Medulla Oblongata; Neurons; Ruthenium Red; Sympathetic Nervous System

1997
Capsazepine, a vanilloid receptor antagonist, inhibits nicotinic acetylcholine receptors in rat trigeminal ganglia.
    Neuroscience letters, 1997, May-30, Volume: 228, Issue:1

    Topics: Animals; Capsaicin; Electric Conductivity; Nicotine; Nicotinic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Drug; Receptors, Nicotinic; Trigeminal Ganglion

1997
Antinociception induced by civamide, an orally active capsaicin analogue.
    Pain, 1997, Volume: 71, Issue:3

    Topics: Administration, Oral; Analgesics; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Hot Temperature; Male; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Stereoisomerism; Substance P

1997
Enhancement of rat trigeminal ganglion neuron responses to piperine in a low-pH environment and block by capsazepine.
    Brain research, 1997, Jun-27, Volume: 761, Issue:1

    Topics: Alkaloids; Animals; Anticonvulsants; Benzodioxoles; Binding, Competitive; Capsaicin; Female; Hydrogen-Ion Concentration; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Protons; Rats; Rats, Sprague-Dawley; Trigeminal Ganglion

1997
Capsazepine block of voltage-activated calcium channels in adult rat dorsal root ganglion neurones in culture.
    British journal of pharmacology, 1997, Volume: 121, Issue:7

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Female; Ganglia, Spinal; Male; omega-Conotoxin GVIA; Peptides; Rats; Rats, Sprague-Dawley; Rats, Wistar

1997
Eugenol activates Ca(2+)-permeable currents in rat dorsal root ganglion cells.
    Journal of dental research, 1997, Volume: 76, Issue:11

    Topics: Animals; Animals, Newborn; Calcium Channel Agonists; Calcium Channels; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Eugenol; Female; Ganglia, Spinal; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Drug

1997
Ruthenium red and capsazepine antinociceptive effect in formalin and capsaicin models of pain in mice.
    Neuroscience letters, 1997, Oct-10, Volume: 235, Issue:1-2

    Topics: Analgesics; Animals; Capsaicin; Dose-Response Relationship, Drug; Formaldehyde; Injections, Intradermal; Injections, Intraventricular; Male; Mice; Naloxone; Pain; Ruthenium Red

1997
Peripheral CGRP release as a marker for neurogenic inflammation: a model system for the study of neuropeptide secretion in rat paw skin.
    Pain, 1997, Volume: 73, Issue:2

    Topics: Animals; Basal Metabolism; Biomarkers; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Hindlimb; Male; Nerve Endings; Neuritis; Neuropeptides; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Skin

1997
Inflammatory mediators at acidic pH activate capsaicin receptors in cultured sensory neurons from newborn rats.
    Journal of neurophysiology, 1998, Volume: 79, Issue:2

    Topics: Animals; Animals, Newborn; Bradykinin; Capsaicin; Cells, Cultured; Coculture Techniques; Dinoprostone; Drug Synergism; Ganglia, Spinal; Hippocampus; Hydrogen-Ion Concentration; Inflammation; Ion Channel Gating; Neuroglia; Neurons, Afferent; Rats; Receptors, Drug; Serotonin; Stimulation, Chemical

1998
Identification of the L-menthol binding site in guinea-pig lung membranes.
    British journal of pharmacology, 1998, Volume: 123, Issue:3

    Topics: Animals; Benzazepines; Binding Sites; Camphor; Capsaicin; Cell Membrane; Eugenol; Guinea Pigs; In Vitro Techniques; Lung; Male; Menthol; Radioligand Assay; Tritium

1998
A non-pungent resiniferatoxin analogue, phorbol 12-phenylacetate 13 acetate 20-homovanillate, reveals vanilloid receptor subtypes on rat trigeminal ganglion neurons.
    Neuroscience, 1998, Volume: 84, Issue:2

    Topics: Animals; Capsaicin; Cells, Cultured; Diterpenes; Kinetics; Membrane Potentials; Neurons, Afferent; Neurotoxins; Patch-Clamp Techniques; Phorbol Esters; Rats; Rats, Sprague-Dawley; Receptors, Drug; Structure-Activity Relationship; Trigeminal Ganglion

1998
Specific vanilloid responses in C6 rat glioma cells.
    Brain research. Molecular brain research, 1998, Volume: 56, Issue:1-2

    Topics: Animals; Calcium Radioisotopes; Capsaicin; Cell Differentiation; Cell Division; Diterpenes; Glioma; Neurotoxins; Rats; Receptors, Drug; Tumor Cells, Cultured

1998
Capsaicin treatment induces muscarinic hyperreactivity in guinea pig trachea: a warning.
    European journal of pharmacology, 1998, Apr-24, Volume: 347, Issue:2-3

    Topics: Animals; Bronchoconstriction; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Receptors, Muscarinic; Receptors, Tachykinin; Trachea

1998
The cAMP transduction cascade mediates the prostaglandin E2 enhancement of the capsaicin-elicited current in rat sensory neurons: whole-cell and single-channel studies.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Aug-15, Volume: 18, Issue:16

    Topics: Animals; Capsaicin; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Electric Conductivity; Ion Channel Gating; Ion Channels; Neurons, Afferent; Osmolar Concentration; Rats; Rats, Sprague-Dawley

1998
Capsaicin receptors mediate free radical-induced activation of cardiac afferent endings.
    Cardiovascular research, 1998, Volume: 38, Issue:2

    Topics: Adrenergic Fibers; Animals; Bradykinin; Capsaicin; Coloring Agents; Free Radicals; Heart; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, Drug; Ruthenium Red; Sensory Receptor Cells; Stellate Ganglion; Vagus Nerve; Xanthine; Xanthine Oxidase

1998
Mechanism of acid-induced mesenteric hyperemia in rats.
    Life sciences, 1998, Volume: 63, Issue:18

    Topics: Animals; Blood Pressure; Capsaicin; Duodenum; Hydrochloric Acid; Hyperemia; Laser-Doppler Flowmetry; Male; Mesenteric Arteries; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Ruthenium Red

1998
Capsaicin-induced desensitization is prevented by capsazepine but not by ruthenium red in guinea pig bronchi.
    European journal of pharmacology, 1998, Dec-04, Volume: 362, Issue:2-3

    Topics: Animals; Bronchi; Calcium; Capsaicin; Coloring Agents; Guinea Pigs; Male; Muscle Contraction; Muscle Relaxation; Ruthenium Red

1998
A capsaicin-receptor antagonist, capsazepine, reduces inflammation-induced hyperalgesic responses in the rat: evidence for an endogenous capsaicin-like substance.
    Neuroscience, 1998, Volume: 86, Issue:2

    Topics: Animals; Capsaicin; Carrageenan; Functional Laterality; Hindlimb; Hyperalgesia; Inflammation; Male; Neurons; Pain; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reflex; Spinal Cord

1998
Stimulation of airway sensory nerves by cyclosporin A and FK506 in guinea-pig isolated bronchus.
    British journal of pharmacology, 1998, Volume: 125, Issue:7

    Topics: Animals; Bronchi; Bronchoconstriction; Capsaicin; Cyclosporine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Immunosuppressive Agents; In Vitro Techniques; Muscle, Smooth; Neurons, Afferent; Neuropeptides; Receptors, Cholinergic; Tacrolimus

1998
Anandamide transport inhibition by the vanilloid agonist olvanil.
    European journal of pharmacology, 1999, Jan-01, Volume: 364, Issue:1

    Topics: Amidohydrolases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acids; Astrocytoma; Biological Transport; Brain; Capsaicin; Depression, Chemical; Endocannabinoids; Humans; Polyunsaturated Alkamides; Rats; Receptors, Drug; Tumor Cells, Cultured

1999
Inhibition by a capsaicin antagonist (capsazepine) of capsaicin-induced swimming capacity increase in mice.
    Bioscience, biotechnology, and biochemistry, 1998, Volume: 62, Issue:12

    Topics: Animals; Capsaicin; Chromatography, High Pressure Liquid; Epinephrine; Male; Mice; Physical Exertion; Receptors, Drug; Swimming

1998
Mechanisms of capsaicin- and lactic acid-induced bronchoconstriction in the newborn dog.
    The Journal of physiology, 1999, Mar-01, Volume: 515 ( Pt 2)

    Topics: Animals; Animals, Newborn; Bronchi; Bronchoconstriction; Capsaicin; Dogs; Lactic Acid; Lung; Lung Compliance; Nerve Fibers; Receptors, Drug; Reflex

1999
Modulation by nitric oxide (NO) of capsaicin-induced calcium uptake into rat dorsal root ganglion neurons.
    Biochemistry and molecular biology international, 1999, Volume: 47, Issue:3

    Topics: Animals; Calcium; Capsaicin; Dithionitrobenzoic Acid; Dithiothreitol; Ganglia, Spinal; Neurons; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Nitroprusside; Rats; Rats, Sprague-Dawley; Spermine; Verapamil

1999
Systemically administered capsazepine prevents the capsaicin-induced functional desensitization and loss of substance P-like immunoreactivity (SP-LI) in guinea-pig bronchi.
    Life sciences, 1999, Volume: 64, Issue:14

    Topics: Animals; Bronchi; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; Male; Substance P

1999
A non-pungent triprenyl phenol of fungal origin, scutigeral, stimulates rat dorsal root ganglion neurons via interaction at vanilloid receptors.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Animals; Basidiomycota; Binding, Competitive; Calcium; Calcium Radioisotopes; Capsaicin; Cells, Cultured; Diterpenes; Dose-Response Relationship, Drug; Eye; Female; Ganglia, Spinal; Humans; Irritants; Male; Membrane Potentials; Membranes; Neurons; Patch-Clamp Techniques; Phenols; Rats; Rats, Sprague-Dawley; Receptors, Drug; Spinal Cord; Taste; Tongue; Tritium

1999
Action of capsaicin on dorsal root-evoked synaptic transmission to substantia gelatinosa neurons in adult rat spinal cord slices.
    Brain research, 1999, Jun-05, Volume: 830, Issue:2

    Topics: Animals; Capsaicin; Evoked Potentials; Ganglia, Spinal; In Vitro Techniques; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Spinal Cord; Substantia Gelatinosa; Synaptic Transmission

1999
Respiratory action of capsaicin microinjected into the nucleus of the solitary tract: involvement of vanilloid and tachykinin receptors.
    British journal of pharmacology, 1999, Volume: 127, Issue:2

    Topics: Anesthesia; Animals; Benzamides; Capsaicin; Dose-Response Relationship, Drug; Indoles; Isoindoles; Male; Microinjections; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Respiratory Mechanics; Solitary Nucleus; Tidal Volume

1999
Rat peripheral nerve components release calcitonin gene-related peptide and prostaglandin E2 in response to noxious stimuli: evidence that nervi nervorum are nociceptors.
    Neuroscience, 1999, Volume: 92, Issue:1

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Dinoprostone; Electric Stimulation; Inflammation Mediators; Male; Nociceptors; Pain; Peripheral Nerves; Rats; Rats, Wistar; Ruthenium Red; Stimulation, Chemical

1999
Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide.
    Nature, 1999, Jul-29, Volume: 400, Issue:6743

    Topics: Animals; Arachidonic Acids; Basilar Artery; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium Channels; Capsaicin; Cell Line; Endocannabinoids; Female; Guinea Pigs; Hepatic Artery; In Vitro Techniques; Neurons, Afferent; Peptide Fragments; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Recombinant Proteins; Vasodilator Agents; Xenopus

1999
Acid-sensing pathways of rat duodenum.
    The American journal of physiology, 1999, Volume: 277, Issue:2

    Topics: Acids; Animals; Bradykinin; Capsaicin; Chemoreceptor Cells; Duodenum; Hyperemia; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug; Regional Blood Flow; Time Factors

1999
The cloned rat vanilloid receptor VR1 mediates both R-type binding and C-type calcium response in dorsal root ganglion neurons.
    Molecular pharmacology, 1999, Volume: 56, Issue:3

    Topics: Animals; Biological Transport; Calcium; Calcium-Binding Proteins; Capsaicin; Cell Membrane; Cells, Cultured; CHO Cells; Cricetinae; Diterpenes; Ganglia, Spinal; Humans; Neurons; Nociceptors; Rats; Receptors, Drug; Transfection; Tritium; TRPV Cation Channels; Vanillic Acid

1999
Similarities and differences between the responses of rat sensory neurons to noxious heat and capsaicin.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Dec-15, Volume: 19, Issue:24

    Topics: Animals; Calcium; Capsaicin; Cell Survival; Cells, Cultured; Electrophysiology; Hot Temperature; Ion Channels; Neurons, Afferent; Rats; Ruthenium Red

1999
Inhibition of rapid heat responses in nociceptive primary sensory neurons of rats by vanilloid receptor antagonists.
    Journal of neurophysiology, 1999, Volume: 82, Issue:6

    Topics: Animals; Capsaicin; Dose-Response Relationship, Drug; Electrophysiology; Female; Ganglia, Spinal; Hot Temperature; Male; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Drug; Ruthenium Red; Signal Transduction; Solutions

1999
Inhibitory effect of capsaicin on cholinergic transmission in ovine airways: evidence for non-cholinergic contractions.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Acetylcholine; Animals; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptides, Cyclic; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-2; Serotonin; Sheep; Substance P; Synaptic Transmission; Trachea

1999
Stimulation of dichlorofluorescin oxidation by capsaicin and analogues in RAW 264 monocyte/macrophages: lack of involvement of the vanilloid receptor.
    Biochemical pharmacology, 2000, Mar-01, Volume: 59, Issue:5

    Topics: Acetylcysteine; Animals; Antioxidants; Capsaicin; Carcinogens; Chromans; Fluoresceins; Macrophages; Mice; Monocytes; Oxidation-Reduction; Polysorbates; Reactive Oxygen Species; Receptors, Drug; Surface-Active Agents; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Vitamin K

2000
Modulation of capsaicin-sensitive nerve activation by low pH solutions in guinea-pig lung.
    Pharmacology & toxicology, 2000, Volume: 86, Issue:1

    Topics: Animals; Bronchoconstriction; Buffers; Calcitonin Gene-Related Peptide; Capsaicin; Cyclooxygenase Inhibitors; Diclofenac; Drug Synergism; Female; Guinea Pigs; Hydrogen-Ion Concentration; Lactic Acid; Lung; Male; Neurons, Afferent

2000
Anandamide: an endogenous activator of the vanilloid receptor.
    Trends in pharmacological sciences, 2000, Volume: 21, Issue:4

    Topics: Animals; Arachidonic Acids; Cannabinoids; Capsaicin; Endocannabinoids; Humans; Ligands; Polyunsaturated Alkamides; Receptors, Drug

2000
Interactions of inflammatory mediators and low pH not influenced by capsazepine in rat cutaneous nociceptors.
    Neuroreport, 2000, Apr-07, Volume: 11, Issue:5

    Topics: Animals; Bradykinin; Capsaicin; Dinoprostone; Drug Interactions; Ganglia, Spinal; Hydrogen-Ion Concentration; Inflammation; Inflammation Mediators; Male; Nerve Fibers; Nociceptors; Oxytocics; Protons; Rats; Rats, Wistar; Serotonin; Signal Transduction; Skin

2000
Cytotoxicity of capsaicin in monkey kidney cells: lack of antagonistic effects of capsazepine and Ruthenium red.
    Archives of toxicology, 2000, Volume: 74, Issue:1

    Topics: Animals; Calcium; Capsaicin; Chlorocebus aethiops; Chromatography, High Pressure Liquid; DNA; Kidney; Mitochondria; Protein Synthesis Inhibitors; Receptors, Drug; Ruthenium Red; Spectrometry, Fluorescence; TRPV Cation Channels; Tyrosine; Vero Cells

2000
Direct activation of capsaicin receptors by products of lipoxygenases: endogenous capsaicin-like substances.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, May-23, Volume: 97, Issue:11

    Topics: Animals; Capsaicin; Cell Line; Cells, Cultured; Dinoprostone; Eicosanoids; Ganglia, Spinal; Humans; Hydroxyeicosatetraenoic Acids; Inflammation; Ion Channel Gating; Leukotriene B4; Leukotrienes; Ligands; Lipid Peroxides; Lipoxygenase; Molecular Structure; Neurons, Afferent; Prostaglandin D2; Prostaglandin H2; Prostaglandins H; Rats; Receptors, Drug; Structure-Activity Relationship

2000
Voltage- and time-dependent properties of the recombinant rat vanilloid receptor (rVR1).
    The Journal of physiology, 2000, Jun-15, Volume: 525 Pt 3

    Topics: Action Potentials; Animals; Barium; Calcium; Capsaicin; Cells, Cultured; Ganglia, Spinal; Humans; Ion Channel Gating; Kidney; Kinetics; Magnesium; Neurons; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Inbred Strains; Receptors, Drug; Recombinant Proteins; Time Factors; Transfection

2000
Inflammatory mediators release calcitonin gene-related peptide from dorsal root ganglion neurons of the rat.
    Neuroscience, 2000, Volume: 98, Issue:1

    Topics: Acids; Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cells, Cultured; Dinoprostone; Female; Free Radical Scavengers; Ganglia, Spinal; Hydrogen-Ion Concentration; Inflammation Mediators; Kallidin; Male; Neurons; Rats; Rats, Wistar; Receptors, Drug; Serotonin; Stimulation, Chemical

2000
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Animals; Calcium; Capsaicin; Cell Line; Diterpenes; DNA, Recombinant; Dose-Response Relationship, Drug; Fluorometry; Humans; Hydrogen-Ion Concentration; Ligands; Phorbol Esters; Polycyclic Sesquiterpenes; Rats; Receptors, Drug; Ruthenium Red; Sesquiterpenes; Transfection

2000
Involvement of kinins, mast cells and sensory neurons in the plasma exudation and paw oedema induced by staphylococcal enterotoxin B in the mouse.
    European journal of pharmacology, 2000, Jul-07, Volume: 399, Issue:2-3

    Topics: Animals; Benzamides; Bradykinin; Capillary Permeability; Capsaicin; Diabetes Mellitus, Experimental; Edema; Enterotoxins; Hindlimb; Kinins; Male; Mast Cells; Mice; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Pyrilamine; Quinuclidines; Receptors, Neurokinin-2

2000
Low-threshold heat response antagonized by capsazepine in chick sensory neurons, which are capsaicin-insensitive.
    The European journal of neuroscience, 2000, Volume: 12, Issue:10

    Topics: Animals; Capsaicin; Cell Size; Cells, Cultured; Chickens; Cobalt; Ganglia, Spinal; Hot Temperature; Ion Channels; Male; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Ruthenium Red; Thermosensing

2000
Induction of apoptosis by capsaicin in A172 human glioblastoma cells.
    Cancer letters, 2000, Dec-08, Volume: 161, Issue:1

    Topics: Apoptosis; Brain Neoplasms; Calcium; Capsaicin; Dose-Response Relationship, Drug; Glioblastoma; Humans; Kinetics; Lipid Peroxidation; Reactive Oxygen Species; Receptors, Drug; Tumor Cells, Cultured

2000
Functional and desensitizing effects of the novel synthetic vanilloid-like agent 12-phenylacetate 13-acetate 20-homovanillate (PPAHV) in the perfused rat hindlimb.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Capsaicin; Dose-Response Relationship, Drug; Hindlimb; Male; Oxygen Consumption; Perfusion; Phorbol Esters; Rats; Rats, Wistar; Vascular Resistance; Vasoconstriction

2000
In vivo pharmacology of SDZ 249-665, a novel, non-pungent capsaicin analogue.
    Pain, 2000, Dec-15, Volume: 89, Issue:1

    Topics: Analgesics; Animals; Behavior, Animal; Blinking; Blood Pressure; Bronchoconstriction; Capsaicin; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Tolerance; Eye; Female; Ganglia, Spinal; Guinea Pigs; Hindlimb; Hyperalgesia; Irritants; Male; Mice; Mice, Inbred Strains; Nociceptors; Nose; Odorants; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Turpentine; Urea

2000
Differential effects of capsaicin on rat visceral sensory neurons.
    Neuroscience, 2000, Volume: 101, Issue:3

    Topics: Action Potentials; Animals; Calcium; Capsaicin; Cells, Cultured; Intracellular Fluid; Male; Neurons, Afferent; Nociceptors; Nodose Ganglion; Potassium Channels; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium Channels; Tetrodotoxin; TRPV Cation Channels; Visceral Afferents

2000
ACTH inhibits the capsaicin-evoked release of CGRP from rat adrenal afferent nerves.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 280, Issue:1

    Topics: Adrenocorticotropic Hormone; Aldosterone; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, Drug; TRPV Cation Channels; Zona Glomerulosa

2001
Anandamide activates peripheral nociceptors in normal and arthritic rat knee joints.
    British journal of pharmacology, 2001, Volume: 132, Issue:3

    Topics: Animals; Arachidonic Acids; Arthritis, Experimental; Calcium Channel Blockers; Capsaicin; Disease Models, Animal; Drug Interactions; Endocannabinoids; Knee Joint; Male; Nociceptors; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Drug; Treatment Outcome; TRPV Cation Channels

2001
Structure-activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens.
    British journal of pharmacology, 2001, Volume: 132, Issue:3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Biological Transport; Calcium; Calcium Channel Blockers; Cannabinoids; Capsaicin; CHO Cells; Cricetinae; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Morpholines; Muscle Contraction; Naphthalenes; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Structure-Activity Relationship; Transfection; TRPV Cation Channels; Vas Deferens

2001
Anandamide excites central terminals of dorsal root ganglion neurons via vanilloid receptor-1 activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Feb-15, Volume: 21, Issue:4

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Ganglia, Spinal; In Vitro Techniques; Male; Neurons, Afferent; Polyunsaturated Alkamides; Presynaptic Terminals; Rats; Receptors, Cannabinoid; Receptors, Drug; Spinal Cord; Substance P; TRPV Cation Channels

2001
Regional differences in anandamide- and methanandamide-induced membrane potential changes in rat mesenteric arteries.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:2

    Topics: Animals; Arachidonic Acids; Benzoxazines; Biological Factors; Calcium Channel Blockers; Cannabinoids; Capsaicin; Electrophysiology; Endocannabinoids; Endothelium, Vascular; Membrane Potentials; Mesenteric Arteries; Morpholines; Muscle, Smooth, Vascular; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Drug; Rimonabant; Vasodilator Agents

2001
Sensory pathways and cyclooxygenase regulate mucus gel thickness in rat duodenum.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 280, Issue:3

    Topics: Animals; Bradykinin; Capsaicin; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Duodenum; Enzyme Inhibitors; Injections, Intravenous; Intestinal Mucosa; Mucus; Perfusion; Prostaglandin-Endoperoxide Synthases; Rats; Signal Transduction

2001
Pharmacological differences between the human and rat vanilloid receptor 1 (VR1).
    British journal of pharmacology, 2001, Volume: 132, Issue:5

    Topics: Amino Acid Sequence; Animals; Calcium; Capsaicin; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Female; Hot Temperature; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Molecular Sequence Data; Phorbol Esters; Rats; Receptors, Drug; Ruthenium Red; Species Specificity; Xenopus

2001
Comparison of intracellular calcium signals evoked by heat and capsaicin in cultured rat dorsal root ganglion neurons and in a cell line expressing the rat vanilloid receptor, VR1.
    Neuroscience, 2001, Volume: 102, Issue:1

    Topics: Animals; Calcium; Calcium Signaling; Capsaicin; Cells, Cultured; Coloring Agents; Cricetinae; Female; Ganglia, Spinal; Hot Temperature; Intracellular Fluid; Membrane Potentials; Neurons; Ovary; Rats; Rats, Sprague-Dawley; Receptors, Drug; Ruthenium Red; TRPV Cation Channels

2001
Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology.
    European journal of pharmacology, 2001, Apr-06, Volume: 417, Issue:1-2

    Topics: Alkaloids; Aniline Compounds; Arachidonic Acids; Benzophenanthridines; Calcium; Capsaicin; Cell Line; Diterpenes; Dose-Response Relationship, Drug; Endocannabinoids; Enzyme Inhibitors; Fluorescence; Fluorometry; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Phenanthridines; Polycyclic Sesquiterpenes; Polyunsaturated Alkamides; Protein Kinase C; Receptors, Drug; Ruthenium Red; Sesquiterpenes; Time Factors; Xanthenes

2001
Capsazepine, a vanilloid receptor antagonist, inhibits the expression of inducible nitric oxide synthase gene in lipopolysaccharide-stimulated RAW264.7 macrophages through the inactivation of nuclear transcription factor-kappa B.
    International immunopharmacology, 2001, Volume: 1, Issue:4

    Topics: Animals; Capsaicin; Cell Line; Gene Expression Regulation, Enzymologic; Lipopolysaccharides; Macrophages; Mice; NF-kappa B; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Receptors, Drug; RNA, Messenger

2001
Capsaicin-induced relaxation in rabbit coronary artery.
    The Journal of veterinary medical science, 2001, Volume: 63, Issue:5

    Topics: 4-Aminopyridine; Animals; Calcium; Capsaicin; Coronary Vessels; Dinoprost; Drug Interactions; Fluorescent Dyes; Fura-2; In Vitro Techniques; Isometric Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Peptides; Potassium Channel Blockers; Potassium Channels; Rabbits; Ruthenium Red

2001
Genital grooming and emesis induced by vanilloids in Suncus murinus, the house musk shrew.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Animals; Behavior, Animal; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Grooming; Injections, Intraventricular; Male; Sexual Behavior, Animal; Shrews; Time Factors; Vomiting

2001
Temperature-dependent activation of recombinant rat vanilloid VR1 receptors expressed in HEK293 cells by capsaicin and anandamide.
    European journal of pharmacology, 2001, Jul-06, Volume: 423, Issue:2-3

    Topics: Animals; Arachidonic Acids; Calcium; Cannabinoid Receptor Modulators; Capsaicin; Cell Line; Dose-Response Relationship, Drug; Endocannabinoids; Gene Expression; Humans; Polyunsaturated Alkamides; Rats; Receptors, Drug; Recombinant Proteins; Ruthenium Red; Temperature

2001
Effects of capsaicin on Ca(2+) release from the intracellular Ca(2+) stores in the dorsal root ganglion cells of adult rats.
    Biochemical and biophysical research communications, 2001, Aug-03, Volume: 285, Issue:5

    Topics: Animals; Bradykinin; Caffeine; Calcium; Calcium Channels; Capsaicin; Cells, Cultured; Cytophotometry; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Ganglia, Spinal; Inositol 1,4,5-Trisphosphate Receptors; Intracellular Fluid; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Receptors, Drug; Ryanodine Receptor Calcium Release Channel; Signal Transduction; Type C Phospholipases

2001
Vanilloid receptor expression and capsaicin excitation of rat dental primary afferent neurons.
    Journal of dental research, 2001, Volume: 80, Issue:6

    Topics: Animals; Capsaicin; Carbocyanines; Cells, Cultured; Dental Pulp; Electrophysiology; Fluorescent Dyes; Male; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Trigeminal Ganglion

2001
The capsaicin VR1 receptor mediates substance P release in toxin A-induced enteritis in rats.
    Peptides, 2001, Volume: 22, Issue:9

    Topics: Acute-Phase Reaction; Animals; Bacterial Toxins; Capsaicin; Clostridioides difficile; Dose-Response Relationship, Drug; Drug Interactions; Endocytosis; Enteritis; Enterotoxins; Ileum; Immunohistochemistry; Intestinal Secretions; Male; Neurogenic Inflammation; Neurons; Peroxidase; Rats; Receptors, Drug; Substance P; Time Factors

2001
A possible role of lipoxygenase in the activation of vanilloid receptors by anandamide in the guinea-pig bronchus.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonic Acids; Bronchi; Calcium Channel Blockers; Capsaicin; Cyclohexanols; Dose-Response Relationship, Drug; Endocannabinoids; Fatty Acids, Unsaturated; Guinea Pigs; Hydrazines; In Vitro Techniques; Indomethacin; Lipoxygenase; Muscle Contraction; Oxazepines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Thiorphan

2001
Differential effects of anandamide on acetylcholine release in the guinea-pig ileum mediated via vanilloid and non-CB1 cannabinoid receptors.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: Acetylcholine; Animals; Arachidonic Acids; Camphanes; Capsaicin; Cyclohexanols; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methacholine Chloride; Muscle Contraction; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2001
Propofol activates vanilloid receptor channels expressed in human embryonic kidney 293 cells.
    Neuroscience letters, 2001, Oct-12, Volume: 312, Issue:1

    Topics: Anesthetics, Intravenous; Binding Sites; Calcium; Calcium Signaling; Capsaicin; Cells, Cultured; Diterpenes; Dose-Response Relationship, Drug; Humans; Membrane Potentials; Nervous System; Pain; Patch-Clamp Techniques; Propofol; Receptors, Drug

2001
Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Amidohydrolases; Arachidonic Acids; Binding, Competitive; Biological Transport; Calcium; Cannabidiol; Capsaicin; Cell Line; Cell Membrane; Cytosol; Dose-Response Relationship, Drug; Endocannabinoids; Gene Expression; Humans; Hydrolysis; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug

2001
Mechanisms of anandamide-induced vasorelaxation in rat isolated coronary arteries.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Amides; Animals; Arachidonic Acids; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Ethanolamines; Gap Junctions; Glycyrrhetinic Acid; In Vitro Techniques; Indoles; Indomethacin; Male; Palmitic Acids; Peptides; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Serotonin; Tetraethylammonium; Vasodilation

2001
Capsaicin vanilloid receptor-1 mediates substance P release in experimental pancreatitis.
    American journal of physiology. Gastrointestinal and liver physiology, 2001, Volume: 281, Issue:5

    Topics: Amylases; Animals; Capsaicin; Endocytosis; Male; Mice; Mice, Inbred C57BL; Pancreas; Pancreatitis; Peroxidase; Receptors, Drug; Receptors, Neurokinin-1; Severity of Illness Index; Substance P; TRPV Cation Channels

2001
Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 4-Aminopyridine; Animals; Apamin; Arachidonic Acid; Arachidonic Acids; Barium; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Coronary Vessels; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Fatty Acids, Unsaturated; Glyburide; In Vitro Techniques; Indomethacin; Miconazole; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptides; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Potassium; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Receptors, Drug; Rimonabant; Sheep; Tetraethylammonium; Vasoconstrictor Agents; Vasodilation

2001
Capsaicin-evoked CGRP release from rat buccal mucosa: development of a model system for studying trigeminal mechanisms of neurogenic inflammation.
    The European journal of neuroscience, 2001, Volume: 14, Issue:7

    Topics: Animals; Bradykinin; Calcimycin; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Histamine; Inflammation Mediators; Ionophores; Male; Mouth Mucosa; Neurogenic Inflammation; Nociceptors; Organ Culture Techniques; Pain Measurement; Potassium Chloride; Rats; Rats, Sprague-Dawley; Serotonin; Trigeminal Nerve

2001
Stimulatory effect of centrally injected capsaicin, an agonist of vanilloid receptors, on gastric acid secretion in rats.
    European journal of pharmacology, 2001, Oct-12, Volume: 428, Issue:3

    Topics: Animals; Capsaicin; Dose-Response Relationship, Drug; Gastric Acid; Gastric Mucosa; Injections, Intraventricular; Male; Rats; Rats, Wistar; Receptors, Drug; Ruthenium; Stomach; Time Factors; Vagotomy; Vagus Nerve

2001
Noxious heat-induced CGRP release from rat sciatic nerve axons in vitro.
    The European journal of neuroscience, 2001, Volume: 14, Issue:8

    Topics: Animals; Axons; Calcitonin Gene-Related Peptide; Capsaicin; Coloring Agents; Dose-Response Relationship, Drug; Ganglia, Spinal; Hot Temperature; Male; Nociceptors; Pain; Potassium; Rats; Rats, Wistar; Receptors, Drug; Ruthenium Red; Sciatic Nerve

2001
Inhibition of rat C6 glioma cell proliferation by endogenous and synthetic cannabinoids. Relative involvement of cannabinoid and vanilloid receptors.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:3

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Arachidonic Acids; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Cell Division; Glioma; Piperidines; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Tumor Cells, Cultured

2001
Involvement of vanilloid receptor VR1 and prostanoids in the acid-induced writhing responses of mice.
    Life sciences, 2001, Nov-02, Volume: 69, Issue:24

    Topics: Acetic Acid; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Benzoquinones; Bradykinin; Capsaicin; Disease Models, Animal; Female; Indomethacin; Lactic Acid; Male; Mice; Mice, Inbred ICR; Pain; Pain Measurement; Propionates; Prostaglandins; Receptors, Drug; Receptors, Prostaglandin

2001
Acidic stimuli activates two distinct pathways in taste receptor cells from rat fungiform papillae.
    Brain research, 2001, Dec-27, Volume: 923, Issue:1-2

    Topics: Acid Sensing Ion Channels; Acids; Adjuvants, Immunologic; Amiloride; Animals; Calcium; Capsaicin; Chemoreceptor Cells; Cholera Toxin; Diuretics; Dose-Response Relationship, Drug; Female; GTP-Binding Proteins; Male; Membrane Proteins; Nerve Tissue Proteins; Pertussis Toxin; Protons; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; Sodium Channels; Stimulation, Chemical; Tachyphylaxis; Taste; Taste Buds; Virulence Factors, Bordetella

2001
CH-19 sweet, nonpungent cultivar of red pepper, increased body temperature in mice with vanilloid receptors stimulation by capsiate.
    Journal of nutritional science and vitaminology, 2001, Volume: 47, Issue:4

    Topics: Animals; Body Temperature; Capsaicin; Capsicum; Male; Mice; Receptors, Drug; Stimulation, Chemical

2001
Capsaicin-, resiniferatoxin-, and olvanil-induced adrenaline secretions in rats via the vanilloid receptor.
    Bioscience, biotechnology, and biochemistry, 2001, Volume: 65, Issue:11

    Topics: Adrenal Glands; Animals; Capsaicin; Diterpenes; Epinephrine; Rats; Rats, Sprague-Dawley; Receptors, Drug

2001
Functional vanilloid receptors in cultured normal human epidermal keratinocytes.
    Biochemical and biophysical research communications, 2002, Feb-15, Volume: 291, Issue:1

    Topics: Acids; Calcium; Capsaicin; Cells, Cultured; Epidermal Cells; Epidermis; Humans; Hydrogen-Ion Concentration; Intracellular Fluid; Keratinocytes; Receptors, Drug

2002
Pharmacological characterization of vanilloid receptor located in the brain.
    Brain research. Molecular brain research, 2002, Jan-31, Volume: 98, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain Chemistry; Capsaicin; Diterpenes; Ganglia, Spinal; Hippocampus; Kinetics; Locus Coeruleus; Macaca fascicularis; Neurons, Afferent; Organ Specificity; Preoptic Area; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; Spinal Cord; Structure-Activity Relationship; TRPV Cation Channels

2002
Relaxant effect of capsazepine in the isolated rat ileum.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 365, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Calcium Channels, L-Type; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Gastrointestinal Transit; Ileum; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptors, Drug

2002
Protease-activated receptor-2 activation causes EDHF-like coronary vasodilation: selective preservation in ischemia/reperfusion injury: involvement of lipoxygenase products, VR1 receptors, and C-fibers.
    Circulation research, 2002, Mar-08, Volume: 90, Issue:4

    Topics: Acetylcholine; Animals; Biological Factors; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Lipoxygenase; Male; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion Injury; Nerve Fibers; Oligopeptides; Potassium; Potassium Channel Blockers; Rats; Rats, Wistar; Receptor, PAR-2; Receptors, Drug; Receptors, Thrombin; Trypsin; Vasodilation

2002
3-D-QSAR analysis of N-(3-acyloxy-2-benzylpropyl)-N'-dihydroxytetrahydrobenzazepine and tetrahydroisoquinoline and N-(3-acyloxy-2-benzylpropyl)-N'-(4-hydroxy-3-methoxybenzyl) thioureas analogues as potent vanilloid receptor ligands.
    Bioorganic & medicinal chemistry, 2002, Volume: 10, Issue:5

    Topics: Analgesics; Animals; Benzazepines; Capsaicin; Cells, Cultured; Isoquinolines; Ligands; Models, Molecular; Protein Binding; Quantitative Structure-Activity Relationship; Rats; Receptors, Drug; Thiourea

2002
Stimulation of pulmonary vagal C-fibres by anandamide in anaesthetized rats: role of vanilloid type 1 receptors.
    The Journal of physiology, 2002, Mar-15, Volume: 539, Issue:Pt 3

    Topics: Afferent Pathways; Animals; Arachidonic Acids; Capsaicin; Cardiovascular System; Chemoreceptor Cells; Dose-Response Relationship, Drug; Electrophysiology; Endocannabinoids; Lung; Male; Morpholines; Nerve Fibers; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reflex; TRPV Cation Channels; Vagus Nerve

2002
Interaction between vanilloid and glutamate receptors in the central modulation of nociception.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Capsaicin; Chromones; Excitatory Amino Acid Antagonists; Male; Pain; Periaqueductal Gray; Phosphoserine; Piperidines; Protein Binding; Pyrazoles; Pyridines; Rats; Rats, Wistar; Receptors, Drug; Receptors, Glutamate; Riluzole; Rimonabant; Time Factors

2002
Capsazepine partially inhibits neurally mediated gastric mucus secretion following activation of protease-activated receptor 2.
    Clinical and experimental pharmacology & physiology, 2002, Volume: 29, Issue:4

    Topics: Animals; Capsaicin; Gastric Mucosa; Male; Neural Inhibition; Neurons, Afferent; Rats; Rats, Wistar; Receptor, PAR-2; Receptors, Drug; Receptors, Thrombin; TRPV Cation Channels

2002
Ethanol elicits and potentiates nociceptor responses via the vanilloid receptor-1.
    Nature neuroscience, 2002, Volume: 5, Issue:6

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Ethanol; Ganglia, Spinal; Hot Temperature; Humans; Male; Neurons, Afferent; Nociceptors; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Drug; Recombinant Proteins; Sensory Thresholds; Substance P; Thermoreceptors; Trigeminal Ganglion; TRPV Cation Channels

2002
Gastric hyperemic response induced by acid back-diffusion in rat stomachs following barrier disruption -- relation to vanilloid type-1 receptors.
    Medical science monitor : international medical journal of experimental and clinical research, 2002, Volume: 8, Issue:5

    Topics: Animals; Capsaicin; Diffusion; Gastric Acid; Gastric Mucosa; Hydrogen; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug; Ruthenium Red; Stomach; Stomach Ulcer; Taurocholic Acid; Time Factors; TRPV Cation Channels

2002
A heat-sensitive TRP channel expressed in keratinocytes.
    Science (New York, N.Y.), 2002, Jun-14, Volume: 296, Issue:5575

    Topics: Amino Acid Sequence; Animals; Animals, Newborn; Blotting, Northern; Capsaicin; Cation Transport Proteins; Cell Line; Cells, Cultured; CHO Cells; Cloning, Molecular; Cricetinae; Epidermal Cells; Epidermis; Ganglia, Spinal; Hot Temperature; Humans; In Situ Hybridization; Ion Channels; Keratinocytes; Membrane Potentials; Mice; Molecular Sequence Data; Nerve Endings; Neurons; Patch-Clamp Techniques; RNA, Messenger; Ruthenium Red; Signal Transduction; Spinal Cord; Temperature; TRPV Cation Channels

2002
Ischemia/reperfusion-induced increase in the hepatic level of prostacyclin is mainly mediated by activation of capsaicin-sensitive sensory neurons in rats.
    The Journal of laboratory and clinical medicine, 2002, Volume: 139, Issue:4

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cyclooxygenase 1; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Epoprostenol; Guanidines; Indomethacin; Isoenzymes; Liver; Liver Circulation; Male; Membrane Proteins; Miotics; Neurons, Afferent; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitrobenzenes; Peptide Fragments; Peroxidase; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Reperfusion Injury; Specific Pathogen-Free Organisms; Sulfonamides; Transaminases; Tumor Necrosis Factor-alpha

2002
DRASIC contributes to pH-gated currents in large dorsal root ganglion sensory neurons by forming heteromultimeric channels.
    Journal of neurophysiology, 2002, Volume: 87, Issue:6

