calmidazolium has been researched along with trifluoperazine in 138 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 66 (47.83) | 18.7374 |
1990's | 52 (37.68) | 18.2507 |
2000's | 16 (11.59) | 29.6817 |
2010's | 3 (2.17) | 24.3611 |
2020's | 1 (0.72) | 2.80 |
Authors | Studies |
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Mio, M; Tasaka, K; Yoshida, T | 1 |
Silver, PJ; Stout, MA | 1 |
Corvol, P; Della Bruna, R; Kurtz, A; Pinet, F | 1 |
Blank, JA; Waite, LC | 1 |
Wagner, PD; Wu, YN | 1 |
Chafouleas, JG; Gehm, BD; Laquerre, S; McConnell, DG; Pepperl, DJ; Pinke, RM; Schultz, DA | 1 |
Ito, A; Kishima, K; Kuno, T; Mukai, H; Tanaka, C | 1 |
Ichikawa, M; Matsumoto, G; Urayama, M | 1 |
Abrams, TW; Kandel, ER; Karl, KA | 1 |
Frizzell, RA; Worrell, RT | 1 |
Murad, F; Schmidt, HH | 1 |
Bernardes, CF; Docampo, R; Hoffmann, ME; Vercesi, AE | 1 |
Geguchadze, RN; Gusev, NB | 1 |
Henshaw, EC; Kumar, RV; Panniers, R; Wolfman, A | 1 |
Johnson, AL; Levorse, JM; Tilly, JL | 1 |
Aprille, JR; Dransfield, DT; Nosek, MT | 1 |
Goodman, HM; Schwartz, Y | 1 |
Geguchadze, RN; Gusev, NB; Krylatov, AV | 1 |
Benaim, G; de Meis, L | 1 |
Girsch, SJ; Peracchia, C | 1 |
Grosman, N | 1 |
Jørgensen, PL; Karlish, SJ; Klaerke, DA | 1 |
Matsumura, Y; Morimoto, S; Sasaki, Y; Shinyama, H; Uriu, T | 1 |
Kleis-San Francisco, S; Schuetz, AW | 1 |
Loretz, CA | 1 |
Isenberg, G; Klöckner, U | 1 |
Suko, J; Wyskovsky, W | 1 |
Dasarathy, Y; Fanburg, BL | 1 |
Lugnier, C; Schaeffer, P; Stoclet, JC | 1 |
Ambudkar, IS; Baum, BJ; Horn, VJ | 1 |
Gadd, GM; Sabie, FT | 1 |
Brumley, LM; Wallace, RW | 1 |
Koch, P; Leidig, A; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wilhelm, D | 1 |
Bright, EC; Colombani, PM; Hess, AD; Wells, M | 1 |
Rossi, NF; Schrier, RW | 1 |
Honn, KV; Nelson, KK; Onoda, JM; Taylor, JD | 1 |
Sobieszek, A | 1 |
Combest, WL; Gilbert, LI; Meller, VH; Smith, WA | 1 |
Aitken, RJ; Clarkson, JS; Henderson, CJ; Hulme, MJ | 1 |
Doroshenko, PA; Kostyuk, PG; Luk'yanetz, EA | 1 |
De Meis, L; Gómez Puyou, A; Tuena de Gómez Puyou, M | 1 |
Bright, EC; Colombani, PM; Hess, AD; Monastyrskyj, O | 1 |
Monteforte, PB; Silver, PJ | 1 |
Hait, WN; Lee, GL | 1 |
Durkin, JP; Whitfield, JF | 1 |
Tallant, EA; Wallace, RW | 1 |
Malik, KU; Weis, MT | 1 |
Cooke, BA; Sullivan, MH | 2 |
Carr, BR; Mason, JI; Rainey, WE | 1 |
Kramar, D; Olson, DM; Smieja, Z | 1 |
Celada, A; Schreiber, RD | 1 |
Gerritsen, ME; Nganele, DM; Rodrigues, AM | 1 |
Ahlijanian, MK; Cooper, DM | 1 |
Lucchesi, PA; Scheid, CR | 1 |
Amoss, MS; Kile, JP | 1 |
Breitbart, H; Rubinstein, S | 1 |
Block, GD; Khalsa, SB | 1 |
Busse, R; Lückhoff, A; Mülsch, A; Pohl, U; Winter, I | 1 |
Lydan, MA; O'Day, DH | 1 |
Little, DK; Moreland, RS; Moreland, S | 1 |
Divo, AA; Geary, TG; Jensen, JB | 1 |
Brostrom, CO; Brostrom, MA; Wolfe, SE | 1 |
Meissner, G | 1 |
Danks, JA; Larkins, RG; Prince, RL; Shaw, M; Taft, JL | 1 |
Connolly, JA; Tai, HH | 1 |
Cooper, CL; Malik, KU; Shaffer, JE | 1 |
Anelli, G; Berruti, G; Camatini, M | 1 |
Borsa, J; Einspenner, M; Hickie, RA; Sargent, MD | 1 |
Bell, PD | 1 |
Barr, R; Craig, TA; Crane, FL; Stone, B | 1 |
DeRiemer, SA; Kaczmarek, LK; Schweitzer, B | 1 |
Jarvis, B; Louis, CF; Turnquist, J | 1 |
Van Belle, H | 1 |
Adunyah, ES; Carafoli, E; Niggli, V | 1 |
Ashraf, M; Peterson, RN; Russell, LD | 1 |
Anderson, KW; Coll, RJ; Murphy, AJ | 1 |
Bader, H; Gietzen, K; Sadorf, I | 1 |
Nakatani, HY | 1 |
Wolberg, G; Zimmerman, TP | 1 |
Hofmann, F; Zimmer, M | 1 |
Crane, FL; Morré, DJ; Sun, IL | 1 |
Collard, KJ; Leung, MT | 1 |
Nicholls, D; Snelling, R | 1 |
Johnson, JD; Wittenauer, LA | 1 |
Kimura, J | 1 |
Barrington, M; Majewski, H | 1 |
Gukovskaya, AS; Pandol, SJ | 1 |
Docampo, R | 1 |
Cooperstein, SJ; Watkins, DT | 2 |
Lefevre, F; Philippot, J; Rouot, B; Sainte-Marie, J; Vidal, M | 1 |
Alling, C; Larsson, C | 1 |
Goko, H; Matsuoka, A | 1 |
Biondi, C; Buzzi, M; Ferretti, ME; Pareschi, MC | 1 |
Carter, C; Nicolas, C | 1 |
Iqbal, Z; Sze, PY | 1 |
Müller, TH; Swandulla, D; Zeilhofer, HU | 1 |
Shiraishi, N; Waalkes, MP | 1 |
Duncan, G; Gandolfi, SA; Sanderson, J | 1 |
Cotter, DA; Lydan, MA; O'Day, DH | 1 |
Barlow, JW; Kolliniatis, E; Scholz, GH; Stockigt, JR; Topliss, DJ | 1 |
Abe, K; Higo, K; Matsuki, N; Nakazawa, K; Saito, H; Tanaka, Y | 1 |
Barbieri, MA; Bertini, F; Isola, EL; Lammel, EM; Wilkowsky, SE | 1 |
Maher, P; Oliver, I; Sinclair, W; Trewavas, A | 1 |
De Graan, PN; De Wit, M; Gispen, WH; Hens, JJ; Marquart, A; Oestreicher, AB | 1 |
Cinotti, GA; Menè, P; Pugliese, F | 1 |
Fukushima, T; Hamada, T; Ono, M; Shibata, S; Shimazoe, T; Watanabe, A; Watanabe, S | 1 |
Droogmans, G; Eggermont, J; Nilius, B; Prenen, J; Van den Bremt, K; Voets, T | 1 |
Balossier, G; Bonhomme, A; Bonhomme, P; Bouchot, A; Burlet, H; Klein, C; Pezzella, N; Pingret, L; Pinon, JM | 1 |
Fusetani, N; Matsumura, K; Nagano, M; Saikawa, W; Tachibana, A; Yamamoto, H | 1 |
Moreland, RS; Rokolya, A; Singer, HA; Walsh, MP | 1 |
Ma, TY; McCloud, E; Ortiz, A; Said, HM | 1 |
Daniel, H; Diehl, D; Herget, M; Kuntz, S; Wenzel, U | 1 |
Chen, J; Hoffman, BB; Hu, ZW; Lin, R | 1 |
Banerjee, C; Bhaduri, A; Sarkar, D | 1 |
Gadea, A; López-Colomé, AM | 1 |
Braiman, A; Gheber, L; Priel, Z; Zagoory, O | 1 |
Goudeau, H; Goudeau, M | 1 |
Dyer, JL; Khan, SZ; Michelangeli, F | 1 |
Sampaio-Maia, B; Soares-Da-Silva, P | 1 |
Gauthier, ML; O'Day, DH | 1 |
Evans, ML; Hasenstein, KH; Stinemetz, CL; Young, LM | 1 |
del Carmen Boyano-Adánez, M; Gustavsson, L | 1 |
Del Carlo, B; Pellegrini, M; Pellegrino, M | 1 |
Fraga, S; Sampaio-Maia, B; Serrão, MP; Soares-da-Silva, P | 1 |
Boulay, G | 1 |
Dohovics, R; Hermann, A; Janáky, R; Oja, SS; Saransaari, P; Varga, V | 1 |
Amorim Jesuino, RS; Daher, BS; de Carvalho, MJ; de Freitas, SM; Felipe, MS; Silva-Pereira, I; Soares, CM | 1 |
Azarashvily, TS; Odinokova, IV; Saris, NE; Teplova, VV | 1 |
Bootman, MD; Collins, TJ; Holmes, AM; McDonald, F; Peppiatt, CM; Roderick, HL; Seo, JT | 1 |
Bang, H; Han, ES; Han, YS; Lee, CS | 1 |
Bellamy, TC; Garthwaite, J; Griffiths, CH; James, LR | 1 |
Lübker, C; Lushington, GH; Richter, M; Schuler, D; Seifert, R; Shen, Y; Tang, WJ | 1 |
Hagemann-Jensen, M; Jensen, H; Lauridsen, F; Skov, S | 1 |
Dulka, K; Gulya, K; Szabo, M | 1 |
Dempsey, S; Jack, C; Miller, CH; Nisa, S; O'Toole, R | 1 |
Kmoníčková, E; Peterková, L; Rimpelová, S; Ruml, T | 1 |
2 review(s) available for calmidazolium and trifluoperazine
Article | Year |
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Functional modulation of cell coupling: evidence for a calmodulin-driven channel gate.
