capsaicin and arvanil

capsaicin has been researched along with arvanil in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (3.03)18.2507
2000's25 (75.76)29.6817
2010's6 (18.18)24.3611
2020's1 (3.03)2.80

Authors

AuthorsStudies
Appendino, G; De Petrocellis, L; Di Marzo, V; Minassi, A; Morello, AS1
Anthes, JC; Correll, CC; Greenfeder, S; Phelps, PT; Umland, S1
Bifulco, M; Bisogno, T; Chuang, H; De Petrocellis, L; Di Marzo, V; Julius, D; Melck, D1
Di Marzo, V; Szallasi, A1
Bisogno, T; Davis, JB; De Petrocellis, L; Di Marzo, V; Pertwee, RG1
Bisogno, T; Breivogel, C; Di Marzo, V; Martin, BR; Melck, D; Patrick, G; Razdan, RK; Szallasi, A; Tao, Q1
Brockie, HC; Craib, SJ; Di Marzo, V; Gibson, TM; Leslie, M; Pashmi, G; Pertwee, RG; Ross, RA1
Bisogno, T; Brandi, I; Dasse, O; Davis, JB; De Petrocellis, L; Di Marzo, V; Jefferson, RG; Mahadevan, A; Martin, BR; Razdan, RK; Winckler, RL1
Bifulco, M; Bisogno, T; De Petrocellis, L; Di Marzo, V; Melck, D; Orlando, P; Vogel, Z; Zagoory, O1
Bisogno, T; Brandi, I; De Petrocellis, L; Di Marzo, V; Grier, MC; Griffin, G; Kulasegram, S; Mahadevan, A; Martin, BR; Razdan, RK; Williams, W1
Baker, D; Bifulco, M; Bisogno, T; Bridges, D; Brooks, JW; Brown, P; Di Marzo, V; Hankey, DJ; Jaggar, SI; Ledent, C; Pryce, G; Rice, AS1
Chiang, HT; Lo, YK; Wu, SN1
Abumrad, NA; Deutsch, DG; Fatade, F; Glaser, ST; Kaczocha, M; Studholme, KM1
Bär, PR; Di Marzo, V; Fezza, F; Maccarrone, M; Nicolay, K; van der Stelt, M; van Zadelhoff, G; Veldhuis, WB; Veldink, GA; Vliegenthart, JF; Wadman, MW1
Appendino, G; de la Vega, L; Di Marzo, V; Macho, A; Munoz, E; Sancho, R1
Aliev, AE; Baker, D; Hiley, R; Hoi, PM; Okuyama, M; Riddall, D; Selwood, DL; Visintin, C1
Anthes, JC; Correll, CC; Phelps, PT1
de Lago, E; Di Marzo, V; Fernández-Ruiz, J; Ramos, JA; Urbani, P1
Andersson, TL; Evilevitch, V; Högestätt, ED; Jönsson, BA; Movahed, P; Wollmer, P; Zygmunt, PM1
Bifulco, M; Bisogno, T; Di Marzo, V; Grimaldi, C; Laezza, C; Lechler, RI; Malfitano, AM; Matarese, G; Pisanti, S1
Cabranes, A; de Lago, E; Di Marzo, V; Fernández-Ruiz, J; Fezza, F; García-Merino, A; Mestre, L; Ramos, JA; Sánchez, A; Valenti, M; Venderova, K1
Appendino, G; Caballero, FJ; De Petrocellis, L; Di Marzo, V; Macho, A; Márquez, N; Minassi, A; Muñoz, E; Schiano-Moriello, A1
Cichewicz, DL; Haller, VL; Welch, SP1
Bifulco, M; De Petrocellis, L; Eletto, D; Gazzerro, P; Husain, S; Laezza, C; Malfitano, AM; Orlando, P; Schwalb, M; Terskiy, A; Toruner, GA; Vitale, E1
Cristino, L; Davison, JS; Di Marzo, V; Guglielmotti, V; Oland, LD; Pittman, QJ; Sharkey, KA; Starowicz, K; Van Sickle, MD1
Kopczyńska, B2
Beattie, RE; Knopp, K; Liu, B; Sher, E; Ursu, D1
Chirasani, SR; Cravatt, BF; Cristino, L; De Petrocellis, L; Di Marzo, V; Dittmar, G; Glass, R; Gurok, U; Imperatore, R; Kettenmann, H; Kumar, J; Lewin, GR; Ligresti, A; Matyash, V; Momma, S; Nuber, UA; Petrosino, S; Purfürst, B; Smith, ES; Stock, K; Synowitz, M; Wälzlein, JH; Wend, P1
Barrière, DA; Blomgren, A; Chapuy, E; Daulhac, L; Eschalier, A; Etienne, M; Högestätt, ED; Libert, F; Mallet, C; Simonsen, C; Zygmunt, PM1
Akers, AT; Brown, KC; Dasgupta, P; Friedman, JR; Hurley, JD; Nolan, NA1
Bartusik-Aebisher, D; Florek-Łuszczki, M; Kołodziejczyk, P; Tutka, P; Wlaź, A; Łuszczki, JJ1
Aldossary, SA; Alsalem, M; Altarifi, A; Azab, B; El-Salem, K; Haddad, M; Jaffal, SM; Kalbouneh, H; Mustafa, AG1