    Topics: Acid Sensing Ion Channels; Acids; Amiloride; Animals; Capsaicin; Diuretics; FMRFamide; Ganglia, Spinal; Hydrogen-Ion Concentration; Ion Channel Gating; Membrane Potentials; Membrane Proteins; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons, Afferent; Neuropeptides; Protons; Sodium Channels

2002
Spinal administration of capsazepine inhibits noxious evoked responses of dorsal horn neurons in non-inflamed and carrageenan inflamed rats.
    Brain research, 2002, May-10, Volume: 935, Issue:1-2

    Topics: Action Potentials; Afferent Pathways; Animals; Capsaicin; Carrageenan; Dose-Response Relationship, Drug; Inflammation; Injections, Spinal; Male; Nerve Fibers; Nerve Fibers, Myelinated; Neural Inhibition; Nociceptors; Pain; Posterior Horn Cells; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Drug

2002
Capsazepine inhibits thermal hyperalgesia but not nociception triggered by protease-activated receptor-2 in rats.
    Japanese journal of pharmacology, 2002, Volume: 89, Issue:2

    Topics: Amino Acid Sequence; Animals; Capsaicin; Hot Temperature; Hyperalgesia; Male; Pain; Peptide Fragments; Rats; Rats, Wistar; Receptor, PAR-2; Receptors, Thrombin

2002
Comparison of capsaicin-evoked calcium transients between rat nodose and jugular ganglion neurons.
    Autonomic neuroscience : basic & clinical, 2002, May-31, Volume: 97, Issue:2

    Topics: Animals; Calcium; Capsaicin; Cell Count; Cells, Cultured; Dose-Response Relationship, Drug; Glomus Jugulare; Neurons; Nodose Ganglion; Rats; Rats, Sprague-Dawley

2002
Effects of peripheral nerve injury on functional spinal VR1 receptors.
    Neuroreport, 2002, Jul-02, Volume: 13, Issue:9

    Topics: Action Potentials; Animals; Capsaicin; Denervation; Dose-Response Relationship, Drug; Down-Regulation; Hyperalgesia; Ligation; Nerve Fibers; Nerve Fibers, Myelinated; Neuralgia; Neuronal Plasticity; Nociceptors; Pain Threshold; Peripheral Nerve Injuries; Peripheral Nerves; Peripheral Nervous System Diseases; Physical Stimulation; Posterior Horn Cells; Rats; Receptors, Drug

2002
Mechanisms underlying tissue selectivity of anandamide and other vanilloid receptor agonists.
    Molecular pharmacology, 2002, Volume: 62, Issue:3

    Topics: Animals; Arachidonic Acids; Bronchi; Bronchial Arteries; Calcium Channel Blockers; Capsaicin; Computer Simulation; Endocannabinoids; Guinea Pigs; Lung; Male; Mesenteric Arteries; Polyunsaturated Alkamides; Receptors, Drug

2002
Mechanisms of acid-induced activation of airway afferent nerve fibres in guinea-pig.
    The Journal of physiology, 2002, Sep-01, Volume: 543, Issue:Pt 2

    Topics: Action Potentials; Animals; Bicarbonates; Bronchi; Buffers; Capsaicin; Citric Acid; Dose-Response Relationship, Drug; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neurons, Afferent; Nodose Ganglion; Protons; Receptors, Drug; Trachea

2002
Effect of piperine, the active ingredient of black pepper, on intestinal secretion in mice.
    Life sciences, 2002, Sep-27, Volume: 71, Issue:19

    Topics: Alkaloids; Animals; Anti-Ulcer Agents; Benzodioxoles; Capsaicin; Castor Oil; Dose-Response Relationship, Drug; Drug Interactions; Injections, Intraperitoneal; Intestinal Secretions; Intestine, Small; Male; Mice; Mice, Inbred ICR; Organ Size; Piperidines; Polyunsaturated Alkamides

2002
Vanilloid receptors presynaptically modulate cranial visceral afferent synaptic transmission in nucleus tractus solitarius.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Sep-15, Volume: 22, Issue:18

    Topics: Animals; Baroreflex; Capsaicin; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Head; In Vitro Techniques; Male; Patch-Clamp Techniques; Pressoreceptors; Presynaptic Terminals; Pyridinium Compounds; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Drug; Receptors, Glutamate; Rhombencephalon; Solitary Nucleus; Synaptic Transmission; Visceral Afferents

2002
Cloning and functional characterization of the guinea pig vanilloid receptor 1.
    Neuropharmacology, 2002, Volume: 43, Issue:3

    Topics: Aequorin; Amino Acid Sequence; Animals; Calcium; Capsaicin; CHO Cells; Chronic Disease; Cloning, Molecular; Cricetinae; Fluorescent Dyes; Fura-2; Guinea Pigs; Heart; Hydrogen-Ion Concentration; Luminescent Measurements; Molecular Sequence Data; Pain; Rats; Receptors, Drug; TRPV Cation Channels

2002
Amiloride-blockable acid-sensing ion channels are leading acid sensors expressed in human nociceptors.
    The Journal of clinical investigation, 2002, Volume: 110, Issue:8

    Topics: Acid Sensing Ion Channels; Adult; Amiloride; Animals; Capsaicin; Female; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Membrane Proteins; Nerve Tissue Proteins; Nociceptors; Oocytes; Pain; Psychophysics; Rats; Receptors, Drug; Recombinant Proteins; Sodium Channels; Xenopus

2002
The putative role of vanilloid receptor-like protein-1 in mediating high threshold noxious heat-sensitivity in rat cultured primary sensory neurons.
    The European journal of neuroscience, 2002, Volume: 16, Issue:8

    Topics: Afferent Pathways; Animals; Calcium Signaling; Capsaicin; Cell Size; Cells, Cultured; Dose-Response Relationship, Drug; Ganglia, Spinal; Hot Temperature; Immunohistochemistry; Male; Membrane Potentials; Neurons, Afferent; Nociceptors; Pain; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, Drug; Ruthenium Red; Synaptic Transmission; Thermosensing; TRPV Cation Channels

2002
Gingerols: a novel class of vanilloid receptor (VR1) agonists.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Animals; Animals, Newborn; Calcium; Capsaicin; Catechols; Cells, Cultured; Dose-Response Relationship, Drug; Fatty Alcohols; Fura-2; Ganglia, Spinal; Membrane Potentials; Neurons; Rats; Receptors, Drug; Time Factors

2002
Anandamide induces cough in conscious guinea-pigs through VR1 receptors.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: Aerosols; Animals; Arachidonic Acids; Calcium; Camphanes; Capsaicin; Cells, Cultured; Consciousness; Cough; Dronabinol; Endocannabinoids; Excitatory Amino Acid Antagonists; Guinea Pigs; Male; Nodose Ganglion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
Upregulation of proinflammatory cytokines and nerve growth factor by intraplantar injection of capsaicin in rats.
    The Journal of physiology, 2002, 11-15, Volume: 545, Issue:1

    Topics: Administration, Topical; Animals; Capsaicin; Cytokines; Denervation; Electric Stimulation; Female; Foot; Inflammation Mediators; Injections; Nerve Growth Factor; Nociceptors; Rats; Sciatic Nerve; Up-Regulation

2002
Synthesis of 2-substituted-pyrrolidinethiourea derivatives and their antagonist effect on vanilloid receptor.
    Bioorganic & medicinal chemistry letters, 2003, Jan-20, Volume: 13, Issue:2

    Topics: Animals; Animals, Newborn; Calcium; Capsaicin; Crystallography, X-Ray; Indicators and Reagents; Models, Molecular; Molecular Conformation; Neurons, Afferent; Pyrrolidines; Rats; Receptors, Drug; Thiourea

2003
The VR1 antagonist capsazepine reverses mechanical hyperalgesia in models of inflammatory and neuropathic pain.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Algorithms; Animals; Anticonvulsants; Capsaicin; Carbamazepine; Dose-Response Relationship, Drug; Guinea Pigs; Hyperalgesia; Inflammation; Male; Mice; Mice, Inbred C57BL; Peripheral Nervous System Diseases; Rats; Rats, Wistar; Receptors, Drug; Sciatic Nerve

2003
Activation of epidermal vanilloid receptor-1 induces release of proinflammatory mediators in human keratinocytes.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Calcium; Calcium Signaling; Capsaicin; Cell Line; Cyclooxygenase 2; Dinoprostone; Humans; Immunoblotting; Inflammation Mediators; Interleukin-8; Isoenzymes; Keratinocytes; Membrane Proteins; Physical Stimulation; Prostaglandin-Endoperoxide Synthases; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Skin

2003
Concentration-dependent dual effect of anandamide on sensory neuropeptide release from isolated rat tracheae.
    Neuroscience letters, 2003, Jan-16, Volume: 336, Issue:2

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; In Vitro Techniques; Male; Neuropeptides; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Reference Values; Reproducibility of Results; Rimonabant; Sensitivity and Specificity; Somatostatin; Substance P; Trachea

2003
R+-methanandamide inhibits tracheal response to endogenously released acetylcholine via capsazepine-sensitive receptors.
    European journal of pharmacology, 2003, Jan-10, Volume: 459, Issue:1

    Topics: Acetylcholine; Animals; Arachidonic Acids; Atropine; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indoles; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Trachea

2003
The actions of anandamide on rat superficial medullary dorsal horn neurons in vitro.
    The Journal of physiology, 2003, Apr-01, Volume: 548, Issue:Pt 1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Capsaicin; Electric Stimulation; Electrophysiology; Endocannabinoids; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; In Vitro Techniques; Medulla Oblongata; Membrane Potentials; Nerve Endings; Patch-Clamp Techniques; Polyunsaturated Alkamides; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Trigeminal Ganglion

2003
Effect of arvanil (N-arachidonoyl-vanillyl-amine), a nonpungent anandamide-capsaicin hybrid, on ion currents in NG108-15 neuronal cells.
    Biochemical pharmacology, 2003, Feb-15, Volume: 65, Issue:4

    Topics: Action Potentials; Animals; Arachidonic Acids; Calcium Channels, L-Type; Capsaicin; Cell Line; Delayed Rectifier Potassium Channels; Drug Interactions; Endocannabinoids; Glycerol; Hybrid Cells; Mice; Neurons; omega-Conotoxin GVIA; Pertussis Toxin; Polyunsaturated Alkamides; Potassium Channels; Potassium Channels, Voltage-Gated; Rats

2003
Anandamide-induced depressor effect in spontaneously hypertensive rats: role of the vanilloid receptor.
    Hypertension (Dallas, Tex. : 1979), 2003, Volume: 41, Issue:3 Pt 2

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Endocannabinoids; Hypertension; Male; Mesenteric Arteries; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2003
Negatively charged 2- and 10-microm particles activate vanilloid receptors, increase cAMP, and induce cytokine release.
    Toxicology and applied pharmacology, 2003, Jan-15, Volume: 186, Issue:2

    Topics: Air Pollutants; Calcium; Capsaicin; Cell Line; Cyclic AMP; Humans; Interleukin-6; Receptors, Drug; Trigeminal Ganglion

2003
Vanilloid receptor-1 containing primary sensory neurones mediate dextran sulphate sodium induced colitis in rats.
    Gut, 2003, Volume: 52, Issue:5

    Topics: Animals; Capsaicin; Colitis, Ulcerative; Colon; Denervation; Dextran Sulfate; Disease Models, Animal; Neurons, Afferent; Peroxidase; Rats; Rats, Sprague-Dawley; Receptors, Drug; Severity of Illness Index; TRPV Cation Channels

2003
State-dependent phosphorylation of epsilon-isozyme of protein kinase C in adult rat dorsal root ganglia after inflammation and nerve injury.
    Journal of neurochemistry, 2003, Volume: 85, Issue:3

    Topics: Animals; Behavior, Animal; Capsaicin; Carrageenan; Disease Models, Animal; Diterpenes; Freund's Adjuvant; Ganglia, Spinal; Hindlimb; Hyperalgesia; Inflammation; Ligation; Male; Neurons; Nociceptors; Pain; Pain Measurement; Peripheral Nervous System Diseases; Phosphorylation; Protein Kinase C; Protein Kinase C-epsilon; Rats; Rats, Sprague-Dawley; Receptors, Drug

2003
Chain-branched acyclic phenethylthiocarbamates as vanilloid receptor antagonists.
    Bioorganic & medicinal chemistry letters, 2003, May-05, Volume: 13, Issue:9

    Topics: Animals; Calcium; Capsaicin; Cells, Cultured; Neurons, Afferent; Rats; Receptors, Drug; Spinal Cord; Structure-Activity Relationship; Thiocarbamates

2003
Peripheral tackykinin and excitatory amino acid receptors mediate hyperalgesia induced by Phoneutria nigriventer venom.
    European journal of pharmacology, 2003, Apr-25, Volume: 467, Issue:1-3

    Topics: Animals; Capsaicin; Edema; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hindlimb; Hyperalgesia; Male; Pain Threshold; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Drug; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Spider Venoms

2003
Inhibitory effect of the plant flavonoid galangin on rat vas deferens in vitro.
    Life sciences, 2003, May-16, Volume: 72, Issue:26

    Topics: Animals; Atropine; Capsaicin; Electric Stimulation; Enzyme Inhibitors; Flavonoids; Hexamethonium; Humans; In Vitro Techniques; Male; Molecular Structure; Muscarinic Antagonists; Naloxone; Narcotic Antagonists; NG-Nitroarginine Methyl Ester; Nicotinic Antagonists; Phenylephrine; Rats; Rats, Wistar; Receptors, Tachykinin; Vas Deferens; Vasoconstrictor Agents

2003
Presynaptic facilitation of glutamatergic synapses to dopaminergic neurons of the rat substantia nigra by endogenous stimulation of vanilloid receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Apr-15, Volume: 23, Issue:8

    Topics: Animals; Arachidonic Acids; Calcium; Calcium Channel Blockers; Capsaicin; Diterpenes; Dopamine; Dose-Response Relationship, Drug; Endocannabinoids; Excitatory Postsynaptic Potentials; GABA Antagonists; Glutamic Acid; In Vitro Techniques; Mesencephalon; Neurons; Patch-Clamp Techniques; Polyunsaturated Alkamides; Presynaptic Terminals; Rats; Rats, Wistar; Receptors, Drug; RNA, Messenger; Substantia Nigra; Synapses; Synaptic Transmission; Tetrodotoxin

2003
Differential effects of intraplantar capsazepine and ruthenium red on capsaicin-induced desensitization in mice.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 75, Issue:1

    Topics: Animals; Behavior, Animal; Capsaicin; Dose-Response Relationship, Drug; Foot; Injections; Male; Mice; Nociceptors; Pain; Receptors, Drug; Ruthenium Red

2003
The effects of local and intravenous anesthetics on recombinant rat VR1 vanilloid receptors.
    Anesthesia and analgesia, 2003, Volume: 96, Issue:6

    Topics: Anesthetics, Intravenous; Anesthetics, Local; Animals; Calcium; Capsaicin; Cell Line; Fluorescent Dyes; Fura-2; Humans; Rats; Receptors, Drug; Recombinant Proteins

2003
Involvement of capsaicin-sensitive sensory nerves in cardioprotection of rutaecarpine in rats.
    Regulatory peptides, 2003, Jun-15, Volume: 114, Issue:1

    Topics: Alkaloids; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cardiotonic Agents; Creatine Kinase; Heart; Indole Alkaloids; Male; Myocardial Infarction; Myocardial Reperfusion Injury; Neurons, Afferent; Organ Size; Quinazolines; Rats; Rats, Wistar

2003
Adrenergic regulation of capsaicin-sensitive neurons in dental pulp.
    Journal of endodontics, 2003, Volume: 29, Issue:6

    Topics: Adrenergic alpha-Agonists; Analysis of Variance; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cattle; Clonidine; Dental Pulp; Epinephrine; Ion Channels; Nerve Fibers, Unmyelinated; Nociceptors; Pain; Receptors, Adrenergic, alpha; Receptors, Drug

2003
Calcium signaling in single peripheral sensory nerve terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Jun-15, Volume: 23, Issue:12

    Topics: Action Potentials; Anesthetics, Local; Animals; Calcium; Calcium Channel Blockers; Calcium Signaling; Capsaicin; Cornea; Electric Stimulation; Fluorescent Dyes; In Vitro Techniques; Microscopy, Confocal; Neurons, Afferent; Peripheral Nerves; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Sodium Channel Blockers; Stimulation, Chemical

2003
Mechanisms of sensitization of the response of single dorsal root ganglion cells from adult rat to noxious heat.
    The European journal of neuroscience, 2003, Volume: 18, Issue:3

    Topics: Animals; Capsaicin; Ganglia, Spinal; Hot Temperature; Nerve Growth Factor; Neurons; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptor, trkA; Receptors, Drug; Tachyphylaxis; Type C Phospholipases

2003
Proton-induced calcitonin gene-related peptide release from rat sciatic nerve axons, in vitro, involving TRPV1.
    The European journal of neuroscience, 2003, Volume: 18, Issue:4

    Topics: Animals; Axons; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Hot Temperature; Hydrogen-Ion Concentration; Immunoenzyme Techniques; Male; Organ Culture Techniques; Potassium; Protons; Rats; Rats, Wistar; Receptors, Drug; Ruthenium Red; Sciatic Nerve

2003
Capsaicin-sensitive neurogenic sensory vasodilatation in the dura mater of the rat.
    The Journal of physiology, 2003, Nov-01, Volume: 552, Issue:Pt 3

    Topics: Administration, Topical; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Drug Resistance; Dura Mater; Humans; Male; Microscopy, Electron; Neurons, Afferent; Peptide Fragments; Rats; Rats, Wistar; Regional Blood Flow; Vasodilation

2003
Expression of vanilloid receptors in rat gastric epithelial cells: role in cellular protection.
    Biochemical pharmacology, 2003, Sep-15, Volume: 66, Issue:6

    Topics: Acids; Animals; Capsaicin; Diterpenes; Epithelial Cells; Ethanol; Gastric Mucosa; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug; RNA, Messenger; TRPV Cation Channels

2003
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
    Peptides, 2003, Volume: 24, Issue:7

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins

2003
Hypotensive effect of anandamide through the activation of CB1 and VR1 spinal receptors in urethane-anesthetized rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:4

    Topics: Anesthesia, Intravenous; Anesthetics, Intravenous; Animals; Antihypertensive Agents; Arachidonic Acids; Benzoxazines; Blood Pressure; Calcium Channel Blockers; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Ganglionic Blockers; Heart Rate; Hemodynamics; Hexamethonium; Injections, Spinal; Male; Morpholines; Naphthalenes; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; Spinal Cord; Urethane

2003
Activation of vanilloid receptor 1 (VR1) by eugenol.
    Journal of dental research, 2003, Volume: 82, Issue:10

    Topics: Animals; Calcium; Calcium Channels; Capsaicin; Cell Line; Chelating Agents; Electrophysiology; Eugenol; Fura-2; Humans; Neurons, Afferent; Patch-Clamp Techniques; Rats; Receptors, Drug; Ruthenium Red; Trigeminal Ganglion

2003
Signal transduction for inhibition of inducible nitric oxide synthase and cyclooxygenase-2 induction by capsaicin and related analogs in macrophages.
    British journal of pharmacology, 2003, Volume: 140, Issue:6

    Topics: Animals; Capsaicin; Cell Line; Cyclooxygenase 2; Dinoprostone; Diterpenes; DNA-Binding Proteins; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Induction; Ganglia, Spinal; I-kappa B Kinase; Interferon-gamma; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Lipopolysaccharides; Macrophages; Male; Mitogen-Activated Protein Kinases; Neurotoxins; NF-kappa B; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Prostaglandin-Endoperoxide Synthases; Protein Serine-Threonine Kinases; Rats; Rats, Sprague-Dawley; Receptors, Drug; RNA, Messenger; Signal Transduction; STAT1 Transcription Factor; Tetradecanoylphorbol Acetate; Trans-Activators; Transcription Factor AP-1

2003
Albaconol from the mushroom Albatrellus confluens induces contraction and desensitization in guinea pig trachea.
    Planta medica, 2003, Volume: 69, Issue:8

    Topics: Agaricales; Analgesics; Animals; Bridged Bicyclo Compounds; Calcium; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Phenols; Phytotherapy; Receptors, Drug; Trachea

2003
Vanilloid type 1 receptors (VR1) on trigeminal sensory nerve fibres play a minor role in neurogenic dural vasodilatation, and are involved in capsaicin-induced dural dilation.
    British journal of pharmacology, 2003, Volume: 140, Issue:4

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Dura Mater; Electric Stimulation; Injections, Intravenous; Male; Microscopy, Video; Neurons, Afferent; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Drug; Trigeminal Nerve; Vasodilation

2003
Stimulation by capsaicin of duodenal HCO3(-) secretion via afferent neurons and vanilloid receptors in rats: comparison with acid-induced HCO3(-) response.
    Digestive diseases and sciences, 2003, Volume: 48, Issue:9

    Topics: Animals; Bicarbonates; Capsaicin; Coloring Agents; Duodenum; Enzyme Inhibitors; Immunohistochemistry; Intestinal Mucosa; Male; Neurons, Afferent; NG-Nitroarginine Methyl Ester; Rats; Rats, Sprague-Dawley; Receptors, Drug; Regional Blood Flow; Ruthenium Red

2003
Neurokinin release produced by capsaicin acting on the central terminals and axons of primary afferents: relationship with N-methyl-D-aspartate and GABA(B) receptors.
    Neuroscience, 2003, Volume: 121, Issue:3

    Topics: Afferent Pathways; Analysis of Variance; Anesthetics, Local; Animals; Axons; Baclofen; Calcium; Capsaicin; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Functional Laterality; GABA Agonists; Immunohistochemistry; In Vitro Techniques; Indoles; Isoindoles; Lidocaine; Microscopy, Confocal; Neurokinin-1 Receptor Antagonists; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Spinal Nerve Roots; Time Factors

2003
Use of a fluorescent imaging plate reader--based calcium assay to assess pharmacological differences between the human and rat vanilloid receptor.
    Journal of biomolecular screening, 2002, Volume: 7, Issue:5

    Topics: Amino Acid Sequence; Animals; Biological Assay; Calcium; Capsaicin; Cells, Cultured; Diterpenes; Fluorescence; Humans; Kinetics; Ligands; Molecular Sequence Data; Rats; Receptors, Drug; Ruthenium Red; Sequence Homology, Amino Acid; Species Specificity

2002
Capsazepine protects against neuronal injury caused by oxygen glucose deprivation by inhibiting I(h).
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Nov-05, Volume: 23, Issue:31

    Topics: Animals; Capsaicin; Cell Death; Cell Hypoxia; Cells, Cultured; Cyclic Nucleotide-Gated Cation Channels; Cytoprotection; Dose-Response Relationship, Drug; Glucose; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Neuroprotective Agents; Patch-Clamp Techniques; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Drug

2003
Insulin induces cobalt uptake in a subpopulation of rat cultured primary sensory neurons.
    The European journal of neuroscience, 2003, Volume: 18, Issue:9

    Topics: Animals; Capsaicin; Cell Count; Cell Culture Techniques; Cobalt; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ganglia, Spinal; Immunohistochemistry; Insulin; Neomycin; Neurons, Afferent; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Receptor, Insulin; Receptors, Drug; Ruthenium Red; Staurosporine; TRPV Cation Channels; Type C Phospholipases; Tyrphostins

2003
Cannabinoids inhibit the release of [3H]glutamate from rodent hippocampal synaptosomes via a novel CB1 receptor-independent action.
    The European journal of neuroscience, 2003, Volume: 18, Issue:7

    Topics: Analgesics; Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Chromatography, High Pressure Liquid; Cyclohexanols; Dose-Response Relationship, Drug; Drug Interactions; Glutamic Acid; Hippocampus; Male; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Radioactivity; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; Synaptosomes; Tritium

2003
A novel neuroimmune mechanism in cannabinoid-mediated attenuation of nerve growth factor-induced hyperalgesia.
    Anesthesiology, 2003, Volume: 99, Issue:6

    Topics: Analgesics; Animals; Arachidonic Acids; Cannabinoids; Capsaicin; Cell Movement; Endocannabinoids; Hyperalgesia; Male; Nerve Growth Factor; Neutrophils; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rimonabant

2003
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.
    Neuropharmacology, 2004, Volume: 46, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acids; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Anilides; Aniline Compounds; Animals; Calcium; Capsaicin; Carrier Proteins; Cell Line; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Hot Temperature; Humans; Intracellular Signaling Peptides and Proteins; Kidney; Membrane Potentials; N-Methylaspartate; Neuropeptides; Norepinephrine; Orexins; Patch-Clamp Techniques; Protein Binding; Radioligand Assay; Rats; Receptors, Drug; Serotonin Receptor Agonists; Xanthenes

2004
Design of a high-affinity competitive antagonist of the vanilloid receptor selective for the calcium entry-linked receptor population.
    Molecular pharmacology, 2004, Volume: 65, Issue:2

    Topics: Animals; Binding, Competitive; Calcium; Capsaicin; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Design; Receptors, Calcium-Sensing; Receptors, Drug; Thiourea; TRPV Cation Channels

2004
Effects of the vanilloid agonist olvanil and antagonist capsazepine on rat behaviors.
    Progress in neuro-psychopharmacology & biological psychiatry, 2004, Volume: 28, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Capsaicin; Dose-Response Relationship, Drug; Maze Learning; Rats; Rats, Sprague-Dawley; Receptors, Drug; Swimming

2004
Activation of capsaicin-sensitive sensory neurons by carvedilol, a nonselective beta-blocker, in spontaneous hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bisoprolol; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Carvedilol; Cells, Cultured; Drug Interactions; Female; Humans; Hypertension; Kidney; Male; Mice; Neurons, Afferent; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Regional Blood Flow

2004
Identification of species-specific determinants of the action of the antagonist capsazepine and the agonist PPAHV on TRPV1.
    The Journal of biological chemistry, 2004, Apr-23, Volume: 279, Issue:17

    Topics: Amino Acid Sequence; Animals; Calcium; Capsaicin; CHO Cells; Cricetinae; Diterpenes; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Guinea Pigs; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Ions; Kinetics; Ligands; Methionine; Models, Chemical; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Phenotype; Phorbol Esters; Protein Structure, Tertiary; Rats; Receptors, Drug; Species Specificity; Time Factors

2004
Modulation of trigeminal sensory neuron activity by the dual cannabinoid-vanilloid agonists anandamide, N-arachidonoyl-dopamine and arachidonyl-2-chloroethylamide.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: Aminobutyrates; Animals; Arachidonic Acid; Arachidonic Acids; Calcitonin Gene-Related Peptide; Calcium Channels; Capsaicin; Dinoprostone; Diterpenes; Dopamine; Endocannabinoids; Ganglia, Spinal; Male; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Drug; Staurosporine; Trigeminal Ganglion; TRPC Cation Channels; TRPV Cation Channels

2004
Multiple actions of anandamide on neonatal rat cultured sensory neurones.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Calcium Channels; Calcium Signaling; Capsaicin; Cells, Cultured; Drug Synergism; Endocannabinoids; Fura-2; Ganglia, Spinal; Neurons, Afferent; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium Chloride; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; TRPV Cation Channels

2004
An investigation of the effects of ruthenium red, nitric oxide and endothelin-1 on infrared receptor activity in a crotaline snake.
    Neuroscience, 2004, Volume: 124, Issue:4

    Topics: Animals; Blood Vessels; Capsaicin; Electrophysiology; Endothelin-1; Female; Male; Nitric Oxide Donors; Nitroprusside; Receptors, Drug; Ruthenium Red; Temperature; Thermoreceptors; Trimeresurus

2004
An efficient parallel synthesis of capsazepine and capsazepine analogs.
    Combinatorial chemistry & high throughput screening, 2004, Volume: 7, Issue:2

    Topics: Benzazepines; Capsaicin; Molecular Structure

2004
Characterization of capsaicin-induced, capsazepine-insensitive relaxation of ileal smooth muscle of rats.
    European journal of pharmacology, 2004, Mar-08, Volume: 487, Issue:1-3

    Topics: Acetylcholine; Animals; Calcium; Calcium Channel Blockers; Capsaicin; Chelating Agents; Egtazic Acid; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nifedipine; Phosphorylation; Potassium; Rats; Rats, Wistar

2004
Inhibitory effect of ginger (Zingiber officinale) on rat ileal motility in vitro.
    Life sciences, 2004, Apr-23, Volume: 74, Issue:23

    Topics: Acetylcholine; Animals; Capsaicin; Dose-Response Relationship, Drug; Drug Antagonism; Electric Stimulation; Gastrointestinal Motility; Ileum; Male; Organ Culture Techniques; Phytotherapy; Plant Extracts; Plants, Medicinal; Rats; Rats, Wistar; Zingiber officinale

2004
Involvement of vanilloid-like receptors in the effects of anandamide on motor behavior and nigrostriatal dopaminergic activity: in vivo and in vitro evidence.
    Brain research, 2004, May-08, Volume: 1007, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Capsaicin; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Drug Interactions; Electrochemistry; Endocannabinoids; In Vitro Techniques; Ion Channels; Male; Motor Activity; Neurons; Polyunsaturated Alkamides; Potassium; Rats; Rats, Wistar; Receptors, Drug; Stereotyped Behavior; TRPV Cation Channels; Tyrosine 3-Monooxygenase

2004
An assessment of vascular pain using the flexor reflex in anesthetized rats.
    Methods and findings in experimental and clinical pharmacology, 2004, Volume: 26, Issue:2

    Topics: Animals; Capsaicin; Dose-Response Relationship, Drug; Electromyography; Hindlimb; Injections, Intra-Arterial; Injections, Spinal; Injections, Subcutaneous; Lidocaine; Male; Morphine; Muscle, Skeletal; Naloxone; Pain Measurement; Procaine; Rats; Rats, Sprague-Dawley; Reflex, Stretch; Time Factors; Toes; Vascular Diseases

2004
The analgesic effect induced by capsaicin is enhanced in inflammatory states.
    Life sciences, 2004, May-14, Volume: 74, Issue:26

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Capsaicin; Carrageenan; Disease Models, Animal; Freund's Adjuvant; Hot Temperature; Hyperalgesia; Inflammation; Male; Mice; Receptors, Drug; Time Factors

2004
Histamine-induced Ca(2+) influx via the PLA(2)/lipoxygenase/TRPV1 pathway in rat sensory neurons.
    Neuroscience letters, 2004, May-06, Volume: 361, Issue:1-3

    Topics: Animals; Calcium; Calcium Signaling; Capsaicin; Cells, Cultured; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Ganglia, Spinal; Histamine; Lipoxygenase; Neurons, Afferent; Nociceptors; Phospholipases A; Pruritus; Rats; Receptors, Drug

2004
Purinergic and vanilloid receptor activation releases glutamate from separate cranial afferent terminals in nucleus tractus solitarius.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, May-19, Volume: 24, Issue:20

    Topics: Adenosine Triphosphate; Afferent Pathways; Animals; Capsaicin; Cell Separation; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Neural Inhibition; Neurons; Nodose Ganglion; Patch-Clamp Techniques; Presynaptic Terminals; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Rats, Sprague-Dawley; Receptors, Drug; Receptors, Purinergic P2; Solitary Nucleus

2004
Effects of TRPV1 receptor antagonists on stimulated iCGRP release from isolated skin of rats and TRPV1 mutant mice.
    Pain, 2004, Volume: 109, Issue:3

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Drug Interactions; Hot Temperature; In Vitro Techniques; Male; Mice; Mice, Knockout; Nociceptors; Pain; Rats; Rats, Wistar; Receptors, Drug; Ruthenium Red; Sensory Receptor Cells; Signal Transduction; Skin

2004
Presynaptic cannabinoid CB(1) receptors are involved in the inhibition of the neurogenic vasopressor response during septic shock in pithed rats.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: Animals; Autonomic Fibers, Postganglionic; Autonomic Fibers, Preganglionic; Blood Pressure; Camphanes; Capsaicin; Decerebrate State; Disease Models, Animal; Electric Stimulation; Germany; Imidazoles; Infusions, Intravenous; Lipopolysaccharides; Male; Norepinephrine; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Shock, Septic; Solvents; Thiourea; Vagotomy; Vasomotor System; Vasopressins

2004
Sex-linked differences in the vasorelaxant effects of anandamide in vascular mesenteric beds: role of oestrogens.
    European journal of pharmacology, 2004, Jun-16, Volume: 493, Issue:1-3

    Topics: Acetylcholine; Animals; Arachidonic Acids; Argentina; Capsaicin; Chile; Cycloheximide; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Estradiol; Estrogens; Female; Male; Mesentery; Muscle, Smooth, Vascular; Nitroprusside; Norepinephrine; Ovariectomy; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Sex Characteristics; Time Factors; Vasodilation

2004
TRPV1 and CB(1) receptor-mediated effects of the endovanilloid/endocannabinoid N-arachidonoyl-dopamine on primary afferent fibre and spinal cord neuronal responses in the rat.
    The European journal of neuroscience, 2004, Volume: 20, Issue:1

    Topics: Animals; Arachidonic Acids; Behavior, Animal; Calcium; Capsaicin; Cells, Cultured; Dopamine; Drug Interactions; Electrophysiology; Male; Membrane Potentials; Nerve Fibers; Pain Measurement; Physical Stimulation; Piperidines; Posterior Horn Cells; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Drug; Rimonabant; Sensory Thresholds; Spinal Cord

2004
Inhibitory effect of the antidepressant St. John's wort (hypericum perforatum) on rat bladder contractility in vitro.
    Urology, 2004, Volume: 64, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Anthracenes; Antidepressive Agents; Atropine; Bridged Bicyclo Compounds; Capsaicin; Depression; Electric Stimulation; Female; Haloperidol; Hypericum; Kaempferols; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Naloxone; Perylene; Phentolamine; Phloroglucinol; Piperidines; Plant Extracts; Propranolol; Pyrazoles; Quercetin; Rats; Rats, Wistar; Rimonabant; Rutin; Terpenes; Tetrodotoxin; Urinary Bladder; Urinary Incontinence; Verapamil

2004
AM404 enhances the spontaneous release of L-glutamate in a manner sensitive to capsazepine in adult rat substantia gelatinosa neurones.
    Brain research, 2004, Aug-27, Volume: 1018, Issue:2

    Topics: Anesthetics, Local; Animals; Arachidonic Acids; Biological Transport; Capsaicin; Drug Interactions; Endocannabinoids; Glutamic Acid; Male; Neurons; Polyunsaturated Alkamides; Rats; Receptors, Drug; Substantia Gelatinosa; Tetrodotoxin

2004
Differential pH and capsaicin responses of Griffonia simplicifolia IB4 (IB4)-positive and IB4-negative small sensory neurons.
    Neuroscience, 2004, Volume: 127, Issue:3

    Topics: Amiloride; Animals; Calcium; Capsaicin; Diuretics; Ganglia, Spinal; Hydrogen-Ion Concentration; Immunohistochemistry; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Plant Lectins; Protons; Rats; Rats, Sprague-Dawley; Receptors, Drug

2004
Regulation of calcitonin gene-related peptide release from rat trigeminal nucleus caudalis slices in vitro.
    Neuroscience letters, 2004, Aug-19, Volume: 366, Issue:3

    Topics: Analysis of Variance; Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cyclooxygenase Inhibitors; Dinoprostone; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Gene Expression Regulation; In Vitro Techniques; Indomethacin; Male; Potassium Chloride; Rats; Rats, Sprague-Dawley; Trigeminal Caudal Nucleus

2004
Evodiamine functions as an agonist for the vanilloid receptor TRPV1.
    Organic & biomolecular chemistry, 2004, Aug-21, Volume: 2, Issue:16

    Topics: Animals; Calcium; Capsaicin; Cations, Divalent; CHO Cells; Cricetinae; Diterpenes; Ligands; Models, Biological; Molecular Conformation; Molecular Structure; Plant Extracts; Quinazolines; TRPV Cation Channels

2004
Capsazepine is a novel activator of the delta subunit of the human epithelial Na+ channel.
    The Journal of biological chemistry, 2004, Oct-22, Volume: 279, Issue:43

    Topics: Amiloride; Animals; Anti-Inflammatory Agents, Non-Steroidal; Capsaicin; Diterpenes; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electrophysiology; Epithelial Sodium Channels; Humans; Hydrogen-Ion Concentration; Neurotoxins; Oocytes; Protein Structure, Tertiary; Protons; Receptors, Drug; Sodium Channels; Xenopus

2004
Vanilloid TRPV1 receptor mediates the antihyperalgesic effect of the nonpsychoactive cannabinoid, cannabidiol, in a rat model of acute inflammation.
    British journal of pharmacology, 2004, Volume: 143, Issue:2

    Topics: Administration, Oral; Animals; Camphanes; Cannabidiol; Capsaicin; Carrageenan; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Therapy, Combination; Hyperalgesia; Inflammation; Italy; Male; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Drug; Rimonabant; Time Factors

2004
Characterization of the human HCN1 channel and its inhibition by capsazepine.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: Animals; Benzazepines; Capsaicin; Cell Line; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Electric Stimulation; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channels; Pyrimidines; Time Factors; Transfection

2004
Nociceptin inhibits vanilloid TRPV-1-mediated neurosensitization induced by fenoterol in human isolated bronchi.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:3

    Topics: Adrenergic beta-Agonists; Bronchi; Bronchoconstriction; Capsaicin; Drug Interactions; Endothelin-1; Female; Fenoterol; Humans; Ion Channels; Male; Middle Aged; Nociceptin; Opioid Peptides; Receptors, Drug; TRPV Cation Channels; Vasodilator Agents

2004
Transient receptor potential vanilloid subfamily 1 expressed in pancreatic islet beta cells modulates insulin secretion in rats.
    Biochemical and biophysical research communications, 2004, Aug-13, Volume: 321, Issue:1

    Topics: Animals; Capsaicin; Cell Line, Tumor; DNA Primers; Ganglia, Spinal; Gene Expression Regulation; Insulin; Insulin Secretion; Insulinoma; Ion Channels; Islets of Langerhans; Male; Pancreatic Neoplasms; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; TRPV Cation Channels

2004
Capsazepine elevates intracellular Ca2+ in human osteosarcoma cells, questioning its selectivity as a vanilloid receptor antagonist.
    Life sciences, 2004, Oct-08, Volume: 75, Issue:21

    Topics: Calcium; Calcium Signaling; Capsaicin; Cell Division; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Fluorescent Dyes; Fura-2; Humans; Osteosarcoma; Pyrrolidinones; Receptors, Drug; Thapsigargin; Type C Phospholipases

2004
Capsaicin, a spicy component of hot pepper, induces apoptosis by activation of the peroxisome proliferator-activated receptor gamma in HT-29 human colon cancer cells.
    Journal of medicinal food, 2004,Fall, Volume: 7, Issue:3

    Topics: Antineoplastic Agents; Apoptosis; Benzhydryl Compounds; Capsaicin; Cell Division; Cell Survival; Colonic Neoplasms; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; HT29 Cells; Humans; Phenols; PPAR gamma; Receptors, Drug; TRPV Cation Channels

2004
Distinct thymocyte subsets express the vanilloid receptor VR1 that mediates capsaicin-induced apoptotic cell death.
    Cell death and differentiation, 2004, Volume: 11, Issue:12

    Topics: Animals; Apoptosis; Calcium Signaling; Capsaicin; Caspases; CD4 Antigens; CD4-Positive T-Lymphocytes; CD5 Antigens; Cell Membrane; Cells, Cultured; DNA Fragmentation; Dose-Response Relationship, Drug; Intracellular Membranes; Lymphocyte Subsets; Male; Mitochondria; Necrosis; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Drug; RNA, Messenger; T-Lymphocytes

2004
Lipopolysaccharide fever is initiated via a capsaicin-sensitive mechanism independent of the subtype-1 vanilloid receptor.
    British journal of pharmacology, 2004, Volume: 143, Issue:8

    Topics: Animals; Body Temperature; Capsaicin; Diterpenes; Eating; Fever; Lipopolysaccharides; Male; Rats; Rats, Long-Evans; Receptors, Drug; TRPV Cation Channels