Topics: Amino Acid Sequence; Animals; Aquaporins; Calcium Channel Blockers; Calmodulin; Cell Communication; Crystallization; Eye Proteins; Freeze Fracturing; Imidazoles; Intercellular Junctions; Ion Channels; Lens, Crystalline; Liposomes; Liver; Membrane Glycoproteins; Membrane Potentials; Microscopy, Electron; Models, Molecular; Permeability; Protein Conformation; Trifluoperazine | 1985 |
Sarco/Endoplasmic Reticulum Calcium ATPase Inhibitors: Beyond Anticancer Perspective.
Topics: Animals; Antineoplastic Agents; Enzyme Inhibitors; Gene Regulatory Networks; Humans; Neoplasms; Protein Structure, Secondary; Sarcoplasmic Reticulum Calcium-Transporting ATPases | 2020 |
136 other study(ies) available for calmidazolium and trifluoperazine
Article | Year |
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Cortisol secretion induced by substance P from bovine adrenocortical cells and its inhibition by calmodulin inhibitors.
Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Animals; Calcium; Calmodulin; Cattle; Cyclic AMP; Dose-Response Relationship, Drug; Hydrocortisone; Imidazoles; Neurokinin A; Neurokinin B; Signal Transduction; Substance P; Sulfonamides; Trifluoperazine | 1992 |
Calcium transport by sarcoplasmic reticulum of vascular smooth muscle: II. Effects of calmodulin and calmodulin inhibitors.
Topics: Actomyosin; Aluminum; Animals; Biological Transport, Active; Calcium; Calmodulin; Cells, Cultured; Imidazoles; Muscle, Smooth, Vascular; Oxalates; Oxalic Acid; Rats; Rats, Inbred Strains; Sarcoplasmic Reticulum; Sulfonamides; Trifluoperazine | 1992 |
Calmodulin antagonists stimulate renin secretion and inhibit renin synthesis in vitro.
Topics: Animals; Calmodulin; Cells, Cultured; Cycloheximide; Imidazoles; Juxtaglomerular Apparatus; Kinetics; Male; Mice; Mice, Inbred C57BL; Protein Biosynthesis; Renin; Sulfonamides; Sulfur Radioisotopes; Trifluoperazine | 1992 |
Effects of calmodulin antagonists on calcium transport by chorioallantoic membranes of developing chicken embryos.
Topics: Allantois; Animals; Biological Transport, Active; Calcium; Calmodulin; Chick Embryo; Chorion; Imidazoles; In Vitro Techniques; Trifluoperazine | 1992 |
Effects of phosphatase inhibitors and a protein phosphatase on norepinephrine secretion by permeabilized bovine chromaffin cells.
Topics: Adrenal Medulla; Animals; Calcium; Cattle; Cell Membrane Permeability; Ethers, Cyclic; Imidazoles; Naphthalenes; Norepinephrine; Okadaic Acid; Organophosphorus Compounds; Phosphoprotein Phosphatases; Phosphorylation; Proteins; Trifluoperazine | 1991 |
Activation of bovine rod outer segment phosphatidylinositol-4,5-bisphosphate phospholipase C by calmodulin antagonists does not depend on calmodulin.
Topics: Animals; Calmodulin; Cattle; Enzyme Activation; Haloperidol; Imidazoles; Kinetics; p-Methoxy-N-methylphenethylamine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Phosphatidylinositols; Phosphoinositide Phospholipase C; Phosphoric Diester Hydrolases; Rod Cell Outer Segment; Substrate Specificity; Sulfonamides; Trifluoperazine; Type C Phospholipases | 1991 |
Calmodulin antagonists differentiate between Ni(2+)- and Mn(2+)-stimulated phosphatase activity of calcineurin.
Topics: 4-Nitrophenylphosphatase; Animals; Brain; Calcineurin; Calmodulin; Calmodulin-Binding Proteins; Cattle; Imidazoles; Kinetics; Manganese; Nickel; Phosphoprotein Phosphatases; Sulfonamides; Thioridazine; Trifluoperazine | 1991 |
Anticalmodulin drugs block the sodium gating current of squid giant axons.
Topics: Animals; Axons; Biological Transport, Active; Calmodulin; Chlorpromazine; Decapodiformes; Diazepam; Imidazoles; Ion Channel Gating; Membrane Potentials; Phenothiazines; Potassium; Quinacrine; Sodium; Sulfonamides; Trifluoperazine | 1991 |
Biochemical studies of stimulus convergence during classical conditioning in Aplysia: dual regulation of adenylate cyclase by Ca2+/calmodulin and transmitter.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Aplysia; Calcium; Calmodulin; Conditioning, Classical; Egtazic Acid; Enzyme Activation; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Neurotransmitter Agents; Serotonin; Time Factors; Trifluoperazine | 1991 |
CaMKII mediates stimulation of chloride conductance by calcium in T84 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Line; Chloride Channels; Colon; Imidazoles; Ion Channels; Ionomycin; Isoquinolines; Kinetics; Membrane Proteins; Peptide Fragments; Phloretin; Piperazines; Protein Kinase C; Protein Kinases; Sphingosine; Trifluoperazine | 1991 |
Purification and characterization of a human NO synthase.
Topics: Amino Acid Oxidoreductases; Animals; Arginine; Calmodulin; Cerebellum; Chromatography, Affinity; Chromatography, Gel; Egtazic Acid; Electrophoresis, Polyacrylamide Gel; Humans; Imidazoles; Kinetics; Molecular Weight; Nitric Oxide Synthase; Nitroarginine; omega-N-Methylarginine; Rats; Temporal Lobe; Trifluoperazine | 1991 |
Regulation of intracellular calcium homeostasis in Trypanosoma cruzi. Effects of calmidazolium and trifluoperazine.
Topics: Animals; Biological Transport; Calcium; Calmodulin; Cell Membrane Permeability; Cytosol; Homeostasis; Imidazoles; Membrane Potentials; Oxygen; Spectrometry, Fluorescence; Trifluoperazine; Trypanosoma cruzi | 1991 |
[The effect of various low molecular weight compounds on the cation-binding properties of troponin with the heart].
