Page last updated: 2024-09-04

canertinib dihydrochloride and ruboxistaurin

canertinib dihydrochloride has been researched along with ruboxistaurin in 1 studies

Compound Research Comparison

Studies
(canertinib dihydrochloride)
Trials
(canertinib dihydrochloride)
Recent Studies (post-2010)
(canertinib dihydrochloride)
Studies
(ruboxistaurin)
Trials
(ruboxistaurin)
Recent Studies (post-2010) (ruboxistaurin)
311362032956

Protein Interaction Comparison

ProteinTaxonomycanertinib dihydrochloride (IC50)ruboxistaurin (IC50)
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)0.6484
Protein kinase C gamma typeHomo sapiens (human)0.3
Protein kinase C alpha typeRattus norvegicus (Norway rat)0.32
Protein kinase C beta typeHomo sapiens (human)0.0054
Protein kinase C delta typeRattus norvegicus (Norway rat)0.32
Protein kinase C epsilon typeRattus norvegicus (Norway rat)0.32
Protein kinase C zeta typeRattus norvegicus (Norway rat)0.32
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.2
Protein kinase C alpha typeHomo sapiens (human)0.36
Protein kinase C eta typeHomo sapiens (human)0.052
Protein kinase C gamma typeRattus norvegicus (Norway rat)0.32
Protein kinase C beta typeRattus norvegicus (Norway rat)0.32
Protein kinase C epsilon typeHomo sapiens (human)0.6
Protein kinase C delta typeHomo sapiens (human)0.25
Protein kinase C eta typeRattus norvegicus (Norway rat)0.32
Homeodomain-interacting protein kinase 1Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 4Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 2Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 3Homo sapiens (human)0.1
Protein kinase C theta typeRattus norvegicus (Norway rat)0.32

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Russu, WA; Shallal, HM1

Other Studies

1 other study(ies) available for canertinib dihydrochloride and ruboxistaurin

ArticleYear
Discovery, synthesis, and investigation of the antitumor activity of novel piperazinylpyrimidine derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:6

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Molecular Structure; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; Stereoisomerism; Structure-Activity Relationship

2011