2004
Vanilloid receptor TRPV1, sensory C-fibers, and vascular autoregulation: a novel mechanism involved in myogenic constriction.
    Circulation research, 2004, Nov-12, Volume: 95, Issue:10

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Capsaicin; Cation Transport Proteins; CHO Cells; Cricetinae; Endothelium, Vascular; Gadolinium; Ganglia, Sympathetic; Guanethidine; Hydroxyeicosatetraenoic Acids; Ion Channels; Male; Mesenteric Arteries; Mice; Mice, Knockout; Models, Cardiovascular; Models, Neurological; Nerve Fibers, Unmyelinated; Nociceptors; Peptides, Cyclic; Piperidines; Pressure; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Ruthenium Red; Sodium Channel Blockers; Splanchnic Circulation; Stress, Mechanical; Sympathectomy, Chemical; Tetrodotoxin; TRPV Cation Channels; Vascular Resistance; Vasoconstriction

2004
Inhibition of the vanilloid receptor subtype-1 attenuates TNBS-colitis.
    Journal of gastrointestinal surgery : official journal of the Society for Surgery of the Alimentary Tract, 2004, Volume: 8, Issue:7

    Topics: Animals; Capsaicin; Colitis; Colon; Nociceptors; Peroxidase; Rats; Rats, Sprague-Dawley; Receptors, Drug; Trinitrobenzenesulfonic Acid; TRPV Cation Channels

2004
Human brain endothelium: coexpression and function of vanilloid and endocannabinoid receptors.
    Brain research. Molecular brain research, 2004, Dec-06, Volume: 132, Issue:1

    Topics: Arachidonic Acids; Blood-Brain Barrier; Brain; Camphanes; Cannabinoid Receptor Agonists; Cannabinoid Receptor Modulators; Capsaicin; Cell Adhesion Molecules; Cells, Cultured; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Endothelium, Vascular; Glycerides; Humans; Ion Channels; Microcirculation; Microfilament Proteins; Phosphoproteins; Phosphorylation; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; RNA, Messenger; TRPV Cation Channels

2004
Evidence that TRPM8 is an androgen-dependent Ca2+ channel required for the survival of prostate cancer cells.
    Cancer research, 2004, Nov-15, Volume: 64, Issue:22

    Topics: Androgens; Apoptosis; Base Sequence; Calcium; Capsaicin; Cell Survival; DNA Primers; Humans; Immunohistochemistry; Ion Channels; Ion Transport; Male; Menthol; Neoplasm Proteins; Prostatic Neoplasms; Sequence Homology, Nucleic Acid; TRPM Cation Channels

2004
Combined determination with functional and morphological studies of origin of nerve fibers expressing transient receptor potential vanilloid 1 in the myenteric plexus of the rat jejunum.
    Autonomic neuroscience : basic & clinical, 2004, Nov-30, Volume: 116, Issue:1-2

    Topics: Action Potentials; Analysis of Variance; Animals; Autonomic Denervation; Calcitonin Gene-Related Peptide; Capsaicin; Drug Interactions; Immunohistochemistry; In Vitro Techniques; Ion Channels; Jejunum; Male; Muscle Relaxation; Myenteric Plexus; Nerve Fibers; Rats; Rats, Wistar; Substance P; TRPV Cation Channels

2004
Capsazepine, a vanilloid antagonist, abolishes tonic responses induced by 20-HETE on guinea pig airway smooth muscle.
    American journal of physiology. Lung cellular and molecular physiology, 2005, Volume: 288, Issue:3

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Bronchi; Calcium; Calcium Channels; Capsaicin; Cyclohexanones; Cytochrome P-450 CYP4A; Female; Guinea Pigs; Hydroxyeicosatetraenoic Acids; In Vitro Techniques; Intracellular Membranes; Lipoprotein Lipase; Male; Muscle Contraction; Muscle, Smooth; Protease Inhibitors; Receptors, Drug; Time Factors; Trachea

2005
Involvement of CGRP in the inhibitory effect of rutaecarpine on vasoconstriction induced by anaphylaxis in guinea pig.
    Regulatory peptides, 2005, Feb-15, Volume: 125, Issue:1-3

    Topics: Alkaloids; Anaphylaxis; Animals; Antigens; Aorta, Thoracic; Calcitonin Gene-Related Peptide; Capsaicin; Diphenhydramine; Female; Guinea Pigs; Indole Alkaloids; Male; Quinazolines; Receptors, Drug; Time Factors; TRPV Cation Channels; Vasoconstriction; Vasodilator Agents

2005
Vanilloid receptor 1 antagonists attenuate disease severity in dextran sulphate sodium-induced colitis in mice.
    Neurogastroenterology and motility, 2004, Volume: 16, Issue:6

    Topics: Animals; Anticoagulants; Capsaicin; Colitis; Dextran Sulfate; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Inflammatory Bowel Diseases; Ion Channels; Mice; Mice, Inbred BALB C; Peroxidase; TRPV Cation Channels

2004
Anandamide-evoked activation of vanilloid receptor 1 contributes to the development of bladder hyperreflexia and nociceptive transmission to spinal dorsal horn neurons in cystitis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Dec-15, Volume: 24, Issue:50

    Topics: Acrolein; Animals; Arachidonic Acids; Capsaicin; Cyclophosphamide; Cystitis; Endocannabinoids; Female; Hydrolysis; Ion Channels; Pain; Polyunsaturated Alkamides; Posterior Horn Cells; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Reflex, Abnormal; TRPV Cation Channels; Urinary Bladder

2004
Protective effects of evodiamine on myocardial ischemia-reperfusion injury in rats.
    Planta medica, 2004, Volume: 70, Issue:12

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cardiotonic Agents; Creatine Kinase; Evodia; Infusions, Intravenous; Male; Myocardial Reperfusion Injury; Myocardium; Phytotherapy; Plant Extracts; Quinazolines; Rats; Rats, Sprague-Dawley; Tumor Necrosis Factor-alpha

2004
TRPV1b, a functional human vanilloid receptor splice variant.
    Molecular pharmacology, 2005, Volume: 67, Issue:4

    Topics: Amino Acid Sequence; Capsaicin; Cloning, Molecular; Humans; Ion Channels; Molecular Sequence Data; Ruthenium Red; Structure-Activity Relationship; Temperature; Trigeminal Ganglion; TRPV Cation Channels

2005
2-aminoethoxydiphenyl borate stimulates pulmonary C neurons via the activation of TRPV channels.
    American journal of physiology. Lung cellular and molecular physiology, 2005, Volume: 288, Issue:5

    Topics: Animals; Blood Pressure; Boron Compounds; Capsaicin; Cation Transport Proteins; Coloring Agents; Heart Rate; Ion Channels; Lung; Nerve Fibers, Unmyelinated; Nodose Ganglion; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reflex; Respiratory Mechanics; Ruthenium Red; TRPV Cation Channels

2005
Lafutidine-induced increase in intracellular ca(2+) concentrations in PC12 and endothelial cells.
    Journal of pharmacological sciences, 2005, Volume: 97, Issue:1

    Topics: Acetamides; Animals; Calcium; Calcium Chloride; Capsaicin; Dose-Response Relationship, Drug; Endothelial Cells; Humans; Imidazoles; Immunoblotting; Intracellular Fluid; PC12 Cells; Piperidines; Pyridines; Rats; Thapsigargin; Time Factors

2005
Vagal selective effects of ruthenium red on the jejunal afferent fibre response to ischaemia in the rat.
    Neurogastroenterology and motility, 2005, Volume: 17, Issue:1

    Topics: Animals; Capsaicin; Ischemia; Jejunum; Male; Nerve Fibers; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reperfusion Injury; Ruthenium Red; Vagotomy; Vagus Nerve

2005
Capsaicin exhibits neuroprotective effects in a model of transient global cerebral ischemia in Mongolian gerbils.
    British journal of pharmacology, 2005, Volume: 144, Issue:5

    Topics: Animals; Capsaicin; Cell Survival; Disease Models, Animal; Electroencephalography; Gerbillinae; Hippocampus; Ischemic Attack, Transient; Male; Memory; Motor Activity; Neuroprotective Agents; Pyramidal Cells; Receptors, Drug

2005
AM404, an inhibitor of anandamide reuptake decreases Fos-immunoreactivity in the spinal cord of neuropathic rats after non-noxious stimulation.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Dose-Response Relationship, Drug; Endocannabinoids; Immunohistochemistry; Indoles; Male; Physical Stimulation; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Spinal Cord

2005
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Antiemetics; Butanols; Capsaicin; Cyclooxygenase Inhibitors; Dihydroergotamine; Diphenhydramine; Diterpenes; Domperidone; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Indomethacin; Malates; Methysergide; Metoclopramide; Migraine Disorders; Ondansetron; Piperidines; Ruthenium Red; Scopolamine; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Sumatriptan; Time Factors; Tropanes; Vomiting

2005
Effects of piperine, the pungent component of black pepper, at the human vanilloid receptor (TRPV1).
    British journal of pharmacology, 2005, Volume: 144, Issue:6

    Topics: Alkaloids; Benzodioxoles; Capsaicin; Cell Line; Humans; Hydrogen-Ion Concentration; Patch-Clamp Techniques; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Receptors, Drug; Ruthenium Red; Structure-Activity Relationship

2005
Characterization and comparison of recombinant human and rat TRPV1 receptors: effects of exo- and endocannabinoids.
    British journal of anaesthesia, 2005, Volume: 94, Issue:5

    Topics: Animals; Arachidonic Acids; Calcium; Cannabinoid Receptor Modulators; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Ion Channels; Polyunsaturated Alkamides; Rats; Recombinant Proteins; Species Specificity; Temperature; TRPV Cation Channels

2005
Transient receptor potential vanilloid (TRPV-1) promotes neurogenic inflammation in the pancreas via activation of the neurokinin-1 receptor (NK-1R).
    Pancreas, 2005, Volume: 30, Issue:3

    Topics: Animals; Capsaicin; Ceruletide; Coloring Agents; Evans Blue; Male; Neuritis; Pancreas; Pancreatitis; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; TRPV Cation Channels

2005
Role of sensory neuron in reduction of endotoxin-induced hypotension in rats.
    Critical care medicine, 2005, Volume: 33, Issue:4

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Cyclooxygenase Inhibitors; Disease Models, Animal; Dose-Response Relationship, Drug; Endotoxins; Hypotension; Iloprost; Indomethacin; Interleukin-16; Lung; Neurons, Afferent; Nitric Oxide Synthase; Prospective Studies; Rats; Rats, Wistar; Reference Values; Tumor Necrosis Factor-alpha; Vasodilator Agents

2005
The effects of Delta9-tetrahydrocannabinol in rat mesenteric vasculature, and its interactions with the endocannabinoid anandamide.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Apamin; Arachidonic Acids; Azepines; Barium Compounds; Biological Factors; Calcium; Cannabinoid Receptor Modulators; Capsaicin; Charybdotoxin; Chlorides; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Endocannabinoids; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Vasodilation; Verapamil

2005
Differential responses of bladder lumbosacral and thoracolumbar dorsal root ganglion neurons to purinergic agonists, protons, and capsaicin.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-13, Volume: 25, Issue:15

    Topics: Adenosine Triphosphate; Amiloride; Amino Acids; Animals; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Ganglia, Spinal; Hydrogen-Ion Concentration; Immunohistochemistry; Lectins; Lumbosacral Region; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Phenols; Polycyclic Compounds; Protons; Purinergic Agonists; Purinergic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic; Sodium Channel Blockers; Thoracic Vertebrae; Time Factors; TRPV Cation Channels; Urinary Bladder

2005
Protective effects of Delta(9)-tetrahydrocannabinol against N-methyl-d-aspartate-induced AF5 cell death.
    Brain research. Molecular brain research, 2005, Apr-04, Volume: 134, Issue:2

    Topics: alpha-Tocopherol; Animals; Benzimidazoles; Benzoxazines; Blotting, Northern; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Capsaicin; Cell Count; Cell Death; Cell Lineage; Dizocilpine Maleate; DNA, Single-Stranded; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Excitatory Amino Acid Agonists; Immunohistochemistry; In Situ Nick-End Labeling; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Neuroprotective Agents; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Ruthenium; Tetrazolium Salts; Thiazoles; TRPC Cation Channels

2005
Vanilloid receptor expressed in the sarcoplasmic reticulum of rat skeletal muscle.
    Biochemical and biophysical research communications, 2005, Jul-08, Volume: 332, Issue:3

    Topics: Animals; Calcium; Calcium-Transporting ATPases; Capsaicin; Cell Line; Gene Expression; Ion Channels; Microscopy, Confocal; Microscopy, Electron; Muscle, Skeletal; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; TRPV Cation Channels

2005
Peripheral, but not central effects of cannabidiol derivatives: mediation by CB(1) and unidentified receptors.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Body Temperature; Camphanes; Cannabidiol; Capsaicin; Drug Interactions; Ear, External; Gastrointestinal Motility; Inflammation; Mice; Mice, Inbred ICR; Mice, Inbred Strains; Motor Activity; Pain Measurement; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant

2005
Evidence that (-)-7-hydroxy-4'-dimethylheptyl-cannabidiol activates a non-CB(1), non-CB(2), non-TRPV1 target in the mouse vas deferens.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzoxazines; Cannabidiol; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Capsaicin; In Vitro Techniques; Isometric Contraction; Male; Mice; Morpholines; Naloxone; Naphthalenes; Phenylephrine; Piperidines; Pyrazoles; Rimonabant; Ruthenium Red; TRPV Cation Channels; Vas Deferens; Yohimbine

2005
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. I. Effect on TRC volume and Na+ flux.
    The Journal of general physiology, 2005, Volume: 125, Issue:6

    Topics: Amiloride; Anilides; Animals; Capsaicin; Cell Size; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Cytosol; Diuretics; Ethanol; Female; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Taste; Temperature; Tongue

2005
Ethanol modulates the VR-1 variant amiloride-insensitive salt taste receptor. II. Effect on chorda tympani salt responses.
    The Journal of general physiology, 2005, Volume: 125, Issue:6

    Topics: Algorithms; Amiloride; Anilides; Animals; Capsaicin; Cell Membrane; Cell Polarity; Central Nervous System Depressants; Chorda Tympani Nerve; Cinnamates; Diterpenes; Diuretics; Ethanol; Female; In Vitro Techniques; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Receptors, Drug; Sodium; Sodium Chloride; Stimulation, Chemical; Taste; Taste Threshold; Temperature; Tongue

2005
Characterization of rat transient receptor potential vanilloid 1 receptors lacking the N-glycosylation site N604.
    Neuroreport, 2005, Jun-21, Volume: 16, Issue:9

    Topics: Analysis of Variance; Animals; Asparagine; Capsaicin; Cell Line; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Glycosylation; Humans; Hydrogen-Ion Concentration; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Point Mutation; Rats; Threonine; Transfection; TRPV Cation Channels

2005
Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat.
    Neuroscience letters, 2005, Sep-09, Volume: 385, Issue:2

    Topics: Analgesics; Anilides; Animals; Capsaicin; Cells, Cultured; Cinnamates; Dose-Response Relationship, Drug; Drug Interactions; Hypothermia; Ion Channels; Male; Mice; Mice, Inbred BALB C; Neurons, Afferent; Nociceptors; Pain; Peripheral Nervous System; Rats; Rats, Wistar; Sensory Receptor Cells; Substance P; Trigeminal Ganglion; TRPV Cation Channels

2005
Capsaicin regulates voltage-dependent sodium channels by altering lipid bilayer elasticity.
    Molecular pharmacology, 2005, Volume: 68, Issue:3

    Topics: Capsaicin; Gramicidin; Kinetics; Lipid Bilayers; Patch-Clamp Techniques; Scattering, Radiation; Sodium Channels

2005
Pharmacological characterization of the TRPV1 receptor antagonist JYL1421 (SC0030) in vitro and in vivo in the rat.
    European journal of pharmacology, 2005, Jul-04, Volume: 517, Issue:1-2

    Topics: Animals; Blood Pressure; Body Temperature; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Ion Channels; Male; Neurons; Neuropeptides; Rats; Rats, Wistar; Somatostatin; Substance P; Sulfonamides; Thiourea; Trachea; TRPV Cation Channels

2005
Characteristics of propofol-evoked vascular pain in anaesthetized rats.
    British journal of anaesthesia, 2005, Volume: 95, Issue:3

    Topics: Analgesics, Opioid; Anesthetics, Intravenous; Anesthetics, Local; Animals; Capsaicin; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Electromyography; Indomethacin; Injections, Intra-Arterial; Male; Muscle, Skeletal; Pain; Procaine; Propofol; Rats; Rats, Sprague-Dawley; Reflex

2005
Capsazepine, a vanilloid receptor antagonist, inhibits allergen-induced tracheal contraction.
    European journal of pharmacology, 2005, Jul-25, Volume: 518, Issue:1

    Topics: Allergens; Animals; Capsaicin; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Ovalbumin; Receptors, Drug; Trachea

2005
Vascular effects of anandamide and N-acylvanillylamines in the human forearm and skin microcirculation.
    British journal of pharmacology, 2005, Volume: 146, Issue:2

    Topics: Adult; Arachidonic Acids; Benzylamines; Capsaicin; Endocannabinoids; Female; Forearm; Humans; Laser-Doppler Flowmetry; Male; Microcirculation; Middle Aged; Muscle, Skeletal; Plethysmography; Polyunsaturated Alkamides; Regional Blood Flow; Skin; TRPV Cation Channels

2005
Icilin activates the delta-subunit of the human epithelial Na+ channel.
    Molecular pharmacology, 2005, Volume: 68, Issue:4

    Topics: Amiloride; Animals; Capsaicin; Epithelial Sodium Channels; Humans; Protons; Pyrimidinones; Sodium Channel Agonists; Sodium Channels; Xenopus laevis

2005
Heat and mechanical hyperalgesia in mice model of cancer pain.
    Pain, 2005, Volume: 117, Issue:1-2

    Topics: Animals; Body Temperature; Capsaicin; Cell Count; Cell Line, Tumor; Cell Size; Disease Models, Animal; Dose-Response Relationship, Drug; Ganglia, Spinal; Humans; Hyperalgesia; Immunohistochemistry; Male; Mice; Mice, Inbred C3H; Neoplasm Transplantation; Neoplasms; Pain; Pain Measurement; Pain Threshold; Reaction Time; Staining and Labeling; Time Factors; TRPV Cation Channels

2005
Multiple types of sensory neurons respond to irritating volatile organic compounds (VOCs): calcium fluorimetry of trigeminal ganglion neurons.
    Pain, 2005, Volume: 117, Issue:1-2

    Topics: Aldehydes; Animals; Animals, Newborn; Calcium; Capsaicin; Central Nervous System Depressants; Diagnostic Imaging; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Fluorometry; Neurons; Organic Chemicals; Potassium Chloride; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Trigeminal Ganglion

2005
Synergistic interactions between airway afferent nerve subtypes regulating the cough reflex in guinea-pigs.
    The Journal of physiology, 2005, Dec-01, Volume: 569, Issue:Pt 2

    Topics: Administration, Inhalation; Animals; Bradykinin; Bronchial Spasm; Capsaicin; Citric Acid; Cough; Guinea Pigs; Lung; Male; Mechanoreceptors; Microinjections; Nerve Fibers, Unmyelinated; Neurons, Afferent; Nociceptors; Reflex; Substance P; Tachykinins

2005
Cannabidiol reverses MK-801-induced disruption of prepulse inhibition in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:4

    Topics: Analysis of Variance; Animals; Behavior, Animal; Cannabidiol; Capsaicin; Clozapine; Conditioning, Classical; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Inhibition, Psychological; Male; Mice; Reflex, Startle; Serotonin Antagonists

2006
TRPV1 activation results in disruption of the blood-brain barrier in the rat.
    British journal of pharmacology, 2005, Volume: 146, Issue:4

    Topics: Animals; Blood-Brain Barrier; Brain Ischemia; Capillaries; Capillary Permeability; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Male; Microspheres; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Starch; Substance P; Tetrazoles; Time Factors; TRPV Cation Channels

2005
Anandamide elicits an acute release of nitric oxide through endothelial TRPV1 receptor activation in the rat arterial mesenteric bed.
    The Journal of physiology, 2005, Oct-15, Volume: 568, Issue:Pt 2

    Topics: Anilides; Animals; Arachidonic Acids; Cannabinoid Receptor Antagonists; Capsaicin; Cinnamates; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Artery, Superior; Nitric Oxide; Nitroarginine; Perfusion; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; RNA, Messenger; TRPV Cation Channels; Vasodilation

2005
Diuresis and natriuresis caused by activation of VR1-positive sensory nerves in renal pelvis of rats.
    Hypertension (Dallas, Tex. : 1979), 2005, Volume: 46, Issue:4

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Denervation; Diuresis; Dose-Response Relationship, Drug; Kidney Cortex; Kidney Pelvis; Male; Natriuresis; Neurons, Afferent; Rats; Rats, Wistar; Regional Blood Flow; TRPV Cation Channels

2005
Attenuation of acid induced oesophagitis in VR-1 deficient mice.
    Gut, 2006, Volume: 55, Issue:1

    Topics: Acute Disease; Animals; Anti-Ulcer Agents; Capsaicin; Endocytosis; Esophagitis; Famotidine; Hydrogen-Ion Concentration; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Confocal; Omeprazole; Peroxidase; Receptors, Neurokinin-1; Severity of Illness Index; TRPV Cation Channels

2006
Mechanisms involved in the nociception produced by peripheral protein kinase c activation in mice.
    Pain, 2005, Volume: 117, Issue:1-2

    Topics: Adrenergic beta-Antagonists; Analgesics; Animals; Antibodies; Behavior, Animal; Blotting, Western; Bradykinin; Calcitonin Gene-Related Peptide; Capsaicin; Chelating Agents; Dipeptides; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Extracellular Signal-Regulated MAP Kinases; Guanethidine; Indoles; Male; Mice; Nociceptors; Pain; Pain Measurement; Peptide Fragments; Propranolol; Protein Kinase C; Ruthenium Red; Salicylates; Sympatholytics; Tetradecanoylphorbol Acetate; Time Factors

2005
Inhibition of fatty-acid amide hydrolase enhances cannabinoid stress-induced analgesia: sites of action in the dorsolateral periaqueductal gray and rostral ventromedial medulla.
    Neuropharmacology, 2005, Volume: 49, Issue:8

    Topics: Amidohydrolases; Analgesia; Animals; Arachidonic Acids; Cannabinoids; Capsaicin; Carrier Proteins; Cytosol; Endocannabinoids; Male; Medulla Oblongata; Mice; Microinjections; Pain Measurement; Periaqueductal Gray; Phospholipases A; Phospholipases A2; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Stress, Psychological; TRPV Cation Channels

2005
VR1-mediated depressor effects during high-salt intake: role of anandamide.
    Hypertension (Dallas, Tex. : 1979), 2005, Volume: 46, Issue:4

    Topics: Animals; Arachidonic Acids; Blood Pressure; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Dose-Response Relationship, Drug; Drug Combinations; Endocannabinoids; Male; Mesenteric Arteries; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Sodium, Dietary; Time Factors; TRPV Cation Channels

2005
Cooling-induced contraction of the rat gastric fundus: mediation via transient receptor potential (TRP) cation channel TRPM8 receptor and Rho-kinase activation.
    Clinical and experimental pharmacology & physiology, 2005, Volume: 32, Issue:10

    Topics: Amides; Animals; Calcium; Calcium Channel Blockers; Capsaicin; Cold Temperature; Enzyme Activation; Enzyme Inhibitors; Gastric Fundus; Gene Expression; Genistein; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Male; Maleimides; Muscle Contraction; Nifedipine; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; RNA, Messenger; TRPM Cation Channels

2005
Inflammatory mediators convert anandamide into a potent activator of the vanilloid type 1 transient receptor potential receptor in nociceptive primary sensory neurons.
    Neuroscience, 2005, Volume: 136, Issue:2

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Bradykinin; Capsaicin; Cells, Cultured; Cobalt; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Endocannabinoids; Enzyme Inhibitors; Inflammation Mediators; Neurons, Afferent; Nociceptors; Polyunsaturated Alkamides; Protein Kinase C; Rats; Rats, Sprague-Dawley; TRPV Cation Channels; Type C Phospholipases

2005
Endocannabinoids activate transient receptor potential vanilloid 1 receptors to reduce hyperdopaminergia-related hyperactivity: therapeutic implications.
    Biological psychiatry, 2006, Mar-15, Volume: 59, Issue:6

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Attention Deficit Disorder with Hyperactivity; Cannabinoid Receptor Modulators; Capsaicin; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Endocannabinoids; Mice; Mice, Knockout; Motor Activity; Polyunsaturated Alkamides; Receptor, Cannabinoid, CB1; Serotonin; Signal Transduction; TRPV Cation Channels

2006
Vanilloid type 1 receptor and the acid-sensing ion channel mediate acid phosphate activation of muscle afferent nerves in rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2006, Volume: 100, Issue:2

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Baroreflex; Blood Pressure; Capsaicin; Decerebrate State; Diterpenes; Dose-Response Relationship, Drug; Hindlimb; Male; Membrane Proteins; Muscle, Skeletal; Nerve Tissue Proteins; Neurons, Afferent; Phosphoric Acids; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Sodium Channels; Sympathetic Nervous System; TRPV Cation Channels

2006
TRPV1 desensitisation and endogenous vanilloid involvement in the enhanced analgesia induced by capsaicin in inflamed tissues.
    Brain research bulletin, 2005, Nov-30, Volume: 67, Issue:6

    Topics: Adjuvants, Immunologic; Analgesics; Animals; Capsaicin; Freund's Adjuvant; Hyperalgesia; Inflammation; Male; Mice; Pain; Pain Measurement; TRPV Cation Channels

2005
Analgesic effects of capsazepine and resiniferatoxin on bone cancer pain in mice.
    Neuroscience letters, 2006, Jan-23, Volume: 393, Issue:1

    Topics: Analgesics; Analysis of Variance; Animals; Bone Neoplasms; Capsaicin; Cell Line; Disease Models, Animal; Diterpenes; Dose-Response Relationship, Drug; Freund's Adjuvant; Functional Laterality; Inflammation; Mice; Mice, Inbred C3H; Osteosarcoma; Pain; Pain Measurement; Reaction Time; Time Factors

2006
Effect of capsazepine on cytosolic Ca(2+) levels and proliferation of human prostate cancer cells.
    Toxicology in vitro : an international journal published in association with BIBRA, 2006, Volume: 20, Issue:5

    Topics: Calcium; Capsaicin; Cell Line, Tumor; Cell Proliferation; Cytosol; Dose-Response Relationship, Drug; Egtazic Acid; Humans; Male; Prostatic Neoplasms; TRPV Cation Channels; Type C Phospholipases

2006
TRPV1 gene knockout impairs postischemic recovery in isolated perfused heart in mice.
    Circulation, 2005, Dec-06, Volume: 112, Issue:23

    Topics: Animals; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Heart; In Vitro Techniques; Mice; Mice, Knockout; Myocardial Ischemia; Neurokinin-1 Receptor Antagonists; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Recovery of Function; Reperfusion Injury; Substance P; TRPV Cation Channels

2005
Facilitation and inhibition by capsaicin of cholinergic neurotransmission in the guinea-pig small intestine.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:4

    Topics: Acetylcholine; Animals; Capsaicin; Electric Stimulation; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Myenteric Plexus; Receptors, Cell Surface; TRPV Cation Channels

2006
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Apamin; Barium; Benzopyrans; Caffeine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Charybdotoxin; Diclofenac; Dimethyl Sulfoxide; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanethidine; Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nitroarginine; Papaverine; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Protein Serine-Threonine Kinases; Pyrazoles; Receptor, Cannabinoid, CB1; rho-Associated Kinases; Tetraethylammonium; Vasodilator Agents

2006
A novel mechanism contributing to development of Dahl salt-sensitive hypertension: role of the transient receptor potential vanilloid type 1.
    Hypertension (Dallas, Tex. : 1979), 2006, Volume: 47, Issue:3

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Ganglia, Spinal; Hypertension; Injections, Intravenous; Kidney; Male; Mesenteric Arteries; Neurons, Afferent; Rats; Rats, Inbred Dahl; Sodium Chloride, Dietary; TRPV Cation Channels; Vascular Resistance

2006
Stimulation by bradykinin of HCO3- secretion in rat gastroduodenal mucosa.
    Medical science monitor : international medical journal of experimental and clinical research, 2006, Volume: 12, Issue:1

    Topics: Animals; Bicarbonates; Bradykinin; Bradykinin B2 Receptor Antagonists; Capsaicin; Duodenum; Enzyme Inhibitors; Gastric Mucosa; Indomethacin; Intestinal Mucosa; Male; NG-Nitroarginine Methyl Ester; Pyridines; Rats; Rats, Sprague-Dawley

2006
Induction of apoptosis in prostate tumor PC-3 cells and inhibition of xenograft prostate tumor growth by the vanilloid capsaicin.
    Apoptosis : an international journal on programmed cell death, 2006, Volume: 11, Issue:1

    Topics: Androgens; Animals; Apoptosis; Capsaicin; Cell Line, Tumor; Cell Proliferation; Drug Resistance, Neoplasm; Gene Expression; Humans; Male; Mice; Mice, Nude; Neoplasm Transplantation; Prostatic Neoplasms; Reactive Oxygen Species; Transplantation, Heterologous; TRPV Cation Channels

2006
Role of cannabinoid receptors in Delta-9-tetrahydrocannabinol suppression of IL-12p40 in mouse bone marrow-derived dendritic cells infected with Legionella pneumophila.
    European journal of pharmacology, 2006, Feb-17, Volume: 532, Issue:1-2

    Topics: Animals; Bone Marrow Cells; Capsaicin; Cells, Cultured; Dendritic Cells; Dose-Response Relationship, Drug; Dronabinol; Enzyme-Linked Immunosorbent Assay; Gene Expression; Hallucinogens; Interleukin-12; Legionella pneumophila; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Pertussis Toxin; Protein Subunits; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; RNA, Messenger; TRPV Cation Channels

2006
Characterization of acid signaling in rat vagal pulmonary sensory neurons.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 291, Issue:1

    Topics: Acid Sensing Ion Channels; Acids; Amiloride; Animals; Capsaicin; Evoked Potentials; Hydrogen-Ion Concentration; Jugular Veins; Lung; Membrane Proteins; Nerve Tissue Proteins; Neurons, Afferent; Nodose Ganglion; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Channel Blockers; Sodium Channels; Stimulation, Chemical; TRPV Cation Channels

2006
Vanilloid VR1 receptor is involved in rimonabant-induced neuroprotection.
    British journal of pharmacology, 2006, Volume: 147, Issue:5

    Topics: Animals; Avoidance Learning; Brain Ischemia; Cannabinoid Receptor Antagonists; Capsaicin; Electroencephalography; Gerbillinae; Male; Motor Activity; Neuroprotective Agents; Piperidines; Pyrazoles; Rimonabant; TRPV Cation Channels

2006
Methanandamide hyperpolarizes gastric arteries by stimulation of TRPV1 receptors on perivascular CGRP containing nerves.
    Journal of cardiovascular pharmacology, 2006, Volume: 47, Issue:2

    Topics: Abdomen; Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Cannabinoids; Capsaicin; Electrophysiology; Female; Kinetics; Membrane Potentials; Mesenteric Arteries; Microelectrodes; Muscle, Smooth, Vascular; Peripheral Nervous System; Rats; Rats, Wistar; Receptors, Drug; TRPV Cation Channels

2006
Ethanol dilates coronary arteries and increases coronary flow via transient receptor potential vanilloid 1 and calcitonin gene-related peptide.
    Cardiovascular research, 2006, Jun-01, Volume: 70, Issue:3

    Topics: Animals; Arteries; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Endothelium, Vascular; Ethanol; Guinea Pigs; Humans; Peptide Fragments; Perfusion; Receptors, Calcitonin Gene-Related Peptide; Regional Blood Flow; Swine; Tissue Culture Techniques; TRPV Cation Channels; Vasodilator Agents

2006
Participation of the spinal TRPV1 receptors in formalin-evoked pain transduction: a study using a selective TRPV1 antagonist, iodo-resiniferatoxin.
    The Journal of pharmacy and pharmacology, 2006, Volume: 58, Issue:4

    Topics: Animals; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Spinal Cord; TRPV Cation Channels

2006
Protease-activated receptor-2 activation exaggerates TRPV1-mediated cough in guinea pigs.
    Journal of applied physiology (Bethesda, Md. : 1985), 2006, Volume: 101, Issue:2

    Topics: Animals; Capsaicin; Citric Acid; Cough; Cyclic AMP-Dependent Protein Kinases; Cyclooxygenase Inhibitors; Diterpenes; Guinea Pigs; Indomethacin; Inflammation; Isoquinolines; Male; Neurons, Afferent; Protein Kinase C; Protein Kinase Inhibitors; Receptor, PAR-2; Saline Solution, Hypertonic; Sulfonamides; TRPV Cation Channels; Trypsin

2006
Mediator mechanisms involved in TRPV1 and P2X receptor-mediated, ROS-evoked bradypneic reflex in anesthetized rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2006, Volume: 101, Issue:2

    Topics: Adenosine Deaminase; Adenosine Triphosphate; Animals; Apyrase; Arachidonic Acid; Capsaicin; Cyclooxygenase Inhibitors; Hydrogen Peroxide; Hyperventilation; Hypoventilation; Indomethacin; Lipoxygenase Inhibitors; Male; Oxidants; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, Purinergic P2; Receptors, Purinergic P2X; Reflex; Respiratory Mechanics; TRPV Cation Channels

2006
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:4

    Topics: Amidohydrolases; Anilides; Animals; Arachidonic Acids; Body Temperature; Capsaicin; Cinnamates; Endocannabinoids; Hypothermia; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; TRPV Cation Channels

2006
Gastro-protective action of lafutidine mediated by capsaicin-sensitive afferent neurons without interaction with TRPV1 and involvement of endogenous prostaglandins.
    World journal of gastroenterology, 2006, May-21, Volume: 12, Issue:19

    Topics: 6-Ketoprostaglandin F1 alpha; Acetamides; Animals; Calcium; Capsaicin; Dinoprostone; Dose-Response Relationship, Drug; Gastric Mucosa; Histamine H2 Antagonists; Humans; Indomethacin; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; NG-Nitroarginine Methyl Ester; Piperidines; Prostaglandins; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Epoprostenol; Stomach; Stomach Diseases; TRPV Cation Channels

2006
Effects of capsazepine on human small airway responsiveness unravel a novel class of bronchorelaxants.
    Pulmonary pharmacology & therapeutics, 2007, Volume: 20, Issue:3

    Topics: Acetylcholine; Adrenergic beta-Antagonists; Atropine; Bronchi; Bronchodilator Agents; Capsaicin; Cholinergic Agents; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; Histamine; Humans; In Vitro Techniques; Indomethacin; Leukotriene D4; Molecular Structure; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nifedipine; Peptides; Potassium Channels, Calcium-Activated; Propranolol; Prostaglandin D2; TRPV Cation Channels; Vasodilator Agents

2007
Antithrombin reduces endotoxin-induced hypotension by enhancing pulmonary sensory neuron activation in rats.
    Thrombosis and haemostasis, 2006, Volume: 95, Issue:6

    Topics: Animals; Antithrombins; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Carbazoles; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Cyclooxygenase Inhibitors; Disease Models, Animal; Endocannabinoids; Endotoxins; Ganglia, Spinal; Gene Expression Regulation; Hypotension; Indoles; Indomethacin; Lung; Male; Neurons, Afferent; Nitrates; Nitric Oxide Synthase Type II; Nitrites; Peptide Fragments; Polyunsaturated Alkamides; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; RNA, Messenger; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2006
Tactile allodynia initiated by local subcutaneous endothelin-1 is prolonged by activation of TRPV-1 receptors.
    Experimental biology and medicine (Maywood, N.J.), 2006, Volume: 231, Issue:6

    Topics: Animals; Behavior, Animal; Capsaicin; Diterpenes; Dose-Response Relationship, Drug; Endothelin-1; Injections, Subcutaneous; Male; Nociceptors; Pain; Rats; Rats, Sprague-Dawley; Reaction Time; Receptor, Endothelin A; Touch; TRPV Cation Channels

2006
Effect of intracochlear perfusion of vanilloids on cochlear neural activity in the guinea pig.
    Hearing research, 2006, Volume: 218, Issue:1-2

    Topics: Animals; Capsaicin; Cochlea; Cochlear Microphonic Potentials; Cochlear Nerve; Evoked Potentials, Auditory; Female; Guinea Pigs; Male; Perfusion; TRPV Cation Channels

2006
Role of substance P in hydrogen sulfide-induced pulmonary inflammation in mice.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 291, Issue:5

    Topics: Air Pollutants; Animals; Anti-Inflammatory Agents, Non-Steroidal; Biphenyl Compounds; Capsaicin; Female; Hydrogen Sulfide; Inflammation Mediators; Lung; Male; Mice; Mice, Inbred BALB C; Mice, Mutant Strains; Neurokinin-1 Receptor Antagonists; Peroxidase; Pneumonia; Protein Precursors; Substance P; Tachykinins; TRPV Cation Channels

2006
A role for vanilloid receptor 1 (TRPV1) and endocannabinnoid signalling in the regulation of spontaneous and L-DOPA induced locomotion in normal and reserpine-treated rats.
    Neuropharmacology, 2006, Volume: 51, Issue:3

    Topics: Adrenergic Uptake Inhibitors; Analysis of Variance; Animals; Arachidonic Acids; Behavior, Animal; Benzamides; Benzyl Compounds; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Levodopa; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Reserpine; Signal Transduction; TRPV Cation Channels

2006
Carbonic anhydrases and mucosal vanilloid receptors help mediate the hyperemic response to luminal CO2 in rat duodenum.
    Gastroenterology, 2006, Volume: 131, Issue:1

    Topics: Amiloride; Animals; Benzolamide; Blood Flow Velocity; Capsaicin; Carbon Dioxide; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Disease Models, Animal; Duodenum; Epithelial Cells; Gene Expression; Hydrogen-Ion Concentration; Hyperemia; Intestinal Mucosa; Intracellular Fluid; Laser-Doppler Flowmetry; Male; Methazolamide; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA; Sodium-Calcium Exchanger; TRPV Cation Channels

2006
TRPV1 receptors and nasal trigeminal chemesthesis.
    Chemical senses, 2006, Volume: 31, Issue:9

    Topics: Animals; Calcium; Capsaicin; Cell Line; Humans; Irritants; Male; Rats; Rats, Sprague-Dawley; Smell; Stimulation, Chemical; Transfection; Trigeminal Nerve; TRPV Cation Channels

2006
Transient receptor potential vanilloid subtype 1 mediates microglial cell death in vivo and in vitro via Ca2+-mediated mitochondrial damage and cytochrome c release.
    Journal of immunology (Baltimore, Md. : 1950), 2006, Oct-01, Volume: 177, Issue:7

    Topics: Animals; Blotting, Western; Calcium; Capsaicin; Cell Death; Cell Line; Cytochromes c; Diterpenes; Enzyme Inhibitors; Humans; Immunohistochemistry; In Situ Nick-End Labeling; In Vitro Techniques; Microglia; Mitochondria; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Substantia Nigra; TRPV Cation Channels

2006
Cannabinoid (CB1) receptor activation inhibits trigeminovascular neurons.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:1

    Topics: Animals; Arachidonic Acids; Benzoxazines; Blood Pressure; Capsaicin; Endocannabinoids; Male; Migraine Disorders; Morpholines; Naphthalenes; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; RNA, Messenger; Trigeminal Nerve; TRPV Cation Channels

2007
Synergistic antinociceptive effects of anandamide, an endocannabinoid, and nonsteroidal anti-inflammatory drugs in peripheral tissue: a role for endogenous fatty-acid ethanolamides?
    European journal of pharmacology, 2006, Nov-21, Volume: 550, Issue:1-3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acids; Capsaicin; Chromatography, High Pressure Liquid; Cyclooxygenase 2 Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Edema; Endocannabinoids; Formaldehyde; Ibuprofen; Lactones; Male; Mass Spectrometry; Nitrobenzenes; Pain Measurement; Peripheral Nervous System; Polyunsaturated Alkamides; Rats; Rats, Wistar; Sulfonamides; Sulfones; TRPV Cation Channels

