Page last updated: 2024-09-04

canertinib and lapatinib ditosylate

canertinib has been researched along with lapatinib ditosylate in 1 studies

Compound Research Comparison

Studies
(canertinib)
Trials
(canertinib)
Recent Studies (post-2010)
(canertinib)
Studies
(lapatinib ditosylate)
Trials
(lapatinib ditosylate)
Recent Studies (post-2010) (lapatinib ditosylate)
124965704

Protein Interaction Comparison

ProteinTaxonomycanertinib (IC50)lapatinib ditosylate (IC50)
Epidermal growth factor receptorHomo sapiens (human)0.0302
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.0242
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)0.0163

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alberti, JG; Alligood, KJ; Caferro, TR; Chamberlain, SD; Dickerson, SH; Dickson, HD; Emerson, HK; Gerding, RM; Griffin, RJ; Hubbard, RD; Keith, BR; Mullin, RJ; Petrov, KG; Reno, MJ; Rheault, TR; Rusnak, DW; Sammond, DM; Smith, SC; Stevens, KL; Uehling, DE; Waterson, AG; Wood, ER1

Other Studies

1 other study(ies) available for canertinib and lapatinib ditosylate

ArticleYear
Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2-d]pyrimidines as EGFR and ErbB-2 inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Jan-01, Volume: 19, Issue:1

    Topics: Administration, Oral; Animals; Antineoplastic Agents; ErbB Receptors; Mice; Pharmacokinetics; Pyrimidines; Pyrrolidines; Receptor, ErbB-2; Structure-Activity Relationship

2009