Page last updated: 2024-09-04

canertinib dihydrochloride and mln8054

canertinib dihydrochloride has been researched along with mln8054 in 1 studies

Compound Research Comparison

Studies
(canertinib dihydrochloride)
Trials
(canertinib dihydrochloride)
Recent Studies (post-2010)
(canertinib dihydrochloride)
Studies
(mln8054)
Trials
(mln8054)
Recent Studies (post-2010) (mln8054)
3113661342

Protein Interaction Comparison

ProteinTaxonomycanertinib dihydrochloride (IC50)mln8054 (IC50)
Aurora kinase AHomo sapiens (human)0.0398
Aurora kinase BMus musculus (house mouse)0.172
Tyrosine-protein kinase LckHomo sapiens (human)3.2
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.33
Platelet-derived growth factor receptor alphaHomo sapiens (human)0.7943
Aurora kinase AMus musculus (house mouse)0.0085
Aurora kinase BHomo sapiens (human)1.6916
Aurora kinase CHomo sapiens (human)0.0118

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Russu, WA; Shallal, HM1

Other Studies

1 other study(ies) available for canertinib dihydrochloride and mln8054

ArticleYear
Discovery, synthesis, and investigation of the antitumor activity of novel piperazinylpyrimidine derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:6

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Molecular Structure; Piperazines; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; Stereoisomerism; Structure-Activity Relationship

2011