2006
Capsaicin inhibits catecholamine secretion and synthesis by blocking Na+ and Ca2+ influx through a vanilloid receptor-independent pathway in bovine adrenal medullary cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 374, Issue:2

    Topics: Adrenal Medulla; Analgesics, Non-Narcotic; Animals; Benzaldehydes; Calcium; Calcium Radioisotopes; Capsaicin; Carbachol; Catecholamines; Cattle; Cells, Cultured; Cholinergic Agonists; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Histamine; Ion Transport; Ruthenium Red; Signal Transduction; Sodium; Sodium Radioisotopes; TRPV Cation Channels; Tyrosine 3-Monooxygenase; Veratridine

2006
TRPV1 is a novel target for omega-3 polyunsaturated fatty acids.
    The Journal of physiology, 2007, Jan-15, Volume: 578, Issue:Pt 2

    Topics: Animals; Binding, Competitive; Calcium; Capsaicin; Cell Line; Cell Membrane; Diterpenes; Fatty Acids, Omega-3; Fatty Acids, Omega-6; Female; Humans; Hydrogen-Ion Concentration; Linoleic Acid; Male; Membrane Fluidity; Membrane Potentials; Mice; Mice, Inbred C57BL; Oocytes; Pain; Rats; RNA, Complementary; TRPV Cation Channels; Xenopus laevis

2007
Anandamide mediates hyperdynamic circulation in cirrhotic rats via CB(1) and VR(1) receptors.
    British journal of pharmacology, 2006, Volume: 149, Issue:7

    Topics: Animals; Arachidonic Acids; Bile Ducts; Blood Flow Velocity; Blood Pressure; Blotting, Western; Capsaicin; Cardiac Output; Disease Models, Animal; Endocannabinoids; Hyperemia; Indoles; Liver Circulation; Liver Cirrhosis, Biliary; Male; Mesenteric Artery, Superior; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Splanchnic Circulation; Time Factors; TRPV Cation Channels; Vascular Resistance; Vasodilation; Vasodilator Agents

2006
Differential mechanisms mediating depressor and diuretic effects of anandamide.
    Journal of hypertension, 2006, Volume: 24, Issue:11

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcium Channel Blockers; Capsaicin; Diuresis; Dose-Response Relationship, Drug; Endocannabinoids; Kidney; Kidney Medulla; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1

2006
Involvement of endothelial cell-derived CGRP in heat stress-induced protection of endothelial function.
    Vascular pharmacology, 2007, Volume: 46, Issue:4

    Topics: Animals; Aorta, Thoracic; Calcitonin Gene-Related Peptide; Capsaicin; Cell Survival; Cells, Cultured; Disease Models, Animal; Endothelial Cells; Endothelium, Vascular; Heat Stress Disorders; Humans; Lysophosphatidylcholines; Male; Mesenteric Arteries; Peptide Fragments; Rats; Rats, Sprague-Dawley; RNA, Messenger; Time Factors; TRPV Cation Channels; Vasodilation

2007
The non-psychoactive cannabis constituent cannabidiol is an orally effective therapeutic agent in rat chronic inflammatory and neuropathic pain.
    European journal of pharmacology, 2007, Feb-05, Volume: 556, Issue:1-3

    Topics: Administration, Oral; Animals; Cannabidiol; Cannabinoid Receptor Antagonists; Cannabis; Capsaicin; Chronic Disease; Dinoprostone; Freund's Adjuvant; Hyperalgesia; Inflammation; Lipid Peroxides; Male; NF-kappa B; Nitric Oxide; Nitric Oxide Synthase; Pain; Pain Measurement; Rats; Rats, Wistar; Sciatic Neuropathy; Tumor Necrosis Factor-alpha

2007
Vanilloid receptor agonists and antagonists are mitochondrial inhibitors: how vanilloids cause non-vanilloid receptor mediated cell death.
    Biochemical and biophysical research communications, 2007, Mar-02, Volume: 354, Issue:1

    Topics: Anilides; Animals; Apoptosis; Capsaicin; Carcinoma, Non-Small-Cell Lung; Cells, Cultured; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Humans; Hydrogen Peroxide; Lung Neoplasms; Membrane Potentials; Mitochondria, Heart; Oxygen Consumption; Rats; TRPV Cation Channels

2007
Vanilloid (subtype 1) receptor-modulatory drugs inhibit [3H]batrachotoxinin-A 20-alpha-benzoate binding to Na+ channels.
    Basic & clinical pharmacology & toxicology, 2007, Volume: 100, Issue:2

    Topics: Animals; Aspartic Acid; Batrachotoxins; Brain; Capsaicin; gamma-Aminobutyric Acid; Glutamic Acid; Male; Mice; Mice, Inbred Strains; Potassium Chloride; Sodium Channels; Synaptosomes; Tritium; TRPV Cation Channels; Veratridine

2007
Mouse colon sensory neurons detect extracellular acidosis via TRPV1.
    American journal of physiology. Cell physiology, 2007, Volume: 292, Issue:5

    Topics: Acidosis; Amiloride; Animals; Capsaicin; Cell Size; Cells, Cultured; Colon; Evoked Potentials; Extracellular Fluid; Ganglia, Spinal; Hydrogen-Ion Concentration; Kinetics; Lumbosacral Plexus; Male; Mechanotransduction, Cellular; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; Pain; Patch-Clamp Techniques; Sodium Channel Blockers; Thoracic Nerves; TRPV Cation Channels

2007
TRPV1 is involved in stretch-evoked contractile changes in the rat autonomous bladder model: a study with piperine, a new TRPV1 agonist.
    Neurourology and urodynamics, 2007, Volume: 26, Issue:3

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Indicators and Reagents; Mechanotransduction, Cellular; Muscle Contraction; Piperidines; Polyunsaturated Alkamides; Pressure; Rats; Rats, Wistar; Ruthenium Red; Stress, Mechanical; TRPV Cation Channels; Urinary Bladder

2007
Pharmacological characterization of receptor types mediating the dilator action of anandamide on blood vessels of the rat knee joint.
    Life sciences, 2007, Mar-27, Volume: 80, Issue:16

    Topics: Amidohydrolases; Analysis of Variance; Animals; Arachidonic Acids; Benzamides; Blood Vessels; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Endocannabinoids; Flurbiprofen; Hindlimb; Indoles; Joints; Morpholines; Polyunsaturated Alkamides; Pyrazoles; Rats; Regional Blood Flow; TRPV Cation Channels; Vasodilation

2007
Heat sensitization in skin and muscle nociceptors expressing distinct combinations of TRPV1 and TRPV2 protein.
    Journal of neurophysiology, 2007, Volume: 97, Issue:4

    Topics: Animals; Capsaicin; Colon; Histocytochemistry; Hot Temperature; Male; Muscle, Skeletal; Muscle, Smooth; Muscles; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neurofilament Proteins; Neurons, Afferent; Nociceptors; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Signal Transduction; Skin; TRPV Cation Channels

2007
Pharmacological characterisation of capsaicin-induced relaxations in human and porcine isolated arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adolescent; Adult; Aged; Analgesics, Non-Narcotic; Animals; Arteries; Calcitonin Gene-Related Peptide; Capsaicin; Coronary Vessels; Cyclic AMP; Dipeptides; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Middle Aged; NG-Nitroarginine Methyl Ester; Piperazines; Piperidines; Potassium Channel Blockers; Potassium Chloride; Protein Kinase Inhibitors; Quinazolines; Swine; Vasodilation

2007
Capsicum ethanol extracts and capsaicin enhance interleukin-2 and interferon-gamma production in cultured murine Peyer's patch cells ex vivo.
    Life sciences, 2007, Apr-03, Volume: 80, Issue:17

    Topics: Administration, Oral; Analgesics, Non-Narcotic; Animals; Capsaicin; Capsicum; Cell Proliferation; Cells, Cultured; Concanavalin A; Dose-Response Relationship, Drug; Drug Antagonism; Drug Combinations; Ethanol; Interferon-gamma; Interleukin-2; Male; Mice; Mice, Inbred C57BL; Peyer's Patches; Plant Extracts; T-Lymphocyte Subsets; TRPV Cation Channels

2007
Capsaicin induces the production of IL-6 in human upper respiratory epithelial cells.
    Life sciences, 2007, Apr-03, Volume: 80, Issue:17

    Topics: Analgesics, Non-Narcotic; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Humans; Interleukin-6; Respiratory Mucosa; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; TRPV Cation Channels

2007
Endocannabinoid regulates blood pressure via activation of the transient receptor potential vanilloid type 1 in Wistar rats fed a high-salt diet.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:2

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Cannabinoid Receptor Modulators; Capsaicin; Endocannabinoids; Hypertension; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Sodium Chloride, Dietary; TRPV Cation Channels

2007
Novel agonistic action of mustard oil on recombinant and endogenous porcine transient receptor potential V1 (pTRPV1) channels.
    Biochemical pharmacology, 2007, May-15, Volume: 73, Issue:10

    Topics: Animals; Calcium; Capsaicin; Cells, Cultured; Ganglia, Spinal; Humans; Membrane Potentials; Mustard Plant; Neurons; Plant Oils; Rats; Recombinant Proteins; Sus scrofa; Swine; TRPV Cation Channels

2007
TRPV1 mediates histamine-induced itching via the activation of phospholipase A2 and 12-lipoxygenase.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Feb-28, Volume: 27, Issue:9

    Topics: Animals; Arachidonate 12-Lipoxygenase; Calcium; Capsaicin; Cells, Cultured; Enzyme Activation; Ganglia, Spinal; Histamine; Mice; Mice, Inbred C57BL; Neurons; Phospholipases A; Phospholipases A2; Rats; TRPV Cation Channels

2007
Capsaicin-induced mucus secretion in rat airways assessed in vivo and non-invasively by magnetic resonance imaging.
    British journal of pharmacology, 2007, Volume: 150, Issue:8

    Topics: Animals; Aza Compounds; Benzamides; Bronchoalveolar Lavage Fluid; Capsaicin; Cromolyn Sodium; Goblet Cells; Lung; Magnetic Resonance Imaging; Male; Mucus; Neurons, Afferent; Rats; Rats, Inbred BN; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Time Factors; TRPV Cation Channels

2007
Discovery of a potent and long-acting bronchorelaxing capsazepinoid, RESPIR 4-95.
    Pulmonary pharmacology & therapeutics, 2008, Volume: 21, Issue:1

    Topics: Adrenergic beta-2 Receptor Agonists; Bronchodilator Agents; Calcium Channel Blockers; Capsaicin; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Leukotriene D4; Lung; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Tetrahydroisoquinolines

2008
Activation of recombinant human TRPV1 receptors expressed in SH-SY5Y human neuroblastoma cells increases [Ca(2+)](i), initiates neurotransmitter release and promotes delayed cell death.
    Journal of neurochemistry, 2007, Volume: 102, Issue:3

    Topics: Arachidonic Acids; Calcium; Calcium Signaling; Capsaicin; Cell Culture Techniques; Cell Death; Cell Line, Tumor; Cell Proliferation; Diterpenes; Dopamine; Endocannabinoids; Humans; Models, Biological; Neuroblastoma; Neurons; Norepinephrine; Polyunsaturated Alkamides; Recombinant Proteins; Synaptic Transmission; Transfection; TRPV Cation Channels; Up-Regulation

2007
AM404 decreases Fos-immunoreactivity in the spinal cord in a model of inflammatory pain.
    Brain research, 2007, Jun-04, Volume: 1152

    Topics: Animals; Arachidonic Acids; Capsaicin; Endocannabinoids; Immunohistochemistry; Indoles; Inflammation; Male; Pain; Pain Measurement; Piperidines; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-fos; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Spinal Cord; TRPV Cation Channels

2007
Transient receptor potential vanilloid-1 mediates heat-shock-induced matrix metalloproteinase-1 expression in human epidermal keratinocytes.
    The Journal of investigative dermatology, 2007, Volume: 127, Issue:10

    Topics: Calcium Signaling; Capsaicin; Cell Line; Cells, Cultured; Gene Expression Regulation; Hot Temperature; Humans; Keratinocytes; Male; Matrix Metalloproteinase 1; RNA, Messenger; RNA, Small Interfering; Ruthenium Red; TRPV Cation Channels

2007
Atrial natriuretic peptide reduces ischemia/reperfusion-induced spinal cord injury in rats by enhancing sensory neuron activation.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Anilides; Animals; Atrial Natriuretic Factor; Calcitonin Gene-Related Peptide; Capsaicin; Carbazoles; Cells, Cultured; Cinnamates; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Indoles; Indomethacin; Male; Neurons, Afferent; Peroxidase; Psychomotor Performance; Pyrroles; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Spinal Cord; Spinal Cord Diseases; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2007
Transient receptor potential vanilloid 1 antagonist, capsazepine, improves survival in a rat hemorrhagic shock model.
    Annals of surgery, 2007, Volume: 245, Issue:6

    Topics: Analysis of Variance; Animals; Capsaicin; Catecholamines; Disease Models, Animal; Dose-Response Relationship, Drug; Immunoenzyme Techniques; Male; Rats; Rats, Sprague-Dawley; Shock, Hemorrhagic; Survival Rate

2007
The role of TRPV1 receptors in the antinociceptive effect of anandamide at spinal level.
    Pain, 2008, Volume: 134, Issue:3

    Topics: Analgesics; Animals; Arachidonic Acids; Capsaicin; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; Hyperalgesia; Injections, Spinal; Male; Polyunsaturated Alkamides; Rats; Rats, Wistar; Spinal Cord; TRPV Cation Channels

2008
Capsaicin-induced avoidance behavior in the terrestrial Gastropoda Megalobulimus abbreviatus: evidence for TRPV-1 signaling and opioid modulation in response to chemical noxious stimuli.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2007, Volume: 148, Issue:2

    Topics: Administration, Topical; Analgesics, Opioid; Animals; Behavior, Animal; Capsaicin; Dose-Response Relationship, Drug; Hot Temperature; Morphine; Naloxone; Narcotic Antagonists; Pain Measurement; Pain Threshold; Reaction Time; Receptors, Opioid; Ruthenium Red; Signal Transduction; Snails; TRPV Cation Channels

2007
Surfactant-induced TRPV1 activity--a novel mechanism for eye irritation?
    Toxicological sciences : an official journal of the Society of Toxicology, 2007, Volume: 99, Issue:1

    Topics: Animal Testing Alternatives; Calcium; Calcium Signaling; Capsaicin; Cell Line, Tumor; Dose-Response Relationship, Drug; Eye Diseases; Fluorescent Antibody Technique, Indirect; Humans; Irritants; Neuroblastoma; Neurons, Afferent; Sodium Dodecyl Sulfate; Surface-Active Agents; TRPV Cation Channels

2007
Effects of anandamide and noxious heat on intracellular calcium concentration in nociceptive drg neurons of rats.
    Journal of neurophysiology, 2007, Volume: 98, Issue:2

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Calcium; Calcium Channel Blockers; Capsaicin; Chelating Agents; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Egtazic Acid; Endocannabinoids; Extracellular Fluid; Ganglia, Spinal; Hot Temperature; Neurons; Physical Stimulation; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2007
Role of capsaicin-sensitive sensory nerves in protease-activated receptor-2-mediated contraction of rat urinary bladder.
    European journal of pharmacology, 2007, Aug-13, Volume: 569, Issue:1-2

    Topics: Acetylcholine; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Capsaicin; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Neurons, Afferent; Oligopeptides; Rats; Rats, Wistar; Receptor, PAR-2; Trypsin; Urinary Bladder

2007
Involvement of the endocannabinoid system in retinal damage after high intraocular pressure-induced ischemia in rats.
    Investigative ophthalmology & visual science, 2007, Volume: 48, Issue:7

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Benzamides; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cell Count; Chromatography, High Pressure Liquid; Endocannabinoids; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Hydrolysis; Intraocular Pressure; Male; Ocular Hypertension; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reperfusion Injury; Retinal Diseases; Retinal Ganglion Cells; Retinal Vessels; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Thy-1 Antigens; TRPV Cation Channels

2007
Fatty acyl amides of endogenous tetrahydroisoquinolines are active at the recombinant human TRPV1 receptor.
    Bioorganic & medicinal chemistry, 2007, Sep-15, Volume: 15, Issue:18

    Topics: Amides; Calcium; Capsaicin; Cells, Cultured; Fatty Acids; Humans; Kidney; Recombinant Proteins; Tetrahydroisoquinolines; TRPV Cation Channels

2007
Bladder afferent sensitivity in wild-type and TRPV1 knockout mice.
    The Journal of physiology, 2007, Sep-01, Volume: 583, Issue:Pt 2

    Topics: Action Potentials; Animals; Capsaicin; Hydrochloric Acid; Male; Mechanotransduction, Cellular; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; Pressure; Time Factors; TRPV Cation Channels; Urinary Bladder

2007
A potential role for the vanilloid receptor TRPV1 in the therapeutic effect of curcumin in dinitrobenzene sulphonic acid-induced colitis in mice.
    Neurogastroenterology and motility, 2007, Volume: 19, Issue:8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzenesulfonates; Capsaicin; Cell Membrane; Colitis; Curcumin; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Oocytes; Peroxidase; Severity of Illness Index; TRPV Cation Channels; Xenopus

2007
The anandamide transport inhibitor AM404 reduces ethanol self-administration.
    The European journal of neuroscience, 2007, Volume: 26, Issue:2

    Topics: Alcohol Drinking; Animals; Arachidonic Acids; Capsaicin; Central Nervous System Depressants; Conditioning, Operant; Depression, Chemical; Endocannabinoids; Ethanol; Extinction, Psychological; Hypothermia; Male; Motor Activity; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Reinforcement, Psychology; Saccharin; Self Administration; TRPV Cation Channels

2007
Effect of capsaicin on plasma and tissue levels of insulin-like growth factor-I in spontaneously hypertensive rats.
    Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society, 2008, Volume: 18, Issue:1

    Topics: Animals; Antihypertensive Agents; Calcitonin Gene-Related Peptide; Capsaicin; Cyclic AMP; Ganglia, Spinal; Hypertension; Insulin-Like Growth Factor I; Neurons, Afferent; Rats; Rats, Inbred SHR; Rats, Inbred WKY

2008
Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Aorta, Abdominal; Apamin; Arachidonic Acids; Benzamides; Calcitonin Gene-Related Peptide; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Charybdotoxin; Dose-Response Relationship, Drug; Endocannabinoids; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Isoindoles; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptide Fragments; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sulfonamides; Vasodilation

2007
TRPV1-mediated diuresis and natriuresis induced by hypertonic saline perfusion of the renal pelvis.
    American journal of nephrology, 2007, Volume: 27, Issue:5

    Topics: Afferent Pathways; Animals; Capsaicin; Diuresis; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Isoindoles; Kidney; Kidney Pelvis; Male; Natriuresis; Neurokinin-1 Receptor Antagonists; Perfusion; Potassium Chloride; Rats; Rats, Wistar; Saline Solution, Hypertonic; Solutions; TRPV Cation Channels

2007
Involvement of a capsaicin-sensitive TRPV1-independent mechanism in lipopolysaccharide-induced fever in chickens.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2007, Volume: 148, Issue:3

    Topics: Analgesics, Non-Narcotic; Animals; Animals, Newborn; Body Temperature; Capsaicin; Cells, Cultured; Chickens; Fever; Lipopolysaccharides; Macrophages, Peritoneal; Male; Nitric Oxide; Nitrites; Time Factors; TRPV Cation Channels

2007
Hydroxy-alpha-sanshool activates TRPV1 and TRPA1 in sensory neurons.
    The European journal of neuroscience, 2007, Volume: 26, Issue:5

    Topics: Amides; Analysis of Variance; Animals; Animals, Newborn; Calcium; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Humans; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; Patch-Clamp Techniques; Plant Extracts; Rats; Rats, Sprague-Dawley; Taste; Transfection; Transient Receptor Potential Channels; TRPV Cation Channels

2007
Delta 9-tetrahydrocannabinol inhibits electrically-evoked CGRP release and capsaicin-sensitive sensory neurogenic vasodilatation in the rat mesenteric arterial bed.
    British journal of pharmacology, 2007, Volume: 152, Issue:5

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Dronabinol; Electric Stimulation; Indoles; Male; Mesenteric Arteries; Methoxamine; Neurons, Afferent; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Ruthenium Red; Time Factors; Vasodilation

2007
Acid-induced modulation of airway basal tone and contractility: role of acid-sensing ion channels (ASICs) and TRPV1 receptor.
    Life sciences, 2007, Sep-08, Volume: 81, Issue:13

    Topics: Acid Sensing Ion Channels; Acidosis; Amiloride; Animals; Capsaicin; Enzyme Inhibitors; Guinea Pigs; Hydrogen-Ion Concentration; Male; Membrane Proteins; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Nerve Tissue Proteins; Poisons; Receptors, Tachykinin; Sensory Receptor Cells; Sodium Channel Blockers; Sodium Channels; Tetrodotoxin; Trachea; TRPV Cation Channels

2007
Anti-dyskinetic effects of cannabinoids in a rat model of Parkinson's disease: role of CB(1) and TRPV1 receptors.
    Experimental neurology, 2007, Volume: 208, Issue:1

    Topics: Amidohydrolases; Animals; Antiparkinson Agents; Arachidonic Acids; Basal Ganglia; Benzamides; Benzoxazines; Cannabinoids; Capsaicin; Carbamates; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Endocannabinoids; Levodopa; Male; Morpholines; Naphthalenes; Oxidopamine; Parkinson Disease, Secondary; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2007
Voltage is a partial activator of rat thermosensitive TRP channels.
    The Journal of physiology, 2007, Dec-01, Volume: 585, Issue:Pt 2

    Topics: Allosteric Regulation; Animals; Capsaicin; Cell Line; Diterpenes; Electric Stimulation; Hot Temperature; Humans; Ion Channel Gating; Kidney; Membrane Potentials; Models, Chemical; Neurons, Afferent; Protein Kinase C; Rats; Sensory System Agents; TRPM Cation Channels; TRPV Cation Channels

2007
Transient receptor potential vanilloid 1 (TRPV1) channels in cultured rat Sertoli cells regulate an acid sensing chloride channel.
    Biochemical pharmacology, 2008, Jan-15, Volume: 75, Issue:2

    Topics: Animals; Calcium; Capsaicin; Cells, Cultured; Chloride Channels; Hydrogen-Ion Concentration; Ibuprofen; Male; Rats; Rats, Wistar; Sertoli Cells; TRPV Cation Channels

2008
Roles of TRPV1 and neuropeptidergic receptors in dorsal root reflex-mediated neurogenic inflammation induced by intradermal injection of capsaicin.
    Molecular pain, 2007, Oct-25, Volume: 3

    Topics: Analgesics; Animals; Bicuculline; Calcitonin Gene-Related Peptide; Capsaicin; Edema; GABA Antagonists; Injections, Intradermal; Neurogenic Inflammation; Peptide Fragments; Rats; Receptors, Neurokinin-1; Reflex; Spinal Nerve Roots; Substance P; TRPV Cation Channels; Vasodilation

2007
Quebrachitol-induced gastroprotection against acute gastric lesions: role of prostaglandins, nitric oxide and K+ ATP channels.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2008, Volume: 15, Issue:5

    Topics: Animals; Arginine; Capsaicin; Diazoxide; Dose-Response Relationship, Drug; Ethanol; Glyburide; Indomethacin; Inositol; KATP Channels; Male; Mice; Misoprostol; Molecular Structure; NG-Nitroarginine Methyl Ester; Nitric Oxide; Phytotherapy; Prostaglandins; Stomach Ulcer

2008
Involvement of peripheral TRPV1 in TMJ hyperalgesia induced by ethanol withdrawal.
    Life sciences, 2007, Nov-30, Volume: 81, Issue:23-24

    Topics: Animals; Capsaicin; Central Nervous System Depressants; Ethanol; Formaldehyde; Male; Pain Measurement; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Temporomandibular Joint Dysfunction Syndrome; TRPV Cation Channels

2007
Increased depressor response to N-arachidonoyl-dopamine during high salt intake: role of the TRPV1 receptor.
    Journal of hypertension, 2007, Volume: 25, Issue:12

    Topics: Animals; Arachidonic Acids; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Dopamine; Male; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Rimonabant; Sodium Chloride, Dietary; TRPV Cation Channels

2007
TRPV1 receptor signaling mediates afferent nerve sensitization during colitis-induced motility disorders in rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2008, Volume: 294, Issue:1

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Colitis; Disease Models, Animal; Dose-Response Relationship, Drug; Ganglia, Spinal; Gastric Emptying; Gastrointestinal Motility; Gastroparesis; Intestinal Mucosa; Intestines; Male; Muscle Relaxation; Neurons, Afferent; Peptide Fragments; Pyrazines; Pyridines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; RNA, Messenger; Signal Transduction; Time Factors; Trinitrobenzenesulfonic Acid; TRPV Cation Channels

2008
Transient receptor potential vanilloid type 1 channels act as mechanoreceptors and cause substance P release and sensory activation in rat kidneys.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:2

    Topics: Action Potentials; Animals; Blood Pressure; Capsaicin; Cell Membrane; Cytosol; Diterpenes; Electrophysiology; Female; Kidney; Kidney Pelvis; Mechanoreceptors; Models, Biological; Neurokinin-1 Receptor Antagonists; Perfusion; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory System Agents; Substance P; TRPV Cation Channels; Ubiquitin Thiolesterase

2008
SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ring.
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: Bronchodilator Agents; Capsaicin; Catechols; Chlorine Compounds; Humans; Molecular Structure; Respiration; Structure-Activity Relationship

2008
SAR studies of capsazepinoid bronchodilators. Part 1: The importance of the catechol moiety and aspects of the B-ring structure.
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: Bronchodilator Agents; Capsaicin; Catechols; Humans; Models, Molecular; Molecular Structure; Respiration; Structure-Activity Relationship

2008
TRPM8 mechanism of cold allodynia after chronic nerve injury.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Dec-12, Volume: 27, Issue:50

    Topics: Animals; Capsaicin; Cells, Cultured; Chronic Disease; Cold Temperature; Disease Models, Animal; Female; Ganglia, Spinal; Hyperalgesia; Ligation; Male; Menthol; Neurons, Afferent; Pain Measurement; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sciatic Neuropathy; Skin; TRPM Cation Channels

2007
Effect of increasing temperature on TRPV1-mediated responses in isolated rat pulmonary sensory neurons.
    American journal of physiology. Lung cellular and molecular physiology, 2008, Volume: 294, Issue:3

    Topics: Acrylamides; Animals; Boron Compounds; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Evoked Potentials; Hexamethonium; Hydrogen-Ion Concentration; Hyperthermia, Induced; Lung; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Temperature; TRPV Cation Channels; Vagus Nerve

2008
Cardiac oxidative stress and electrophysiological changes in rats exposed to concentrated ambient particles are mediated by TRP-dependent pulmonary reflexes.
    Toxicological sciences : an official journal of the Society of Toxicology, 2008, Volume: 102, Issue:2

    Topics: Action Potentials; Air Pollutants; Animals; Autonomic Nervous System; Capsaicin; Drug Interactions; Edema; Edema, Cardiac; Heart Diseases; Heart Rate; Inhalation Exposure; Lipid Peroxidation; Oxidative Stress; Particle Size; Particulate Matter; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2008
Capsazepine, a synthetic vanilloid that converts the Na,K-ATPase to Na-ATPase.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Feb-05, Volume: 105, Issue:5

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Capsaicin; Cation Transport Proteins; Cations, Monovalent; Kinetics; Ligands; Sodium; Sodium-Potassium-Exchanging ATPase

2008
SAR studies of capsazepinoid bronchodilators 3: The thiourea part (coupling region) and the 2-(4-chlorophenyl)ethyl moiety (C-region).
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: Bronchodilator Agents; Capsaicin; Chlorine Compounds; Humans; Hydrophobic and Hydrophilic Interactions; Lipids; Molecular Structure; Respiration; Structure-Activity Relationship; Thiourea

2008
Pronociceptive response elicited by TRPA1 receptor activation in mice.
    Neuroscience, 2008, Mar-18, Volume: 152, Issue:2

    Topics: Analgesics; Anilides; Animals; Behavior, Animal; Capsaicin; Cinnamates; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Isothiocyanates; Male; Mice; Pain; Pain Measurement; Ruthenium Red; Time Factors; Transient Receptor Potential Channels; TRPA1 Cation Channel

2008
Increased GFR and renal excretory function by activation of TRPV1 in the isolated perfused kidney.
    Pharmacological research, 2008, Volume: 57, Issue:3

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Colorimetry; Dose-Response Relationship, Drug; Glomerular Filtration Rate; In Vitro Techniques; Kidney; Male; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Radioimmunoassay; Rats; Rats, Wistar; Sodium; Substance P; TRPV Cation Channels

2008
TRPV1 mediates cell death in rat synovial fibroblasts through calcium entry-dependent ROS production and mitochondrial depolarization.
    Biochemical and biophysical research communications, 2008, May-16, Volume: 369, Issue:4

    Topics: Animals; Apoptosis; Arthritis, Experimental; Calcium; Capsaicin; Cytosol; Fibroblasts; Hyperplasia; Male; Membrane Potential, Mitochondrial; NADPH Oxidases; Onium Compounds; Rats; Rats, Wistar; Reactive Oxygen Species; Synovial Membrane; TRPV Cation Channels

2008
TRPV1-mediated protection against endotoxin-induced hypotension and mortality in rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2008, Volume: 294, Issue:5

    Topics: Animals; Blood Pressure; Capsaicin; Catecholamines; Endotoxins; Heart Rate; Hypotension; Isoindoles; Lipopolysaccharides; Male; Neurons, Afferent; Rats; Rats, Wistar; Receptors, Neurokinin-1; Substance P; TRPV Cation Channels

2008
Lafutidine facilitates calcitonin gene-related peptide (CGRP) nerve-mediated vasodilation via vanilloid-1 receptors in rat mesenteric resistance arteries.
    Journal of pharmacological sciences, 2008, Volume: 106, Issue:3

    Topics: Acetamides; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Drug Synergism; Electric Stimulation; Male; Mesenteric Arteries; Peripheral Nervous System; Piperidines; Pyridines; Rats; Rats, Wistar; Ruthenium Red; TRPV Cation Channels; Vasodilation

2008
Dependence of regulatory volume decrease on transient receptor potential vanilloid 4 (TRPV4) expression in human corneal epithelial cells.
    Cell calcium, 2008, Volume: 44, Issue:4

    Topics: Calcium; Capsaicin; Cell Line; Coloring Agents; Epithelium, Corneal; Gene Knockdown Techniques; Humans; Hypotonic Solutions; Isotonic Solutions; Ringer's Solution; RNA, Small Interfering; Ruthenium Red; TRPV Cation Channels

2008
Interdependent regulation of afferent renal nerve activity and renal function: role of transient receptor potential vanilloid type 1, neurokinin 1, and calcitonin gene-related peptide receptors.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:3

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Ganglia, Spinal; Isoindoles; Kidney Pelvis; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Fragments; Quinuclidines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Substance P; TRPV Cation Channels

2008
Impaired capsaicin-induced relaxation of coronary arteries in a porcine model of the metabolic syndrome.
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 294, Issue:6

    Topics: Animals; Calcium; Capsaicin; Coronary Vessels; Disease Models, Animal; Dose-Response Relationship, Drug; Down-Regulation; Endothelium, Vascular; Enzyme Inhibitors; Male; Manganese; Metabolic Syndrome; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Obesity; Potassium Channel Blockers; Potassium Channels; Swine; Swine, Miniature; TRPV Cation Channels; Vasodilation; Vasodilator Agents

2008
Segmental regulation of sodium and water excretion by TRPV1 activation in the kidney.
    Journal of cardiovascular pharmacology, 2008, Volume: 51, Issue:5

    Topics: Animals; Blood Pressure; Body Water; Capsaicin; Cations, Monovalent; Creatinine; Glomerular Filtration Rate; Kidney; Lithium; Lithium Chloride; Male; Natriuresis; Nerve Fibers; Rats; Rats, Wistar; Renal Circulation; Sodium; TRPV Cation Channels

2008
Role of TRPV1 channels in renal haemodynamics and function in Dahl salt-sensitive hypertensive rats.
    Experimental physiology, 2008, Volume: 93, Issue:8

    Topics: Animals; Blood Pressure; Capsaicin; Disease Models, Animal; Glomerular Filtration Rate; Hypertension; Kidney; Rats; Rats, Inbred Dahl; Sodium; TRPV Cation Channels

2008
Antistress effect of TRPV1 channel on synaptic plasticity and spatial memory.
    Biological psychiatry, 2008, Aug-15, Volume: 64, Issue:4

    Topics: Anilides; Animals; Animals, Newborn; Behavior, Animal; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Male; Memory; Neuronal Plasticity; Neurons; Rats; Rats, Wistar; Space Perception; Synaptic Transmission; TRPV Cation Channels

2008
Involvement of TRPV1 in nociceptive behavior in a rat model of cancer pain.
    The journal of pain, 2008, Volume: 9, Issue:8

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Capsaicin; Carcinoma, Squamous Cell; Cell Line, Tumor; Foot Diseases; Ganglia, Spinal; Hyperalgesia; Immunohistochemistry; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Morphine; Neoplasms, Experimental; Nociceptors; Pain; Pain Measurement; Pain Threshold; Rats; Rats, Inbred F344; Ruthenium Red; TRPV Cation Channels

2008
In vivo pharmacological evaluation of compound 48/80-induced airways oedema by MRI.
    British journal of pharmacology, 2008, Volume: 154, Issue:5

    Topics: Androstadienes; Animals; Anti-Inflammatory Agents; Aza Compounds; Benzamides; Bronchoalveolar Lavage Fluid; Budesonide; Capsaicin; Cell Degranulation; Cromolyn Sodium; Disease Models, Animal; Drug Evaluation, Preclinical; Indomethacin; Lung; Magnetic Resonance Imaging; Male; Mast Cells; Naphthoquinones; ortho-Aminobenzoates; p-Methoxy-N-methylphenethylamine; Proteins; Pulmonary Edema; Rats; Rats, Inbred BN; Respiratory System Agents; Time Factors; Wortmannin

2008
The analgesic drug, tramadol, acts as an agonist of the transient receptor potential vanilloid-1.
    Anesthesia and analgesia, 2008, Volume: 106, Issue:6

    Topics: Analgesics, Opioid; Animals; Calcium; Capsaicin; CHO Cells; Cricetinae; Cricetulus; Cytophotometry; Dose-Response Relationship, Drug; Tachyphylaxis; Tramadol; Transfection; TRPV Cation Channels; Up-Regulation

2008
SA13353 (1-[2-(1-Adamantyl)ethyl]-1-pentyl-3-[3-(4-pyridyl)propyl]urea) inhibits TNF-alpha production through the activation of capsaicin-sensitive afferent neurons mediated via transient receptor potential vanilloid 1 in vivo.
    European journal of pharmacology, 2008, Jul-07, Volume: 588, Issue:2-3

    Topics: Animals; Arthritis, Experimental; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Lipopolysaccharides; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; Pyridines; Rats; Rats, Inbred Lew; Somatostatin; TRPV Cation Channels; Tumor Necrosis Factor-alpha; Urea

2008
Dorsal root ganglion neurons innervating skeletal muscle respond to physiological combinations of protons, ATP, and lactate mediated by ASIC, P2X, and TRPV1.
    Journal of neurophysiology, 2008, Volume: 100, Issue:3

    Topics: Acid Sensing Ion Channels; Adenosine Triphosphate; Amiloride; Analysis of Variance; Animals; Calcium; Capsaicin; Cells, Cultured; Cnidarian Venoms; Dose-Response Relationship, Drug; Drug Interactions; Ganglia, Spinal; Hydrogen-Ion Concentration; Lactic Acid; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Nerve Tissue Proteins; Neurons; Protons; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Receptors, Purinergic P2; Receptors, Purinergic P2X; Sodium Channels; TRPV Cation Channels

2008
Behavioral and electrophysiological evidence for the differential functions of TRPV1 at early and late stages of chronic inflammatory nociception in rats.
    Neurochemical research, 2008, Volume: 33, Issue:10

    Topics: Animals; Capsaicin; Chronic Disease; Electric Stimulation; Evoked Potentials; Freund's Adjuvant; Hot Temperature; Hyperalgesia; Inflammation; Injections, Spinal; Male; Pain; Physical Stimulation; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Spinal Cord; TRPV Cation Channels

2008
Sustained increase of Ca+2 oscillations after chronic TRPV1 receptor activation with capsaicin in cultured spinal neurons.
    Brain research, 2008, Jul-07, Volume: 1218

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Calcium; Capsaicin; Cells, Cultured; CREB-Binding Protein; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Female; Humans; Mice; Mice, Inbred C57BL; Neurons; Pregnancy; Ruthenium Red; Sodium Channel Blockers; Spinal Cord; Tetrodotoxin; TRPV Cation Channels

2008
Transient receptor potential vanilloid 1-mediated expression and secretion of endothelial cell-derived calcitonin gene-related peptide.
    Regulatory peptides, 2008, Oct-09, Volume: 150, Issue:1-3

    Topics: Calcitonin Gene-Related Peptide; Capsaicin; Cell Survival; Cells, Cultured; Culture Media; Endothelial Cells; Endothelium, Vascular; Fever; Humans; Lysophosphatidylcholines; Radioimmunoassay; RNA, Messenger; TRPV Cation Channels; Umbilical Veins

2008
Attenuation of anxiety-related behaviour after the antagonism of transient receptor potential vanilloid type 1 channels in the rat ventral hippocampus.
    Behavioural pharmacology, 2008, Volume: 19, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Avoidance Learning; Behavior, Animal; Capsaicin; Hippocampus; Male; Maze Learning; Rats; Rats, Wistar; TRPV Cation Channels

2008
TRPV1 mediates the uterine capsaicin-induced NMDA NR2B-dependent cross-organ reflex sensitization in anesthetized rats.
    American journal of physiology. Renal physiology, 2008, Volume: 295, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Anesthesia; Animals; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Muscle, Smooth; Neurons, Afferent; Pelvic Pain; Phosphorylation; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reflex; Spinal Cord; TRPV Cation Channels; Uterus

2008
CO2 chemosensing in rat oesophagus.
    Gut, 2008, Volume: 57, Issue:12

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Benzolamide; Capsaicin; Carbon Dioxide; Carbonic Anhydrase Inhibitors; Epithelial Cells; Esophageal pH Monitoring; Esophagus; Gastroesophageal Reflux; Hyperemia; Male; Methazolamide; Mucous Membrane; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Sodium Channels; TRPV Cation Channels

2008
Facilitation of contextual fear memory extinction and anti-anxiogenic effects of AM404 and cannabidiol in conditioned rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2008, Volume: 18, Issue:12

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Arachidonic Acids; Behavior, Animal; Cannabidiol; Capsaicin; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Administration Schedule; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Injections, Intraventricular; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; TRPV Cation Channels

2008
[Protective effect of capsaicin on against myocardial ischemia-reperfusion injury of rat in vivo].
    Sichuan da xue xue bao. Yi xue ban = Journal of Sichuan University. Medical science edition, 2008, Volume: 39, Issue:4

    Topics: Animals; Capsaicin; Creatine Kinase, MB Form; Heart Rate; Male; Myocardial Reperfusion Injury; Random Allocation; Rats; Rats, Sprague-Dawley; Ventricular Function, Left

2008
Excitatory and inhibitory urinary bladder reflexes induced by stimulation of cervicovaginal capsaicin-sensitive sensory fibers in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2009, Volume: 379, Issue:2

    Topics: Animals; Atropine; Capsaicin; Cervix Uteri; Female; Ganglionectomy; Guanethidine; Hexamethonium; Muscle Contraction; Muscle, Smooth; Nerve Fibers; Rats; Rats, Wistar; Reflex; Sensory Receptor Cells; TRPV Cation Channels; Urinary Bladder; Urination; Vagina

2009
TRPV1 channels facilitate glutamate transmission in the striatum.
    Molecular and cellular neurosciences, 2009, Volume: 40, Issue:1