Topics: Animals; Calcium; Cations; Cattle; Fluorescence Polarization; Heart; Imidazoles; Molecular Weight; Myocardium; Nicardipine; p-Methoxy-N-methylphenethylamine; Substrate Specificity; Trifluoperazine; Troponin | 1991 |
Inhibition of protein synthesis by antagonists of calmodulin in Ehrlich ascites tumor cells.
Topics: Animals; Calmodulin; Carcinoma, Ehrlich Tumor; Cell-Free System; Centrifugation, Density Gradient; Imidazoles; Methionine; Peptide Chain Initiation, Translational; Polyribosomes; Protein Biosynthesis; Protein Synthesis Inhibitors; RNA, Transfer; Sulfonamides; Sulfur Radioisotopes; Trifluoperazine | 1991 |
Role of calcium in the regulation of theca cell androstenedione production in the domestic hen.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Androstenedione; Animals; Calcimycin; Calcium; Calmodulin; Chickens; Colforsin; Dose-Response Relationship, Drug; Female; Imidazoles; Luteinizing Hormone; Theca Cells; Trifluoperazine; Verapamil | 1991 |
Calcium stimulates ATP-Mg/Pi carrier activity in rat liver mitochondria.
Topics: Adenine Nucleotides; Adenosine Triphosphate; Animals; Calcium Chloride; Calmodulin; Carrier Proteins; Cells, Cultured; Chlorpromazine; Egtazic Acid; Glucagon; Imidazoles; Kinetics; Liver; Magnesium; Male; Mitochondria, Liver; Neomycin; Phosphates; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine; Vasopressins | 1990 |
Refractoriness to the insulin-like effects of growth hormone depends upon calcium.
Topics: Adipose Tissue; Animals; Calcimycin; Calcium; Calmodulin; Egtazic Acid; Glucose; Growth Hormone; Imidazoles; Insulin; Male; Rats; Signal Transduction; Trifluoperazine; Verapamil | 1990 |
Drug interaction with cardiac and skeletal muscle troponin C.
Topics: Allosteric Site; Animals; Calcium; Calmodulin; Cardiotonic Agents; Cattle; Heart; Imidazoles; Magnesium; Muscles; Myocardium; Nicardipine; p-Methoxy-N-methylphenethylamine; Piperazines; Protein Binding; Protein Conformation; Pyridones; Rabbits; Trifluoperazine; Troponin; Troponin C | 1990 |
Similarities between the effects of dimethyl sulfoxide and calmodulin on the red blood cell Ca2(+)-ATPase.
Topics: Adenosine Triphosphate; Animals; Binding Sites; Calcium; Calcium-Transporting ATPases; Calmodulin; Cattle; Dimethyl Sulfoxide; Enzyme Activation; Erythrocyte Membrane; Humans; Imidazoles; p-Methoxy-N-methylphenethylamine; Phosphates; Trifluoperazine | 1990 |
Effect of calmidazolium (R24571) on histamine release from isolated rat mast cells.
Topics: Animals; Calcimycin; Calmodulin; Chlorpromazine; Flupenthixol; Glucose; Histamine Release; Imidazoles; Imipramine; In Vitro Techniques; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Rats; Rats, Inbred Strains; Trifluoperazine | 1986 |
Reconstitution in phospholipid vesicles of calcium-activated potassium channel from outer renal medulla.
Topics: Animals; Calcium; Calmodulin; Imidazoles; Ion Channels; Kidney Medulla; Liposomes; Loop of Henle; Membrane Potentials; Potassium; Quinidine; Rubidium; Swine; Trifluoperazine | 1987 |
Inhibitory effects of calcium channel agonists on renin release from rat kidney cortical slices.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dose-Response Relationship, Drug; Imidazoles; Ion Channels; Kidney Cortex; Male; Nifedipine; Pyridines; Rats; Rats, Inbred Strains; Renin; Trifluoperazine; Verapamil | 1987 |
Sources of calcium and the involvement of calmodulin during steroidogenesis and oocyte maturation in follicles of Rana pipiens.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Calmodulin; Female; Gallic Acid; Imidazoles; Lanthanum; Oocytes; Ovarian Follicle; Progesterone; Rana pipiens; Sulfonamides; Trifluoperazine | 1987 |
Regulation of goby intestinal ion absorption by the calcium messenger system.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcimycin; Calcium; Calmodulin; Female; Fishes; Imidazoles; Intestinal Absorption; Ion Channels; Male; Microscopy, Electron; Trifluoperazine | 1987 |
Calmodulin antagonists depress calcium and potassium currents in ventricular and vascular myocytes.
Topics: Animals; Calcium; Calmodulin; Cattle; Guinea Pigs; Heart; Imidazoles; Ion Channels; Myocardium; Portal Vein; Potassium; Tetrodotoxin; Trifluoperazine | 1987 |
Drug-induced calcium release from sarcoplasmic reticulum of skeletal muscle.
Topics: Animals; Calcium; Calmodulin; Imidazoles; In Vitro Techniques; Ion Channels; Kinetics; p-Methoxy-N-methylphenethylamine; Rabbits; Sarcoplasmic Reticulum; Sulfonamides; Trifluoperazine | 1988 |
Elevation of angiotensin converting enzyme by 3-isobutyl-1-methylxanthine in cultured endothelial cells: a possible role for calmodulin.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Calmodulin; Cattle; Cells, Cultured; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; Egtazic Acid; Endothelium, Vascular; Imidazoles; Indomethacin; Peptidyl-Dipeptidase A; Propranolol; Theophylline; Trifluoperazine; Verapamil; Xanthines | 1988 |
Interaction of calmodulin and calcium antagonists with [3H]diltiazem and [3H]nitrendipine binding sites.
Topics: Animals; Bepridil; Calcium Channel Blockers; Calcium Channels; Calmodulin; Diltiazem; Imidazoles; Phosphodiesterase Inhibitors; Pyrrolidines; Rats; Receptors, Nicotinic; Sulfonamides; Trifluoperazine | 1988 |
ATP-dependent Ca2+ transport in the rat parotid basolateral plasma membrane is regulated by calmodulin.
Topics: Animals; Biological Transport, Active; Calcium; Calmodulin; Cell Membrane; Cell Membrane Permeability; Egtazic Acid; Imidazoles; In Vitro Techniques; Kinetics; Male; Parotid Gland; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine | 1989 |
Involvement of a Ca2+-calmodulin interaction in the yeast-mycelial (Y-M) transition of Candida albicans.
Topics: Calcimycin; Calcium; Calmodulin; Candida albicans; Hydrogen-Ion Concentration; Imidazoles; Morphogenesis; Trifluoperazine | 1989 |
Calmodulin and protein kinase C antagonists also inhibit the Ca2+-dependent protein protease, calpain I.
Topics: Bee Venoms; Calmodulin; Calpain; Erythrocytes; Humans; Imidazoles; Kinetics; Melitten; Protein Kinase C; Sulfonamides; Trifluoperazine | 1989 |
Effect of calmodulin antagonists on contraction and 45Ca movements in rat aorta.
Topics: Animals; Aorta, Thoracic; Calcium; Calcium Radioisotopes; Calmodulin; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine | 1989 |
Drug-drug interaction between cyclosporine and agents affecting calcium-dependent lymphocyte proliferation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium Channel Blockers; Cells, Cultured; Cyclosporins; Drug Interactions; Humans; Imidazoles; Isoquinolines; Lymphocyte Activation; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine; Verapamil | 1989 |
Anti-calmodulin agents affect osmotic and angiotensin II-induced vasopressin release.
Topics: Angiotensin II; Animals; Arginine Vasopressin; Calmodulin; Culture Techniques; Hypothalamus; Imidazoles; Male; Osmolar Concentration; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine | 1989 |
In vivo characterization of combination antitumor chemotherapy with calcium channel blockers and cis-diamminedichloroplatinum(II).
Topics: Animals; Calcium Channel Blockers; Cisplatin; Diltiazem; Drug Evaluation, Preclinical; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Imidazoles; Lung Neoplasms; Melanoma, Experimental; Mice; Nicardipine; Nifedipine; Trifluoperazine; Verapamil | 1989 |
Calmodulin antagonist action in smooth-muscle myosin phosphorylation. Different mechanisms for trifluoperazine and calmidazolium inhibition.
