Page last updated: 2024-09-03

caprylates and bisindolylmaleimide i

caprylates has been researched along with bisindolylmaleimide i in 3 studies

Compound Research Comparison

Studies
(caprylates)
Trials
(caprylates)
Recent Studies (post-2010)
(caprylates)
Studies
(bisindolylmaleimide i)
Trials
(bisindolylmaleimide i)
Recent Studies (post-2010) (bisindolylmaleimide i)
5,0611002,3391,1981174

Protein Interaction Comparison

ProteinTaxonomycaprylates (IC50)bisindolylmaleimide i (IC50)
Chain A, Protein kinase C, iotaHomo sapiens (human)5.8
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)9
G2/mitotic-specific cyclin-B2Homo sapiens (human)2.3
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.5
Protein kinase C gamma typeHomo sapiens (human)0.03
Protein kinase C beta typeHomo sapiens (human)0.0054
Cyclin-dependent kinase 1Homo sapiens (human)2.3
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.068
Cyclin-dependent kinase 4Homo sapiens (human)0.99
G2/mitotic-specific cyclin-B1Homo sapiens (human)2.3
Lethal factorBacillus anthracis1.5
Protein kinase C alpha typeHomo sapiens (human)0.0055
Glycogen synthase kinase-3 betaRattus norvegicus (Norway rat)0.36
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoformOryctolagus cuniculus (rabbit)0.7
G1/S-specific cyclin-D1Homo sapiens (human)0.99
Protein kinase C eta typeHomo sapiens (human)0.0066
G1/S-specific cyclin-E1Homo sapiens (human)0.99
Cyclin-dependent kinase 2Homo sapiens (human)0.99
cAMP-dependent protein kinase catalytic subunit alpha Rattus norvegicus (Norway rat)2
Protein kinase C iota typeHomo sapiens (human)3.463
Glycogen synthase kinase-3 betaHomo sapiens (human)0.19
Protein kinase C epsilon typeHomo sapiens (human)0.0067
Protein kinase C theta typeHomo sapiens (human)0.0061
Protein kinase C zeta typeHomo sapiens (human)5.8
Protein kinase C delta typeHomo sapiens (human)0.0096
Peroxisome proliferator-activated receptor alphaHomo sapiens (human)0.006
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)7.3
G2/mitotic-specific cyclin-B3Homo sapiens (human)2.3
Serine/threonine-protein kinase LMTK3Homo sapiens (human)0.0001

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujikawa, H; Kanno, T; Nagata, T; Nishizaki, T; Tanaka, A; Yaguchi, T; Yamamoto, H; Yamamoto, S1
Kanno, T; Nishizaki, T; Tanaka, A1
Nishizaki, T1

Other Studies

3 other study(ies) available for caprylates and bisindolylmaleimide i

ArticleYear
8-[2-(2-pentyl-cyclopropylmethyl)-cyclopropyl]-octanoic acid stimulates GABA release from interneurons projecting to CA1 pyramidal neurons in the rat hippocampus via pre-synaptic alpha7 acetylcholine receptors.
    Journal of neurochemistry, 2005, Volume: 95, Issue:3

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Caprylates; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Indoles; Interneurons; Male; Maleimides; Membrane Potentials; Neural Pathways; Oocytes; Organ Culture Techniques; Patch-Clamp Techniques; Presynaptic Terminals; Protein Kinase C; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Nicotinic; Xenopus

2005
Linoleic acid derivative DCP-LA stimulates vesicular transport of α7 ACh receptors towards surface membrane.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2012, Volume: 30, Issue:1

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Caprylates; Cell Membrane; Female; Hippocampus; In Vitro Techniques; Indoles; Male; Maleimides; Membrane Potentials; Protein Kinase C; Protein Transport; Rats; Rats, Wistar; Receptors, Nicotinic; Synaptosomes; Transport Vesicles; Xenopus laevis

2012
PKCε Increases Extracellular Elastin and Fibulin-5/DANCE in Dermal Fibroblasts.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2018, Volume: 46, Issue:1

    Topics: Caprylates; Cells, Cultured; Dermis; Elastin; Extracellular Matrix Proteins; Fibroblasts; Humans; Immunoassay; Indoles; Maleimides; Matrix Metalloproteinase 9; Matrix Metalloproteinase Inhibitors; Protein Kinase C-epsilon; Ribosomal Protein S6 Kinases, 70-kDa; RNA Interference; RNA, Small Interfering; TOR Serine-Threonine Kinases; Tropoelastin; Up-Regulation

2018