Page last updated: 2024-09-04

canertinib dihydrochloride and pd168393

canertinib dihydrochloride has been researched along with pd168393 in 1 studies

Compound Research Comparison

Studies
(canertinib dihydrochloride)
Trials
(canertinib dihydrochloride)
Recent Studies (post-2010)
(canertinib dihydrochloride)
Studies
(pd168393)
Trials
(pd168393)
Recent Studies (post-2010) (pd168393)
3113661033

Protein Interaction Comparison

ProteinTaxonomycanertinib dihydrochloride (IC50)pd168393 (IC50)
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)1.0702
Epidermal growth factor receptorHomo sapiens (human)0.0143
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.0334
Tyrosine-protein kinase FynHomo sapiens (human)0.1543
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.073
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)0.0011
Tyrosine-protein kinase BlkHomo sapiens (human)5.47
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)0.5757
Tyrosine-protein kinase JAK3Homo sapiens (human)3.14
Tyrosine-protein kinase BTKHomo sapiens (human)5.83
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)0.0047

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bridges, AJ; Denny, WA; Elliott, WL; Fry, DW; McNamara, DJ; Nelson, JM; Roberts, BJ; Sherwood, V; Showalter, HD; Smaill, JB; Vincent, PW; Zhou, H1

Other Studies

1 other study(ies) available for canertinib dihydrochloride and pd168393

ArticleYear
Tyrosine kinase inhibitors. 18. 6-Substituted 4-anilinoquinazolines and 4-anilinopyrido[3,4-d]pyrimidines as soluble, irreversible inhibitors of the epidermal growth factor receptor.
    Journal of medicinal chemistry, 2001, Feb-01, Volume: 44, Issue:3

    Topics: Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; Enzyme Inhibitors; ErbB Receptors; Inhibitory Concentration 50; Mice; Phosphorylation; Pyrimidines; Quinazolines; Solubility; Structure-Activity Relationship; Transplantation, Heterologous; Tumor Cells, Cultured

2001