Reviews

1 review(s) available for capsaicin and arvanil

ArticleYear
New perspectives on enigmatic vanilloid receptors.
    Trends in neurosciences, 2000, Volume: 23, Issue:10

    Topics: Animals; Arachidonic Acids; Brain Chemistry; Cannabinoid Receptor Modulators; Capsaicin; Diterpenes; Drug Design; Endocannabinoids; Forecasting; Ganglia, Spinal; Glycerides; Humans; Ligands; Nerve Tissue Proteins; Neurons, Afferent; Polyunsaturated Alkamides; Rats; Receptors, Cannabinoid; Receptors, Drug; Structure-Activity Relationship

2000

Other Studies

32 other study(ies) available for capsaicin and arvanil

ArticleYear
N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor.
    Journal of medicinal chemistry, 2002, Aug-15, Volume: 45, Issue:17

    Topics: Amides; Animals; Binding Sites; Capsaicin; Cell Line; Fatty Acids; Ganglia, Spinal; Humans; In Vitro Techniques; Rats; Receptors, Drug; Terpenes; Vanillic Acid

2002
Cloning and pharmacological characterization of mouse TRPV1.
    Neuroscience letters, 2004, Nov-03, Volume: 370, Issue:1

    Topics: Amino Acid Sequence; Animals; Calcium; Capsaicin; Cell Line; Cloning, Molecular; Cyclic AMP-Dependent Protein Kinases; Diterpenes; Enzyme Activation; Guinea Pigs; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Intracellular Space; Ion Channels; Mice; Phorbol Esters; Phosphorylation; Rabbits; Rats; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; TRPV Cation Channels

2004
Unsaturated long-chain N-acyl-vanillyl-amides (N-AVAMs): vanilloid receptor ligands that inhibit anandamide-facilitated transport and bind to CB1 cannabinoid receptors.
    Biochemical and biophysical research communications, 1999, Aug-19, Volume: 262, Issue:1

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Binding Sites; Biological Transport; Capsaicin; Cell Division; Cell Line; Cell Membrane; Diffusion; Electric Conductivity; Endocannabinoids; Fatty Acids, Unsaturated; Humans; Ligands; Mice; Oocytes; Polyunsaturated Alkamides; Rats; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Xenopus laevis

1999
Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity.
    FEBS letters, 2000, Oct-13, Volume: 483, Issue:1

    Topics: Animals; Arachidonic Acids; Binding, Competitive; Biological Transport; Calcium; Capsaicin; Cell Line; Dose-Response Relationship, Drug; Endocannabinoids; Humans; Ligands; Polyunsaturated Alkamides; Rats; Receptors, Cannabinoid; Receptors, Drug; TRPV Cation Channels; Tumor Cells, Cultured

2000
Neurobehavioral activity in mice of N-vanillyl-arachidonyl-amide.
    European journal of pharmacology, 2000, Oct-20, Volume: 406, Issue:3