Topics: Animals; Calmodulin; Enzyme Inhibitors; Imidazoles; Kinetics; Muscle, Smooth; Myosin Subfragments; Myosin-Light-Chain Kinase; Myosins; Phosphorylation; Trifluoperazine | 1989 |
A calmodulin-sensitive adenylate cyclase in the prothoracic glands of the tobacco hornworm, Manduca sexta.
Topics: Adenylyl Cyclases; Animals; Calcium; Calcium Channels; Calmodulin; Cyclic AMP; Guanosine Triphosphate; Imidazoles; Insect Hormones; Insecta; Thorax; Trifluoperazine | 1988 |
Analysis of calmodulin acceptor proteins and the influence of calmodulin antagonists on human spermatozoa.
Topics: Calcium; Calmodulin; Calmodulin-Binding Proteins; Cyclic AMP; Humans; Imidazoles; Male; Sperm-Ovum Interactions; Trifluoperazine | 1988 |
Modulation of calcium current by calmodulin antagonists.
Topics: Animals; Calcium Channels; Calmodulin; Chlorpromazine; Helix, Snails; Imidazoles; In Vitro Techniques; Membrane Potentials; Neurons; Trifluoperazine | 1988 |
Inhibition of mitochondrial F1 ATPase and sarcoplasmic reticulum ATPase by hydrophobic molecules.
Topics: Biological Transport, Active; Calcium; Calcium-Transporting ATPases; Imidazoles; Mitochondria; Phenanthrolines; Phosphates; Proton-Translocating ATPases; Sarcoplasmic Reticulum; Solubility; Solvents; Submitochondrial Particles; Trifluoperazine | 1988 |
Subcellular action of cyclosporine: interaction between CsA and calmodulin antagonists.
Topics: Calmodulin; Cyclosporins; Drug Interactions; Humans; Imidazoles; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Sulfonamides; Trifluoperazine | 1987 |
Differential effects of pharmacological modulators of cardiac myofibrillar ATPase activity in normal and myopathic (BIO 14.6) hamsters.
Topics: Adenosine Triphosphatases; Animals; Anti-Arrhythmia Agents; Bepridil; Calcium; Calcium Channel Blockers; Cricetinae; Disease Models, Animal; Electrophoresis, Polyacrylamide Gel; Heart Failure; Imidazoles; Male; Myocardium; Myofibrils; Perhexiline; Pyrrolidines; Trifluoperazine | 1988 |
Inhibition of growth of C6 astrocytoma cells by inhibitors of calmodulin.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Astrocytoma; Calmodulin; Cell Division; Cell Line; Chlorpromazine; Imidazoles; Melitten; Pimozide; Rats; Structure-Activity Relationship; Trifluoperazine | 1985 |
Transforming NRK cells with avian sarcoma virus reduces the extracellular Ca2+ requirement without affecting the calcicalmodulin requirement for the G1/S transition.
Topics: Animals; Avian Sarcoma Viruses; Calcium; Calmodulin; Cell Line; Cell Transformation, Neoplastic; Cell Transformation, Viral; Culture Media; DNA Replication; Imidazoles; Interphase; Oncogene Protein pp60(v-src); Phenotype; Rats; Sulfonamides; Temperature; Trifluoperazine; Viral Proteins | 1985 |
Characterization of a calmodulin-dependent protein phosphatase from human platelets.
Topics: Animals; Blood Platelets; Brain; Calcium-Binding Proteins; Calmodulin; Calmodulin-Binding Proteins; Humans; Hydrogen-Ion Concentration; Imidazoles; Kinetics; Macromolecular Substances; Molecular Weight; Phosphoprotein Phosphatases; Swine; Trifluoperazine; Troponin; Troponin C; Trypsin | 1985 |
Beta adrenergic receptor-stimulated prostaglandin synthesis in the isolated rabbit heart: relationship to extra- and intracellular calcium.
Topics: 6-Ketoprostaglandin F1 alpha; Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Calcium Channel Blockers; Calmodulin; Dinoprostone; Dose-Response Relationship, Drug; Gallic Acid; Heart; Heart Rate; Imidazoles; Isoproterenol; Male; Myocardium; Prostaglandins; Prostaglandins E; Rabbits; Receptors, Adrenergic, beta; Trifluoperazine | 1985 |
Modulation and role of Ca2+ in LH and LHRH agonist action in rat Leydig cells.
Topics: Animals; Calcium; Chlorpromazine; Cyclic AMP; Gonadotropin-Releasing Hormone; Imidazoles; Leydig Cells; Lipoxygenase Inhibitors; Luteinizing Hormone; Male; Rats; Testosterone; Trifluoperazine | 1986 |
The role of calmodulin antagonists on steroidogenesis by fetal zone cells of the human fetal adrenal gland.
Topics: Adrenal Glands; Adrenocorticotropic Hormone; Bucladesine; Calmodulin; Cells, Cultured; Chlorpromazine; Cyclic AMP; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Embryo, Mammalian; Fetus; Humans; Hydrocortisone; Imidazoles; Kinetics; Pregnenolone; Trifluoperazine | 1987 |
Identification of calmodulin-like activity in term human amnion: effect of calmodulin inhibitors on prostaglandin biosynthesis.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Amnion; Calcimycin; Calcium; Calmodulin; Cytosol; Dinoprostone; Female; Humans; Imidazoles; Microsomes; Pregnancy; Prostaglandins E; Sulfonamides; Trifluoperazine | 1987 |
Role of protein kinase C and intracellular calcium mobilization in the induction of macrophage tumoricidal activity by interferon-gamma.
Topics: Aminoquinolines; Calcimycin; Calcium; Cytotoxicity, Immunologic; Imidazoles; Interferon-gamma; Macrophage Activation; Macrophages; Neoplasms, Experimental; Protein Kinase C; Tetradecanoylphorbol Acetate; Trifluoperazine | 1986 |
Calcium ionophore (A23187)- and arachidonic acid-stimulated prostaglandin release from microvascular endothelial cells: effects of calcium antagonists and calmodulin inhibitors.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Cells, Cultured; Coronary Vessels; Endothelium; Imidazoles; Kinetics; Microcirculation; Prostaglandins; Rabbits; Trifluoperazine; Valinomycin | 1987 |
Antagonism of calmodulin-stimulated adenylate cyclase by trifluoperazine, calmidazolium and W-7 in rat cerebellar membranes.
Topics: Adenylyl Cyclases; Animals; Calmodulin; Cerebellum; Chlorpromazine; Dose-Response Relationship, Drug; Egtazic Acid; Imidazoles; Membranes; Rats; Sulfonamides; Trifluoperazine | 1987 |
Effects of the anti-calmodulin drugs calmidazolium and trifluoperazine on 45Ca transport in plasmalemmal vesicles from gastric smooth muscle.
Topics: Adenosine Triphosphate; Animals; Bufo marinus; Calcium; Calcium Radioisotopes; Calmodulin; Cell Membrane; Cell Membrane Permeability; Imidazoles; Muscle, Smooth; Stomach; Swine; Trifluoperazine | 1988 |
Calmodulin antagonist effects on GnRH and secretogogue-induced release of bovine LH.
Topics: Animals; Calcimycin; Calmodulin; Cattle; Dinoprostone; Female; Gonadotropin-Releasing Hormone; Imidazoles; Luteinizing Hormone; Male; Pituitary Gland, Anterior; Prostaglandins E; Sulfonamides; Trifluoperazine | 1988 |
Effect of calmodulin antagonists on calcium pump of ram spermatozoa plasma membrane.
Topics: Animals; Calcium; Calmodulin; Cell Membrane; Egtazic Acid; Gallopamil; Imidazoles; Male; p-Methoxy-N-methylphenethylamine; Sheep; Spermatozoa; Trifluoperazine | 1988 |
Phase-shifts of the Bulla ocular circadian pacemaker in the presence of calmodulin antagonists.
Topics: Animals; Calmodulin; Circadian Rhythm; Imidazoles; Mollusca; Sulfonamides; Trifluoperazine | 1988 |
Fendiline and calmidazolium enhance the release of endothelium-derived relaxant factor and of prostacyclin from cultured endothelial cells.
