caffeine and rolipram

caffeine has been researched along with rolipram in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19903 (13.64)18.7374
1990's9 (40.91)18.2507
2000's3 (13.64)29.6817
2010's6 (27.27)24.3611
2020's1 (4.55)2.80

Authors

AuthorsStudies
Browne, RG; Howard, HR; Koe, BK; Lebel, LA; Sarges, R; Seymour, PA1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Balliano, TL; Barbosa, G; Carvalho, VF; da Silva, BA; de Souza, ET; Lima, LM; Martins, IRR; Martins, MA; Medeiros, MM; Moraes Junior, MO; Nunes, IKDC; Silva, PMR; Silva, SWD1
Bolton, TB; Hering, S; Hughes, AD1
Harvey, JA; Winsky, L1
Rowlands, MW1
Fredholm, BB; Johansson, B; Svenningsson, P1
Byrd, LD; Howell, LL1
Anselmi, E; Catret, M; Cortes, D; D'Ocon, P; Ivorra, MD; Lugnier, C1
Howell, LL1
Eigler, A; Endres, S; Greten, TF; Haslberger, C; Sinha, B; Sullivan, GW1
Howell, LL; Landrum, AM1
Aardal, S; Helle, KB; Lillestłl, IK1
Chen, JF; Coelho, JE; Fredholm, BB; Fu, Y; Karaoz, U; Tillman, A; Weng, Z; Yu, L; Zhang, X1
Fujimoto, K; Kaneda, T; Kubota, T; Nakajyo, S; Shimizu, K; Urakawa, N1
Ballanyi, K; Ruangkittisakul, A1
Bersani, I; Fehrholz, M; Kramer, BW; Kunzmann, S; Speer, CP1
Fehrholz, M; Kunzmann, S; Speer, CP1
Haji, A; Kimura, S; Ohi, Y1
Muñoz, MD; Solís, JM1

Other Studies

22 other study(ies) available for caffeine and rolipram

ArticleYear
4-Amino[1,2,4]triazolo[4,3-a]quinoxalines. A novel class of potent adenosine receptor antagonists and potential rapid-onset antidepressants.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:8

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antidepressive Agents; Behavior, Animal; Caffeine; Cats; Cell Membrane; Cerebral Cortex; Chemical Phenomena; Chemistry; Corpus Striatum; Male; Molecular Structure; Motor Activity; Purinergic Antagonists; Quinoxalines; Rats; Receptors, Purinergic; Sleep; Structure-Activity Relationship; Triazoles

1990
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Identifying off-target effects and hidden phenotypes of drugs in human cells.
    Nature chemical biology, 2006, Volume: 2, Issue:6

    Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship

2006
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Discovery of sulfonyl hydrazone derivative as a new selective PDE4A and PDE4D inhibitor by lead-optimization approach on the prototype LASSBio-448: In vitro and in vivo preclinical studies.
    European journal of medicinal chemistry, 2020, Oct-15, Volume: 204

    Topics: Animals; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Design; Enzyme Inhibitors; Humans; Hydrazones; Hypersensitivity; Lung; Male; Mice

2020
The action of caffeine on inward barium current through voltage-dependent calcium channels in single rabbit ear artery cells.
    Pflugers Archiv : European journal of physiology, 1990, Volume: 416, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Arteries; Barium; Caffeine; Calcium Channels; Cell Membrane; Ear; Electric Conductivity; Female; Ion Channels; Male; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Purinones; Pyrrolidinones; Rabbits; Rolipram; Xanthines

1990
Effects of N6-(L-phenylisopropyl)adenosine, caffeine, theophylline and rolipram on the acquisition of conditioned responses in the rabbit.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Adenosine; Animals; Caffeine; Conditioning, Classical; Dose-Response Relationship, Drug; Drug Interactions; Female; Male; Phenylisopropyladenosine; Pyrrolidinones; Rabbits; Rolipram; Theophylline

1987
Caffeine and panic attacks.
    The British journal of psychiatry : the journal of mental science, 1987, Volume: 150

    Topics: Adult; Caffeine; Fear; Humans; Male; Panic; Phosphodiesterase Inhibitors; Pyrrolidinones; Rolipram

1987
Effect of different xanthines and phosphodiesterase inhibitors on c-fos expression in rat striatum.
    Acta physiologica Scandinavica, 1995, Volume: 154, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Caffeine; Dose-Response Relationship, Drug; Drug Administration Schedule; In Situ Hybridization; Male; Neostriatum; Nicotinic Acids; Phosphodiesterase Inhibitors; Proto-Oncogene Proteins c-fos; Purinones; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram; Xanthines

1995
Effects of CGS 15943, a nonxanthine adenosine antagonist, on behavior in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:1

    Topics: Animals; Behavior, Animal; Caffeine; Drug Interactions; Drug Synergism; Male; Purinergic P1 Receptor Antagonists; Pyrrolidinones; Quinazolines; Receptors, Purinergic P1; Rolipram; Saimiri; Time Factors; Triazoles