    Topics: Analgesics; Animals; Arachidonic Acids; Behavior, Animal; Brain; Cannabinoid Receptor Modulators; Capsaicin; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Endocannabinoids; Glycerides; Male; Mice; Mice, Inbred ICR; Polyunsaturated Alkamides; Receptors, Cannabinoid; Receptors, Drug

2000
Structure-activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens.
    British journal of pharmacology, 2001, Volume: 132, Issue:3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Biological Transport; Calcium; Calcium Channel Blockers; Cannabinoids; Capsaicin; CHO Cells; Cricetinae; Drug Interactions; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Male; Mice; Morpholines; Muscle Contraction; Naphthalenes; Phenylmethylsulfonyl Fluoride; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Radioligand Assay; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Structure-Activity Relationship; Transfection; TRPV Cation Channels; Vas Deferens

2001
Highly selective CB(1) cannabinoid receptor ligands and novel CB(1)/VR(1) vanilloid receptor "hybrid" ligands.
    Biochemical and biophysical research communications, 2001, Feb-23, Volume: 281, Issue:2

    Topics: Animals; Arachidonic Acids; Benzoxazines; Binding, Competitive; Calcium; Capsaicin; Cell Line; Cyclohexanols; Cytosol; Dose-Response Relationship, Drug; Endocannabinoids; Humans; Ligands; Membranes; Morpholines; Naphthalenes; Polyunsaturated Alkamides; Rats; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Structure-Activity Relationship; Tritium; TRPV Cation Channels; Tumor Cells, Cultured

2001
Palmitoylethanolamide inhibits the expression of fatty acid amide hydrolase and enhances the anti-proliferative effect of anandamide in human breast cancer cells.
    The Biochemical journal, 2001, Aug-15, Volume: 358, Issue:Pt 1

    Topics: Amides; Amidohydrolases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Arachidonic Acids; Blotting, Western; Breast Neoplasms; Camphanes; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Cell Division; Colforsin; COS Cells; Cyclic AMP; Dose-Response Relationship, Drug; Endocannabinoids; Ethanolamines; Glycerides; Humans; Hydrolysis; Inhibitory Concentration 50; Palmitic Acids; Polyunsaturated Alkamides; Protein Binding; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; Transfection; Tumor Cells, Cultured

2001
A structure/activity relationship study on arvanil, an endocannabinoid and vanilloid hybrid.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:3

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Behavior, Animal; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Carrier Proteins; Cytosol; Endocannabinoids; Guanosine 5'-O-(3-Thiotriphosphate); Mice; Motor Activity; Pain Measurement; Polyunsaturated Alkamides; Rats; Receptors, Cannabinoid; Receptors, Drug

2002
Arvanil-induced inhibition of spasticity and persistent pain: evidence for therapeutic sites of action different from the vanilloid VR1 receptor and cannabinoid CB(1)/CB(2) receptors.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: Animals; Arachidonic Acids; Benzoxazines; Camphanes; Cannabinoid Receptor Modulators; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Genotype; Mice; Mice, Inbred Strains; Mice, Knockout; Morpholines; Multiple Sclerosis; Muscle Spasticity; Naphthalenes; Pain; Pain Measurement; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

2002
Effect of arvanil (N-arachidonoyl-vanillyl-amine), a nonpungent anandamide-capsaicin hybrid, on ion currents in NG108-15 neuronal cells.
    Biochemical pharmacology, 2003, Feb-15, Volume: 65, Issue:4

    Topics: Action Potentials; Animals; Arachidonic Acids; Calcium Channels, L-Type; Capsaicin; Cell Line; Delayed Rectifier Potassium Channels; Drug Interactions; Endocannabinoids; Glycerol; Hybrid Cells; Mice; Neurons; omega-Conotoxin GVIA; Pertussis Toxin; Polyunsaturated Alkamides; Potassium Channels; Potassium Channels, Voltage-Gated; Rats

2003
Evidence against the presence of an anandamide transporter.
    Proceedings of the National Academy of Sciences of the United States of America, 2003, Apr-01, Volume: 100, Issue:7