Topics: Adenosine Triphosphate; Animals; Biological Products; Calcium; Calmodulin; Cattle; Cells, Cultured; Endothelium, Vascular; Epoprostenol; Fendiline; Imidazoles; Nitric Oxide; Phenethylamines; Trifluoperazine | 1988 |
Different developmental functions for calmodulin in Dictyostelium: trifluoperazine and R24571 both inhibit cell and pronuclear fusion but enhance gamete formation.
Topics: Calmodulin; Cell Fusion; Cell Nucleus; Dictyostelium; Gametogenesis; Imidazoles; Membrane Fusion; Trifluoperazine; Zygote | 1988 |
Calmodulin antagonists inhibit latch bridges in detergent skinned swine carotid media.
Topics: Adenosine Triphosphate; Animals; Calcium; Calmodulin; Carotid Arteries; Cytidine Triphosphate; Detergents; Imidazoles; In Vitro Techniques; Magnesium; Muscle Contraction; Myosins; Osmolar Concentration; Phosphorylation; Sulfonamides; Swine; Trifluoperazine | 1987 |
Effect of calmodulin inhibitors on viability and mitochondrial potential of Plasmodium falciparum in culture.
Topics: Calmodulin; Chlorpromazine; Imidazoles; Mitochondria; Plasmodium falciparum; Trifluoperazine | 1986 |
Mechanisms of action of inhibitors of prolactin secretion in GH3 pituitary cells. I. Ca2+-dependent inhibition of amino acid incorporation.
Topics: Acetylcholine; Amino Acids; Animals; Bromocriptine; Calcium; Carbachol; Cell Line; Chlorpromazine; Imidazoles; Magnesium; Nifedipine; Pituitary Neoplasms; Prolactin; Protein Processing, Post-Translational; Rats; Trifluoperazine; Verapamil | 1986 |
Evidence of a role for calmodulin in the regulation of calcium release from skeletal muscle sarcoplasmic reticulum.
Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Radioisotopes; Calmodulin; Cattle; Imidazoles; Kinetics; Magnesium; Muscles; p-Methoxy-N-methylphenethylamine; Rabbits; Sarcoplasmic Reticulum; Trifluoperazine | 1986 |
A role for calmodulin in renal production of 1,25-dihydroxyvitamin D3.
Topics: Animals; Calcifediol; Calcitriol; Calcium; Calmodulin; Chickens; Imidazoles; Kidney Tubules; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Sulfonamides; Trifluoperazine; Vitamin D Deficiency | 1986 |
Calmodulin and acetylcholine receptor clustering in embryonic chick myotubes.
Topics: Animals; Calmodulin; Cell Membrane; Chick Embryo; Imidazoles; Kinetics; Muscles; Receptors, Cholinergic; Trifluoperazine | 1986 |
Mechanism of action of angiotensin II and bradykinin on prostaglandin synthesis and vascular tone in the isolated rat kidney. Effect of Ca++ antagonists and calmodulin inhibitors.
Topics: 6-Ketoprostaglandin F1 alpha; Angiotensin II; Animals; Bradykinin; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Dantrolene; Diltiazem; Dinoprostone; Gallic Acid; Imidazoles; Indomethacin; Kidney; Male; Nicotinic Acids; Nimodipine; Prostaglandins E; Quinacrine; Rats; Rats, Inbred Strains; Ryanodine; Stimulation, Chemical; Sulfonamides; Trifluoperazine; Vasoconstriction | 1985 |
Effects of calmodulin and lipoxygenase inhibitors on LH (lutropin)- and LHRH (luliberin)-agonist-stimulated steroidogenesis in rat Leydig cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Calmodulin; Imidazoles; In Vitro Techniques; Indomethacin; Leydig Cells; Lipoxygenase Inhibitors; Luteinizing Hormone; Male; Propionates; Pyrazoles; Rats; Testosterone; Trifluoperazine | 1985 |
The effects of anticalmodulin drugs on the ultrastructure of boar spermatozoa.
Topics: Acrosome; Animals; Calmodulin; Fluorescein-5-isothiocyanate; Fluoresceins; Imidazoles; Lectins; Male; Microscopy, Electron; Microscopy, Fluorescence; Plant Lectins; Spermatozoa; Sulfonamides; Swine; Thiocyanates; Trifluoperazine | 1985 |
Selective cytotoxicity of calmidazolium and trifluoperazine for cycling versus noncycling C3H10T1/2 cells in vitro.
Topics: Animals; Calmodulin; Cell Cycle; Cell Survival; Cell Transformation, Neoplastic; Dose-Response Relationship, Drug; Flow Cytometry; Imidazoles; Mice; Trifluoperazine | 1986 |
Tubuloglomerular feedback responses in the rat during calmodulin inhibition.
Topics: Animals; Calmodulin; Feedback; Glomerular Filtration Rate; Imidazoles; Kidney Glomerulus; Kidney Tubules; Male; Rats; Trifluoperazine | 1986 |
Evidence for Ca++-calmodulin control of transplasmalemma electron transport in carrot cells.
Topics: Calcium; Calmodulin; Cell Membrane; Electron Transport; Ferricyanides; Fluphenazine; Gallic Acid; Imidazoles; Oxidation-Reduction; Pimozide; Plants; Spectrophotometry; Trifluoperazine | 1985 |
Inhibitors of calcium-dependent enzymes prevent the onset of afterdischarge in the peptidergic bag cell neurons of Aplysia.
Topics: Animals; Aplysia; Evoked Potentials; Imidazoles; Neurons; Protein Kinase Inhibitors; Reaction Time; Sulfonamides; Trifluoperazine | 1985 |
Inhibition of calmodulin-dependent and independent cardiac sarcoplasmic reticulum activities by R24571.
Topics: Adenosine Triphosphatases; Animals; Ca(2+) Mg(2+)-ATPase; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Dogs; Enzyme Inhibitors; Imidazoles; Kinetics; Myocardium; Phosphorylation; Protein Kinases; Sarcoplasmic Reticulum; Trifluoperazine | 1983 |
The effect of drugs on calmodulin and its interaction with phosphodiesterase.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Animals; Antipsychotic Agents; Calmodulin; Enzyme Activation; Imidazoles; Penfluridol; Rats; Structure-Activity Relationship; Trifluoperazine | 1984 |
The anticalmodulin drugs trifluoperazine and R24571 remove the activation of the purified erythrocyte Ca2+-ATPase by acidic phospholipids and by controlled proteolysis.
Topics: Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Humans; Imidazoles; Kinetics; Phosphatidylcholines; Phospholipids; Trifluoperazine | 1982 |
Effect of calmodulin antagonists on CA2+ uptake by boar spermatozoa.
Topics: Animals; Biological Transport, Active; Calcium; Calcium Channel Blockers; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Cell Membrane; Imidazoles; Kinetics; Male; Spermatozoa; Swine; Trifluoperazine; Verapamil | 1983 |
Inhibition of skeletal muscle sarcoplasmic reticulum CaATPase activity by calmidazolium.
Topics: Adenosine Triphosphate; Animals; Calcium-Transporting ATPases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Imidazoles; Kinetics; Mathematics; Muscles; Phosphorylation; Propranolol; Quercetin; Rabbits; Sarcoplasmic Reticulum; Trifluoperazine | 1984 |
A model for the regulation of the calmodulin-dependent enzymes erythrocyte Ca2+-transport ATPase and brain phosphodiesterase by activators and inhibitors.
Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Animals; Brain; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Cattle; Enzyme Activation; Erythrocytes; Humans; Imidazoles; Models, Biological; Penfluridol; Phosphoric Diester Hydrolases; Trifluoperazine | 1982 |
Inhibition of photosynthetic oxygen evolution by calmodulin-type inhibitors and other calcium-antagonists.
Topics: Calcium; Calmodulin; Chlorpromazine; Imidazoles; Metals; Oxygen; Photochemistry; Photosynthesis; Photosynthetic Reaction Center Complex Proteins; Photosystem II Protein Complex; Plant Proteins; Plants; Trifluoperazine | 1984 |
Effects of calmodulin antagonists on immune mouse lymphocytes.