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Capsaicin; Corpus Striatum; Endocannabinoids; gamma-Aminobutyric Acid; Glutamic Acid; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Patch-Clamp Techniques; Polyunsaturated Alkamides; Protein Kinase C; Sensory System Agents; Synaptic Transmission; Tetradecanoylphorbol Acetate; TRPV Cation Channels

2009
Reciprocal changes in vanilloid (TRPV1) and endocannabinoid (CB1) receptors contribute to visceral hyperalgesia in the water avoidance stressed rat.
    Gut, 2009, Volume: 58, Issue:2

    Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Corticosterone; Defecation; Electromyography; Endocannabinoids; Ganglia, Spinal; Hyperalgesia; Immunohistochemistry; Intestinal Mucosa; Male; Microscopy, Fluorescence; Models, Animal; Morpholines; Naphthalenes; Pain Threshold; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Spectrum Analysis; Stress, Psychological; TRPV Cation Channels

2009
Differential effects of topically applied formalin and aromatic compounds on neurogenic-mediated microvascular leakage in rat skin.
    Toxicology, 2009, Jan-08, Volume: 255, Issue:1-2

    Topics: Administration, Topical; Animals; Antipruritics; Capillary Leak Syndrome; Capsaicin; Cell Degranulation; Disinfectants; Dose-Response Relationship, Drug; Formaldehyde; Hydrocarbons, Aromatic; Ketotifen; Male; Mast Cells; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Rats, Wistar; Regional Blood Flow; Skin

2009
Capsaicin, a component of red peppers, induces expression of androgen receptor via PI3K and MAPK pathways in prostate LNCaP cells.
    FEBS letters, 2009, Jan-05, Volume: 583, Issue:1

    Topics: Anilides; Capsaicin; Capsicum; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cinnamates; Diterpenes; Gene Silencing; Humans; Male; Mitogen-Activated Protein Kinase Kinases; Phosphatidylinositol 3-Kinases; Prostate; Receptors, Androgen; RNA, Small Interfering; TRPV Cation Channels

2009
Modulation of anxiety-like behaviour by Transient Receptor Potential Vanilloid Type 1 (TRPV1) channels located in the dorsolateral periaqueductal gray.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2009, Volume: 19, Issue:3

    Topics: Analysis of Variance; Animals; Anxiety; Behavior, Animal; Capsaicin; Conflict, Psychological; Dose-Response Relationship, Drug; Drinking; Male; Maze Learning; Periaqueductal Gray; Rats; Rats, Wistar; Time Factors; TRPV Cation Channels

2009
Salt intake augments hypotensive effects of transient receptor potential vanilloid 4: functional significance and implication.
    Hypertension (Dallas, Tex. : 1979), 2009, Volume: 53, Issue:2

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Ganglia, Spinal; Hypertension; Hypotension; Kidney; Male; Mesenteric Arteries; Phorbol Esters; Rats; Rats, Wistar; Ruthenium Red; Salt Tolerance; Sodium Chloride, Dietary; Substance P; TRPV Cation Channels

2009
Contribution of transient receptor potential vanilloid subtype 1 to the analgesic and antihyperalgesic activity of nefopam in rodents.
    Pharmacology, 2009, Volume: 83, Issue:2

    Topics: Analgesics, Non-Narcotic; Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cells, Cultured; Ganglia, Spinal; Hyperalgesia; Intracellular Fluid; Mice; Nefopam; Potassium Chloride; Rats; Sensory Receptor Cells; Sensory System Agents; TRPV Cation Channels

2009
Antiaversive effects of cannabinoids: is the periaqueductal gray involved?
    Neural plasticity, 2009, Volume: 2009

    Topics: Animals; Anti-Anxiety Agents; Cannabidiol; Cannabinoids; Capsaicin; Microinjections; Periaqueductal Gray; Rats; Receptor, Cannabinoid, CB1; Stress, Physiological; Synaptic Transmission; TRPV Cation Channels

2009
N-acyldopamines control striatal input terminals via novel ligand-gated cation channels.
    Neuropharmacology, 2009, Volume: 56, Issue:3

    Topics: Animals; Arachidonic Acids; Boron Compounds; Capsaicin; Cations; Corpus Striatum; Dopamine; Endocannabinoids; Glutamic Acid; Ion Channels; Ligands; Male; Mice; Mice, Mutant Strains; Polyunsaturated Alkamides; Presynaptic Terminals; Rats; Rats, Wistar; Synaptosomes; TRPV Cation Channels

2009
Nociceptive vascular reflexes evoked by scorpion venom modulate cardiorespiratory parameters involving vanilloid receptor 1 in anaesthetised rats.
    Neuroscience letters, 2009, Feb-27, Volume: 451, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Blood Pressure; Blood Vessels; Capsaicin; Cardiovascular Physiological Phenomena; Drug Interactions; Heart Rate; Injections, Intra-Arterial; Lidocaine; Male; Nociceptors; Rats; Receptors, Serotonin, 5-HT3; Reflex; Respiratory Physiological Phenomena; Scorpion Venoms; Sensory Receptor Cells; Serotonin; Time Factors; TRPV Cation Channels; Visceral Afferents

2009
Activation of sensory neurons reduces ischemia/reperfusion-induced acute renal injury in rats.
    Anesthesiology, 2009, Volume: 110, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Acute Disease; Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capillary Permeability; Capsaicin; Chemokine CCL2; Denervation; Immunohistochemistry; Indomethacin; Kidney; Kidney Diseases; Male; Peptide Fragments; Peroxidase; Rats; Rats, Wistar; Renal Circulation; Reperfusion Injury; Sensory Receptor Cells; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2009
Capsaicin-induced glutamate release is implicated in nociceptive processing through activation of ionotropic glutamate receptors and group I metabotropic glutamate receptor in primary afferent fibers.
    Journal of pharmacological sciences, 2009, Volume: 109, Issue:2

    Topics: Animals; Capsaicin; Glutamic Acid; Hyperalgesia; Male; Nerve Fibers; Nociceptors; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Sensory System Agents; Time Factors; TRPV Cation Channels

2009
A novel role for the TRPV1 channel in UV-induced matrix metalloproteinase (MMP)-1 expression in HaCaT cells.
    Journal of cellular physiology, 2009, Volume: 219, Issue:3

    Topics: Base Sequence; Calcium Signaling; Capsaicin; Cell Line; DNA, Complementary; Humans; Keratinocytes; Matrix Metalloproteinase 1; Models, Biological; Protein Kinase C; RNA, Messenger; RNA, Small Interfering; Skin; Skin Aging; Transfection; TRPV Cation Channels; Ultraviolet Rays

2009
Excitation of cutaneous C nociceptors by intraplantar administration of anandamide.
    Brain research, 2009, May-01, Volume: 1268

    Topics: Action Potentials; Anilides; Animals; Arachidonic Acids; Calcium Channel Blockers; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Endocannabinoids; Hindlimb; Hot Temperature; Male; Nociceptors; Pain; Pain Measurement; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Skin; Tibial Nerve; TRPV Cation Channels

2009
Enhancement of the hypotensive effects of intrathecally injected endocannabinoids by the entourage compound palmitoylethanolamide.
    European journal of pharmacology, 2009, May-21, Volume: 610, Issue:1-3

    Topics: Amides; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Capsaicin; Dose-Response Relationship, Drug; Drug Synergism; Endocannabinoids; Ethanolamines; Heart Rate; Injections, Spinal; Male; Palmitic Acids; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2009
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Capsaicin; Efferent Pathways; Endocannabinoids; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Pyridazines; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Tetrodotoxin; Vagus Nerve

2009
Ethanol aggravates itch-related scratching in hairless mice developing atopic dermatitis.
    European journal of pharmacology, 2009, Jun-02, Volume: 611, Issue:1-3

    Topics: Administration, Oral; Animals; Capsaicin; Dermatitis, Atopic; Dibucaine; Ethanol; Female; Mice; Mice, Hairless; N-Methylaspartate; Naltrexone; Petrolatum; Pruritus; Skin Temperature

2009
Functional type I vanilloid receptor expression by substantia gelatinosa neurons of trigeminal subnucleus caudalis in mice.
    Neuroscience letters, 2009, Mar-20, Volume: 452, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Brain Stem; Capsaicin; Central Nervous System Stimulants; Convulsants; Excitatory Amino Acid Antagonists; In Vitro Techniques; Male; Membrane Potentials; Mice; Neurokinin-1 Receptor Antagonists; Neurons; Picrotoxin; Sensory System Agents; Sodium Channel Blockers; Strychnine; Substantia Gelatinosa; Tetrodotoxin; TRPV Cation Channels; Tryptophan

2009
Involvement of increased expression of transient receptor potential melastatin 8 in oxaliplatin-induced cold allodynia in mice.
    Neuroscience letters, 2009, Jul-17, Volume: 458, Issue:2

    Topics: Animals; Capsaicin; Cold Temperature; Diterpenes; Ganglia, Spinal; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Organoplatinum Compounds; Oxaliplatin; Pain Measurement; Pain Threshold; Physical Stimulation; RNA, Messenger; Time Factors; TRPM Cation Channels; Up-Regulation

2009
Anxiolytic-like effects induced by blockade of transient receptor potential vanilloid type 1 (TRPV1) channels in the medial prefrontal cortex of rats.
    Psychopharmacology, 2009, Volume: 205, Issue:2

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Maze Learning; Morphine; Narcotics; Pain Measurement; Pain Threshold; Prefrontal Cortex; Rats; Rats, Wistar; Reaction Time; TRPV Cation Channels; Water Deprivation

2009
Role of ET(A) and ET(B) endothelin receptors on endothelin-1-induced potentiation of nociceptive and thermal hyperalgesic responses evoked by capsaicin in rats.
    Neuroscience letters, 2009, Jul-03, Volume: 457, Issue:3

    Topics: Analysis of Variance; Animals; Capsaicin; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Hindlimb; Hyperalgesia; Male; Oligopeptides; Pain Measurement; Peptides, Cyclic; Physical Stimulation; Piperidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Sensory System Agents; Temperature; TRPV Cation Channels

2009
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, May-13, Volume: 29, Issue:19

    Topics: Amino Acids; Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Polyunsaturated Alkamides; Propionates; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; Ruthenium Red; Synaptic Transmission; Transient Receptor Potential Channels; TRPM Cation Channels; TRPV Cation Channels; Xanthenes

2009
Activation of TRPV1 and TRPA1 leads to muscle nociception and mechanical hyperalgesia.
    Pain, 2009, Volume: 144, Issue:3

    Topics: Acrylamides; Afferent Pathways; Animals; Ankyrins; Bridged Bicyclo Compounds, Heterocyclic; Calcium Channels; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Facial Pain; Hyperalgesia; Injections, Intramuscular; Male; Masticatory Muscles; Mustard Plant; Nociceptors; Pain Measurement; Pain Threshold; Plant Oils; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Sensory System Agents; Trigeminal Ganglion; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2009
Essential role for TRPV1 in stress-induced (mast cell-dependent) colonic hypersensitivity in maternally separated rats.
    Neurogastroenterology and motility, 2009, Volume: 21, Issue:10

    Topics: Animals; Blotting, Western; Capsaicin; Catheterization; Colon; Drinking Behavior; Female; Immunohistochemistry; Macrophages; Mast Cells; Maternal Deprivation; Nerve Growth Factor; Pregnancy; Pyrrolidines; Rats; Rats, Long-Evans; Stress, Psychological; T-Lymphocytes; Transcription, Genetic; TRPV Cation Channels; Urea

2009
TRPM8, a versatile channel in human sperm.
    PloS one, 2009, Jun-30, Volume: 4, Issue:6

    Topics: Acrosome Reaction; Calcium; Capsaicin; Chemotaxis; Fluorescent Antibody Technique, Indirect; Humans; Male; Models, Biological; Progesterone; Pyrazines; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Sperm Motility; Spermatozoa; TRPM Cation Channels

2009
Characterization of the endocannabinoid system in human spermatozoa and involvement of transient receptor potential vanilloid 1 receptor in their fertilizing ability.
    Endocrinology, 2009, Volume: 150, Issue:10

    Topics: Acrosome Reaction; Amidohydrolases; Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Capsaicin; Cricetinae; Endocannabinoids; Humans; Infertility, Male; Male; Phospholipase D; Polyunsaturated Alkamides; Progesterone; Receptor, Cannabinoid, CB1; Spermatozoa; TRPV Cation Channels

2009
Evidence of TRPV1 receptor and PKC signaling pathway in the antinociceptive effect of amyrin octanoate.
    Brain research, 2009, Oct-27, Volume: 1295

    Topics: Acetic Acid; Analgesics; Analysis of Variance; Animals; Capsaicin; Dose-Response Relationship, Drug; Female; Hot Temperature; Hyperalgesia; Male; Mice; Motor Activity; Neurons; Oleanolic Acid; Opioid Peptides; Pain; Pain Measurement; Physical Stimulation; Protein Kinase C; Psychomotor Performance; Rats; Rats, Wistar; Serotonin; Signal Transduction; TRPV Cation Channels

2009
Capsaicin protects mouse neuromuscular junctions from the neuroparalytic effects of botulinum neurotoxin a.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Acetylcholine; Animals; Body Weight; Botulinum Toxins, Type A; Capsaicin; Cell Line; Electrophysiology; Immunohistochemistry; In Vitro Techniques; Mice; Microscopy, Confocal; Motor Neurons; Muscle Strength; Muscle, Skeletal; Nerve Endings; Neuromuscular Agents; Neuromuscular Junction; Neuroprotective Agents; Synapses; TRPV Cation Channels

2009
Endogenous expression of TRPV1 channel in cultured human melanocytes.
    Journal of dermatological science, 2009, Volume: 56, Issue:2

    Topics: Calcium; Capsaicin; Cells, Cultured; Humans; Immunohistochemistry; Melanins; Melanocytes; Membrane Potentials; Monophenol Monooxygenase; TRPV Cation Channels

2009
AT(1) receptor blockers increase insulin-like growth factor-I production by stimulating sensory neurons in spontaneously hypertensive rats.
    Translational research : the journal of laboratory and clinical medicine, 2009, Volume: 154, Issue:3

    Topics: Angiotensin II Type 1 Receptor Blockers; Animals; Benzimidazoles; Benzoates; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Cells, Cultured; Ganglia, Spinal; Hypertension; Imidazoles; Insulin-Like Growth Factor I; Kidney; Losartan; Male; Myocardium; Nifedipine; Peptidyl-Dipeptidase A; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptor, Angiotensin, Type 1; RNA, Messenger; Sensory Receptor Cells; Telmisartan; Tetrazoles; Valine; Valsartan; Vasodilator Agents

2009
Importance of the non-selective cation channel TRPV1 for microglial reactive oxygen species generation.
    Journal of neuroimmunology, 2009, Nov-30, Volume: 216, Issue:1-2

    Topics: Animals; Capsaicin; Cell Line; Cell Respiration; Diterpenes; Encephalitis; Gliosis; Ion Channel Gating; Lanthanum; Membrane Potentials; Mice; Microglia; NADPH Oxidases; Organ Culture Techniques; Oxidative Stress; Reactive Oxygen Species; Respiratory Burst; Ruthenium Red; TRPV Cation Channels

2009
Deletion of vanilloid receptor (TRPV1) in mice alters behavioral effects of ethanol.
    Neuropharmacology, 2009, Volume: 56, Issue:4

    Topics: Alcohol Drinking; Animals; Capsaicin; Central Nervous System Depressants; Choice Behavior; Ethanol; Mice; Mice, Inbred C57BL; Mice, Knockout; Postural Balance; Substance Withdrawal Syndrome; Taste; TRPV Cation Channels

2009
Evidence for a potential role for TRPV1 receptors in the dorsolateral periaqueductal gray in the attenuation of the anxiolytic effects of cannabinoids.
    Progress in neuro-psychopharmacology & biological psychiatry, 2009, Nov-13, Volume: 33, Issue:8

    Topics: Analgesics; Analysis of Variance; Animals; Anxiety; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Endocannabinoids; Male; Microinjections; Morpholines; Naphthalenes; Periaqueductal Gray; Polyunsaturated Alkamides; Rats; Rats, Wistar; Time Factors; TRPV Cation Channels

2009
Mediating roles of the vanilloid receptor TRPV1 in activation of rat primary afferent nociceptive neurons by formaldehyde.
    Sheng li xue bao : [Acta physiologica Sinica], 2009, Oct-25, Volume: 61, Issue:5

    Topics: Acetanilides; Action Potentials; Animals; Capsaicin; Formaldehyde; Ganglia, Spinal; Nociceptors; Pain; Pain Measurement; Patch-Clamp Techniques; Purines; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2009
Hydrogen sulfide promotes transient receptor potential vanilloid 1-mediated neurogenic inflammation in polymicrobial sepsis.
    Critical care medicine, 2010, Volume: 38, Issue:2

    Topics: Alkynes; Animals; Capsaicin; Cystathionine gamma-Lyase; Glycine; Hydrogen Sulfide; Liver; Lung; Male; Mice; Multiple Organ Failure; Neurogenic Inflammation; Peroxidase; Sepsis; Sulfides; Transient Receptor Potential Channels; TRPV Cation Channels

2010
Protective effect of anacardic acids from cashew (Anacardium occidentale) on ethanol-induced gastric damage in mice.
    Chemico-biological interactions, 2010, Jan-05, Volume: 183, Issue:1

    Topics: Anacardic Acids; Anacardium; Animals; Anti-Ulcer Agents; Antioxidants; Capsaicin; Catalase; Ethanol; Gastric Mucosa; KATP Channels; Male; Malondialdehyde; Mice; Nitric Oxide; Prostaglandins; Rats; Rats, Wistar; Stomach Ulcer; Superoxide Dismutase

2010
Differential role of the menthol-binding residue Y745 in the antagonism of thermally gated TRPM8 channels.
    Molecular pain, 2009, Nov-03, Volume: 5

    Topics: Animals; Capsaicin; Clotrimazole; Cold Temperature; Humans; Imidazoles; Ion Channel Gating; Menthol; Mice; Models, Molecular; Molecular Dynamics Simulation; Mutant Proteins; Mutation; Phenotype; Pyrazines; Pyridines; Structure-Activity Relationship; TRPM Cation Channels; Tyrosine

2009
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: Acrylamides; Administration, Oral; Alkaloids; Anilides; Animals; Avoidance Learning; Benzodioxoles; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazines; Pyridines; Taste; TRPM Cation Channels; TRPV Cation Channels

2010
Behavioral assessment and identification of a molecular marker in a salicylate-induced tinnitus in rats.
    Neuroscience, 2010, Feb-17, Volume: 165, Issue:4

    Topics: Animals; Auditory Pathways; Behavior, Animal; Biomarkers; Capsaicin; Disease Models, Animal; Male; Membrane Transport Modulators; Neuropsychological Tests; Rats; Rats, Wistar; RNA, Messenger; Salicylates; Spiral Ganglion; Time Factors; Tinnitus; TRPV Cation Channels; Up-Regulation

2010
Effects of transient receptor potential (TRP) channel agonists and antagonists on slowly adapting type II mechanoreceptors in the rat sinus hair follicle.
    Journal of the peripheral nervous system : JPNS, 2009, Volume: 14, Issue:4

    Topics: Acrolein; Action Potentials; Animals; Ankyrins; Calcium Channels; Camphor; Capsaicin; Evoked Potentials; Hair Follicle; In Vitro Techniques; Isothiocyanates; Male; Mechanoreceptors; Menthol; Physical Stimulation; Pyrimidinones; Rats; Rats, Wistar; Ruthenium Red; Time Factors; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2009
Gastroprotective effect of barbatusin and 3-beta-hydroxy-3-deoxibarbatusin, quinonoid diterpenes isolated from Plectranthus grandis, in ethanol-induced gastric lesions in mice.
    Journal of ethnopharmacology, 2010, Feb-17, Volume: 127, Issue:3

    Topics: Acetylcysteine; Animals; Anti-Ulcer Agents; Antioxidants; Capsaicin; Disease Models, Animal; Diterpenes; Ethanol; Gastric Mucosa; Glyburide; Indomethacin; Male; Mice; Mucus; NG-Nitroarginine Methyl Ester; Phytotherapy; Plant Extracts; Plant Leaves; Plectranthus; Quinones; Stomach; Stomach Ulcer; Sulfhydryl Compounds; Thiobarbiturates

2010
2-APB and capsazepine-induced Ca2+ influx stimulates clathrin-dependent endocytosis in alveolar epithelial cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2010, Volume: 25, Issue:1

    Topics: Alveolar Epithelial Cells; Animals; Boron Compounds; Calcium; Capsaicin; Cell Line; Cells, Cultured; Clathrin; Endocytosis; Male; Rats; Rats, Sprague-Dawley

2010
Glycolic acid induces keratinocyte proliferation in a skin equivalent model via TRPV1 activation.
    Journal of dermatological science, 2010, Volume: 57, Issue:2

    Topics: Adenosine Triphosphate; Calcium; Capsaicin; Cell Proliferation; Cells, Cultured; Diterpenes; Glycolates; Humans; Immunohistochemistry; Keratinocytes; Skin, Artificial; TRPV Cation Channels

2010
Neuroprotection induced by vitamin E against oxidative stress in hippocampal neurons: involvement of TRPV1 channels.
    Molecular nutrition & food research, 2010, Volume: 54, Issue:4

    Topics: alpha-Tocopherol; Animals; Calcium; Capsaicin; Cell Death; Cells, Cultured; Diterpenes; Electric Conductivity; Ferrous Compounds; Glutamic Acid; Hippocampus; Neurons; Neuroprotective Agents; Oxidative Stress; Rats; Rats, Sprague-Dawley; Synaptic Transmission; TRPV Cation Channels

2010
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: Analysis of Variance; Angiotensin II; Anilides; Animals; Capsaicin; Chelating Agents; Cinnamates; Diuretics, Osmotic; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; In Vitro Techniques; Male; Mannitol; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Piperidines; Pyrazines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Supraoptic Nucleus; TRPV Cation Channels; Vasoconstrictor Agents

2010
The TRPV1 ion channel antagonist capsazepine inhibits osteoclast and osteoblast differentiation in vitro and ovariectomy induced bone loss in vivo.
    Bone, 2010, Volume: 46, Issue:4

    Topics: Analysis of Variance; Animals; Apoptosis; Blotting, Western; Bone Resorption; Capsaicin; Cell Differentiation; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Female; Macrophages; Mice; Osteoblasts; Osteoclasts; Osteogenesis; Ovariectomy; RANK Ligand; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; TRPV Cation Channels

2010
Direct activation of transient receptor potential V1 by nickel ions.
    Pflugers Archiv : European journal of physiology, 2010, Volume: 459, Issue:5

    Topics: Animals; Capsaicin; Cell Line; Cricetinae; Ganglia, Spinal; Gene Expression Regulation; Humans; Mice; Neurons; Nickel; Rats; Ruthenium Red; Temperature; Trigeminal Ganglion; TRPV Cation Channels

2010
The dual fatty acid amide hydrolase/TRPV1 blocker, N-arachidonoyl-serotonin, relieves carrageenan-induced inflammation and hyperalgesia in mice.
    Pharmacological research, 2010, Volume: 61, Issue:6

    Topics: Amidohydrolases; Analgesics; Animals; Anti-Inflammatory Agents; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Carrageenan; Hyperalgesia; Inflammation; Mice; Receptor, Cannabinoid, CB1; Serotonin; TRPV Cation Channels

2010
The TRPv1 receptor is a mediator of the exercise pressor reflex in rats.
    The Journal of physiology, 2010, Apr-01, Volume: 588, Issue:Pt 7

    Topics: Animals; Blood Pressure; Capsaicin; Diterpenes; Heart Rate; Hindlimb; Male; Muscle Contraction; Muscle, Skeletal; Physical Conditioning, Animal; Rats; Rats, Sprague-Dawley; Reflex; Ruthenium Red; TRPV Cation Channels

2010
Characterization of a calcitonin gene-related peptide release assay in rat isolated distal colon.
    Archives of pharmacal research, 2009, Volume: 32, Issue:12

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Anti-Allergic Agents; Benzalkonium Compounds; Calcitonin Gene-Related Peptide; Capsaicin; Colon; Hydrogen-Ion Concentration; In Vitro Techniques; Inflammation Mediators; Ketotifen; Male; Mast Cells; Nerve Tissue Proteins; Neurons, Afferent; p-Methoxy-N-methylphenethylamine; Rats; Rats, Sprague-Dawley; Sodium Channels; Solutions; TRPV Cation Channels

2009
Opposing effects of cannabinoids and vanilloids on evoked quantal release at the frog neuromuscular junction.
    Neuroscience letters, 2010, Apr-05, Volume: 473, Issue:2

    Topics: Acetylcholine; Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Capsaicin; Morpholines; Naphthalenes; Neuromuscular Junction; Piperidines; Pyrazoles; Rana catesbeiana; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2010
[Modulation of the smooth muscle contractions of the rat vas deferens by TRPM8 channel agonist menthol].
    Fiziolohichnyi zhurnal (Kiev, Ukraine : 1994), 2009, Volume: 55, Issue:6

    Topics: Animals; Calcium; Calcium-Transporting ATPases; Capsaicin; Carbachol; Cold Temperature; In Vitro Techniques; Intracellular Membranes; Isotonic Solutions; Male; Menthol; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Receptors, Adrenergic; Receptors, Muscarinic; Sarcoplasmic Reticulum; TRPM Cation Channels; Vas Deferens

2009
Role of TRPV1 channels in boar spermatozoa acquisition of fertilizing ability.
    Molecular and cellular endocrinology, 2010, Jul-29, Volume: 323, Issue:2

    Topics: Actins; Animals; Calcium; Capsaicin; Female; Fertilization; Fluorescent Dyes; Male; Membrane Potentials; Sperm Capacitation; Spermatozoa; Swine; TRPV Cation Channels

2010
Functional roles of TRPV1 channels in lower urinary tract irritated by acetic acid: in vivo evaluations of the sex difference in decerebrate unanesthetized mice.
    American journal of physiology. Renal physiology, 2010, Volume: 298, Issue:6

    Topics: Acetic Acid; Administration, Intravesical; Animals; Capsaicin; Decerebrate State; Female; Irritants; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Neurons, Afferent; Neurons, Efferent; Pressure; Reflex; Time Factors; TRPV Cation Channels; Urethra; Urinary Bladder; Urination

2010
TRPA1 receptor induced relaxation of the human urethra involves TRPV1 and cannabinoid receptor mediated signals, and cyclooxygenase activation.
    The Journal of urology, 2010, Volume: 183, Issue:5

    Topics: Acrolein; Analysis of Variance; Arginine; Calcium Channels; Capsaicin; Cyclohexanols; Female; Humans; Immunohistochemistry; Indomethacin; Isothiocyanates; Male; Middle Aged; Nerve Tissue Proteins; Receptors, Cannabinoid; Signal Transduction; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels; Urethra

2010
Functional vanilloid receptor-1 in human submandibular glands.
    Journal of dental research, 2010, Volume: 89, Issue:7

    Topics: Adult; Aged; Aquaporin 5; Calcium; Capsaicin; Cell Line; Cell Membrane; Cytoplasm; Extracellular Signal-Regulated MAP Kinases; Female; Humans; Male; Middle Aged; Mucous Membrane; Phosphorylation; Saliva; Salivary Ducts; Serous Membrane; Submandibular Gland; TRPV Cation Channels; Young Adult

2010
Accelerated senescence of endothelial progenitor cells in hypertension is related to the reduction of calcitonin gene-related peptide.
    Journal of hypertension, 2010, Volume: 28, Issue:5

    Topics: Adult; Adult Stem Cells; Angiotensin II; Animals; Base Sequence; Calcitonin Gene-Related Peptide; Capsaicin; Cellular Senescence; DNA Primers; Endothelial Cells; Female; Humans; Hypertension; In Vitro Techniques; Indole Alkaloids; Male; Middle Aged; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; RNA, Messenger; TRPV Cation Channels

2010
Effects of topical application of alpha-D-glucosylglycerol on dermal levels of insulin-like growth factor-i in mice and on facial skin elasticity in humans.
    Bioscience, biotechnology, and biochemistry, 2010, Volume: 74, Issue:4

    Topics: Administration, Topical; Animals; Capsaicin; Carbazoles; Dermis; Elasticity; Face; Female; Ganglia, Spinal; Genes; Glucosides; Humans; Insulin-Like Growth Factor I; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons, Afferent; Pyrroles; RNA, Messenger; Sensory Receptor Cells; Skin; TRPV Cation Channels

2010
Screening of OATP1B1/3 and OCT1 inhibitors in cryopreserved hepatocytes in suspension.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2010, Jul-11, Volume: 40, Issue:4

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Bepridil; Biological Transport; Capsaicin; Cryopreservation; Cyproheptadine; Dantrolene; Drug Evaluation, Preclinical; Drug Interactions; Enzyme Inhibitors; Estradiol; Hepatocytes; Humans; Isoenzymes; Liver-Specific Organic Anion Transporter 1; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Rats; Solute Carrier Organic Anion Transporter Family Member 1B3; Species Specificity; Structure-Activity Relationship

2010
1-Nitro-2-phenylethane, the main constituent of the essential oil of Aniba canelilla, elicits a vago-vagal bradycardiac and depressor reflex in normotensive rats.
    European journal of pharmacology, 2010, Jul-25, Volume: 638, Issue:1-3

    Topics: Animals; Aorta; Atropine Derivatives; Benzene Derivatives; Bradycardia; Capsaicin; Cryptocarya; Dose-Response Relationship, Drug; Herb-Drug Interactions; Hypotension; In Vitro Techniques; Male; Oils, Volatile; Ondansetron; Phenylephrine; Rats; Rats, Wistar; Reflex; Vagus Nerve; Vasoconstriction

2010
'TRPing' synaptic ribbon function in the rat pineal gland: neuroendocrine regulation involves the capsaicin receptor TRPV1.
    Neuroendocrinology, 2010, Volume: 92, Issue:2

    Topics: Animals; Bradykinin; Calcium; Capsaicin; Kinesins; Melatonin; Membrane Potentials; Norepinephrine; Pineal Gland; Rats; Rats, Sprague-Dawley; Synapses; TRPV Cation Channels

2010
Existence and distinction of acid-evoked currents in rat astrocytes.
    Glia, 2010, Volume: 58, Issue:12

    Topics: Acid Sensing Ion Channels; Acids; Amiloride; Animals; Animals, Newborn; Astrocytes; Calcium; Capsaicin; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Membrane Potentials; Nerve Tissue Proteins; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Sodium Channels; TRPV Cation Channels

2010
Characterization of in vitro metabolism of capsazepine, a vanilloid transient receptor potential channel antagonist, by liquid chromatography quadrupole ion trap mass spectrometry.
    Biomedical chromatography : BMC, 2011, Volume: 25, Issue:4

    Topics: Animals; Capsaicin; Chromatography, High Pressure Liquid; Dogs; Drug Stability; Mass Spectrometry; Mice; Microsomes, Liver; Rats; TRPV Cation Channels

2011
Emodin down-regulates expression of TRPV1 mRNA and its function in DRG neurons in vitro.
    The American journal of Chinese medicine, 2010, Volume: 38, Issue:4

    Topics: Analgesics; Animals; Calcium; Capsaicin; Cells, Cultured; Down-Regulation; Emodin; Ganglia, Spinal; Gene Expression; Neurons; Plant Extracts; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Rheum; Rhizome; RNA, Messenger; TRPV Cation Channels

2010
Mechanosensitive transient receptor potential vanilloid type 1 channels contribute to vascular remodeling of rat fistula veins.
    Journal of vascular surgery, 2010, Volume: 52, Issue:5

    Topics: Animals; Arginase; Arteriovenous Shunt, Surgical; Benzylamines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Capsaicin; Female; Femoral Artery; Femoral Vein; Hemodynamics; Iliac Vein; Infusion Pumps, Implantable; Infusions, Intravenous; Ligation; Matrix Metalloproteinase 2; Mechanotransduction, Cellular; Nitric Oxide; Nitric Oxide Synthase Type III; Protein Kinase Inhibitors; Rats; Rats, Wistar; RNA, Messenger; Sensory System Agents; Sulfonamides; Time Factors; TRPV Cation Channels

2010
Modulation of single-channel properties of TRPV1 by phosphorylation.
    The Journal of physiology, 2010, Oct-01, Volume: 588, Issue:Pt 19

    Topics: Algorithms; Capsaicin; Dose-Response Relationship, Drug; Electrophysiological Phenomena; Enzyme Activation; HEK293 Cells; Humans; Ion Channel Gating; Kinetics; Nerve Growth Factor; Patch-Clamp Techniques; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Staurosporine; Tetradecanoylphorbol Acetate; Transfection; TRPV Cation Channels

2010
Amphiphile regulation of ion channel function by changes in the bilayer spring constant.
    Proceedings of the National Academy of Sciences of the United States of America, 2010, Aug-31, Volume: 107, Issue:35

    Topics: Algorithms; Capsaicin; Cell Line; Cell Membrane; Genistein; Gramicidin; Humans; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Ion Channel Gating; Ion Channels; Isoflavones; Kinetics; Lipid Bilayers; Membrane Potentials; Membrane Proteins; Octoxynol; Phloretin; Phosphatidylcholines; Protein Conformation

2010
Effects of capsazepine, a transient receptor potential vanilloid type 1 antagonist, on morphine-induced antinociception, tolerance, and dependence in mice.
    British journal of anaesthesia, 2010, Volume: 105, Issue:5

    Topics: Analgesics, Opioid; Animals; Capsaicin; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Synergism; Drug Tolerance; Male; Mice; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Pain; Substance Withdrawal Syndrome; TRPV Cation Channels

2010
TRPV1 activation is required for hypertonicity-stimulated inflammatory cytokine release in human corneal epithelial cells.
    Investigative ophthalmology & visual science, 2011, Volume: 52, Issue:1

    Topics: Blotting, Western; Calcium; Capsaicin; Cells, Cultured; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Epithelium, Corneal; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Fura-2; Humans; Hypertonic Solutions; Interleukin-6; Interleukin-8; Microscopy, Fluorescence; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Signal Transduction; Stress, Physiological; Sulfonamides; Thiourea; Time Factors; TRPV Cation Channels

2011
Evidence for CGRP re-uptake in rat dura mater encephali.
    British journal of pharmacology, 2010, Volume: 161, Issue:8

    Topics: Animals; Antibodies, Monoclonal; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Capsaicin; Dipeptides; Dura Mater; Male; Peptide Fragments; Piperazines; Quinazolines; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells

2010
Phosphorylation of ERK in the spinal dorsal horn following pancreatic pronociceptive stimuli with proteinase-activated receptor-2 agonists and hydrogen sulfide in rats: evidence for involvement of distinct mechanisms.
    Journal of neuroscience research, 2010, Nov-01, Volume: 88, Issue:14

    Topics: Animals; Calcium Channel Blockers; Capsaicin; Down-Regulation; Extracellular Signal-Regulated MAP Kinases; Hydrogen Sulfide; Male; MAP Kinase Signaling System; Nociceptors; Pain, Intractable; Pancreatic Ducts; Phosphorylation; Posterior Horn Cells; Rats; Rats, Wistar; Receptor, PAR-2

2010
TRPV1 receptors are involved in protein nitration and Müller cell reaction in the acutely axotomized rat retina.
    Experimental eye research, 2010, Volume: 91, Issue:5

    Topics: Animals; Axotomy; Capsaicin; Cell Count; Fluoresceins; Fluorescent Antibody Technique, Indirect; Fluorescent Dyes; Glial Fibrillary Acidic Protein; In Situ Nick-End Labeling; Lipid Peroxidation; Neuroglia; Nitric Oxide; Nitrosation; Optic Nerve; Organic Chemicals; Rats; Rats, Wistar; Retinal Ganglion Cells; TRPV Cation Channels

2010
The proteinase/proteinase-activated receptor-2/transient receptor potential vanilloid-1 cascade impacts pancreatic pain in mice.
    Life sciences, 2010, Nov-20, Volume: 87, Issue:19-22

    Topics: Acute Disease; Animals; Benzamidines; Capsaicin; Ceruletide; Disease Models, Animal; Gene Expression Regulation; Guanidines; Hyperalgesia; Male; Mice; Oligopeptides; Pain; Pancreatitis; Proto-Oncogene Proteins c-fos; Receptor, PAR-2; Spinal Cord; TRPV Cation Channels

2010
TRPV1 agonist capsaicin attenuates lung ischemia-reperfusion injury in rabbits.
    The Journal of surgical research, 2012, Volume: 173, Issue:1

    Topics: Animals; Blood Gas Analysis; Bronchoalveolar Lavage Fluid; Calcitonin Gene-Related Peptide; Capsaicin; Lung; Male; Malondialdehyde; Models, Animal; Neutrophils; Oxidative Stress; Peroxidase; Rabbits; Reperfusion Injury; TRPV Cation Channels

2012
dsRNA-induced expression of thymic stromal lymphopoietin (TSLP) in asthmatic epithelial cells is inhibited by a small airway relaxant.
    Pulmonary pharmacology & therapeutics, 2011, Volume: 24, Issue:1

    Topics: Anti-Inflammatory Agents; Asthma; Bronchi; Capsaicin; Cell Survival; Cells, Cultured; Cytokines; Dexamethasone; Epithelial Cells; Humans; I-kappa B Proteins; NF-KappaB Inhibitor alpha; RNA, Double-Stranded; RNA, Messenger; Thymic Stromal Lymphopoietin; Tumor Necrosis Factor-alpha

2011
Bring on the heat: transient receptor potential vanilloid type-1 (TRPV-1) channels as a sensory link for local thermal hyperaemia.
    The Journal of physiology, 2010, Nov-01, Volume: 588, Issue:Pt 21

    Topics: Anesthetics, Local; Capsaicin; Hot Temperature; Humans; Hyperemia; Lidocaine; Lidocaine, Prilocaine Drug Combination; Nitric Oxide; Prilocaine; Regional Blood Flow; Sensory Receptor Cells; Skin; TRPV Cation Channels

2010
TRPA1 receptors mediate environmental irritant-induced meningeal vasodilatation.
    Pain, 2011, Volume: 152, Issue:1

    Topics: Acetanilides; Acrolein; Animals; Animals, Newborn; Ankyrins; Calcitonin Gene-Related Peptide; Calcium Channels; Capsaicin; Cells, Cultured; Dose-Response Relationship, Drug; Formaldehyde; Garlic; Laser-Doppler Flowmetry; Meningeal Arteries; Mustard Plant; Neurons; Peptide Fragments; Plant Oils; Purines; Rats; Sensory System Agents; Substance P; Trigeminal Ganglion; TRPA1 Cation Channel; TRPC Cation Channels; Vasodilation

2011
The M-channel blocker linopirdine is an agonist of the capsaicin receptor TRPV1.
    Journal of pharmacological sciences, 2010, Volume: 114, Issue:3

    Topics: Animals; Calcium; Capsaicin; Ganglia, Spinal; HEK293 Cells; Hot Temperature; Humans; Indoles; KCNQ Potassium Channels; Neurons; Nociceptors; Pyridines; Rats; Rats, Wistar; TRPV Cation Channels

2010
Diabetic rats show reduced cardiac-somatic reflex evoked by intrapericardial capsaicin.
    European journal of pharmacology, 2011, Jan-25, Volume: 651, Issue:1-3

    Topics: Animals; Biomechanical Phenomena; Blood Glucose; Body Weight; Capsaicin; Diabetes Mellitus; Electric Stimulation; Electromyography; Heart; Injections; Male; Pericardium; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Temperature; TRPV Cation Channels

2011
Atomic force microscopy of microvillous cell surface dynamics at fixed and living alveolar type II cells.
    Analytical and bioanalytical chemistry, 2011, Volume: 399, Issue:7

    Topics: Alveolar Epithelial Cells; Animals; Boron Compounds; Calcium; Capsaicin; Cell Membrane; Cells, Cultured; Cytoskeletal Proteins; Endocytosis; Glutaral; Imaging, Three-Dimensional; Lung; Male; Microscopy, Atomic Force; Microscopy, Confocal; Microscopy, Electron, Scanning; Microvilli; Rats; Rats, Sprague-Dawley