    Topics: Arachidonic Acids; Astrocytoma; Biological Transport; Cannabinoids; Capsaicin; Carrier Proteins; Endocannabinoids; Humans; Immunohistochemistry; Kinetics; Neuroblastoma; Polyunsaturated Alkamides; Tumor Cells, Cultured

2003
Neuroprotection by the endogenous cannabinoid anandamide and arvanil against in vivo excitotoxicity in the rat: role of vanilloid receptors and lipoxygenases.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, May-15, Volume: 23, Issue:10

    Topics: Animals; Animals, Newborn; Arachidonic Acids; Blood Cells; Brain; Brain Chemistry; Brain Mapping; Cannabinoid Receptor Modulators; Cannabinoids; Capsaicin; Endocannabinoids; Ethanolamines; Fatty Acids, Unsaturated; Lipoxygenase; Male; Masoprocol; Nerve Degeneration; Neuroprotective Agents; Ouabain; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Drug

2003
The CB1/VR1 agonist arvanil induces apoptosis through an FADD/caspase-8-dependent pathway.
    British journal of pharmacology, 2003, Volume: 140, Issue:6

    Topics: Adaptor Proteins, Signal Transducing; Apoptosis; Capsaicin; Carrier Proteins; Caspase 8; Caspase Inhibitors; Caspases; Cells, Cultured; Cysteine Proteinase Inhibitors; DNA Fragmentation; Dose-Response Relationship, Drug; Fas Ligand Protein; Fas-Associated Death Domain Protein; Humans; In Situ Nick-End Labeling; Jurkat Cells; Membrane Glycoproteins; Models, Biological; Reactive Oxygen Species; Receptor, Cannabinoid, CB1; Receptors, Drug; Signal Transduction; T-Lymphocytes; Time Factors; Transcription, Genetic

2003
Membrane receptor probes: solid-phase synthesis of biotin-Asp-PEG-arvanil derivatives.
    Organic letters, 2005, Apr-28, Volume: 7, Issue:9

    Topics: Aspartic Acid; Biotin; Biotinylation; Capsaicin; Cross-Linking Reagents; Molecular Probes; Molecular Structure; Photoaffinity Labels; Receptors, Cannabinoid

2005
Cloning and functional characterization of dog transient receptor potential vanilloid receptor-1 (TRPV1).
    European journal of pharmacology, 2005, Apr-18, Volume: 513, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Biological Transport; Calcium; Capsaicin; Cell Line; Cloning, Molecular; Diterpenes; DNA, Complementary; Dogs; Dopamine; Dose-Response Relationship, Drug; Fluorometry; Genetic Vectors; Genotype; Humans; Molecular Sequence Data; Mutation, Missense; Phorbol Esters; Phylogeny; Pyrazines; Pyridines; Receptors, Drug; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Transfection

2005
Arvanil, a hybrid endocannabinoid and vanilloid compound, behaves as an antihyperkinetic agent in a rat model of Huntington's disease.
    Brain research, 2005, Jul-19, Volume: 1050, Issue:1-2

    Topics: Animals; Brain Chemistry; Capsaicin; Convulsants; Disease Models, Animal; Dopamine; gamma-Aminobutyric Acid; Glutamic Acid; Huntington Disease; Hyperkinesis; Male; Motor Activity; Nitro Compounds; Propionates; Rats; Rats, Sprague-Dawley

2005
Vascular effects of anandamide and N-acylvanillylamines in the human forearm and skin microcirculation.
    British journal of pharmacology, 2005, Volume: 146, Issue:2

    Topics: Adult; Arachidonic Acids; Benzylamines; Capsaicin; Endocannabinoids; Female; Forearm; Humans; Laser-Doppler Flowmetry; Male; Microcirculation; Middle Aged; Muscle, Skeletal; Plethysmography; Polyunsaturated Alkamides; Regional Blood Flow; Skin; TRPV Cation Channels

2005
Arvanil inhibits T lymphocyte activation and ameliorates autoimmune encephalomyelitis.
    Journal of neuroimmunology, 2006, Volume: 171, Issue:1-2