Topics: Animals; Calmodulin; Cell Line; Chlorpromazine; Cytotoxicity, Immunologic; Enzyme Inhibitors; Imidazoles; Kinetics; Leukemia, Experimental; Lymphocytes; Mice; Pimozide; Structure-Activity Relationship; Sulfonamides; Trifluoperazine | 1984 |
Calmodulin antagonists inhibit activity of myosin light-chain kinase independent of calmodulin.
Topics: Animals; Calmodulin; Cattle; Imidazoles; Myosin-Light-Chain Kinase; Myosins; Protein Binding; Protein Kinase Inhibitors; Spectrometry, Fluorescence; Sulfonamides; Trifluoperazine | 1984 |
Calmodulin-NADH semidehydroascorbate oxidoreductase interactions of clathrin coated vesicles.
Topics: Animals; Calmodulin; Clathrin; Enzyme Inhibitors; Golgi Apparatus; Imidazoles; Kinetics; Liver; Microsomes, Liver; NADH, NADPH Oxidoreductases; Pimozide; Rats; Subcellular Fractions; Trifluoperazine | 1983 |
The effect of trifluoperazine and R 24 571 on the K+-evoked release of 5-hydroxytryptamine from superfused synaptosomes.
Topics: Animals; Imidazoles; In Vitro Techniques; Male; Potassium; Potassium Radioisotopes; Rats; Rats, Inbred Strains; Serotonin; Synaptosomes; Trifluoperazine | 1983 |
The calmodulin antagonists, trifluoperazine and R24571, depolarize the mitochondria within guinea pig cerebral cortical synaptosomes.
Topics: Animals; Calcium; Calmodulin; Cell Membrane; Cerebral Cortex; Female; Guinea Pigs; Imidazoles; Intracellular Membranes; Kinetics; Male; Membrane Potentials; Mitochondria; Synaptosomes; Trifluoperazine | 1984 |
A fluorescent calmodulin that reports the binding of hydrophobic inhibitory ligands.
Topics: Anilino Naphthalenesulfonates; Calcium; Calcium-Binding Proteins; Calmodulin; Felodipine; Fluorescent Dyes; Imidazoles; Ligands; Liposomes; Nifedipine; Protein Binding; Spectrometry, Fluorescence; Trifluoperazine | 1983 |
Effects of various calmodulin antagonists on Na/Ca exchange current of single ventricular cells of guinea-pig.
Topics: Animals; Benzimidazoles; Calcium; Calmodulin; Carrier Proteins; Guinea Pigs; Heart Ventricles; Imidazoles; In Vitro Techniques; Intercellular Signaling Peptides and Proteins; Melitten; Myocardium; Peptides; Ruthenium Red; Sodium; Sodium-Calcium Exchanger; Sulfonamides; Trifluoperazine; Wasp Venoms | 1993 |
Trifluoperazine and calmidazolium have multiple actions on the release of noradrenaline from sympathetic nerves of mouse atria.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Atropine; Calmodulin; Desipramine; Electric Stimulation; Enterochromaffin Cells; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Male; Mice; Myocardium; Norepinephrine; Phentolamine; Sympathetic Nervous System; Trifluoperazine | 1994 |
Dual regulation of cGMP formation by calcium in pancreatic acinar cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Oxidoreductases; Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Cyclic GMP; Cytosol; Guanylate Cyclase; Guinea Pigs; Homeostasis; Imidazoles; In Vitro Techniques; Isoquinolines; Kinetics; Nitric Oxide Synthase; Pancreas; Piperazines; Protein Kinase C; Staurosporine; Sulfonamides; Trifluoperazine | 1995 |
Calcium homeostasis in Trypanosoma cruzi.
Topics: Animals; Antimycin A; Biological Transport; Ca(2+) Mg(2+)-ATPase; Calcium; Calmodulin; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cell Membrane; Cell Membrane Permeability; Digitonin; Fura-2; Homeostasis; Imidazoles; Intracellular Membranes; Membrane Potentials; Mitochondria; Ruthenium Red; Trifluoperazine; Trypanosoma cruzi; Vanadates | 1993 |
Ca(++)-calmodulin-dependent phosphorylation and dephosphorylation of rat parotid secretion granules.
Topics: Adenosine Triphosphate; Animals; Calcium; Calmodulin; Cell Fractionation; Cell Membrane; Centrifugation, Density Gradient; Cytoplasmic Granules; Imidazoles; Intracellular Membranes; Membrane Fusion; Molecular Weight; Parotid Gland; Phosphorylation; Rats; Trifluoperazine | 1995 |
A GTP-binding protein modulates a Ca2+ pump present in reticulocyte endocytic vesicles.
Topics: Animals; Benzalkonium Compounds; Blotting, Western; Calcium; Calcium-Transporting ATPases; Calmodulin; Cell Membrane; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Endocytosis; Endosomes; Enzyme Inhibitors; Erythrocytes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Intercellular Signaling Peptides and Proteins; Peptides; Rats; Rats, Sprague-Dawley; Reticulocytes; Trifluoperazine; Vanadates; Wasp Venoms | 1995 |
Calmidazolium inhibits muscarinic receptor-mediated PLC activation in SH-SY5Y cells.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Imidazoles; Inositol 1,4,5-Trisphosphate; Neuroblastoma; Receptors, Muscarinic; Trifluoperazine | 1995 |
N-(6-aminohexyl)-5-chloro-1-naphthalenesulfonamide, a calmodulin antagonist, reverses the inhibitory effect of insulin on lipolysis due to dibutyryl cyclic AMP.
Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Animals; Bucladesine; Calmodulin; Cells, Cultured; Dose-Response Relationship, Drug; Epididymis; Epinephrine; Imidazoles; Insulin; Insulin Antagonists; Kinetics; Lipolysis; Male; Rats; Rats, Sprague-Dawley; Receptor, Insulin; Sulfonamides; Trifluoperazine | 1993 |
Adenylate cyclase activity from Hirudo medicinalis segmental ganglia: modulation by calcium and calmodulin.
Topics: Adenylyl Cyclases; Animals; Calcium; Calmodulin; Drug Synergism; Enzyme Inhibitors; Ganglia, Invertebrate; Imidazoles; Leeches; Serotonin; Trifluoperazine | 1995 |
Autoradiographic distribution and characteristics of high- and low-affinity polyamine-sensitive [3H]ifenprodil sites in the rat brain: possible relationship to NMDAR2B receptors and calmodulin.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Calmodulin; Hippocampus; Imidazoles; Male; Piperidines; Polyamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Sepharose; Spermidine; Spermine; Sulfonamides; Tissue Distribution; Trifluoperazine; Tritium | 1994 |
Ethanol modulates calmodulin-dependent Ca(2+)-activated ATPase in synaptic plasma membranes.
Topics: Alcoholism; Animals; Brain; Calcium-Transporting ATPases; Ethanol; Imidazoles; Kinetics; Male; Ouabain; Rats; Rats, Sprague-Dawley; Reference Values; Synaptic Membranes; Synaptosomes; Trifluoperazine | 1994 |
Inhibition of high voltage-activated calcium currents by L-glutamate receptor-mediated calcium influx.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Calcium Channels; Egtazic Acid; Electric Conductivity; Female; Glutamates; Glutamic Acid; Hypothalamus; Imidazoles; Neurons; Quinoxalines; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Trifluoperazine | 1993 |
Enhancement of metallothionein gene expression in male Wistar (WF/NCr) rats by treatment with calmodulin inhibitors: potential role of calcium regulatory pathways in metallothionein induction.
Topics: Animals; Base Sequence; Cadmium; Cadmium Chloride; Calcimycin; Calmodulin; Chlorides; Chlorpromazine; Gene Expression Regulation; Imidazoles; Kidney; Liver; Male; Metallothionein; Molecular Sequence Data; Rats; Rats, Wistar; RNA, Messenger; Sulfonamides; Testis; Trifluoperazine | 1994 |
Calmodulin antagonists induce changes in lens permeability and transparency.
Topics: Animals; Calcium; Calmodulin; Cataract; Cell Membrane Permeability; Imidazoles; Lens, Crystalline; Membrane Potentials; Rats; Rats, Wistar; Sodium; Sulfonamides; Trifluoperazine | 1994 |
Stage-specific changes in protein phosphorylation during spore germination in Dictyostelium: role of calmodulin.