2011
Endocannabinoid 2-arachidonoylglycerol protects neurons against β-amyloid insults.
    Neuroscience, 2011, Mar-31, Volume: 178

    Topics: Amyloid beta-Peptides; Animals; Apoptosis; Arachidonic Acids; Benzodioxoles; Biphenyl Compounds; Camphanes; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Capsaicin; Cell Culture Techniques; Drug Interactions; Endocannabinoids; Glycerides; Hippocampus; Monoacylglycerol Lipases; Nerve Degeneration; Peptide Fragments; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Signal Transduction

2011
Role of transient receptor potential ankyrin subfamily member 1 in pruritus induced by endothelin-1.
    Neuroscience letters, 2011, Apr-04, Volume: 492, Issue:3

    Topics: Animals; Behavior, Animal; Capsaicin; Endothelin-1; Enzyme Inhibitors; Histamine; Irritants; Male; Mice; Mice, Inbred C57BL; Pruritus; Ruthenium Red; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2011
Disruption of the transient receptor potential vanilloid 1 can affect survival, bacterial clearance, and cytokine gene expression during murine sepsis.
    Anesthesiology, 2011, Volume: 114, Issue:5

    Topics: Animals; Bacterial Load; Capsaicin; Cecum; Cytokines; Disease Models, Animal; Diterpenes; Down-Regulation; Female; Flow Cytometry; Gene Expression; Ligation; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Mice, Knockout; Peritoneal Lavage; Peritoneum; Reverse Transcriptase Polymerase Chain Reaction; Sepsis; Survival Analysis; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2011
TRPM8 in mouse sperm detects temperature changes and may influence the acrosome reaction.
    Journal of cellular physiology, 2011, Volume: 226, Issue:6

    Topics: Acrosome Reaction; Animals; Capsaicin; Humans; Ion Channel Gating; Male; Menthol; Mice; Mice, Knockout; Pyrazines; Pyridines; Pyrimidinones; Spermatozoa; Temperature; Testis; TRPM Cation Channels

2011
TRPV1 receptors modulate retinal development.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 2011, Volume: 29, Issue:4

    Topics: Animals; Animals, Newborn; Apoptosis; Biomarkers; Capsaicin; Caspase 3; Cell Proliferation; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Rats; Retina; TRPV Cation Channels

2011
Human dental pulp fibroblasts express the "cold-sensing" transient receptor potential channels TRPA1 and TRPM8.
    Journal of endodontics, 2011, Volume: 37, Issue:4

    Topics: Acetanilides; Acrolein; Adult; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Capsaicin; Cells, Cultured; Cold Temperature; Cytophotometry; Dental Pulp; Fibroblasts; Humans; Immunohistochemistry; Membrane Proteins; Menthol; Nerve Tissue Proteins; Nociceptors; Physical Stimulation; Purines; Reverse Transcriptase Polymerase Chain Reaction; Thermosensing; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPM Cation Channels; Young Adult

2011
The vanilloid capsaicin induces IL-6 secretion in prostate PC-3 cancer cells.
    Cytokine, 2011, Volume: 54, Issue:3

    Topics: Capsaicin; Carcinoma; Cell Line, Tumor; Cell Survival; Enzyme-Linked Immunosorbent Assay; Extracellular Signal-Regulated MAP Kinases; Humans; Interleukin-6; Male; Phosphatidylinositol 3-Kinases; Prostatic Neoplasms; Signal Transduction; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2011
Capsaicinoids regulate airway anion transporters through Rho kinase- and cyclic AMP-dependent mechanisms.
    American journal of respiratory cell and molecular biology, 2011, Volume: 45, Issue:4

    Topics: Adenylyl Cyclases; Anion Transport Proteins; Antiporters; Capsaicin; Cell Line; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Enzyme-Linked Immunosorbent Assay; Epithelial Cells; Humans; Ion Transport; Membrane Potentials; Membrane Transport Proteins; Patch-Clamp Techniques; Protein Kinase Inhibitors; Respiratory Mucosa; rho-Associated Kinases; SLC4A Proteins; Sodium-Bicarbonate Symporters; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2

2011
Oxaliplatin elicits mechanical and cold allodynia in rodents via TRPA1 receptor stimulation.
    Pain, 2011, Volume: 152, Issue:7

    Topics: Animals; Antineoplastic Agents; Atropine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cells, Cultured; Chromatography, High Pressure Liquid; Cisplatin; Cricetinae; Cricetulus; Dipeptides; Disease Models, Animal; Drug Interactions; Ganglia, Spinal; Gene Expression Regulation; Guinea Pigs; Hyperalgesia; Mice; Mice, Inbred C57BL; Mice, Knockout; Organoplatinum Compounds; Oxaliplatin; Pain Measurement; Piperazines; Pulmonary Artery; Quinazolines; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensory Receptor Cells; Spectrometry, Mass, Electrospray Ionization; Superoxides; Tissue Culture Techniques; Transient Receptor Potential Channels; TRPA1 Cation Channel

2011
The hypothermic response to bacterial lipopolysaccharide critically depends on brain CB1, but not CB2 or TRPV1, receptors.
    The Journal of physiology, 2011, May-01, Volume: 589, Issue:Pt 9

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Body Temperature Regulation; Brain; Camphanes; Capsaicin; Disease Models, Animal; Diterpenes; Endocannabinoids; Female; Hypothermia; Injections, Intraperitoneal; Injections, Intravenous; Injections, Intraventricular; Lipopolysaccharides; Male; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Long-Evans; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Signal Transduction; Sulfonamides; Time Factors; TRPV Cation Channels

2011
Molecular mechanisms of activation of endothelial nitric oxide synthase mediated by transient receptor potential vanilloid type 1.
    Cardiovascular research, 2011, Aug-01, Volume: 91, Issue:3

    Topics: Animals; Apolipoproteins E; Atherosclerosis; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Capsaicin; Cattle; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activation; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphatidylinositol 3-Kinase; Phosphorylation; Proto-Oncogene Proteins c-akt; Quinazolines; RNA Interference; Signal Transduction; Time Factors; Transfection; TRPV Cation Channels

2011
[Apoptosis inhibition of capsaicin on myocardial ischemia-reperfusion injury in rats].
    Sichuan da xue xue bao. Yi xue ban = Journal of Sichuan University. Medical science edition, 2011, Volume: 42, Issue:2

    Topics: Animals; Apoptosis; Capsaicin; Cardiotonic Agents; Male; Myocardial Reperfusion Injury; Myocardium; Random Allocation; Rats; Rats, Sprague-Dawley

2011
Cardioprotection by ischemic postconditioning is lost in isolated perfused heart from diabetic rats: Involvement of transient receptor potential vanilloid 1, calcitonin gene-related peptide and substance P.
    Regulatory peptides, 2011, Aug-08, Volume: 169, Issue:1-3

    Topics: Animals; Blood Flow Velocity; Calcitonin Gene-Related Peptide; Capsaicin; Coronary Vessels; Diabetes Mellitus, Experimental; Heart; In Vitro Techniques; Ischemic Postconditioning; Male; Myocardial Reperfusion Injury; Myocardium; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Rats, Sprague-Dawley; Substance P; TRPV Cation Channels; Ventricular Function

2011
Leukotriene B4 mediates inflammation via TRPV1 in duct obstruction-induced pancreatitis in rats.
    Pancreas, 2011, Volume: 40, Issue:5

    Topics: Animals; Capsaicin; Cholestasis; Disease Models, Animal; Indoles; Inflammation Mediators; Leukotriene B4; Ligation; Lipoxygenase Inhibitors; Male; Models, Biological; Pancreatitis; Peroxidase; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2011
Sensitivity of bronchopulmonary receptors to cold and heat mediated by transient receptor potential cation channel subtypes in an ex vivo rat lung preparation.
    Respiratory physiology & neurobiology, 2011, Aug-15, Volume: 177, Issue:3

    Topics: Acetanilides; Acrolein; Animals; Capsaicin; Cold Temperature; Hot Temperature; In Vitro Techniques; Lung; Male; Menthol; Purines; Rats; Rats, Sprague-Dawley; Respiratory System; Sensory System Agents; TRPM Cation Channels

2011
Mechanisms underlying the protective effect of eugenol in rats with acute doxorubicin cardiotoxicity.
    Archives of pharmacal research, 2011, Volume: 34, Issue:5

    Topics: Animals; Antibiotics, Antineoplastic; Antioxidants; Calcium Signaling; Capsaicin; Cardiotonic Agents; Cardiotoxins; Caspase 3; Doxorubicin; Eugenol; Heart; Heart Failure; Lipid Peroxidation; Male; Myocardium; Nitric Oxide; Oxidative Stress; Random Allocation; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2011
Suppression of tumor necrosis factor-α-induced nuclear factor κB activation and aromatase activity by capsaicin and its analog capsazepine.
    Journal of medicinal food, 2011, Volume: 14, Issue:11

    Topics: Anticarcinogenic Agents; Aromatase; Capsaicin; Capsicum; Cell Line; Humans; Inhibitory Concentration 50; NF-kappa B; Plant Extracts; Transfection; Tumor Necrosis Factor-alpha

2011
Opposite effect of capsaicin and capsazepine on behavioral thermoregulation in insects.
    Journal of comparative physiology. A, Neuroethology, sensory, neural, and behavioral physiology, 2011, Volume: 197, Issue:10

    Topics: Animals; Behavior, Animal; Body Temperature Regulation; Capsaicin; Dose-Response Relationship, Drug; Larva; Sensory System Agents; Tenebrio; Time Factors; TRPV Cation Channels

2011
TRPV1 agonist piperine but not olvanil enhances glutamatergic spontaneous excitatory transmission in rat spinal substantia gelatinosa neurons.
    Biochemical and biophysical research communications, 2011, Jul-15, Volume: 410, Issue:4

    Topics: Alkaloids; Animals; Benzodioxoles; Capsaicin; Excitatory Amino Acid Agents; Glutamates; Neurons; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Rats; Substantia Gelatinosa; Synaptic Transmission; TRPV Cation Channels

2011
Characterization of capsaicin induced responses in mice vas deferens: evidence of CGRP uptake.
    European journal of pharmacology, 2011, Sep-30, Volume: 667, Issue:1-3

    Topics: Animals; Behavior, Animal; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Mice; Protein Transport; TRPV Cation Channels; Vas Deferens

2011
Proteinase-activated receptor 2 sensitizes transient receptor potential vanilloid 1, transient receptor potential vanilloid 4, and transient receptor potential ankyrin 1 in paclitaxel-induced neuropathic pain.
    Neuroscience, 2011, Oct-13, Volume: 193

    Topics: Analysis of Variance; Anilides; Animals; Ankyrins; Antineoplastic Agents, Phytogenic; Capsaicin; Carbazoles; Central Nervous System; Cinnamates; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Estrenes; Gene Expression Regulation; Hyperalgesia; Male; Mice; Mice, Inbred ICR; Neuralgia; Oligopeptides; Paclitaxel; Pain Measurement; Physical Stimulation; Protein Kinase C; Pyrroles; Pyrrolidinones; Receptor, PAR-2; Sulfonamides; Time Factors; TRPV Cation Channels; Tryptases; Type C Phospholipases

2011
Differential effects of TRPV1 receptor ligands against nicotine-induced depression-like behaviors.
    BMC pharmacology, 2011, Jul-18, Volume: 11

    Topics: Animals; Antidepressive Agents; Arachidonic Acids; Capsaicin; Depression; Dopamine; Endocannabinoids; Hindlimb Suspension; Ligands; Male; Mice; Mice, Inbred ICR; Nicotine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Stress, Psychological; Swimming; TRPV Cation Channels

2011
Osmosensitivity of transient receptor potential vanilloid 1 is synergistically enhanced by distinct activating stimuli such as temperature and protons.
    PloS one, 2011, Volume: 6, Issue:7

    Topics: Animals; Aquaporins; Calcium; Capsaicin; HEK293 Cells; Humans; Mercury Compounds; Mice; Mice, Knockout; Protons; Ruthenium Red; Temperature; TRPV Cation Channels; Water-Electrolyte Balance

2011
Capsaicin induces reflex scratching in inflamed skin.
    Pharmacology, 2011, Volume: 88, Issue:1-2

    Topics: Adjuvants, Immunologic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Capsaicin; Dimethyl Sulfoxide; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Freund's Adjuvant; Inflammation; Injections, Intradermal; Male; Mice; Mice, Inbred C57BL; Morphine; Naloxone; Pain; Pruritus; Receptors, Opioid, mu; Reflex; Sensory System Agents; Skin; Time Factors; TRPV Cation Channels

2011
Hydrogen sulfide and neurogenic inflammation in polymicrobial sepsis: involvement of substance P and ERK-NF-κB signaling.
    PloS one, 2011, Volume: 6, Issue:9

    Topics: Animals; Capsaicin; Cell Nucleus; Chemokines; Cytokines; Extracellular Signal-Regulated MAP Kinases; Hydrogen Sulfide; Inflammation; Male; Mice; NF-kappa B; Phosphorylation; Sepsis; Substance P; TRPV Cation Channels

2011
Opposing roles for cannabinoid receptor type-1 (CB₁) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:2

    Topics: Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Drug Interactions; Electric Stimulation; Male; Microinjections; Panic; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2012
Small molecule positive allosteric modulation of TRPV1 activation by vanilloids and acidic pH.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:1

    Topics: Animals; Body Temperature; Calcium; Calcium Radioisotopes; Capsaicin; Dihydropyridines; Electrophysiological Phenomena; HEK293 Cells; Humans; Hydrogen-Ion Concentration; Phosphorylation; Protons; Rats; Serine; TRPV Cation Channels

2012
Transient receptor potential vanilloid 1 channels modulate the anxiolytic effect of diazepam.
    Brain research, 2011, Nov-24, Volume: 1425

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Capsaicin; Diazepam; Dose-Response Relationship, Drug; Injections, Intraventricular; Interpersonal Relations; Male; Mice; Motor Activity; TRPV Cation Channels

2011
Antagonism of the TRPv1 receptor partially corrects muscle metaboreflex overactivity in spontaneously hypertensive rats.
    The Journal of physiology, 2011, Dec-15, Volume: 589, Issue:Pt 24

    Topics: Animals; Baroreflex; Blood Pressure; Capsaicin; Electric Stimulation; Hindlimb; Hypertension; Ischemia; Kidney; Male; Muscle Contraction; Muscle, Skeletal; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Sciatic Nerve; Sympathetic Nervous System; TRPV Cation Channels

2011
Influence of influenza A infection on capsaicin-induced responses in murine airways.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:2

    Topics: Animals; Biphenyl Compounds; Bronchoalveolar Lavage Fluid; Capsaicin; Carbachol; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Indomethacin; Inflammation; Influenza A virus; Isoproterenol; Leukocytes; Male; Mice; Mice, Inbred BALB C; Models, Biological; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Orthomyxoviridae Infections; Piperidines; Prostaglandin Antagonists; Respiratory Mucosa; Specific Pathogen-Free Organisms; Substance P; Trachea; TRPV Cation Channels; Xanthones

2012
Heteromeric heat-sensitive transient receptor potential channels exhibit distinct temperature and chemical response.
    The Journal of biological chemistry, 2012, Mar-02, Volume: 287, Issue:10

    Topics: Animals; Capsaicin; Ganglia, Spinal; HEK293 Cells; Hot Temperature; Humans; Ion Channel Gating; Mice; Sensory Receptor Cells; Sensory System Agents; Thermosensing; TRPV Cation Channels

2012
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
    Journal of neuroinflammation, 2012, Jan-20, Volume: 9

    Topics: Acetylcysteine; Analysis of Variance; Anilides; Animals; Antioxidants; Autoradiography; Bradykinin; Bradykinin B1 Receptor Antagonists; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Gene Expression Regulation; Iodine Isotopes; Male; Microglia; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; RNA, Messenger; Sensory System Agents; Spinal Cord; Superoxides; Tetrahydroisoquinolines; Time Factors; TRPV Cation Channels

2012
Role of TRPV1 in consolidation of fear memories depends on the averseness of the conditioning procedure.
    Neurobiology of learning and memory, 2012, Volume: 97, Issue:4

    Topics: Animals; Avoidance Learning; Capsaicin; Conditioning, Psychological; Fear; Hippocampus; Male; Memory; Rats; Rats, Wistar; Sensory System Agents; TRPV Cation Channels

2012
Gastroprotective potential of frutalin, a D-galactose binding lectin, against ethanol-induced gastric lesions.
    Fitoterapia, 2012, Volume: 83, Issue:3

    Topics: Animals; Anti-Ulcer Agents; Antioxidants; Biomarkers; Capsaicin; Cimetidine; Ethanol; Galactose; Galectins; Gastric Mucosa; Glutathione; Glyburide; Indomethacin; Male; Malondialdehyde; Mice; Mice, Inbred Strains; NG-Nitroarginine Methyl Ester; Oxidative Stress; Phytotherapy; Plant Extracts; Stomach Ulcer

2012
Acute myocardial ischemia enhances the vanilloid TRPV1 and serotonin 5-HT3 receptor-mediated Bezold-Jarisch reflex in rats.
    Pharmacological reports : PR, 2011, Volume: 63, Issue:6

    Topics: Acute Disease; Animals; Capsaicin; Male; Myocardial Ischemia; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Reflex; TRPV Cation Channels; Vagus Nerve Stimulation

2011
Enhanced vasorelaxant effects of the endocannabinoid-like mediator, oleamide, in hypertension.
    European journal of pharmacology, 2012, Jun-05, Volume: 684, Issue:1-3

    Topics: Amidohydrolases; Animals; Aorta; Benzamides; Biomimetic Materials; Cannabinoid Receptor Modulators; Capsaicin; Carbamates; Cyclooxygenase Inhibitors; Endocannabinoids; Endothelium, Vascular; Hypertension; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Oleic Acids; Rats; Receptor, Cannabinoid, CB1; TRPV Cation Channels; Vasodilator Agents

2012
Characterization of a novel splice variant of δ ENaC subunit in human lungs.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Jun-15, Volume: 302, Issue:12

    Topics: Alveolar Epithelial Cells; Amiloride; Amino Acid Sequence; Animals; Biological Transport; Capsaicin; Cloning, Molecular; Electric Conductivity; Epithelial Sodium Channels; Exocytosis; Humans; Hydrogen-Ion Concentration; Ion Channel Gating; Lung; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Respiratory Mucosa; RNA Splicing; Sodium; Xenopus

2012
Vasorelaxation to capsaicin and its effects on calcium influx in arteries.
    European journal of pharmacology, 2012, Apr-15, Volume: 681, Issue:1-3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Abdominal; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Capsaicin; Coronary Vessels; Dose-Response Relationship, Drug; Male; Rats; Rats, Wistar; Swine; TRPV Cation Channels; Vasodilation

2012
A possible participation of transient receptor potential vanilloid type 1 channels in the antidepressant effect of fluoxetine.
    European journal of pharmacology, 2012, Jun-15, Volume: 685, Issue:1-3

    Topics: Animals; Antidepressive Agents, Second-Generation; Capsaicin; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Fenclonine; Fluoxetine; Injections, Intraventricular; Male; Mice; Serotonin; Swimming; TRPV Cation Channels

2012
Capacity of capsazepinoids to relax human small airways and inhibit TLR3-induced TSLP and IFNβ production in diseased bronchial epithelial cells.
    International immunopharmacology, 2012, Volume: 13, Issue:3

    Topics: Adult; Aged; Asthma; Base Sequence; Bronchi; Bronchodilator Agents; Capsaicin; Cells, Cultured; Cytokines; Epithelial Cells; Female; Humans; In Vitro Techniques; Interferon-beta; Male; Middle Aged; Pulmonary Disease, Chronic Obstructive; RNA, Messenger; Thymic Stromal Lymphopoietin; Toll-Like Receptor 3; Young Adult

2012
Transient receptor potential vanilloid 1 receptors mediate acid-induced mucin secretion via Ca2+ influx in human airway epithelial cells.
    Journal of biochemical and molecular toxicology, 2012, Volume: 26, Issue:5

    Topics: Airway Obstruction; Bronchi; Calcium; Capsaicin; Cell Line; Citric Acid; Dose-Response Relationship, Drug; Epithelial Cells; Gene Expression; Humans; In Vitro Techniques; Mucin 5AC; Patch-Clamp Techniques; TRPV Cation Channels

2012
G-protein-mediated inhibition of the Trp channel TRPM1 requires the Gβγ dimer.
    Proceedings of the National Academy of Sciences of the United States of America, 2012, May-29, Volume: 109, Issue:22

    Topics: Amino Acids; Animals; Capsaicin; Cells, Cultured; Excitatory Amino Acid Antagonists; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; HEK293 Cells; Humans; Light; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Protein Binding; Protein Multimerization; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; TRPM Cation Channels; Xanthenes

2012
Transient receptor potential vanilloid-1 regulates osteoprotegerin/RANKL homeostasis in human periodontal ligament cells.
    Journal of periodontal research, 2013, Volume: 48, Issue:1

    Topics: 3T3 Cells; Animals; Bone Remodeling; Calcium; Capsaicin; Cell Culture Techniques; Chelating Agents; Dinoprostone; Dose-Response Relationship, Drug; Egtazic Acid; Estrenes; Homeostasis; Humans; Mice; Osteoblasts; Osteoprotegerin; Periodontal Ligament; Phosphodiesterase Inhibitors; Pyrrolidinones; RANK Ligand; TRPV Cation Channels; Type C Phospholipases

2013
Disruption of TRPV1-mediated coupling of coronary blood flow to cardiac metabolism in diabetic mice: role of nitric oxide and BK channels.
    American journal of physiology. Heart and circulatory physiology, 2012, Jul-15, Volume: 303, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Anilides; Animals; Capsaicin; Cinnamates; Coronary Vessels; Diabetes Mellitus, Type 2; Diabetic Cardiomyopathies; Enzyme Inhibitors; Large-Conductance Calcium-Activated Potassium Channels; Male; Mice; Mice, Inbred C57BL; Microvessels; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptides; TRPV Cation Channels; Vasoconstrictor Agents; Vasodilation

2012
Endothelium-dependent mechanisms of the vasodilatory effect of the endocannabinoid, anandamide, in the rat pulmonary artery.
    Pharmacological research, 2012, Volume: 66, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amidohydrolases; Animals; Anisoles; Apamin; Arachidonic Acids; Benzamides; Benzyl Compounds; Cannabinoid Receptor Antagonists; Capsaicin; Carbamates; Charybdotoxin; Cyclohexanes; Endocannabinoids; Endothelium, Vascular; Imidazoles; Indoles; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Chloride; Prostaglandin-Endoperoxide Synthases; Pulmonary Artery; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Epoprostenol; Tetraethylammonium; TRPV Cation Channels; Vasodilation

2012
N-arachidonoyl-serotonin in the basolateral amygdala increases anxiolytic behavior in the elevated plus maze.
    Behavioural brain research, 2012, Aug-01, Volume: 233, Issue:2

    Topics: Amygdala; Analysis of Variance; Animals; Anxiety Disorders; Arachidonic Acids; Benzamides; Capsaicin; Carbamates; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Exploratory Behavior; Male; Maze Learning; Rats; Rats, Sprague-Dawley; Serotonin; TRPV Cation Channels

2012
TRPV1-mediated calcium signal couples with cannabinoid receptors and sodium-calcium exchangers in rat odontoblasts.
    Cell calcium, 2012, Volume: 52, Issue:2

    Topics: Animals; Arachidonic Acids; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Signaling; Cannabinoid Receptor Antagonists; Capsaicin; Cyclic AMP; Diterpenes; Endocannabinoids; Glycerides; Hydrogen-Ion Concentration; Odontoblasts; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Cannabinoid; Sodium-Calcium Exchanger; Thiourea; TRPV Cation Channels

2012
Involvement of TRPV1 and TRPV4 channels in migration of rat pulmonary arterial smooth muscle cells.
    Pflugers Archiv : European journal of physiology, 2012, Volume: 464, Issue:3

    Topics: Animals; Calcium; Capsaicin; Cell Movement; Cytoskeleton; Morpholines; Myocytes, Smooth Muscle; Phorbol Esters; Pulmonary Artery; Pyrroles; Rats; RNA, Messenger; TRPV Cation Channels

2012
Regulation of particulate matter-induced mucin secretion by transient receptor potential vanilloid 1 receptors.
    Inflammation, 2012, Volume: 35, Issue:6

    Topics: Air Pollutants; Bronchi; Calcium; Capsaicin; Cell Line, Transformed; Chelating Agents; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Environmental Exposure; Epithelial Cells; Exocytosis; Humans; Isoquinolines; Microscopy, Confocal; Mucin 5AC; Mucins; Particulate Matter; Protein Kinase Inhibitors; Sulfonamides; TRPV Cation Channels

2012
Role of KATP channels and TRPV1 receptors in hydrogen sulfide-enhanced gastric emptying of liquid in awake mice.
    European journal of pharmacology, 2012, Oct-15, Volume: 693, Issue:1-3

    Topics: Animals; Capsaicin; Gastric Emptying; Glyburide; Hydrogen Sulfide; KATP Channels; Male; Mice; Muscle Relaxation; Potassium Channel Blockers; Pylorus; TRPV Cation Channels

2012
Capsazepine, a TRPV1 antagonist, sensitizes colorectal cancer cells to apoptosis by TRAIL through ROS-JNK-CHOP-mediated upregulation of death receptors.
    Free radical biology & medicine, 2012, Nov-15, Volume: 53, Issue:10

    Topics: Acetylcysteine; Apoptosis; Apoptosis Regulatory Proteins; Capsaicin; Caspase 3; Caspase 8; Caspase 9; Cell Line, Tumor; Colorectal Neoplasms; Glutathione; Humans; JNK Mitogen-Activated Protein Kinases; Reactive Oxygen Species; Receptors, TNF-Related Apoptosis-Inducing Ligand; RNA Interference; RNA, Small Interfering; TNF-Related Apoptosis-Inducing Ligand; Transcription Factor CHOP; TRPV Cation Channels; Up-Regulation

2012
Peripheral antinociceptive effect of anandamide and drugs that affect the endocannabinoid system on the formalin test in normal and streptozotocin-diabetic rats.
    Neuropharmacology, 2012, Volume: 63, Issue:8

    Topics: Analgesics; Animals; Arachidonic Acids; Behavior, Animal; Capsaicin; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Endocannabinoids; Formaldehyde; Hyperalgesia; Indoles; Male; Pain Measurement; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Cannabinoid

2012
Comparison of the effects of pelargonic acid vanillylamide and capsaicin on human vanilloid receptors.
    Phytotherapy research : PTR, 2013, Volume: 27, Issue:7

    Topics: Animals; Benzylamines; Capsaicin; Fatty Acids; HEK293 Cells; Humans; TRPV Cation Channels

2013
Regulation of MMP-9 by a WIN-binding site in the monocyte-macrophage system independent from cannabinoid receptors.
    PloS one, 2012, Volume: 7, Issue:11

    Topics: Animals; Benzoxazines; Binding Sites; Bone Resorption; Bronchoalveolar Lavage Fluid; Capsaicin; Cell Differentiation; Disease Models, Animal; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation, Enzymologic; Glycosylation; Humans; Macrophages; Matrix Metalloproteinase 9; Mice; Microglia; Monocytes; Morpholines; Naphthalenes; Osteoclasts; Phosphorylation; Pneumonia; PPAR gamma; Receptors, Cannabinoid; rho GTP-Binding Proteins; Signal Transduction; TRPV Cation Channels

2012
Effects of glutamate NMDA and TRPV1 receptor antagonists on the biphasic responses to anandamide injected into the dorsolateral periaqueductal grey of Wistar rats.
    Psychopharmacology, 2013, Volume: 226, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Capsaicin; Dose-Response Relationship, Drug; Endocannabinoids; Male; Maze Learning; Periaqueductal Gray; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; TRPV Cation Channels

2013
The monoterpene (-)-carvone: a novel agonist of TRPV1 channels.
    Cytometry. Part A : the journal of the International Society for Analytical Cytology, 2013, Volume: 83, Issue:2

    Topics: Animals; Calcium Signaling; Capsaicin; Cell Survival; Cyclohexane Monoterpenes; HEK293 Cells; Humans; Monoterpenes; Neurons; Rats; Rats, Wistar; TRPV Cation Channels

2013
Occludin is required for TRPV1-modulated paracellular permeability in the submandibular gland.
    Journal of cell science, 2013, Mar-01, Volume: 126, Issue:Pt 5

    Topics: Animals; Blotting, Western; Capsaicin; Cell Line; Flavonoids; Immunoprecipitation; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Occludin; Phosphorylation; Rats; Reverse Transcriptase Polymerase Chain Reaction; Submandibular Gland; Tight Junctions; TRPV Cation Channels

2013
Cellular mechanism underlying formaldehyde-stimulated Cl- secretion in rat airway epithelium.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Biological Transport; Capsaicin; Cells, Cultured; Chlorides; Colforsin; Epinephrine; Epithelial Cells; Formaldehyde; Imines; Male; Nerve Endings; ortho-Aminobenzoates; Quinuclidines; Rats; Respiratory Mucosa; Substance P; Trachea; TRPV Cation Channels

2013
Role of TRPA1 and TRPV1 in the ROS-dependent sensory irritation of superior laryngeal capsaicin-sensitive afferents by cigarette smoke in anesthetized rats.
    Pulmonary pharmacology & therapeutics, 2013, Volume: 26, Issue:3

    Topics: Acetanilides; Acetylcysteine; Animals; Antioxidants; Apnea; Calcium Channels; Capsaicin; Chelating Agents; Dose-Response Relationship, Drug; Egtazic Acid; Indomethacin; Laryngeal Nerves; Larynx; Neurons, Afferent; Purines; Rats; Reactive Oxygen Species; Smoking; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2013
Role of TRPV1 and P2X receptors in the activation of lung vagal C-fiber afferents by inhaled cigarette smoke in rats.
    Molecular medicine reports, 2013, Volume: 7, Issue:4

    Topics: Animals; Capsaicin; Cholinergic Fibers; Humans; Hydroxyl Radical; Pyridoxal Phosphate; Rats; Reactive Oxygen Species; Receptors, Nicotinic; Receptors, Purinergic P2X; Smoke; Smoking; Thiourea; TRPV Cation Channels

2013
Linalool-rich rosewood oil induces vago-vagal bradycardic and depressor reflex in rats.
    Phytotherapy research : PTR, 2014, Volume: 28, Issue:1

    Topics: Acetanilides; Acyclic Monoterpenes; Animals; Aorta; Atropine Derivatives; Blood Pressure; Bradycardia; Capsaicin; Hypotension; In Vitro Techniques; Lauraceae; Male; Monoterpenes; Oils, Volatile; Ondansetron; Phenylephrine; Plant Oils; Purines; Rats; Rats, Wistar; Reflex

2014
Hydrogen sulfide mediated inhibitory neurotransmission to the pig bladder neck: role of KATP channels, sensory nerves and calcium signaling.
    The Journal of urology, 2013, Volume: 190, Issue:2

    Topics: Acetanilides; Acrylamides; Animals; Bridged Bicyclo Compounds, Heterocyclic; Calcitonin Gene-Related Peptide; Calcium Signaling; Capsaicin; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Glyburide; Guanylate Cyclase; Hydrogen Sulfide; Indomethacin; KATP Channels; Morpholines; Muscle, Smooth; Organothiophosphorus Compounds; Phenylephrine; Pituitary Adenylate Cyclase-Activating Polypeptide; Purines; Pyrazoles; Sensory Receptor Cells; Swine; Synaptic Transmission; Urinary Bladder

2013
The membrane-associated transient receptor potential vanilloid channel is the central heat shock receptor controlling the cellular heat shock response in epithelial cells.
    PloS one, 2013, Volume: 8, Issue:2

    Topics: Capsaicin; Cell Line; Cell Nucleus; DNA-Binding Proteins; Epithelial Cells; Gene Expression Regulation; Heat Shock Transcription Factors; Heat-Shock Response; HSP70 Heat-Shock Proteins; Humans; Protein Binding; Protein Transport; Transcription Factors; TRPV Cation Channels

2013
Expression and functionality of TRPV1 receptor in human MCF-7 and canine CF.41 cells.
    Veterinary and comparative oncology, 2015, Volume: 13, Issue:2

    Topics: Adenocarcinoma; Animals; Breast Neoplasms; Capsaicin; Cell Line, Tumor; Cell Proliferation; Diterpenes; Dogs; Female; Gene Expression Regulation, Neoplastic; Humans; Mammary Neoplasms, Animal; MCF-7 Cells; TRPV Cation Channels

2015
Characterization of functional TRPV1 channels in the sarcoplasmic reticulum of mouse skeletal muscle.
    PloS one, 2013, Volume: 8, Issue:3

    Topics: Animals; Calcium; Capsaicin; Male; Mice; Muscle, Skeletal; Protein Transport; Ryanodine Receptor Calcium Release Channel; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; TRPV Cation Channels

2013
Neuroprotection induced by N-acetylcysteine against cytosolic glutathione depletion-induced Ca2+ influx in dorsal root ganglion neurons of mice: role of TRPV1 channels.
    Neuroscience, 2013, Jul-09, Volume: 242

    Topics: Acetylcysteine; Animals; Buthionine Sulfoximine; Calcium; Calcium Signaling; Capsaicin; Caspase 3; Caspase 9; Cell Survival; Cells, Cultured; Cytosol; Drug Interactions; Ganglia, Spinal; Glutathione; Lipid Peroxidation; Male; Membrane Potentials; Mice; Neurons; Neuroprotective Agents; Oxidative Stress; Reactive Oxygen Species; TRPV Cation Channels

2013
Detection of mouse cough based on sound monitoring and respiratory airflow waveforms.
    PloS one, 2013, Volume: 8, Issue:3

    Topics: Animals; Capsaicin; Codeine; Cough; Female; Mice; Mice, Inbred BALB C; Plethysmography, Whole Body; Pulmonary Ventilation; Respiratory Sounds; Sodium Chloride

2013
Capsaicin regulates the NF-κB pathway in salivary gland inflammation.
    Journal of dental research, 2013, Volume: 92, Issue:6

    Topics: Animals; Anti-Inflammatory Agents; Capsaicin; Cells, Cultured; Cytokines; Epithelial Cells; Escherichia coli; I-kappa B Proteins; Inflammation Mediators; Interleukin-6; Lipopolysaccharides; Mice; NF-kappa B; NF-KappaB Inhibitor alpha; Phosphorylation; Poly I-C; Salivary Ducts; Sialadenitis; Submandibular Gland; Time Factors; Toll-Like Receptors; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2013
TRPM5-dependent amiloride- and benzamil-insensitive NaCl chorda tympani taste nerve response.
    American journal of physiology. Gastrointestinal and liver physiology, 2013, Jul-01, Volume: 305, Issue:1

    Topics: Amiloride; Anilides; Animals; Capsaicin; Chorda Tympani Nerve; Cinnamates; Diterpenes; Mice; Mice, Knockout; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Sodium Chloride; Taste; TRPM Cation Channels; TRPV Cation Channels

2013
Capsicum annuum enhances L-lactate production by Lactobacillus acidophilus: implication in curd formation.
    Journal of dairy science, 2013, Volume: 96, Issue:7

    Topics: Capsaicin; Capsicum; Cultured Milk Products; Hydrogen-Ion Concentration; Lactic Acid; Lactobacillus acidophilus; Temperature

2013
Role of transient receptor potential ion channels and evoked levels of neuropeptides in a formaldehyde-induced model of asthma in BALB/c mice.
    PloS one, 2013, Volume: 8, Issue:5

    Topics: Acetanilides; Animals; Asthma; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Enzyme-Linked Immunosorbent Assay; Formaldehyde; Immunoglobulin E; Immunohistochemistry; Interleukin-1beta; Interleukin-4; Interleukin-6; Lung; Male; Mice; Mice, Inbred BALB C; Neuropeptides; Ovalbumin; Purines; Substance P; Transient Receptor Potential Channels

2013
Anxiogenic-like effect induced by TRPV1 receptor activation within the dorsal periaqueductal gray matter in mice.
    Behavioural brain research, 2013, Aug-01, Volume: 250

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Combinations; Male; Maze Learning; Mice; Microinjections; Periaqueductal Gray; TRPV Cation Channels

2013
Operant behavioral responses to orofacial cold stimuli in rats with chronic constrictive trigeminal nerve injury: effects of menthol and capsazepine.
    Molecular pain, 2013, Jun-14, Volume: 9

    Topics: Animals; Behavior, Animal; Capsaicin; Cold Temperature; Conditioning, Operant; Facial Nerve; Facial Pain; Hyperalgesia; Male; Menthol; Neuralgia; Pain Measurement; Physical Stimulation; Rats; Rats, Sprague-Dawley; Trigeminal Nerve; Trigeminal Nerve Injuries; TRPM Cation Channels

2013
Leptin modulates enteric neurotransmission in the rat proximal colon: an in vitro study.
    Regulatory peptides, 2013, Aug-10, Volume: 185

    Topics: Acetylcholine; Animals; Capsaicin; Cholinergic Agonists; Colon; Enteric Nervous System; Hexamethonium; Humans; In Vitro Techniques; Leptin; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nicotinic Antagonists; Nitric Oxide; Nitric Oxide Synthase; Rats; Rats, Wistar; Synaptic Transmission

2013
Cyclooxygenase-2, prostaglandin E2 glycerol ester and nitric oxide are involved in muscarine-induced presynaptic enhancement at the vertebrate neuromuscular junction.
    The Journal of physiology, 2013, Oct-01, Volume: 591, Issue:19

    Topics: Animals; Arachidonic Acids; Benzoates; Capsaicin; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dinoprostone; Endocannabinoids; Glycerides; Imidazoles; Lizards; Miniature Postsynaptic Potentials; Muscarine; Neuromuscular Junction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Schwann Cells; Sulfonamides; Thiophenes; Xanthones

2013
Optical control of TRPV1 channels.
    Angewandte Chemie (International ed. in English), 2013, Sep-09, Volume: 52, Issue:37

    Topics: Azo Compounds; Capsaicin; Crystallography, X-Ray; Euphorbia; Isomerism; Molecular Conformation; TRPV Cation Channels

2013
Activation of TRPV1 prevents OxLDL-induced lipid accumulation and TNF-α-induced inflammation in macrophages: role of liver X receptor α.
    Mediators of inflammation, 2013, Volume: 2013

    Topics: Animals; Atherosclerosis; Blotting, Western; Calcium; Capsaicin; Cells, Cultured; Chromatin Immunoprecipitation; Inflammation; Lipoproteins, LDL; Liver X Receptors; Macrophages; Mice; Orphan Nuclear Receptors; RNA, Small Interfering; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2013
Intragastric Dai-Kenchu-To, a Japanese herbal medicine, stimulates colonic motility via transient receptor potential cation channel subfamily V member 1 in dogs.
    The Tohoku journal of experimental medicine, 2013, Volume: 230, Issue:4

    Topics: Animals; Capsaicin; Colon; Constipation; Dogs; Drug Evaluation, Preclinical; Gastrointestinal Motility; Herbal Medicine; Infusions, Parenteral; Japan; Medicine, East Asian Traditional; Panax; Plant Extracts; Plants, Medicinal; Stomach; TRPV Cation Channels; Zanthoxylum; Zingiberaceae

2013
Functional expression of TRPV1 and TRPA1 in rat vestibular ganglia.
    Neuroscience letters, 2013, Sep-27, Volume: 552

    Topics: Acetanilides; Acrolein; Animals; Calcium; Capsaicin; Molecular Imaging; Primary Cell Culture; Purines; Rats; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels; Vestibular Nerve

2013
Effect of TRPV1 channel on the proliferation and apoptosis in asthmatic rat airway smooth muscle cells.
    Experimental lung research, 2013, Volume: 39, Issue:7

    Topics: Airway Remodeling; Animals; Apoptosis; Asthma; Calcium; Capsaicin; Cell Proliferation; Cells, Cultured; Disease Models, Animal; Hyperplasia; Male; Myocytes, Smooth Muscle; Ovalbumin; Proliferating Cell Nuclear Antigen; Rats; Rats, Sprague-Dawley; Respiratory System; TRPV Cation Channels