    Topics: Animals; Arachidonic Acids; Blotting, Western; Body Weight; Cannabinoid Receptor Modulators; Capsaicin; CD4-Positive T-Lymphocytes; Cell Line; Cell Proliferation; Cytokines; Disease Models, Animal; Dose-Response Relationship, Drug; Dose-Response Relationship, Immunologic; Drug Interactions; Encephalomyelitis, Autoimmune, Experimental; Endocannabinoids; Enzyme Activation; Female; Flow Cytometry; Humans; Leukocytes, Mononuclear; Lymphocyte Activation; Mice; Myelin Proteolipid Protein; Peptide Fragments; Polyunsaturated Alkamides; Proto-Oncogene Proteins c-akt; Statistics, Nonparametric; Time Factors

2006
Decreased endocannabinoid levels in the brain and beneficial effects of agents activating cannabinoid and/or vanilloid receptors in a rat model of multiple sclerosis.
    Neurobiology of disease, 2005, Volume: 20, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Arachidonic Acids; Basal Ganglia; Brain; Cannabinoid Receptor Modulators; Capsaicin; Cyclic Nucleotide Phosphodiesterases, Type 4; Disease Models, Animal; Encephalomyelitis, Autoimmune, Experimental; Endocannabinoids; Gene Expression; Glycerides; Male; Multiple Sclerosis; Phosphodiesterase Inhibitors; Polyunsaturated Alkamides; Rats; Rats, Inbred Lew; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Rolipram; TRPV Cation Channels

2005
Iodinated N-acylvanillamines: potential "multiple-target" anti-inflammatory agents acting via the inhibition of t-cell activation and antagonism at vanilloid TRPV1 channels.
    Molecular pharmacology, 2006, Volume: 69, Issue:4

    Topics: Amines; Capsaicin; Cell Cycle; Cell Proliferation; Humans; In Situ Nick-End Labeling; Interleukin-2; Iodine; Jurkat Cells; Lymphocyte Activation; NF-kappa B; Plasmids; Promoter Regions, Genetic; T-Lymphocytes; TRPV Cation Channels

2006
Non-cannabinoid CB1, non-cannabinoid CB2 antinociceptive effects of several novel compounds in the PPQ stretch test in mice.
    European journal of pharmacology, 2006, Sep-28, Volume: 546, Issue:1-3

    Topics: Acetaminophen; Amides; Analgesics; Animals; Arachidonic Acids; Benzamides; Benzoquinones; Camphanes; Capsaicin; Carbamates; Dose-Response Relationship, Drug; Dronabinol; Endocannabinoids; Ethanolamines; Hyperalgesia; Male; Mesencephalon; Mice; Mice, Inbred ICR; Narcotic Antagonists; Pain; Palmitic Acids; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid; Rimonabant; Spinal Cord; TRPV Cation Channels

2006
Arvanil and anandamide up-regulate CD36 expression in human peripheral blood mononuclear cells.
    Immunology letters, 2007, Apr-15, Volume: 109, Issue:2

    Topics: Arachidonic Acids; Capsaicin; CD28 Antigens; CD3 Complex; CD36 Antigens; Endocannabinoids; Humans; Leukocytes, Mononuclear; Lymphocyte Activation; Oligonucleotide Array Sequence Analysis; Polyunsaturated Alkamides; Up-Regulation

2007
Arvanil, anandamide and N-arachidonoyl-dopamine (NADA) inhibit emesis through cannabinoid CB1 and vanilloid TRPV1 receptors in the ferret.
    The European journal of neuroscience, 2007, Volume: 25, Issue:9

    Topics: Acrylamides; Animals; Antiemetics; Arachidonic Acids; Area Postrema; Autonomic Pathways; Brain Stem; Bridged Bicyclo Compounds, Heterocyclic; Cannabinoids; Capsaicin; Dopamine; Emetics; Endocannabinoids; Ferrets; Male; Mice; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptor, Cannabinoid, CB1; Solitary Nucleus; TRPV Cation Channels; Vagus Nerve; Vomiting

2007
Role of VR1 and CB1 receptors in modelling of cardio-respiratory response to arvanil, an endocannabinoid and vanilloid hybrid, in rats.
    Life sciences, 2008, Jul-18, Volume: 83, Issue:3-4