Topics: Animals; Calmodulin; Dictyostelium; Fungal Proteins; Imidazoles; Phosphoproteins; Protein Kinases; Spores, Fungal; Trifluoperazine | 1994 |
Influence of calmodulin antagonists and calcium channel blockers on triiodothyronine uptake by rat hepatoma and myoblast cell lines.
Topics: Analysis of Variance; Animals; Cadmium; Calcium; Calcium Channel Blockers; Calmodulin; Cell Line; Diltiazem; Imidazoles; Iodine Radioisotopes; Liver Neoplasms, Experimental; Magnesium; Muscles; Nifedipine; Protein Kinase C; Rats; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine; Triiodothyronine; Tumor Cells, Cultured; Verapamil | 1993 |
Blockade by calmodulin inhibitors of Ca2+ channels in smooth muscle from rat vas deferens.
Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Calmodulin; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nimodipine; Potassium Chloride; Radioligand Assay; Rats; Rats, Wistar; Sulfonamides; Trifluoperazine; Vas Deferens | 1993 |
Trypanosoma cruzi: involvement of intracellular calcium in multiplication and differentiation.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcimycin; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Chelating Agents; Chlorpromazine; Dopamine Antagonists; Egtazic Acid; Enzyme Inhibitors; Gallic Acid; Gallopamil; Imidazoles; Ionomycin; Ionophores; Morphogenesis; Triatoma; Trifluoperazine; Trypanosoma cruzi | 1996 |
The role of calmodulin in the gravitropic response of the Arabidopsis thaliana agr-3 mutant.
Topics: Arabidopsis; Calmodulin; Gravitropism; Imidazoles; Mutation; Plant Roots; Sulfonamides; Trifluoperazine | 1996 |
Evidence for a role of calmodulin in calcium-induced noradrenaline release from permeated synaptosomes: effects of calmodulin antibodies and antagonists.
Topics: Animals; Antibodies; Calcium; Calmodulin; GAP-43 Protein; Imidazoles; Immunoglobulin G; Male; Membrane Glycoproteins; Nerve Tissue Proteins; Norepinephrine; Permeability; Rats; Rats, Wistar; Sulfonamides; Synaptosomes; Trifluoperazine | 1996 |
Regulation of capacitative calcium influx in cultured human mesangial cells: roles of protein kinase C and calmodulin.
Topics: Angiotensin II; Biological Transport; Calcium; Calmodulin; Cells, Cultured; Egtazic Acid; Enzyme Inhibitors; Glomerular Mesangium; Humans; Imidazoles; Ionomycin; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine | 1996 |
The involvement of calmodulin and Ca2+/calmodulin-dependent protein kinase II in the circadian rhythms controlled by the suprachiasmatic nucleus.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Analysis of Variance; Animals; Biomarkers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Circadian Rhythm; Drug Evaluation, Preclinical; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Nerve Tissue Proteins; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Suprachiasmatic Nucleus; Trifluoperazine | 1997 |
Kinetic and pharmacological properties of the calcium-activated chloride-current in macrovascular endothelial cells.
Topics: Animals; Calcium; Calmodulin; Cattle; Chloride Channels; Electrophysiology; Endothelium, Vascular; Epithelium; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Kinetics; Polymerase Chain Reaction; Trifluoperazine | 1997 |
Involvement of calcium and calmodulin in Toxoplasma gondii tachyzoite invasion.
Topics: Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Carcinoma, Squamous Cell; Cytosol; Epithelial Cells; Humans; Imidazoles; Ionophores; Toxoplasma; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1997 |
Calcium-calmodulin-stimulated phosphorylation of rat parotid secretion granule proteins.
Topics: Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Cell Membrane; Cytoplasmic Granules; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Imidazoles; Membrane Fusion; Molecular Weight; Parotid Gland; Parvalbumins; Phosphorylation; Rats; Salivary Proteins and Peptides; Trifluoperazine; Troponin; Trypsin; Vacuoles | 1997 |
Effects of calmodulin inhibitors on cyprid larvae of the barnacle, Balanus amphitrite.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Chlorpromazine; Cyclic AMP; Dose-Response Relationship, Drug; Imidazoles; Immunoblotting; Larva; Metamorphosis, Biological; Myosin-Light-Chain Kinase; Phosphodiesterase Inhibitors; Sulfonamides; Thoracica; Trifluoperazine; Vinca Alkaloids | 1998 |
Protein kinase C--catalyzed calponin phosphorylation in swine carotid arterial homogenate.
Topics: Animals; Antiemetics; Calcium; Calcium-Binding Proteins; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Calmodulin-Binding Proteins; Calponins; Carcinogens; Carotid Arteries; Chelating Agents; Diglycerides; Egtazic Acid; Electrophoresis; Enzyme Inhibitors; Imidazoles; Microfilament Proteins; Okadaic Acid; Organ Culture Techniques; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phosphorus Radioisotopes; Phosphorylation; Protein Kinase C; Staurosporine; Sulfonamides; Swine; Trifluoperazine; Vasodilator Agents | 1998 |
Riboflavin uptake by the human-derived liver cells Hep G2: mechanism and regulation.
Topics: Antiemetics; Biological Transport; Bucladesine; Calcium; Calmodulin; Carcinogens; Carcinoma, Hepatocellular; Carrier Proteins; Cholera Toxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Extracellular Space; Flavins; Genistein; Humans; Imidazoles; Protein Kinase C; Riboflavin; Signal Transduction; Tetradecanoylphorbol Acetate; Trifluoperazine; Tritium; Tumor Cells, Cultured; Vanadates | 1998 |
Regulation of the high-affinity H+/peptide cotransporter in renal LLC-PK1 cells.
Topics: Animals; Biological Transport; Calcium; Carrier Proteins; Cell Survival; Dipeptides; Enzyme Inhibitors; Hydrogen-Ion Concentration; Imidazoles; Kidney Tubules, Proximal; Kinetics; LLC-PK1 Cells; Protein Kinase C; Signal Transduction; Staurosporine; Stereoisomerism; Sulfonamides; Swine; Symporters; Tetradecanoylphorbol Acetate; Trifluoperazine | 1999 |
alpha1-adrenergic receptor activation of c-fos expression in transfected rat-1 fibroblasts: role of Ca2+.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenergic alpha-1 Receptor Antagonists; Animals; Calcium; Calmodulin; Doxazosin; Egtazic Acid; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Genes, fos; Imidazoles; Kinetics; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-fos; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Sulfonamides; Transcription, Genetic; Trifluoperazine | 1999 |
Ca2+ and calmodulin-dependent protein phosphatase from Leishmania donovani.
Topics: Animals; Blotting, Western; Calcineurin; Calcium-Calmodulin-Dependent Protein Kinases; Cyclosporine; Fluphenazine; Humans; Imidazoles; Immunophilins; Leishmania donovani; Protozoan Proteins; Tacrolimus; Tacrolimus Binding Proteins; Trifluoperazine | 1999 |
Regulation of glycine transport in cultured Müller cells by Ca2+/calmodulin-dependent enzymes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Transport Systems, Neutral; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Carrier Proteins; Cell Line; Chick Embryo; Enzyme Inhibitors; Glycine Plasma Membrane Transport Proteins; Imidazoles; Kinetics; Sulfonamides; Trifluoperazine | 1999 |
Role of calcium and calmodulin in ciliary stimulation induced by acetylcholine.
Topics: Acetylcholine; Animals; Calcium; Calcium Signaling; Calmodulin; Cell Movement; Cells, Cultured; Cilia; Enzyme Inhibitors; Epithelium; Esophagus; Imidazoles; Muscarinic Antagonists; Rana ridibunda; Receptors, Muscarinic; Sulfonamides; Trifluoperazine | 2001 |
Voltage dependence of the [Ca2+](i) oscillations system, in the Mg2+ -stimulated oocyte of the prawn Palaemon serratus.
Topics: Animals; Calcium; Calcium Channels; Calcium Signaling; Dopamine Antagonists; Enzyme Inhibitors; Female; Fluorescent Dyes; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Magnesium; Male; Membrane Potentials; Microinjections; Oocytes; Palaemonidae; Patch-Clamp Techniques; Receptors, Cytoplasmic and Nuclear; Sulfonamides; Trifluoperazine | 2001 |
Inhibition of the type 1 inositol 1,4,5-trisphosphate-sensitive Ca2+ channel by calmodulin antagonists.
