Page last updated: 2024-09-03

candoxatril and enalapril

candoxatril has been researched along with enalapril in 4 studies

Compound Research Comparison

Studies
(candoxatril)
Trials
(candoxatril)
Recent Studies (post-2010)
(candoxatril)
Studies
(enalapril)
Trials
(enalapril)
Recent Studies (post-2010) (enalapril)
622956,3111,924859

Protein Interaction Comparison

ProteinTaxonomycandoxatril (IC50)enalapril (IC50)
Angiotensin-converting enzyme Homo sapiens (human)0.3536
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)2.7083
Type-2 angiotensin II receptorRattus norvegicus (Norway rat)1.2
Angiotensin-converting enzymeRattus norvegicus (Norway rat)0.14
Angiotensin-converting enzyme 2 Homo sapiens (human)0.14

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ikuse, T; Kuro, T; Matsumura, Y; Nose, M; Okahara, A1
Jakovski, K; Jovanoska, E; Kostova, E; Maleska, V; Slaninka-Miceska, M; Zafirov, D1
Coppey, LJ; Dake, B; Davidson, EP; Kleinschmidt, TL; Oltman, CL; Yorek, MA1
Eizenberg, Y; Grossman, E; Peleg, E; Shabtai, Z; Sharabi, Y1

Other Studies

4 other study(ies) available for candoxatril and enalapril

ArticleYear
Effects of SA7060, a novel dual inhibitor of neutral endopeptidase and angiotensin-converting enzyme, on deoxycorticosterone acetate-salt-induced hypertension in rats.
    Biological & pharmaceutical bulletin, 2000, Volume: 23, Issue:7

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta; Blood Pressure; Body Weight; Cardiomegaly; Desoxycorticosterone; Enalapril; Heart; Hypertension; Hypertrophy; Indans; Kidney; Kidney Function Tests; Male; Naphthalenes; Neprilysin; Organ Size; Peptidyl-Dipeptidase A; Propionates; Rats; Rats, Sprague-Dawley; Urea

2000
Dual inhibition of angiotensin converting enzyme and neutral endopeptidase produces effective blood pressure control in spontaneously hypertensive rats.
    Bratislavske lekarske listy, 2005, Volume: 106, Issue:12

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Atrial Natriuretic Factor; Blood Pressure; Drug Combinations; Enalapril; Hypertension; Indans; Male; Neprilysin; Propionates; Pyridines; Rats; Rats, Inbred SHR; Thiazepines

2005
Role of the effect of inhibition of neutral endopeptidase on vascular and neural complications in streptozotocin-induced diabetic rats.
    European journal of pharmacology, 2011, Jan-15, Volume: 650, Issue:2-3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Diabetic Neuropathies; Enalapril; Heterocyclic Compounds, 3-Ring; Indans; Male; Neprilysin; Neural Conduction; Propionates; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Streptozocin

2011
Neutral endopeptidase inhibitor versus angiotensin converting enzyme inhibitor in a rat model of the metabolic syndrome.
    Journal of the American Society of Hypertension : JASH, 2014, Volume: 8, Issue:4

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Disease Models, Animal; Enalapril; Indans; Insulin; Male; Metabolic Syndrome; Propionates; Rats; Rats, Sprague-Dawley; Triglycerides

2014