    Topics: Anilides; Animals; Blood Pressure; Cannabinoid Receptor Modulators; Capsaicin; Cinnamates; Disease Models, Animal; Endocannabinoids; Hypertension; Injections, Intravenous; Male; Morpholines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Respiration; Respiration Disorders; Ruthenium Red; Tidal Volume; TRPV Cation Channels

2008
Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicity.
    European journal of pharmacology, 2010, Sep-01, Volume: 641, Issue:2-3

    Topics: Action Potentials; Alkaloids; Animals; Benzodioxoles; Capsaicin; Diterpenes; Ganglia, Spinal; Kinetics; Lipid Metabolism; Male; Neurons, Afferent; Pain; Patch-Clamp Techniques; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Sensory Receptor Cells; Solubility; TRPV Cation Channels; Urea

2010
Midcervical vagotomy precludes respiratory response to novel anti-inflammatory and anti-tumour drug arvanil in rats.
    European journal of pharmacology, 2010, Sep-15, Volume: 643, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Anticarcinogenic Agents; Blood Pressure; Capsaicin; Dose-Response Relationship, Drug; Injections, Intravenous; Male; Rats; Rats, Wistar; Respiratory Mechanics; Respiratory Physiological Phenomena; Tidal Volume; Vagotomy; Vagus Nerve

2010
Neural precursor cells induce cell death of high-grade astrocytomas through stimulation of TRPV1.
    Nature medicine, 2012, Volume: 18, Issue:8

    Topics: Aging; Amides; Amidohydrolases; Animals; Antineoplastic Agents; Apoptosis; Arachidonic Acids; Brain; Brain Neoplasms; Capsaicin; Cell Movement; Culture Media, Conditioned; Dopamine; Endocannabinoids; Ethanolamines; Female; Gene Expression Regulation, Neoplastic; Glioblastoma; Humans; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, SCID; Neoplasm Proteins; Neural Stem Cells; Oleic Acids; Palmitic Acids; Polyunsaturated Alkamides; Real-Time Polymerase Chain Reaction; RNA, Small Interfering; TRPV Cation Channels; Tumor Cells, Cultured

2012
Fatty acid amide hydrolase-dependent generation of antinociceptive drug metabolites acting on TRPV1 in the brain.
    PloS one, 2013, Volume: 8, Issue:8

    Topics: Amidohydrolases; Aminophenols; Analgesics; Animals; Arachidonic Acids; Benzylamines; Brain; Capsaicin; Inhibitory Concentration 50; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nociception; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; TRPV Cation Channels; Vasodilation

2013
Non-pungent long chain capsaicin-analogs arvanil and olvanil display better anti-invasive activity than capsaicin in human small cell lung cancers.
    Cell adhesion & migration, 2017, 01-02, Volume: 11, Issue:1

    Topics: Adenylate Kinase; Animals; Capsaicin; Cell Line, Tumor; Humans; Lung Neoplasms; Neoplasm Invasiveness; Receptor, Cannabinoid, CB1; Signal Transduction; Small Cell Lung Carcinoma; Time Factors; TRPV Cation Channels

2017
Arvanil, olvanil, AM 1172 and LY 2183240 (various cannabinoid CB1 receptor agonists) increase the threshold for maximal electroshock-induced seizures in mice.
    Pharmacological reports : PR, 2018, Volume: 70, Issue:1

    Topics: Animals; Arachidonic Acids; Benzamides; Brain; Brain Waves; Cannabinoid Receptor Agonists; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Heterocyclic Compounds, 1-Ring; Male; Mice; Receptor, Cannabinoid, CB1; Seizures; Signal Transduction; Urea

2018
The desensitization of the transient receptor potential vanilloid 1 by nonpungent agonists and its resensitization by bradykinin.
    Neuroreport, 2020, 08-05, Volume: 31, Issue:11

    Topics: Animals; Bradykinin; Capsaicin; Hyperalgesia; Male; Mice; Mice, Inbred BALB C; Nociception; Receptors, Prostaglandin E, EP3 Subtype; Receptors, Prostaglandin E, EP4 Subtype; Sensory System Agents; TRPV Cation Channels

2020