Topics: Animals; Calcium Channels; Calmodulin; Cerebellum; Chlorpromazine; Dose-Response Relationship, Drug; Fluphenazine; Imidazoles; In Vitro Techniques; Inositol 1,4,5-Trisphosphate Receptors; Microsomes; Phenothiazines; Receptors, Cytoplasmic and Nuclear; Swine; Trifluoperazine | 2001 |
Inhibition of calcium-independent luminal uptake of L-dopa by calmodulin antagonists in immortalized rat capillary cerebral endothelial cells.
Topics: Amino Acids, Cyclic; Aminoisobutyric Acids; Animals; Biological Transport; Calcium Channels, L-Type; Calmodulin; Cell Line; Cell Survival; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP-Dependent Protein Kinases; Endothelium, Vascular; Enzyme Inhibitors; Hydrogen-Ion Concentration; Imidazoles; Inhibitory Concentration 50; Levodopa; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Signal Transduction; Sodium; Telencephalon; Time Factors; Trifluoperazine | 2001 |
Detection of calmodulin-binding proteins and calmodulin-dependent phosphorylation linked to calmodulin-dependent chemotaxis to folic and cAMP in Dictyostelium.
Topics: Animals; Calmodulin; Calmodulin-Binding Proteins; Cell Movement; Chemotaxis; Cyclic AMP; Dictyostelium; Enzyme Inhibitors; Folic Acid; Imidazoles; Phosphorylation; Phosphoserine; Subcellular Fractions; Trifluoperazine | 2001 |
Effect of calmodulin antagonists on the growth and graviresponsiveness of primary roots of maize.
Topics: Biological Transport; Calcium; Calcium Radioisotopes; Calmodulin; Chlorpromazine; Gravitropism; Imidazoles; Indoleacetic Acids; Plant Roots; Time Factors; Trifluoperazine; Tritium; Zea mays | 1992 |
Effect of calmodulin antagonists on phospholipase D activity in SH-SY5Y cells.
Topics: Calmodulin; Carbachol; Cell Line; Cholinergic Agonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycerophospholipids; Imidazoles; Phosphatidic Acids; Phospholipase D; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Trifluoperazine; Tyrosine | 2002 |
Calmodulin antagonists do not inhibit IK(Ca) channels of human erythrocytes.
Topics: Calcium; Calmodulin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Erythrocytes; Humans; Imidazoles; Patch-Clamp Techniques; Potassium Channels, Calcium-Activated; Sulfonamides; Trifluoperazine | 2002 |
Regulation of apical transporter of L-DOPA in human intestinal Caco-2 cells.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Biological Transport; Caco-2 Cells; Calmodulin; Cell Polarity; Dose-Response Relationship, Drug; Humans; Imidazoles; Inhibitory Concentration 50; Levodopa; Logistic Models; Membrane Transport Proteins; Time Factors; Trifluoperazine | 2002 |
Ca(2+)-calmodulin regulates receptor-operated Ca(2+) entry activity of TRPC6 in HEK-293 cells.
Topics: Calcium; Calcium Channels; Calmodulin; Cell Line; Humans; Imidazoles; Ion Channel Gating; Ion Transport; Trifluoperazine; TRPC Cation Channels; TRPC6 Cation Channel | 2002 |
Regulation of glutamatergic neurotransmission in the striatum by presynaptic adenylyl cyclase-dependent processes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Bucladesine; Calcium; Calmodulin; Corpus Striatum; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Feedback; Female; Glutamic Acid; Imidazoles; Imines; Isoenzymes; Isoproterenol; Isoquinolines; Kainic Acid; Male; Mice; N-Methylaspartate; Nerve Tissue Proteins; Propranolol; Receptors, Adrenergic, beta; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Presynaptic; Second Messenger Systems; Sulfonamides; Synaptic Transmission; Trifluoperazine | 2003 |
Functional and genetic characterization of calmodulin from the dimorphic and pathogenic fungus Paracoccidioides brasiliensis.
Topics: Amino Acid Sequence; Base Sequence; Calmodulin; Chelating Agents; DNA, Fungal; Egtazic Acid; Fungal Proteins; Gene Dosage; Genes, Fungal; Genome, Fungal; Imidazoles; Introns; Molecular Sequence Data; Mycelium; Paracoccidioides; Sequence Alignment; Sequence Homology; Trifluoperazine; Yeasts | 2003 |
Interference of calmidazolium with measurement of mitochondrial membrane potential using the tetraphenylphosphonium electrode or the fluorescent probe rhodamine 123.
Topics: Animals; Calcium; Calibration; Calmodulin; Dose-Response Relationship, Drug; Electrochemistry; Electrodes; Enzyme Inhibitors; Fluorescent Dyes; Imidazoles; Indicators and Reagents; Membrane Potentials; Mitochondria, Liver; Onium Compounds; Organophosphorus Compounds; Rats; Rhodamine 123; Signal Transduction; Time Factors; Trifluoperazine | 2004 |
Calmidazolium and arachidonate activate a calcium entry pathway that is distinct from store-operated calcium influx in HeLa cells.
Topics: Arachidonic Acid; Calcium; Calcium Channels; Calcium Signaling; Calmodulin; Cell Line, Tumor; Cytosol; HeLa Cells; Humans; Imidazoles; Sulfonamides; Trifluoperazine | 2004 |
Differential effect of calmodulin antagonists on MG132-induced mitochondrial dysfunction and cell death in PC12 cells.
Topics: Animals; Calcium; Calmodulin; Caspase 3; Caspases; Cell Count; Cell Death; Cell Size; Cell Survival; Cytochromes c; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Glutathione; Imidazoles; Leupeptins; Mitochondrial Diseases; PC12 Cells; Rats; Reactive Oxygen Species; Sulfonamides; Trifluoperazine | 2005 |
Inhibition of nitric oxide-activated guanylyl cyclase by calmodulin antagonists.
Topics: Animals; Calcium; Calmodulin; Cerebellum; Cyclic GMP; Guanylate Cyclase; Imidazoles; Inhibitory Concentration 50; Nitric Oxide; Nitric Oxide Donors; Phenoxybenzamine; Rats; Rats, Wistar; Signal Transduction; Trifluoperazine | 2009 |
Interactions of Bordetella pertussis adenylyl cyclase toxin CyaA with calmodulin mutants and calmodulin antagonists: comparison with membranous adenylyl cyclase I.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Binding, Competitive; Bordetella pertussis; Calmodulin; Catalysis; Cell Membrane; Dose-Response Relationship, Drug; Enzyme Inhibitors; Escherichia coli; Fluorescence Resonance Energy Transfer; Humans; Imidazoles; Models, Molecular; Molecular Structure; Mutation; Protein Binding; Sulfonamides; Trifluoperazine; Virulence; Whooping Cough | 2012 |
Regulation of NKG2D-ligand cell surface expression by intracellular calcium after HDAC-inhibitor treatment.
Topics: Base Sequence; Calcium Signaling; Calmodulin; Calpain; Cell Line, Tumor; Cell Membrane; Depsipeptides; Galectin 1; Gene Knockdown Techniques; GPI-Linked Proteins; Histone Deacetylase Inhibitors; Humans; Imidazoles; Intercellular Signaling Peptides and Proteins; Jurkat Cells; Ligands; Melanoma; RNA, Small Interfering; Trifluoperazine | 2013 |
Calmodulin inhibition regulates morphological and functional changes related to the actin cytoskeleton in pure microglial cells.
Topics: Actin Cytoskeleton; Animals; Blotting, Western; Calcium-Binding Proteins; Calmodulin; Cell Proliferation; Cell Survival; Cells, Cultured; Central Nervous System Agents; Frontal Lobe; Imidazoles; Immunohistochemistry; Intracellular Space; Ki-67 Antigen; Lipopolysaccharides; Microfilament Proteins; Microglia; Phagocytosis; Rats, Sprague-Dawley; Trifluoperazine | 2016 |
Modifying culture conditions in chemical library screening identifies alternative inhibitors of mycobacteria.
Topics: Antitubercular Agents; Cysteine; Drug Evaluation, Preclinical; Mycobacterium; Mycobacterium smegmatis; Organoselenium Compounds; Selenocysteine; Small Molecule Libraries | 2009 |