2013
Medial prefrontal cortex Transient Receptor Potential Vanilloid Type 1 (TRPV1) in the expression of contextual fear conditioning in Wistar rats.
    Psychopharmacology, 2014, Volume: 231, Issue:1

    Topics: Animals; Behavior, Animal; Blood Pressure; Capsaicin; Conditioning, Psychological; Electroshock; Fear; Heart Rate; Male; Microinjections; Prefrontal Cortex; Rats; Rats, Wistar; TRPV Cation Channels

2014
Nonivamide, a capsaicin analog, increases dopamine and serotonin release in SH-SY5Y cells via a TRPV1-independent pathway.
    Molecular nutrition & food research, 2013, Volume: 57, Issue:11

    Topics: Capsaicin; Cell Line, Tumor; Cell Survival; Cyclohexanols; Dopamine; Dose-Response Relationship, Drug; Gene Expression Regulation; Humans; Sensory System Agents; Serotonin; Signal Transduction; TRPV Cation Channels

2013
Allyl isothiocyanate sensitizes TRPV1 to heat stimulation.
    Pflugers Archiv : European journal of physiology, 2014, Volume: 466, Issue:3

    Topics: Action Potentials; Animals; Calcium; Capsaicin; Cells, Cultured; HEK293 Cells; Hot Temperature; Humans; Hyperalgesia; Isothiocyanates; Mice; Mice, Inbred C57BL; Sensory Receptor Cells; Thermosensing; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2014
Capsazepine concentration dependently inhibits currents in HEK 293 cells mediated by human hyperpolarization-activated cyclic nucleotide-gated 2 and 4 channels.
    Experimental biology and medicine (Maywood, N.J.), 2013, Volume: 238, Issue:9

    Topics: Analgesics; Capsaicin; Cyclic Nucleotide-Gated Cation Channels; HEK293 Cells; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Ion Channels; Muscle Proteins; Potassium Channels

2013
TRPV1 antagonist capsazepine suppresses 4-AP-induced epileptiform activity in vitro and electrographic seizures in vivo.
    Experimental neurology, 2013, Volume: 250

    Topics: 4-Aminopyridine; Animals; Anticonvulsants; Capsaicin; Convulsants; Disease Models, Animal; Epilepsy; Evoked Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; TRPV Cation Channels

2013
Activation of transient receptor potential ankyrin 1 by eugenol.
    Neuroscience, 2014, Mar-07, Volume: 261

    Topics: Acetanilides; Analgesics; Animals; Calcium; Calcium Channels; Capsaicin; Eugenol; HEK293 Cells; Humans; Isothiocyanates; Male; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Purines; Rats; Rats, Sprague-Dawley; Sensory System Agents; Transient Receptor Potential Channels; Trigeminal Ganglion; TRPA1 Cation Channel; TRPC Cation Channels

2014
[6]-shogaol induces Ca²⁺ signals by activating the TRPV1 channels in the rat insulinoma INS-1E cells.
    JOP : Journal of the pancreas, 2014, Jan-10, Volume: 15, Issue:1

    Topics: Animals; Calcium Signaling; Capsaicin; Catechols; Cell Line, Tumor; Clone Cells; Dose-Response Relationship, Drug; Glucose; Insulinoma; Islets of Langerhans; Pancreatic Neoplasms; Rats; TRPV Cation Channels

2014
Morphine inhibits acid-sensing ion channel currents in rat dorsal root ganglion neurons.
    Brain research, 2014, Mar-20, Volume: 1554

    Topics: Acetic Acid; Acid Sensing Ion Channel Blockers; Acid Sensing Ion Channels; Action Potentials; Analgesics, Opioid; Animals; Capsaicin; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ganglia, Spinal; In Vitro Techniques; Male; Morphine; Naloxone; Narcotic Antagonists; Neurons; Nociception; Pain; Protons; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; TRPV Cation Channels

2014
Effects of cannabinoid and vanilloid drugs on positive and negative-like symptoms on an animal model of schizophrenia: the SHR strain.
    Schizophrenia research, 2014, Volume: 153, Issue:1-3

    Topics: Analysis of Variance; Animals; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Interpersonal Relations; Male; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Inbred SHR; Rats, Wistar; Rimonabant; Schizophrenia; Schizophrenic Psychology; TRPV Cation Channels

2014
The induction of long-term potentiation in spinal dorsal horn after peripheral nociceptive stimulation and contribution of spinal TRPV1 in rats.
    Neuroscience, 2014, Jun-06, Volume: 269

    Topics: Acrylamides; Animals; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Central Nervous System Agents; Electric Stimulation; Formaldehyde; Freund's Adjuvant; Long-Term Potentiation; Male; Microelectrodes; Nociception; Posterior Horn Cells; Rats, Sprague-Dawley; Sciatic Nerve; TRPV Cation Channels

2014
Electromagnetic radiation (Wi-Fi) and epilepsy induce calcium entry and apoptosis through activation of TRPV1 channel in hippocampus and dorsal root ganglion of rats.
    Metabolic brain disease, 2014, Volume: 29, Issue:3

    Topics: Animals; Apoptosis; Calcium; Capsaicin; Caspase 3; Electromagnetic Radiation; Epilepsy; Ganglia, Spinal; Hippocampus; Male; Neurons; Oxidative Stress; Rats; TRPV Cation Channels

2014
Hypoxic preconditioning protects rat hearts against ischemia-reperfusion injury via the arachidonate12-lipoxygenase/transient receptor potential vanilloid 1 pathway.
    Basic research in cardiology, 2014, Volume: 109, Issue:4

    Topics: 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid; Animals; Arachidonate 12-Lipoxygenase; Caffeic Acids; Capsaicin; Flavanones; Hypoxia; In Vitro Techniques; Isoenzymes; Lipoxygenase Inhibitors; Male; Myocardial Reperfusion Injury; Myocardium; Protein Kinase C; Protein Transport; Rats, Wistar; Sarcolemma; Signal Transduction; Time Factors; TRPV Cation Channels

2014
Inhibition of K+ transport through Na+, K+-ATPase by capsazepine: role of membrane span 10 of the α-subunit in the modulation of ion gating.
    PloS one, 2014, Volume: 9, Issue:5

    Topics: 4-Nitrophenylphosphatase; Animals; Biological Transport; Capsaicin; Catalytic Domain; Cell Membrane; Endopeptidase K; Enzyme Inhibitors; Hydrogen-Ion Concentration; Hydrolysis; Intracellular Space; Ion Channel Gating; Isoxazoles; Myocytes, Cardiac; Potassium; Proteolysis; Rats; Sodium; Sodium-Potassium-Exchanging ATPase; Temperature; Trypsin; Vanadates

2014
Acid mediates a prolonged antinociception via substance P signaling in acid-induced chronic widespread pain.
    Molecular pain, 2014, May-21, Volume: 10

    Topics: Acid Sensing Ion Channels; Acids; Animals; Capsaicin; Chronic Pain; Cnidarian Venoms; Disease Models, Animal; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle, Skeletal; Pain Measurement; Signal Transduction; Substance P; TRPV Cation Channels

2014
Cannabinoid 1 and transient receptor potential vanilloid 1 receptors discretely modulate evoked glutamate separately from spontaneous glutamate transmission.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Jun-11, Volume: 34, Issue:24

    Topics: Action Potentials; Analgesics; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Capsaicin; Dopamine; Excitatory Postsynaptic Potentials; Glutamic Acid; Hot Temperature; In Vitro Techniques; Male; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission; TRPV Cation Channels

2014
QSAR and docking studies on capsazepine derivatives for immunomodulatory and anti-inflammatory activity.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; Biological Availability; Capsaicin; Cell Survival; Cytokines; Drug Evaluation, Preclinical; Female; Immunologic Factors; Macrophages; Mice; Molecular Docking Simulation; Protein Conformation; Quantitative Structure-Activity Relationship; Risk Assessment; Tumor Necrosis Factor-alpha

2014
Spatio-temporal expression and functional involvement of transient receptor potential vanilloid 1 in diabetic mechanical allodynia in rats.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Analysis of Variance; Animals; Blotting, Western; Capsaicin; Diabetic Neuropathies; Fluorescent Antibody Technique; Ganglia, Spinal; Gene Expression Profiling; Gene Expression Regulation; Hyperalgesia; Image Processing, Computer-Assisted; Immunohistochemistry; Rats; Real-Time Polymerase Chain Reaction; Ruthenium Red; Spinal Cord; Streptozocin; Time Factors; TRPV Cation Channels

2014
The ethanol-induced stimulation of rat duodenal mucosal bicarbonate secretion in vivo is critically dependent on luminal Cl-.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Animals; Anion Transport Proteins; Antiporters; Bicarbonates; Body Fluids; Capsaicin; Chlorine; Cystic Fibrosis Transmembrane Conductance Regulator; Duodenum; Ethanol; Gastric Acid; Hexamethonium; Hydrochloric Acid; Intestinal Mucosa; Male; Nicotinic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Sulfate Transporters

2014
Capsaicin induces "brite" phenotype in differentiating 3T3-L1 preadipocytes.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: 3T3-L1 Cells; Adipocytes; Adipocytes, Brown; Adipogenesis; Adipokines; Animals; Biomarkers; Body Weight; Capsaicin; Cell Differentiation; Diet, High-Fat; Gene Expression Regulation; Lipid Metabolism; Mice; Motor Activity; Pain Threshold; Phenotype; PPAR gamma; TRPV Cation Channels

2014
Protons modulate perivascular axo-axonal neurotransmission in the rat mesenteric artery.
    British journal of pharmacology, 2014, Volume: 171, Issue:24

    Topics: Acetylcholine; Adrenergic Neurons; Animals; Atropine; Axons; Calcitonin Gene-Related Peptide; Capsaicin; Cholinergic Agonists; Guanethidine; Hydrogen-Ion Concentration; Mecamylamine; Mesenteric Arteries; Muscarinic Antagonists; Nicotinic Antagonists; Protons; Rats; Ruthenium Red; Sympatholytics; Synaptic Transmission; Vasoconstriction; Vasodilation

2014
Blocking TRPV1 in nucleus accumbens inhibits persistent morphine conditioned place preference expression in rats.
    PloS one, 2014, Volume: 9, Issue:8

    Topics: Animals; Blotting, Western; Capsaicin; Craving; Dose-Response Relationship, Drug; Male; Microscopy, Immunoelectron; Morphine; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Spatial Behavior; TRPV Cation Channels

2014
Effect of TRPV1 channel on proliferation and apoptosis of airway smooth muscle cells of rats.
    Journal of Huazhong University of Science and Technology. Medical sciences = Hua zhong ke ji da xue xue bao. Yi xue Ying De wen ban = Huazhong keji daxue xuebao. Yixue Yingdewen ban, 2014, Volume: 34, Issue:4

    Topics: Animals; Antipruritics; Apoptosis; Bronchi; Calcium Signaling; Capsaicin; Cell Proliferation; Myocytes, Smooth Muscle; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2014
External QX-314 inhibits evoked cranial primary afferent synaptic transmission independent of TRPV1.
    Journal of neurophysiology, 2014, Dec-01, Volume: 112, Issue:11

    Topics: Anesthetics, Local; Animals; Capsaicin; Cranial Nerves; Excitatory Postsynaptic Potentials; Lidocaine; Male; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Reaction Time; TRPV Cation Channels

2014
Palmitoylethanolamide, a naturally occurring lipid, is an orally effective intestinal anti-inflammatory agent.
    British journal of pharmacology, 2015, Volume: 172, Issue:1

    Topics: Administration, Oral; Amides; Animals; Anti-Inflammatory Agents; Benzenesulfonates; Capsaicin; Colitis; Colon; Disease Models, Animal; Endocannabinoids; Ethanolamines; Intestinal Absorption; Male; Mice, Inbred ICR; Oleic Acids; Palmitic Acids; Peroxidase; PPAR alpha; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; RNA, Messenger; TRPV Cation Channels

2015
TRPV1 antagonism by capsazepine modulates innate immune response in mice infected with Plasmodium berghei ANKA.
    Mediators of inflammation, 2014, Volume: 2014

    Topics: Animals; Capsaicin; Flow Cytometry; Interferon-gamma; Interleukin-10; Interleukin-17; Interleukin-4; Interleukin-6; Killer Cells, Natural; Male; Mice; Mice, Inbred C57BL; Plasmodium berghei; TRPV Cation Channels

2014
Role of membrane cholesterol in spontaneous exocytosis at frog neuromuscular synapses: reactive oxygen species-calcium interplay.
    The Journal of physiology, 2014, Nov-15, Volume: 592, Issue:22

    Topics: Acetophenones; Acetylcysteine; Animals; beta-Cyclodextrins; Calcium; Calcium Signaling; Capsaicin; Cholesterol; Cyclosporine; Exocytosis; Neuromuscular Junction; Okadaic Acid; Ranidae; Reactive Oxygen Species; Ruthenium Red; Synaptic Membranes; TRPV Cation Channels

2014
Role of TRPV1 channels in ischemia/reperfusion-induced acute kidney injury.
    PloS one, 2014, Volume: 9, Issue:10

    Topics: Animals; Capsaicin; Eicosanoids; Hydroxyeicosatetraenoic Acids; Kidney; Mice; Mice, Inbred C57BL; Reperfusion Injury; TRPV Cation Channels

2014
Role of TRPV1 and ASIC3 in formalin-induced secondary allodynia and hyperalgesia.
    Pharmacological reports : PR, 2014, Volume: 66, Issue:6

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Blotting, Western; Capsaicin; Cnidarian Venoms; Disease Models, Animal; Dose-Response Relationship, Drug; Formaldehyde; Ganglia, Spinal; Hyperalgesia; Pyridines; Rats; Sulfones; Time Factors; TRPV Cation Channels

2014
Capsaicin modulates acetylcholine release at the myoneural junction.
    European journal of pharmacology, 2014, Dec-05, Volume: 744

    Topics: Acetylcholine; Animals; Capsaicin; Exocytosis; Mice; Mice, Inbred C57BL; Neuromuscular Junction; Phrenic Nerve; TRPV Cation Channels; Vagus Nerve Stimulation

2014
Carvacrol presynaptically enhances spontaneous excitatory transmission and produces outward current in adult rat spinal substantia gelatinosa neurons.
    Brain research, 2014, Dec-10, Volume: 1592

    Topics: Acetanilides; Analgesics; Animals; Capsaicin; Cymenes; Excitatory Amino Acid Agents; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Monoterpenes; Neurons; Neurotransmitter Agents; Nociception; Patch-Clamp Techniques; Permeability; Potassium; Potassium Channel Blockers; Purines; Rats, Sprague-Dawley; Substantia Gelatinosa; Tissue Culture Techniques; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2014
Full-length transient receptor potential vanilloid 1 channels mediate calcium signals and possibly contribute to osmoreception in vasopressin neurones in the rat supraoptic nucleus.
    Cell calcium, 2015, Volume: 57, Issue:1

    Topics: Action Potentials; Animals; Calcium Signaling; Capsaicin; Cells, Cultured; HEK293 Cells; Humans; Male; Mannitol; Neurons; Osmolar Concentration; Oxytocin; Pyrazines; Pyridines; Rats; Rats, Transgenic; Rats, Wistar; Supraoptic Nucleus; Temperature; TRPV Cation Channels

2015
Involvement of TRPV1 channels in the periaqueductal grey on the modulation of innate fear responses.
    Acta neuropsychiatrica, 2015, Volume: 27, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Capsaicin; Cats; Fear; Male; Periaqueductal Gray; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; TRPV Cation Channels

2015
Transient receptor potential vanilloid type 1 is vital for (-)-epigallocatechin-3-gallate mediated activation of endothelial nitric oxide synthase.
    Molecular nutrition & food research, 2015, Volume: 59, Issue:4

    Topics: AMP-Activated Protein Kinases; Anilides; Animals; Calcium; Capsaicin; Catechin; Cell Movement; Cell Proliferation; Cell Survival; Cinnamates; Endothelial Cells; HEK293 Cells; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Neovascularization, Pathologic; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphorylation; Signal Transduction; Tea; TRPV Cation Channels

2015
The role of TRPV1 channels in carrageenan-induced mechanical hyperalgesia in mice.
    Neuroreport, 2015, Feb-11, Volume: 26, Issue:3

    Topics: Analgesics; Animals; Capsaicin; Carrageenan; Disease Models, Animal; Functional Laterality; Hyperalgesia; Inflammation; Male; Mice, Inbred C57BL; Mice, Knockout; Sensory System Agents; Touch; TRPV Cation Channels

2015
Inhibitors of glutamate release from breast cancer cells; new targets for cancer-induced bone-pain.
    Scientific reports, 2015, Feb-11, Volume: 5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Bone and Bones; Breast Neoplasms; Capsaicin; Cell Line, Tumor; Dopamine Agonists; Drug Discovery; Female; Glutamic Acid; High-Throughput Screening Assays; Humans; Inhibitory Concentration 50; Pain; Signal Transduction; Small Molecule Libraries

2015
Expression and function of the epithelial sodium channel δ-subunit in human respiratory epithelial cells in vitro.
    Pflugers Archiv : European journal of physiology, 2015, Volume: 467, Issue:11

    Topics: Capsaicin; Diuretics; Epithelial Cells; Epithelial Sodium Channels; Evans Blue; Gene Knockdown Techniques; Humans; Primary Cell Culture; Pulmonary Alveoli; Pyrimidinones; Respiratory Mucosa; Sodium

2015
Antinociceptive activity of transient receptor potential channel TRPV1, TRPA1, and TRPM8 antagonists in neurogenic and neuropathic pain models in mice.
    Journal of Zhejiang University. Science. B, 2015, Volume: 16, Issue:3

    Topics: Acetanilides; Analgesics; Animals; Benzamides; Capsaicin; Cold Temperature; Disease Models, Animal; Formaldehyde; Hyperalgesia; Isothiocyanates; Male; Mice; Neuralgia; Oximes; Paclitaxel; Pain Measurement; Purines; Thiophenes; Touch; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPM Cation Channels; TRPV Cation Channels

2015
Involvement of apoptosis and calcium accumulation through TRPV1 channels in neurobiology of epilepsy.
    Neuroscience, 2015, May-07, Volume: 293

    Topics: Animals; Apoptosis; Calcium; Capsaicin; Diterpenes; Epilepsy; Ganglia, Spinal; Hippocampus; Male; Neurons; Pentylenetetrazole; Rats; Rats, Wistar; TRPV Cation Channels

2015
Spontaneous L-glutamate release enhancement in rat substantia gelatinosa neurons by (-)-carvone and (+)-carvone which activate different types of TRP channel.
    Biochemical and biophysical research communications, 2015, Apr-10, Volume: 459, Issue:3

    Topics: Acetanilides; Animals; Capsaicin; Cyclohexane Monoterpenes; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Monoterpenes; Neurons; Patch-Clamp Techniques; Purines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Substantia Gelatinosa; Synaptic Transmission; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPC Cation Channels; TRPV Cation Channels

2015
Intracolonic Administration of the TRPA1 Agonist Allyl Isothiocyanate Stimulates Colonic Motility and Defecation in Conscious Dogs.
    Journal of gastrointestinal surgery : official journal of the Society for Surgery of the Alimentary Tract, 2015, Volume: 19, Issue:7

    Topics: Acetanilides; Anastomosis, Surgical; Animals; Atropine; Capsaicin; Colon; Defecation; Denervation; Dogs; Enteric Nervous System; Ganglionic Blockers; Gastrointestinal Motility; Hexamethonium; Ileum; Isothiocyanates; Muscarinic Antagonists; Ondansetron; Purines; Serotonin Antagonists; Transient Receptor Potential Channels

2015
[6]-gingerol induces electrogenic sodium absorption in the rat colon via the capsaicin receptor TRPV1.
    Journal of nutritional science and vitaminology, 2014, Volume: 60, Issue:6

    Topics: Animals; Bumetanide; Capsaicin; Catechols; Colon; Enzyme Inhibitors; Fatty Alcohols; Ileum; Male; Membrane Potentials; Ouabain; Rats; Rats, Sprague-Dawley; Sodium; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Potassium-Exchanging ATPase; TRPV Cation Channels

2014
Impaired capsaicin-induced relaxation in diabetic mesenteric arteries.
    Journal of diabetes and its complications, 2015, Volume: 29, Issue:6

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Diabetes Mellitus, Experimental; Disease Models, Animal; Male; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Peptide Fragments; Rats; Rats, Sprague-Dawley; TRPV Cation Channels; Vasodilation; Vasodilator Agents

2015
Hypericum perforatum Attenuates Spinal Cord Injury-Induced Oxidative Stress and Apoptosis in the Dorsal Root Ganglion of Rats: Involvement of TRPM2 and TRPV1 Channels.
    Molecular neurobiology, 2016, Volume: 53, Issue:6

    Topics: Animals; Apoptosis; Calcium; Capsaicin; Caspases; Cell Survival; Ganglia, Spinal; Glutathione; Glutathione Peroxidase; Hydrogen Peroxide; Hypericum; Ion Channel Gating; Lipid Peroxidation; Male; Membrane Potential, Mitochondrial; Oxidative Stress; Plant Extracts; Rats; Rats, Wistar; Reactive Oxygen Species; Spinal Cord Injuries; TRPM Cation Channels; TRPV Cation Channels

2016
Synovial TRPV1 is upregulated by 17-β-estradiol and involved in allodynia of inflamed temporomandibular joints in female rats.
    Archives of oral biology, 2015, Volume: 60, Issue:9

    Topics: Animals; Blotting, Western; Capsaicin; Cyclooxygenase 2; Estradiol; Female; Freund's Adjuvant; Hyperalgesia; Inflammation; Nerve Growth Factor; Ovariectomy; Random Allocation; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Temporomandibular Joint; Temporomandibular Joint Disorders; Transcriptional Activation; TRPV Cation Channels; Up-Regulation

2015
Role of TRPV1 channels of the dorsal periaqueductal gray in the modulation of nociception and open elevated plus maze-induced antinociception in mice.
    Behavioural brain research, 2015, Oct-01, Volume: 292

    Topics: Animals; Anxiety; Capsaicin; Fear; Male; Maze Learning; Mice; Nociception; Pain; Pain Measurement; Periaqueductal Gray; TRPV Cation Channels

2015
The molecular pathway of ATP-sensitive potassium channel in endothelial cells for mediating arteriole relaxation.
    Life sciences, 2015, Sep-15, Volume: 137

    Topics: Allyl Compounds; Anilides; Animals; Arterioles; Calcium; Capsaicin; Cells, Cultured; Cinnamates; Down-Regulation; Endothelial Cells; KATP Channels; Mesenteric Arteries; Nitric Oxide; Propylamines; Rats; RNA, Small Interfering; TRPV Cation Channels; Vasodilation

2015
Evodiamine suppresses capsaicin-induced thermal hyperalgesia through activation and subsequent desensitization of the transient receptor potential V1 channels.
    Journal of natural medicines, 2016, Volume: 70, Issue:1

    Topics: Alkaloids; Analgesics; Animals; Calcium; Calcium Channels; Capsaicin; Dose-Response Relationship, Drug; Evodia; Ganglia, Spinal; HEK293 Cells; Hot Temperature; Humans; Hyperalgesia; Male; Medicine, Chinese Traditional; Nerve Tissue Proteins; Neurons; Patch-Clamp Techniques; Plant Extracts; Quinazolines; Quinolines; Rats; Rats, Sprague-Dawley; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2016
Sensory nerves contribute to cutaneous vasodilator response to cathodal stimulation in healthy rats.
    Microvascular research, 2015, Volume: 101

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Electrodes; Electrophysiology; Hydrogen-Ion Concentration; Laser-Doppler Flowmetry; Male; Microcirculation; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory Receptor Cells; Skin; Substance P; TRPV Cation Channels; Vasodilation; Vasodilator Agents

2015
Social stress in mice induces urinary bladder overactivity and increases TRPV1 channel-dependent afferent nerve activity.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2015, Sep-15, Volume: 309, Issue:6

    Topics: Aggression; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Male; Mice; Mice, Inbred C57BL; Neurons, Afferent; Social Environment; Stress, Psychological; TRPV Cation Channels; Urethra; Urinary Bladder; Urinary Bladder, Overactive; Urination

2015
Thermosensation and the TRPV channel in Rhodnius prolixus.
    Journal of insect physiology, 2015, Volume: 81

    Topics: Amino Acid Sequence; Animals; Behavior, Animal; Capsaicin; Chagas Disease; Conditioning, Operant; Feeding Behavior; Gene Expression; Hot Temperature; Insect Vectors; Molecular Sequence Data; Rhodnius; Spatial Learning; Temperature; Thermosensing; TRPV Cation Channels

2015
Alterations in CA1 pyramidal neuronal intrinsic excitability mediated by Ih channel currents in a rat model of amyloid beta pathology.
    Neuroscience, 2015, Oct-01, Volume: 305

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Avoidance Learning; CA1 Region, Hippocampal; Capsaicin; Disease Models, Animal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Male; Memory Disorders; Nerve Net; Neurons; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Wistar; Sensory System Agents; TRPV Cation Channels

2015
Action of thymol on spontaneous excitatory transmission in adult rat spinal substantia gelatinosa neurons.
    Neuroscience letters, 2015, Oct-08, Volume: 606

    Topics: Acetanilides; Animals; Capsaicin; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Neurons; Purines; Pyrazines; Pyridines; Rats, Sprague-Dawley; Sodium Channel Blockers; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin; Thymol; TRPA1 Cation Channel; TRPC Cation Channels; TRPM Cation Channels

2015
Medial prefrontal cortex TRPV1 channels modulate the baroreflex cardiac activity in rats.
    British journal of pharmacology, 2015, Volume: 172, Issue:22

    Topics: Animals; Baroreflex; Capsaicin; Heart; Male; Prefrontal Cortex; Rats, Wistar; TRPV Cation Channels

2015
A pathophysiological role of TRPV1 in ischemic injury after transient focal cerebral ischemia in mice.
    Biochemical and biophysical research communications, 2015, Nov-20, Volume: 467, Issue:3

    Topics: Animals; Brain Ischemia; Capsaicin; Mice; Mice, Inbred C57BL; Mice, Knockout; TRPV Cation Channels

2015
Measurement of Ensemble TRPV1 Ion Channel Currents Using Droplet Bilayers.
    PloS one, 2015, Volume: 10, Issue:10

    Topics: Action Potentials; Capsaicin; Humans; Lipid Bilayers; TRPV Cation Channels

2015
[TRPV1 channel-mediated thermogenesis is a common mode for the Chinese pungent-hot or pungent-warm herbs to demonstrate their natures].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2015, Volume: 50, Issue:7

    Topics: Adipose Tissue, Brown; Animals; Capsaicin; Energy Metabolism; Ganglia, Spinal; HEK293 Cells; Humans; Mice; Neurons; Plants, Medicinal; Temperature; Thermogenesis; TRPV Cation Channels

2015
Hydrogen sulfide-induced itch requires activation of Cav3.2 T-type calcium channel in mice.
    Scientific reports, 2015, Nov-25, Volume: 5

    Topics: Acetanilides; Animals; Behavior, Animal; Calcium Channel Blockers; Calcium Channels, T-Type; Capsaicin; Cystathionine beta-Synthase; Cystathionine gamma-Lyase; Disease Models, Animal; Diterpenes; Male; Mibefradil; Mice; Pruritus; Purines; Receptors, Opioid; RNA Interference; Sensory Receptor Cells; Sulfides; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2015
TRPV1 receptors augment basal synaptic transmission in CA1 and CA3 pyramidal neurons in epilepsy.
    Neuroscience, 2016, Feb-09, Volume: 314

    Topics: Animals; Capsaicin; Disease Models, Animal; Epilepsy, Temporal Lobe; Excitatory Postsynaptic Potentials; Hippocampus; Male; Pilocarpine; Pyramidal Cells; Rats, Wistar; RNA, Messenger; TRPV Cation Channels

2016
Tris-hydroxymethyl-aminomethane enhances capsaicin-induced intracellular Ca(2+) influx through transient receptor potential V1 (TRPV1) channels.
    Journal of pharmacological sciences, 2016, Volume: 130, Issue:2

    Topics: Acrylamides; Animals; Calcium; Capsaicin; Cells, Cultured; Cricetinae; Hydrogen-Ion Concentration; Pain; TRPV Cation Channels

2016
Effect of cannabinoids on CGRP release in the isolated rat lumbar spinal cord.
    Neuroscience letters, 2016, Feb-12, Volume: 614

    Topics: Animals; Arachidonic Acids; Benzoxazines; Calcitonin Gene-Related Peptide; Cannabinoid Receptor Agonists; Cannabinoids; Capsaicin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; In Vitro Techniques; Indoles; Lumbosacral Region; Male; Morpholines; Naphthalenes; Rats, Wistar; Receptors, Opioid; Sciatic Nerve; Spinal Cord; TRPV Cation Channels

2016
Activation of TRPV1-dependent calcium oscillation exacerbates seawater inhalation-induced acute lung injury.
    Molecular medicine reports, 2016, Volume: 13, Issue:3

    Topics: Actin Cytoskeleton; Acute Lung Injury; Administration, Inhalation; Animals; Calcium; Calcium Chelating Agents; Calcium Signaling; Capsaicin; Cell Line, Tumor; Cytosol; Disease Progression; Egtazic Acid; Extracellular Space; Fluorescence; Humans; Inflammation Mediators; Interleukin-1beta; Lung; Male; NF-kappa B; Phosphorylation; Proline; Rats, Sprague-Dawley; Seawater; Thiocarbamates; TRPV Cation Channels; Tumor Necrosis Factor-alpha

2016
Evaluation of the antidepressant- and anxiolytic-like activity of α-spinasterol, a plant derivative with TRPV1 antagonistic effects, in mice.
    Behavioural brain research, 2016, Apr-15, Volume: 303

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety; Body Temperature; Capsaicin; Depression; Male; Mice; Motor Activity; Stigmasterol; TRPV Cation Channels

2016
Involvement of TRPV1 in the Olfactory Bulb in Rimonabant-Induced Olfactory Discrimination Deficit.
    The Chinese journal of physiology, 2016, 02-29, Volume: 59, Issue:1

    Topics: Animals; Capsaicin; Male; Mice; Mice, Inbred C57BL; Motor Activity; Olfactory Bulb; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Smell; TRPV Cation Channels

2016
Effect of transient receptor potential vanilloid-1 on cough hypersensitivity induced by particulate matter 2.5.
    Life sciences, 2016, Apr-15, Volume: 151

    Topics: Animals; Capillary Permeability; Capsaicin; Central Nervous System Diseases; Cough; Guinea Pigs; Herpesvirus 1, Suid; Hypersensitivity; Male; Particulate Matter; Respiratory Hypersensitivity; Signal Transduction; Substance P; TRPV Cation Channels; Vagus Nerve

2016
Potentiation of acid-sensing ion channel activity by peripheral group I metabotropic glutamate receptor signaling.
    Pharmacological research, 2016, Volume: 107

    Topics: Acetic Acid; Acid Sensing Ion Channels; Acidosis; Animals; Capsaicin; Ganglia, Spinal; Male; Methoxyhydroxyphenylglycol; Neurons; Pain; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Sodium Channel Blockers; Tetrodotoxin; TRPV Cation Channels

2016
Activation of transient receptor potential vanilloid 1 accelerates re-endothelialization and inhibits neointimal formation after vascular injury.
    Journal of vascular surgery, 2017, Volume: 65, Issue:1

    Topics: Adenosine Triphosphate; Animals; Calcium Chelating Agents; Capsaicin; Carotid Artery Injuries; Cell Movement; Cell Proliferation; Cells, Cultured; Disease Models, Animal; Egtazic Acid; Endothelial Cells; GTP Phosphohydrolases; Human Umbilical Vein Endothelial Cells; Humans; Hyperplasia; Male; Membrane Potential, Mitochondrial; Mice, Inbred C57BL; Mice, Knockout; Mitochondrial Proteins; Neointima; Re-Epithelialization; RNA Interference; Signal Transduction; Transfection; TRPV Cation Channels

2017
Protective role of cannabinoid CB1 receptors and vascular effects of chronic administration of FAAH inhibitor URB597 in DOCA-salt hypertensive rats.
    Life sciences, 2016, Apr-15, Volume: 151

    Topics: Amidohydrolases; Animals; Aorta; Arachidonic Acids; Benzamides; Blood Pressure; Capsaicin; Carbamates; Desoxycorticosterone Acetate; Dose-Response Relationship, Drug; Drug Interactions; Hypertension; Male; Mesenteric Arteries; Morpholines; Phenylephrine; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Sodium Chloride; Vasoconstriction; Vasodilation

2016
Involvement of TRPV1 channels in the activity of the cannabinoid WIN 55,212-2 in an acute rat model of temporal lobe epilepsy.
    Epilepsy research, 2016, Volume: 122

    Topics: Acute Disease; Animals; Anticonvulsants; Benzoxazines; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Electric Stimulation; Epilepsy, Temporal Lobe; Male; Membrane Transport Modulators; Morpholines; Naphthalenes; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2016
Inflammatory stimuli acutely modulate peripheral taste function.
    Journal of neurophysiology, 2016, 06-01, Volume: 115, Issue:6

    Topics: Amiloride; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Body Weight; Capsaicin; Chorda Tympani Nerve; Dose-Response Relationship, Drug; Epithelial Sodium Channel Blockers; Female; Functional Laterality; Interleukin-6; Lipopolysaccharides; Quinine; Rats; Sensory Receptor Cells; Sodium; Sodium Acetate; Sodium Chloride; Taste Buds; Tomography Scanners, X-Ray Computed; Tumor Necrosis Factor-alpha

2016
The Transient Receptor Potential Vanilloid 1 Antagonist Capsazepine Improves the Impaired Lung Mechanics during Endotoxemia.
    Basic & clinical pharmacology & toxicology, 2016, Volume: 119, Issue:5

    Topics: Acute Lung Injury; Animals; Capsaicin; Disease Models, Animal; Endotoxemia; Lipopolysaccharides; Lung; Male; Mice; TRPV Cation Channels

2016
Radiosensitizing Effect of TRPV1 Channel Inhibitors in Cancer Cells.
    Biological & pharmaceutical bulletin, 2016, Jul-01, Volume: 39, Issue:7

    Topics: Acrylamides; Anilides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line, Tumor; Cell Survival; Cinnamates; DNA Damage; Gamma Rays; Humans; Mice; Necrosis; Neoplasms; Pyrazines; Pyridines; Radiation-Sensitizing Agents; TRPV Cation Channels

2016
NMDA receptors are involved in the antidepressant-like effects of capsaicin following amphetamine withdrawal in male mice.
    Neuroscience, 2016, 08-04, Volume: 329

    Topics: Amphetamine; Animals; Antidepressive Agents; Capsaicin; Central Nervous System Stimulants; Depressive Disorder; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome; Time Factors; TRPV Cation Channels

2016
TRPV1 is crucial for proinflammatory STAT3 signaling and thermoregulation-associated pathways in the brain during inflammation.
    Scientific reports, 2016, 05-18, Volume: 6

    Topics: Animals; Body Temperature Regulation; Brain; Capsaicin; Diterpenes; Lipopolysaccharides; Mice; Mice, Knockout; Signal Transduction; STAT3 Transcription Factor; TRPV Cation Channels

2016
Endovanilloids are potential activators of the trigeminovascular nocisensor complex.
    The journal of headache and pain, 2016, Volume: 17

    Topics: Animals; Arachidonic Acids; Calcitonin Gene-Related Peptide; Cannabinoid Receptor Agonists; Capsaicin; Disease Models, Animal; Dopamine; Dose-Response Relationship, Drug; Dura Mater; Endocannabinoids; Enzyme-Linked Immunosorbent Assay; Laser-Doppler Flowmetry; Nociceptors; Peptide Fragments; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Calcitonin Gene-Related Peptide; Regional Blood Flow; Trigeminal Nerve; TRPV Cation Channels

2016
Role of curcumin in protection of gastric mucosa against stress-induced gastric mucosal damage. Involvement of hypoacidity, vasoactive mediators and sensory neuropeptides.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2016, Volume: 67, Issue:2

    Topics: Animals; Anti-Ulcer Agents; Capsaicin; Curcumin; Cyclooxygenase 2; Female; Gastric Acid; Gastric Mucosa; Gastrins; Immersion; Male; Nitric Oxide Synthase Type II; Rats, Wistar; Restraint, Physical; RNA, Messenger; Stomach Ulcer; Stress, Psychological; TRPV Cation Channels; Tumor Necrosis Factor-alpha; Water

2016
Systemic desensitization through TRPA1 channels by capsazepine and mustard oil - a novel strategy against inflammation and pain.
    Scientific reports, 2016, 06-30, Volume: 6

    Topics: Acetanilides; Analgesics; Animals; Anti-Inflammatory Agents; Calcium Signaling; Capsaicin; HEK293 Cells; Humans; Inflammation; Mice; Mice, Knockout; Mustard Plant; Oximes; Pain; Plant Oils; Purines; TRPA1 Cation Channel

2016
TRPV1-mediated presynaptic transmission in basolateral amygdala contributes to visceral hypersensitivity in adult rats with neonatal maternal deprivation.
    Scientific reports, 2016, 07-01, Volume: 6

    Topics: Animals; Basolateral Nuclear Complex; Capsaicin; Excitatory Postsynaptic Potentials; Hypersensitivity; In Vitro Techniques; Male; Maternal Deprivation; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Synapses; Synaptic Transmission; TRPV Cation Channels; Up-Regulation

2016
Co-administration of cannabidiol and capsazepine reduces L-DOPA-induced dyskinesia in mice: Possible mechanism of action.
    Neurobiology of disease, 2016, Volume: 94

    Topics: Animals; Anti-Dyskinesia Agents; Arachidonic Acids; Brain; Cannabidiol; Capsaicin; Cyclooxygenase 2; Dyskinesia, Drug-Induced; Endocannabinoids; Extracellular Signal-Regulated MAP Kinases; Histones; Levodopa; Male; Mice, Inbred C57BL; NF-kappa B; Oxidopamine; Parkinsonian Disorders; Polyunsaturated Alkamides; PPAR gamma; Receptor, Cannabinoid, CB1; TRPV Cation Channels; Tyrosine 3-Monooxygenase

2016
Duloxetine Reduces Oxidative Stress, Apoptosis, and Ca
    Molecular neurobiology, 2017, Volume: 54, Issue:6

    Topics: Animals; Apoptosis; Calcium; Capsaicin; Caspase 3; Caspase 9; Duloxetine Hydrochloride; Ganglia, Spinal; Hippocampus; Ion Channel Gating; Male; Membrane Potential, Mitochondrial; Neurons; ortho-Aminobenzoates; Oxidative Stress; Rats, Wistar; Reactive Oxygen Species; TRPM Cation Channels; TRPV Cation Channels

2017
Capsazepine inhibits JAK/STAT3 signaling, tumor growth, and cell survival in prostate cancer.
    Oncotarget, 2017, Mar-14, Volume: 8, Issue:11

    Topics: A549 Cells; Animals; Antineoplastic Agents; Apoptosis; Capsaicin; Cell Line, Tumor; Cell Proliferation; Cell Survival; Enzyme Activation; Humans; Janus Kinase 1; Ki-67 Antigen; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Invasiveness; Phosphorylation; Prostatic Neoplasms; Protein Tyrosine Phosphatases; Receptor-Like Protein Tyrosine Phosphatases, Class 4; RNA Interference; RNA, Small Interfering; STAT3 Transcription Factor; Vanadates; Xenograft Model Antitumor Assays

2017
Mitogen-Activated Protein Kinase and Intracellular Polyamine Signaling Is Involved in TRPV1 Activation-Induced Cardiac Hypertrophy.
    Journal of the American Heart Association, 2016, 07-29, Volume: 5, Issue:8

    Topics: Analysis of Variance; Animals; Aorta, Thoracic; Arachidonic Acids; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Capsaicin; Cardiomegaly; Cardiotonic Agents; Cells, Cultured; Down-Regulation; Endocannabinoids; Enzyme Inhibitors; Ligation; Male; Mice, Inbred C57BL; Mitogen-Activated Protein Kinase Kinases; Myocytes, Cardiac; Polyamines; Polyunsaturated Alkamides; Rats, Wistar; RNA, Small Interfering; Signal Transduction; TRPV Cation Channels

2016
Inhibition of interleukin-1β-induced endothelial tissue factor expression by the synthetic cannabinoid WIN 55,212-2.
    Oncotarget, 2016, 09-20, Volume: 7, Issue:38

    Topics: Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Cannabinoids; Capsaicin; Cells, Cultured; Ceramides; Human Umbilical Vein Endothelial Cells; Humans; Indoles; Interleukin-1beta; JNK Mitogen-Activated Protein Kinases; Monocytes; Morpholines; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Partial Thromboplastin Time; Phosphorylation; Piperidines; Pyrazoles; RNA, Messenger; Signal Transduction; Sphingomyelin Phosphodiesterase; Thromboplastin; TRPV Cation Channels

2016
Involvement of the TRPV1 receptor in plasma extravasation in airways of rats treated with an angiotensin-converting enzyme inhibitor.
    Pulmonary pharmacology & therapeutics, 2016, Volume: 41

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Animals, Newborn; Bradykinin; Bronchi; Capillary Permeability; Capsaicin; Captopril; Male; Plasma; Rats; Rats, Wistar; Trachea; TRPV Cation Channels

2016
Mechanistic Studies of Capsaicin-Induced Apnea in Rodents.
    American journal of respiratory cell and molecular biology, 2017, Volume: 56, Issue:2

    Topics: Animals; Animals, Newborn; Apnea; Brain Stem; Capsaicin; Mice, Inbred C57BL; Plethysmography; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Spinal Cord; TRPV Cation Channels

2017
TRPV1 Antagonist Suppresses Allergic Conjunctivitis in a Murine Model.
    Ocular immunology and inflammation, 2018, Volume: 26, Issue:3

    Topics: Acetanilides; Animals; Blotting, Western; Capsaicin; Conjunctivitis, Allergic; Disease Models, Animal; Enzyme-Linked Immunosorbent Assay; Eosinophils; Fluorescent Antibody Technique, Indirect; Immunoglobulin E; Male; Mast Cells; Mice; Mice, Inbred BALB C; Ovalbumin; Purines; TRPA1 Cation Channel; TRPV Cation Channels

2018
Pharmacological Properties of Propiverine Contribute to Improving Lower Urinary Tract Dysfunctions in Rats with Spinal Cord Injuries.
    Drug research, 2016, Volume: 66, Issue:9

    Topics: Animals; Atropine; Benzilates; Capsaicin; Female; Muscarinic Antagonists; Rats; Spinal Cord Injuries; Urinary Bladder; Urinary Bladder, Overactive; Verapamil

2016
Gastroprotective and ulcer healing effects of hydroethanolic extract of leaves of Caryocar coriaceum: Mechanisms involved in the gastroprotective activity.
    Chemico-biological interactions, 2017, Jan-05, Volume: 261

    Topics: Animals; Antioxidants; Capsaicin; Chromatography, High Pressure Liquid; Chronic Disease; Disease Models, Animal; Ericales; Ethanol; Female; Flavonoids; Gastrointestinal Motility; Glyburide; Histamine; Indomethacin; Male; Mice; Mucus; Naloxone; NG-Nitroarginine Methyl Ester; Phenols; Phytotherapy; Plant Extracts; Plant Leaves; Protective Agents; Stomach Ulcer; Water; Yohimbine

2017
Effects of a TRPV1 agonist capsaicin on respiratory rhythm generation in brainstem-spinal cord preparation from newborn rats.
    Pflugers Archiv : European journal of physiology, 2017, Volume: 469, Issue:2

    Topics: Acrylamides; Animals; Animals, Newborn; Brain Stem; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Medulla Oblongata; Membrane Potentials; Neurons; Rats; Rats, Wistar; Respiration; Spinal Cord; TRPV Cation Channels; Voltage-Sensitive Dye Imaging

2017
Heat Sensing Receptor TRPV1 Is a Mediator of Thermotaxis in Human Spermatozoa.
    PloS one, 2016, Volume: 11, Issue:12

    Topics: Adult; Azoospermia; Capsaicin; Humans; Infertility, Male; Male; Neoplasms, Germ Cell and Embryonal; Sperm Motility; Spermatozoa; Taxis Response; Testicular Neoplasms; TRPV Cation Channels; Young Adult

2016
Presynaptic facilitation by tetracaine of glutamatergic spontaneous excitatory transmission in the rat spinal substantia gelatinosa - Involvement of TRPA1 channels.
    Brain research, 2017, 02-15, Volume: 1657

    Topics: Acetanilides; Amides; Anesthetics, Local; Animals; Bupivacaine; Capsaicin; Excitatory Postsynaptic Potentials; Glutamic Acid; Levobupivacaine; Male; Neurotransmitter Agents; Pain; Patch-Clamp Techniques; Presynaptic Terminals; Prilocaine; Purines; Pyrazines; Pyridines; Rats, Sprague-Dawley; Ropivacaine; Ruthenium Red; Substantia Gelatinosa; Tetracaine; Tetrodotoxin; Tissue Culture Techniques; TRPA1 Cation Channel; TRPC Cation Channels

2017
Activation of TRPM2 and TRPV1 Channels in Dorsal Root Ganglion by NADPH Oxidase and Protein Kinase C Molecular Pathways: a Patch Clamp Study.
    Journal of molecular neuroscience : MN, 2017, Volume: 61, Issue:3

    Topics: Acetophenones; Action Potentials; Animals; Calcium Signaling; Capsaicin; Cells, Cultured; Cinnamates; Ganglia, Spinal; Indoles; Male; Maleimides; NADPH Oxidases; Neurons; ortho-Aminobenzoates; Oxidative Stress; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; TRPM Cation Channels; TRPV Cation Channels

2017
Nitric oxide, afferent sensory nerves, and antioxidative enzymes in the mechanism of protection mediated by tricarbonyldichlororuthenium(II) dimer and sodium hydrosulfide against aspirin-induced gastric damage.
    Journal of gastroenterology, 2018, Volume: 53, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Aspirin; Blotting, Western; Calcitonin Gene-Related Peptide; Capsaicin; Carbon Monoxide; Gastric Mucosa; Glutathione Peroxidase; Glutathione Peroxidase GPX1; Lipid Peroxidation; Male; Nitric Oxide; Organometallic Compounds; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; Sensory Receptor Cells; Stomach; Sulfides

2018
Role of transient receptor potential vanilloid 1 in the modulation of airway smooth muscle tone and calcium handling.
    American journal of physiology. Lung cellular and molecular physiology, 2017, 06-01, Volume: 312, Issue:6

    Topics: Acetylcholine; Animals; Calcium; Capsaicin; Guinea Pigs; Humans; Immunohistochemistry; Methacholine Chloride; Mice; Muscle Contraction; Muscle, Smooth; RNA, Messenger; Trachea; TRPV Cation Channels

2017
Dynasore blocks evoked release while augmenting spontaneous synaptic transmission from primary visceral afferents.
    PloS one, 2017, Volume: 12, Issue:3

    Topics: Aminopyridines; Animals; Capsaicin; Excitatory Postsynaptic Potentials; Hydrazones; Male; Patch-Clamp Techniques; Piperazines; Rats; Rats, Sprague-Dawley; Solitary Nucleus; Synaptic Transmission; TRPV Cation Channels; Visceral Afferents

2017
Antinociceptive effect of natural and synthetic alkamides involves TRPV1 receptors.
    The Journal of pharmacy and pharmacology, 2017, Volume: 69, Issue:7

    Topics: Amides; Analgesics; Animals; Asteraceae; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Design; Facial Pain; Female; Mice; Pain Measurement; TRPV Cation Channels

2017
Vincristine-induced peripheral neuropathic pain and expression of transient receptor potential vanilloid 1 in rat.
    Journal of pharmacological sciences, 2017, Volume: 133, Issue:4

    Topics: Animals; Antineoplastic Agents, Phytogenic; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Ganglia, Spinal; Gene Expression; Humans; Male; Neuralgia; Neurons; Rats, Wistar; Ruthenium Red; TRPV Cation Channels; Up-Regulation; Vincristine

2017
Role of peripheral and central TRPV1 receptors in facial heat hyperalgesia in streptozotocin-induced diabetic rats.
    Brain research, 2017, Sep-01, Volume: 1670

    Topics: Animals; Capsaicin; Diabetes Mellitus, Experimental; Diterpenes; Face; Facial Pain; Hot Temperature; Hyperalgesia; Male; Pain Threshold; Rats; Rats, Wistar; Trigeminal Ganglion; TRPV Cation Channels

2017
l-Ornithine and l-lysine stimulate gastrointestinal motility via transient receptor potential vanilloid 1.
    Molecular nutrition & food research, 2017, Volume: 61, Issue:11

    Topics: Animals; Arginine; Calcium Signaling; Capsaicin; Down-Regulation; Gastrointestinal Motility; HEK293 Cells; Humans; Intestine, Small; Lysine; Male; Membrane Transport Modulators; Mice, Inbred C57BL; Mice, Knockout; Mice, Mutant Strains; Ornithine; Rats; Recombinant Proteins; Ruthenium Red; TRPV Cation Channels; Up-Regulation

2017
Capsaicin-induced rapid neutrophil leukocyte activation in the rat urinary bladder microcirculatory bed.
    Neurourology and urodynamics, 2018, Volume: 37, Issue:2

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Male; Microcirculation; Neurons, Afferent; Neutrophils; Rats; Rats, Sprague-Dawley; Substance P; Urinary Bladder

2018
4,5-Di-O-Caffeoylquinic Acid from Ligularia fischeri Suppresses Inflammatory Responses Through TRPV1 Activation.
    Phytotherapy research : PTR, 2017, Volume: 31, Issue:10

    Topics: A549 Cells; Asteraceae; Caffeic Acids; Capsaicin; Cell Movement; Cyclooxygenase 2; Humans; Plant Extracts; Quinic Acid; TRPV Cation Channels

2017
Do TRPV1 antagonists increase the risk for skin tumourigenesis? A collaborative in vitro and in vivo assessment.
    Cell biology and toxicology, 2018, Volume: 34, Issue:2

    Topics: Acrylamides; Animals; Anthracenes; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line; Cell Proliferation; Cell Survival; Cocarcinogenesis; Female; Humans; Keratinocytes; Mice; Mice, Hairless; Piperidines; Primary Cell Culture; Pyridines; Pyrrolidines; Risk; Skin Neoplasms; TRPV Cation Channels; Urea

2018
Mechanisms of curcumin-induced gastroprotection against ethanol-induced gastric mucosal lesions.
    Journal of gastroenterology, 2018, Volume: 53, Issue:5

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcitonin Gene-Related Peptide; Capsaicin; CDX2 Transcription Factor; Curcumin; Cyclooxygenase 2 Inhibitors; Denervation; Down-Regulation; Ethanol; Female; Gastric Mucosa; Gastrins; Gene Expression; Heme Oxygenase (Decyclizing); Hypoxia-Inducible Factor 1, alpha Subunit; Indomethacin; Lactones; Male; Nitric Oxide; Nitric Oxide Synthase; Prostaglandins; Pyrazoles; Rats; Rats, Wistar; Regional Blood Flow; RNA, Messenger; Stomach Diseases; Sulfones; Superoxide Dismutase; TRPV Cation Channels; Up-Regulation

2018
Ethanol potentiates heat response in the carotid artery via TRPV1.
    Life sciences, 2017, Nov-01, Volume: 188

    Topics: Animals; Capsaicin; Carotid Arteries; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Hot Temperature; Rabbits; TRPV Cation Channels; Vasoconstriction

2017
Effects of eugenol on respiratory burst generation in newborn rat brainstem-spinal cord preparations.
    Pflugers Archiv : European journal of physiology, 2018, Volume: 470, Issue:2

    Topics: Acetanilides; Action Potentials; Animals; Brain Stem; Capsaicin; Eugenol; GABA-A Receptor Antagonists; Neurons; Purines; Rats; Rats, Wistar; Respiration; Spinal Cord; Transient Receptor Potential Channels

2018
Transient receptor potential vanilloid 1 inhibitors block laparotomy- and opioid-induced infarct size reduction in rats.
    British journal of pharmacology, 2017, Volume: 174, Issue:24

    Topics: Analgesics, Opioid; Animals; Capsaicin; Male; Myocardial Infarction; Pyridines; Rats; Rats, Sprague-Dawley; TRPV Cation Channels

2017
Oxytocin Modulates Nociception as an Agonist of Pain-Sensing TRPV1.
    Cell reports, 2017, Nov-07, Volume: 21, Issue:6

    Topics: Animals; Calcium; Capsaicin; Cells, Cultured; Evoked Potentials; Female; Ganglia, Spinal; HEK293 Cells; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Nociception; Oxytocin; Protein Structure, Quaternary; Receptors, Oxytocin; TRPV Cation Channels

2017
TRPV1 enhances the afferent response to P2X receptor activation in the mouse urinary bladder.
    Scientific reports, 2018, 01-09, Volume: 8, Issue:1

    Topics: Adenosine Triphosphate; Animals; Capsaicin; Cells, Cultured; Ganglia, Spinal; Male; Mice; Mice, Inbred C57BL; Neurons, Afferent; Purinergic P2X Receptor Agonists; Receptors, Purinergic P2X; TRPV Cation Channels; Urinary Bladder; Urothelium

2018
Cannabinoids induce apathetic and impulsive patterns of choice through CB1 receptors and TRPV1 channels.
    Neuropharmacology, 2018, 05-01, Volume: 133

    Topics: Animals; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Cerebral Cortex; Choice Behavior; Dose-Response Relationship, Drug; Impulsive Behavior; Male; Maze Learning; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; TRPV Cation Channels

2018
TRPV1 and the MCP-1/CCR2 Axis Modulate Post-UTI Chronic Pain.
    Scientific reports, 2018, 05-08, Volume: 8, Issue:1

    Topics: Animals; Capsaicin; Chemokine CCL2; Chronic Pain; Disease Models, Animal; Female; Ganglia, Spinal; Gene Expression Regulation; Hyperalgesia; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Pelvic Pain; Receptors, CCR2; Signal Transduction; Toll-Like Receptor 4; TRPV Cation Channels; Urinary Tract Infections; Uropathogenic Escherichia coli

2018
Developmental and behavioral effects in neonatal and adult mice following prenatal activation of endocannabinoid receptors by capsaicin.
    Acta pharmacologica Sinica, 2019, Volume: 40, Issue:3

    Topics: Animals; Behavior, Animal; Benzoxazines; Cannabinoid Receptor Agonists; Capsaicin; Embryonic Development; Female; Injections, Intraperitoneal; Male; Maze Learning; Mice, Inbred BALB C; Morpholines; Naphthalenes; Pregnancy; Prenatal Exposure Delayed Effects; Receptor Cross-Talk; Receptors, Cannabinoid; Rimonabant; TRPV Cation Channels

2019
TRPV1 mediates the anticonvulsant effects of acetaminophen in mice.
    Epilepsy research, 2018, Volume: 145

    Topics: Acetaminophen; Acetanilides; Acrylamides; Animals; Anticonvulsants; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Pentylenetetrazole; Piperidines; Purines; Pyrazoles; Seizures; Time Factors; TRPV Cation Channels

2018
α7 Nicotinic acetylcholine receptor contributes to the alleviation of lung ischemia-reperfusion injury by transient receptor potential vanilloid type 1 stimulation.
    The Journal of surgical research, 2018, Volume: 230

    Topics: Aconitine; alpha7 Nicotinic Acetylcholine Receptor; Animals; Apoptosis; Benzamides; Bridged Bicyclo Compounds; Capsaicin; Disease Models, Animal; Down-Regulation; Humans; Lung; Lung Injury; Male; Mice; Mice, Knockout; Reperfusion Injury; Treatment Outcome; TRPV Cation Channels

2018
Cannabidiol modulates serotonergic transmission and reverses both allodynia and anxiety-like behavior in a model of neuropathic pain.
    Pain, 2019, Volume: 160, Issue:1

    Topics: Action Potentials; Animals; Anxiety; Cannabidiol; Capsaicin; Disease Models, Animal; Exploratory Behavior; Feeding Behavior; Ganglia, Spinal; Hyperalgesia; Lysergic Acid Diethylamide; Male; Maze Learning; Neuralgia; Piperazines; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Swimming

2019
Inhibitions of anandamide transport and FAAH synthesis decrease apoptosis and oxidative stress through inhibition of TRPV1 channel in an in vitro seizure model.
    Molecular and cellular biochemistry, 2019, Volume: 453, Issue:1-2

    Topics: Amidohydrolases; Animals; Apoptosis; Arachidonic Acids; Calcium Signaling; Capsaicin; Cell Line, Tumor; Disease Models, Animal; Endocannabinoids; Hippocampus; Humans; Male; Oxidative Stress; Polyunsaturated Alkamides; Rats; Rats, Wistar; Seizures; TRPV Cation Channels

2019
[6]-Gingerol Induces Amiloride-Sensitive Sodium Absorption in the Rat Colon via the Capsaicin Receptor TRPV1 in Colonic Mucosa.
    Journal of nutritional science and vitaminology, 2018, Volume: 64, Issue:4

    Topics: Amiloride; Animals; Capsaicin; Catechols; Colon; Epithelial Sodium Channel Blockers; Fatty Alcohols; Gastrointestinal Agents; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Membrane Potentials; Membrane Transport Modulators; Muscle, Smooth; Oximes; Rats, Sprague-Dawley; Sodium, Dietary; TRPA1 Cation Channel; TRPV Cation Channels

2018
14,15-epoxyeicosatrienoic acid produced by cytochrome P450s enhances neurite outgrowth of PC12 and rat hippocampal neuronal cells.
    Pharmacology research & perspectives, 2018, Volume: 6, Issue:5

    Topics: 8,11,14-Eicosatrienoic Acid; Animals; Arachidonic Acid; Calcium; Capsaicin; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Embryo, Mammalian; Hippocampus; Neurites; Neuronal Outgrowth; PC12 Cells; Primary Cell Culture; Rats; Rats, Wistar; TRPV Cation Channels

2018
Attenuation of glutamatergic and nitrergic system contributes to the antidepressant-like effect induced by capsazepine in the forced swimming test.
    Behavioural pharmacology, 2019, Volume: 30, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Antidepressive Agents; Apomorphine; Arginine; Capsaicin; Cyclic GMP; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Enzyme Inhibitors; Exploratory Behavior; Glutamic Acid; Male; Microinjections; Nitric Oxide; Nitroprusside; Rats; Receptors, N-Methyl-D-Aspartate; Statistics, Nonparametric; Swimming

2019
Inhibition of Transient Receptor Potential Vanilloid 1 Attenuates Blood-Brain Barrier Disruption after Traumatic Brain Injury in Mice.
    Journal of neurotrauma, 2019, 04-15, Volume: 36, Issue:8

    Topics: Animals; Apoptosis; Blood-Brain Barrier; Brain Injuries, Traumatic; Capsaicin; Endothelial Cells; Male; Mice; Mice, Inbred C57BL; TRPV Cation Channels

2019
TrpV1 receptor activation rescues neuronal function and network gamma oscillations from Aβ-induced impairment in mouse hippocampus in vitro.
    eLife, 2018, 11-12, Volume: 7

    Topics: Action Potentials; Alzheimer Disease; Amyloid beta-Peptides; Animals; CA3 Region, Hippocampal; Capsaicin; Cognition; Electrodes, Implanted; Gamma Rhythm; Gene Expression; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microtomy; Models, Biological; Peptide Fragments; Pyramidal Cells; Recombinant Proteins; Tissue Culture Techniques; TRPV Cation Channels

2018
Troglitazone activates TRPV1 and causes deacetylation of PPARγ in 3T3-L1 cells.
    Biochimica et biophysica acta. Molecular basis of disease, 2019, 02-01, Volume: 1865, Issue:2

    Topics: 3T3-L1 Cells; Acetylation; Adipogenesis; Adipose Tissue; Animals; Bone Morphogenetic Proteins; Capsaicin; CCAAT-Enhancer-Binding Proteins; Diet, High-Fat; Epididymis; Feeding Behavior; Ion Channel Gating; Lipid Metabolism; Male; Mice; PPAR alpha; PPAR gamma; RNA, Messenger; Sirtuin 1; Thermogenesis; Troglitazone; TRPV Cation Channels; Uncoupling Protein 1; Weight Loss

2019
Synthesis and SAR of novel capsazepine analogs with significant anti-cancer effects in multiple cancer types.
    Bioorganic & medicinal chemistry, 2019, 01-01, Volume: 27, Issue:1

    Topics: Animals; Antineoplastic Agents; Capsaicin; Cell Line, Tumor; Cell Proliferation; Female; Humans; Mice, Nude; Molecular Structure; Neoplasms; Structure-Activity Relationship; TRPV Cation Channels; Xenograft Model Antitumor Assays

2019
Effect of Capsaicin and Other Thermo-TRP Agonists on Thermoregulatory Processes in the American Cockroach.
    Molecules (Basel, Switzerland), 2018, Dec-18, Volume: 23, Issue:12

    Topics: Animals; Capsaicin; Cockroaches; Isothiocyanates; Menthol; Temperature; Thymol; TRPV Cation Channels

2018
The investigation of allosteric regulation mechanism of analgesic effect using SD rat taste bud tissue biosensor.
    Biosensors & bioelectronics, 2019, Feb-01, Volume: 126

    Topics: Alginates; Allosteric Regulation; Analgesics; Animals; Arachidonic Acids; Biosensing Techniques; Body Temperature; Capsaicin; Cross-Linking Reagents; Electrochemical Techniques; Endocannabinoids; Fever; Pain; Polyunsaturated Alkamides; Rats, Sprague-Dawley; Starch; Taste Buds; TRPV Cation Channels

2019
Possible involvement of peripheral TRP channels in the hydrogen sulfide-induced hyperalgesia in diabetic rats.
    BMC neuroscience, 2019, Jan-03, Volume: 20, Issue:1

    Topics: Acetanilides; Analgesics; Animals; Capsaicin; Cystathionine beta-Synthase; Diabetes Mellitus, Experimental; Female; Formaldehyde; Hydrogen Sulfide; Hydroxylamine; Hyperalgesia; Imidazoles; Nociception; Purines; Rats, Wistar; Skin; Spinal Nerve Roots; Sulfites; Transient Receptor Potential Channels

2019
Effect of TRPV1 on Activity of Isoforms of Constitutive Nitric Oxide Synthase during Regulation of Bicarbonate Secretion in the Stomach.
    Bulletin of experimental biology and medicine, 2019, Volume: 166, Issue:3

    Topics: Amiloride; Animals; Bicarbonates; Capsaicin; Gastric Mucosa; Gene Expression Regulation; Hydrogen-Ion Concentration; Indazoles; Male; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; Nitroarginine; Osmolar Concentration; Perfusion; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Chloride; Stomach; TRPV Cation Channels; Vagotomy

2019
Accumulation of intramyocyte TRPV1-mediated calcium during heat stress is inhibited by concomitant muscle contractions.
    Journal of applied physiology (Bethesda, Md. : 1985), 2019, 03-01, Volume: 126, Issue:3

    Topics: Animals; Calcium; Capsaicin; Heat Stress Disorders; Heat-Shock Response; Isometric Contraction; Male; Muscle Contraction; Muscle Fibers, Skeletal; Phosphorylation; Rats; Rats, Wistar; TRPV Cation Channels

2019
Molecular and functional insights into Transient Receptor Potential Vanilloid 1 (TRPV1) in bull spermatozoa.
    Theriogenology, 2019, Apr-01, Volume: 128

    Topics: Acrosome Reaction; Animals; Arachidonic Acids; Calcium Channel Blockers; Capsaicin; Cattle; Endocannabinoids; Male; Polyunsaturated Alkamides; Sperm Capacitation; Sperm Motility; Spermatozoa; TRPV Cation Channels

2019
Capsaicin causes robust reduction in glycinergic transmission to rat hypoglossal motor neurons via a TRPV1-independent mechanism.
    Journal of neurophysiology, 2019, 04-01, Volume: 121, Issue:4

    Topics: Animals; Brain Stem; Capsaicin; Female; Glycine; Hypoglossal Nerve; Inhibitory Postsynaptic Potentials; Male; Motor Neurons; Potassium Channels; Rats; Rats, Wistar; TRPV Cation Channels

2019
Baicalein inhibits matrix metalloproteinase 1 expression via activation of TRPV1-Ca-ERK pathway in ultraviolet B-irradiated human dermal fibroblasts.
    Experimental dermatology, 2019, Volume: 28, Issue:5

    Topics: Anthracenes; Antioxidants; Apoptosis; Arachidonate 12-Lipoxygenase; Calcium; Capsaicin; Cytosol; Dermis; Egtazic Acid; Extracellular Signal-Regulated MAP Kinases; Fibroblasts; Flavanones; Humans; Leukotrienes; Matrix Metalloproteinase 1; NF-E2-Related Factor 2; Phosphorylation; Reactive Oxygen Species; Signal Transduction; Skin; Skin Aging; TRPV Cation Channels; Ultraviolet Rays

2019
The novel capsazepine analog, CIDD-99, significantly inhibits oral squamous cell carcinoma in vivo through a TRPV1-independent induction of ER stress, mitochondrial dysfunction, and apoptosis.
    Journal of oral pathology & medicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology, 2019, Volume: 48, Issue:5

    Topics: Animals; Apoptosis; Capsaicin; Carcinoma, Squamous Cell; Cell Line, Tumor; Endoplasmic Reticulum Stress; Female; Humans; Isoquinolines; Male; Mice; Mice, Nude; Mitochondria; Mouth Neoplasms; Rats; Rats, Sprague-Dawley; TRPV Cation Channels; Xenograft Model Antitumor Assays

2019
Involvement of Substance P in the Analgesic Effect of Low-Level Laser Therapy in a Mouse Model of Chronic Widespread Muscle Pain.
    Pain medicine (Malden, Mass.), 2019, 10-01, Volume: 20, Issue:10

    Topics: Acids; Animals; Capsaicin; Chronic Pain; Cnidarian Venoms; Disease Models, Animal; Dose-Response Relationship, Drug; Fibromyalgia; Laser Therapy; Low-Level Light Therapy; Mice; Mice, Inbred C57BL; Mice, Knockout; Musculoskeletal Pain; Protein Precursors; Signal Transduction; Substance P; Tachykinins; TRPV Cation Channels

2019
Analgesic transient receptor potential vanilloid-1-active compounds inhibit native and recombinant T-type calcium channels.
    British journal of pharmacology, 2019, Volume: 176, Issue:13

    Topics: Analgesics; Animals; Calcium Channel Blockers; Calcium Channels, T-Type; Capsaicin; Diterpenes; Ganglia, Spinal; HEK293 Cells; Humans; Neurons; Rats, Sprague-Dawley; TRPV Cation Channels

2019
Dry eye sensitizes cool cells to capsaicin-induced changes in activity via TRPV1.
    Journal of neurophysiology, 2019, 06-01, Volume: 121, Issue:6

    Topics: Animals; Capsaicin; Cornea; Dry Eye Syndromes; Electrophysiological Phenomena; Lacrimal Apparatus; Menthol; Neurons, Afferent; Rats; Sensory System Agents; Trigeminal Ganglion; TRPM Cation Channels; TRPV Cation Channels

2019
Selective Action of N-Arachidonoyl Dopamine on Viability and Proliferation of Stromal Cells from Eutopic and Ectopic Endometrium.
    Bulletin of experimental biology and medicine, 2019, Volume: 167, Issue:1

    Topics: Camphanes; Cannabinoid Receptor Antagonists; Capsaicin; Cell Proliferation; Cell Survival; Dopamine; Endometriosis; Endometrium; Female; Humans; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Stromal Cells

2019
Intrathecal lentivirus-mediated RNA interference targeting nerve growth factor attenuates myocardial ischaemia-reperfusion injury in rat.
    British journal of anaesthesia, 2019, Volume: 123, Issue:4

    Topics: Animals; Arrhythmias, Cardiac; Capsaicin; Cardiotonic Agents; Ganglia, Spinal; Genetic Therapy; Injections, Spinal; Lentivirus; MAP Kinase Signaling System; Myocardial Infarction; Myocardial Reperfusion Injury; Nerve Growth Factor; Patch-Clamp Techniques; PC12 Cells; Rats; Rats, Sprague-Dawley; RNA, Small Interfering; TRPV Cation Channels

2019
Transient receptor potential vanilloid 1 mediates cocaine reinstatement via the D1 dopamine receptor in the nucleus accumbens.
    Journal of psychopharmacology (Oxford, England), 2019, Volume: 33, Issue:12

    Topics: Animals; Behavior, Animal; Benzazepines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Capsaicin; Cocaine; Conditioning, Psychological; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Nucleus Accumbens; Receptors, Dopamine D1; TRPV Cation Channels

2019
The Role of the Activation of the TRPV1 Receptor and of Nitric Oxide in Changes in Endothelial and Cardiac Function and Biomarker Levels in Hypertensive Rats.
    International journal of environmental research and public health, 2019, 09-25, Volume: 16, Issue:19

    Topics: Animals; Biomarkers; Biopterins; Blood Pressure; Capsaicin; Drug Evaluation, Preclinical; Heart; Hypertension; Male; Myocardium; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type III; Oxidative Stress; Proto-Oncogene Proteins c-akt; Rats; Rats, Wistar; TRPV Cation Channels; Vascular Resistance

2019
Cannabidiol increases the nociceptive threshold in a preclinical model of Parkinson's disease.
    Neuropharmacology, 2020, Volume: 163

    Topics: Amidohydrolases; Analgesics; Animals; Benzamides; Brain; Cannabidiol; Capsaicin; Carbamates; Celecoxib; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Nociception; Oxidopamine; Pain; Parkinson Disease; Piperidines; Pyrazoles; Thienamycins

2020
The
    Toxins, 2019, 11-27, Volume: 11, Issue:12

    Topics: Animals; Arthropod Venoms; Behavior, Animal; Calcium Signaling; Capsaicin; Female; Ganglia, Spinal; Larva; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Nociceptors; Pain; Pain Measurement; Sebaceous Glands; TRPV Cation Channels

2019
Ca2+-permeable TRPV1 pain receptor knockout rescues memory deficits and reduces amyloid-β and tau in a mouse model of Alzheimer's disease.
    Human molecular genetics, 2020, 01-15, Volume: 29, Issue:2

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Animals; Calcium; Calcium Channels; Capsaicin; Chelating Agents; Disease Models, Animal; Egtazic Acid; Hippocampus; Learning; Memory Disorders; Mice; Mice, Knockout; Nociceptors; tau Proteins; TRPV Cation Channels

2020
Mechanism underlying the negative inotropic effect in rat left ventricle in hyperthermia: the role of TRPV1.
    The journal of physiological sciences : JPS, 2020, Feb-05, Volume: 70, Issue:1

    Topics: Animals; Capsaicin; Fever; Gene Expression Regulation; Heart Rate; Rats; TRPV Cation Channels; Ventricular Function, Left

2020
Effects of inhalation of sevoflurane at different concentrations on TRPV1 in airways of rats at different developmental stages.
    Life sciences, 2020, May-15, Volume: 249

    Topics: Administration, Inhalation; Age Factors; Anesthetics, Inhalation; Animals; Blood Gas Analysis; Body Weight; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Neurokinin A; Neurokinin B; Rats; Rats, Sprague-Dawley; Respiration; Sevoflurane; Substance P; Trachea; TRPV Cation Channels

2020
Amelioration from the ocular irritant Capsaicin: development and assessment of a Capsazepine
    Expert opinion on drug delivery, 2020, Volume: 17, Issue:6

    Topics: Animals; Capsaicin; Chitosan; Cornea; Female; Gels; Humans; Irritants; Male; Poloxamer; Rabbits; Rats; Rats, Wistar

2020
Role of TRPV1/TRPV3 channels in olanzapine-induced metabolic alteration: Possible involvement in hypothalamic energy-sensing, appetite regulation, inflammation and mesolimbic pathway.
    Toxicology and applied pharmacology, 2020, 09-01, Volume: 402

    Topics: Animals; Appetite Regulation; Capsaicin; Coloring Agents; Energy Metabolism; Female; Furans; Gene Expression Regulation; Glucose Tolerance Test; Hypoglycemic Agents; Hypothalamus; Inflammation; Metformin; Mice; Mice, Inbred BALB C; Motor Activity; Olanzapine; Ruthenium Red; Sensory System Agents; TRPV Cation Channels

2020
Antinociceptive activity of 3β-6β-16β-trihydroxylup-20 (29)-ene triterpene isolated from Combretum leprosum leaves in adult zebrafish (Danio rerio).
    Biochemical and biophysical research communications, 2020, 12-10, Volume: 533, Issue:3

    Topics: Acid Sensing Ion Channels; Amiloride; Analgesics; Animals; Camphor; Capsaicin; Combretum; Dose-Response Relationship, Drug; Female; Ketamine; Locomotion; Male; Methylene Blue; Naloxone; NG-Nitroarginine Methyl Ester; Nociception; Pain; Pain Measurement; Plant Extracts; Plant Leaves; Receptors, N-Methyl-D-Aspartate; Ruthenium Red; Triterpenes; TRPV Cation Channels; Zebrafish; Zebrafish Proteins

2020
Antiallodynic effect of PhAR-DBH-Me involves cannabinoid and TRPV1 receptors.
    Pharmacology research & perspectives, 2020, Volume: 8, Issue:5

    Topics: Animals; Antineoplastic Agents; Arachidonic Acids; Azabicyclo Compounds; Cannabinoid Receptor Antagonists; Capsaicin; Cisplatin; Endocannabinoids; Female; Hyperalgesia; Injections, Intraperitoneal; Ligation; Models, Animal; Neuralgia; Oleic Acids; Polyunsaturated Alkamides; Rats; Rats, Wistar; Spinal Nerves; TRPV Cation Channels; Vagus Nerve Stimulation

2020
Chronic intermittent hypoxia impairs diuretic and natriuretic responses to volume expansion in rats with preserved low-pressure baroreflex control of the kidney.
    American journal of physiology. Renal physiology, 2021, 01-01, Volume: 320, Issue:1

    Topics: Animals; Arterial Pressure; Baroreflex; Blood Volume; Capsaicin; Chronic Disease; Disease Models, Animal; Diuresis; Heart Rate; Hypoxia; Infusions, Intravenous; Kidney; Male; Natriuresis; Rats, Wistar; Saline Solution; Sympathetic Nervous System; Time Factors; TRPV Cation Channels; Urodynamics

2021
Comparison of joint degeneration and pain in male and female mice in DMM model of osteoarthritis.
    Osteoarthritis and cartilage, 2021, Volume: 29, Issue:5

    Topics: Animals; Behavior, Animal; Capsaicin; Cartilage, Articular; Disease Models, Animal; Female; Ganglia, Spinal; Male; Mice, Inbred C57BL; Microscopy, Fluorescence; Osteoarthritis; Pain; Sensory System Agents; Sex Factors; Stifle; TRPV Cation Channels

2021
CB2 cannabinoid receptor agonist selectively inhibits the mechanosensitivity of mucosal afferents in the guinea pig bladder.
    American journal of physiology. Renal physiology, 2021, 05-01, Volume: 320, Issue:5

    Topics: Animals; Arachidonic Acids; Camphanes; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Capsaicin; Endocannabinoids; Female; Guinea Pigs; Ligands; Mechanotransduction, Cellular; Mucous Membrane; Muscle, Smooth; Neurons, Afferent; Pyrazoles; Receptor, Cannabinoid, CB2; TRPV Cation Channels; Urinary Bladder

2021
Inhibitory effect of intrathecally administered AM404, an endocannabinoid reuptake inhibitor, on neuropathic pain in a rat chronic constriction injury model.
    Pharmacological reports : PR, 2021, Volume: 73, Issue:3

    Topics: Animals; Arachidonic Acids; Capsaicin; Constriction; Disease Models, Animal; Endocannabinoids; Hyperalgesia; Indoles; Male; Neuralgia; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rotarod Performance Test; Spinal Cord; TRPV Cation Channels

2021
Capsazepine decreases corneal pain syndrome in severe dry eye disease.
    Journal of neuroinflammation, 2021, May-11, Volume: 18, Issue:1

    Topics: Animals; Capsaicin; Cornea; Dry Eye Syndromes; Male; Mice; Mice, Inbred C57BL; Pain; Syndrome; TRPV Cation Channels

2021
Role of the Transient Receptor Potential Vanilloid Type 1 (TRPV1) in the Regulation of Nitric Oxide Release in Wistar Rat Aorta.
    Oxidative medicine and cellular longevity, 2021, Volume: 2021

    Topics: Animals; Aorta; Biopterins; Capsaicin; Cyclic GMP; Endothelial Cells; Male; Malondialdehyde; Nitric Oxide; Nitric Oxide Synthase Type III; Oxidative Stress; Rats; Rats, Wistar; TRPV Cation Channels

2021
TRPV1 and TRPA1 Channels Are Both Involved Downstream of Histamine-Induced Itch.
    Biomolecules, 2021, 08-06, Volume: 11, Issue:8

    Topics: Acetanilides; Animals; Calcium; Capsaicin; Female; Ganglia, Spinal; Gene Expression; Histamine; Male; Methylhistamines; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Molecular Imaging; Primary Cell Culture; Pruritus; Purines; Ruthenium Red; Sensory Receptor Cells; Signal Transduction; TRPA1 Cation Channel; TRPV Cation Channels

2021
Inhibition of Spinal TRPV1 Reduces NMDA Receptor 2B Phosphorylation and Produces Anti-Nociceptive Effects in Mice with Inflammatory Pain.
    International journal of molecular sciences, 2021, Oct-16, Volume: 22, Issue:20

    Topics: Analgesics; Animals; Capsaicin; Carrageenan; Disease Models, Animal; Glutamic Acid; Hyperalgesia; Inflammation; Male; Mice; Mice, Inbred ICR; Pain; Phosphorylation; Receptors, N-Methyl-D-Aspartate; Spinal Cord; TRPV Cation Channels

2021
Membrane Interactivity of Capsaicin Antagonized by Capsazepine.
    International journal of molecular sciences, 2022, Apr-02, Volume: 23, Issue:7

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Capsaicin; Lipid Bilayers; Membranes

2022
Intrarectal Capsazepine Administration Modulates Colonic Mucosal Health in Mice.
    International journal of molecular sciences, 2022, Aug-24, Volume: 23, Issue:17

    Topics: Animals; Capsaicin; Colon; Inflammatory Bowel Diseases; Mice; Pain; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPV Cation Channels

2022
Bioflavonoid exerts analgesic and anti-inflammatory effects via transient receptor potential 1 channel in a rat model.
    Arquivos de neuro-psiquiatria, 2022, Volume: 80, Issue:9

    Topics: Acute Pain; Analgesics; Animals; Anti-Inflammatory Agents; Capsaicin; Flavonoids; Kaempferols; Rats; Transient Receptor Potential Channels; TRPV Cation Channels

2022
Capsazepine (CPZ) Inhibits TRPC6 Conductance and Is Protective in Adriamycin-Induced Nephropathy and Diabetic Glomerulopathy.
    Cells, 2023, 01-10, Volume: 12, Issue:2

    Topics: Animals; Capsaicin; Diabetes Mellitus; Diabetic Nephropathies; Doxorubicin; Mice; Mice, Knockout; Transient Receptor Potential Channels; TRPC Cation Channels; TRPC6 Cation Channel

2023
Neuroprotective effect of transient receptor potential Vanilloid 1 agonist capsaicin in Alzheimer's disease model induced with okadaic acid.
    International immunopharmacology, 2023, Volume: 118

    Topics: Alzheimer Disease; Animals; Antineoplastic Agents; Capsaicin; Humans; Neuroprotective Agents; Okadaic Acid; Rats; TRPV Cation Channels

2023
L-Carnitine Suppresses Transient Receptor Potential Vanilloid Type 1 Activation in Human Corneal Epithelial Cells.
    International journal of molecular sciences, 2023, Jul-23, Volume: 24, Issue:14

    Topics: Antineoplastic Agents; Calcium; Capsaicin; Carnitine; Epithelial Cells; Humans; TRPV Cation Channels

2023