1993
Investigations of the dual contractile/relaxant properties showed by antioquine in rat aorta.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Alkaloids; Animals; Aorta, Thoracic; Benzylisoquinolines; Caffeine; Calcium; Calcium Channel Blockers; Cattle; Cytosol; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; Radioligand Assay; Rats; Rats, Wistar; Receptors, Drug; Rolipram

1993
Effects of adenosine agonists on ventilation during hypercapnia, hypoxia and hyperoxia in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Carbon Dioxide; Female; Hypercapnia; Hypoxia; Macaca mulatta; Male; Oxygen; Phenethylamines; Plethysmography; Pyrrolidinones; Receptors, Purinergic; Respiration; Respiratory Function Tests; Rolipram

1993
Endogenous adenosine curtails lipopolysaccharide-stimulated tumour necrosis factor synthesis.
    Scandinavian journal of immunology, 1997, Volume: 45, Issue:2

    Topics: Adenosine; Adenosine Deaminase; Caffeine; Dipyridamole; Humans; Inosine; Leukocytes, Mononuclear; Lipopolysaccharides; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Antagonists; Pyrrolidinones; Rolipram; Tumor Necrosis Factor-alpha; Xanthines

1997
Effects of chronic caffeine administration on respiration and schedule-controlled behavior in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 283, Issue:1

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Caffeine; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Tolerance; Female; Macaca mulatta; Male; Pyrrolidinones; Respiration; Rolipram; Theophylline

1997
Relaxing effects of cyclic GMP and cyclic AMP-enhancing agents on the long-lasting contraction to endothelin-1 in the porcine coronary artery.
    Scandinavian journal of clinical and laboratory investigation, 1998, Volume: 58, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atrial Natriuretic Factor; Caffeine; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Endothelin-1; In Vitro Techniques; Isradipine; Milrinone; Muscle, Smooth, Vascular; Papaverine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Purinones; Pyrrolidinones; Rolipram; Swine; Vasoactive Intestinal Peptide; Vasoconstriction; Vasodilation; Verapamil; Vinca Alkaloids

1998
Uncovering multiple molecular targets for caffeine using a drug target validation strategy combining A 2A receptor knockout mice with microarray profiling.
    Physiological genomics, 2009, May-13, Volume: 37, Issue:3

    Topics: Animals; Bicuculline; Caffeine; Central Nervous System Stimulants; Cluster Analysis; Dose-Response Relationship, Drug; Female; GABA Antagonists; Gene Expression Profiling; Gene Expression Regulation; Male; Mice; Mice, Knockout; Neostriatum; Oligonucleotide Array Sequence Analysis; Phosphodiesterase Inhibitors; Receptor, Adenosine A2A; Reverse Transcriptase Polymerase Chain Reaction; Rolipram

2009
Effects of rolipram on U46619-induced contraction and cyclic nucleotide content in the porcine coronary artery.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2010, Volume: 46, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Aorta; Caffeine; Calcium; Carotid Arteries; Coronary Vessels; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle Tonus; Nucleotides, Cyclic; Phosphodiesterase Inhibitors; Potassium; Rolipram; Swine; Vasoconstrictor Agents

2010
Methylxanthine reversal of opioid-evoked inspiratory depression via phosphodiesterase-4 blockade.
    Respiratory physiology & neurobiology, 2010, Jul-31, Volume: 172, Issue:3

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Analgesics, Opioid; Animals; Animals, Newborn; Caffeine; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Fentanyl; In Vitro Techniques; Interneurons; Nerve Net; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Opioid, mu; Respiratory Insufficiency; Respiratory Physiological Phenomena; Rolipram; Theophylline; Xanthines

2010
Synergistic effect of caffeine and glucocorticoids on expression of surfactant protein B (SP-B) mRNA.
    PloS one, 2012, Volume: 7, Issue:12

    Topics: Caffeine; Cell Line, Tumor; Dexamethasone; Drug Synergism; Flow Cytometry; Gene Expression Regulation; Glucocorticoids; Homeostasis; Humans; Immunoblotting; Promoter Regions, Genetic; Pulmonary Surfactant-Associated Protein B; Receptors, Glucocorticoid; RNA, Messenger; Rolipram; Transcription Factors

2012
Caffeine and rolipram affect Smad signalling and TGF-β1 stimulated CTGF and transgelin expression in lung epithelial cells.
    PloS one, 2014, Volume: 9, Issue:5

    Topics: Airway Remodeling; Caffeine; Cell Line, Tumor; Connective Tissue Growth Factor; Down-Regulation; Epithelial Cells; Gene Expression Regulation; Humans; Lung; Microfilament Proteins; Muscle Proteins; Promoter Regions, Genetic; Rolipram; Signal Transduction; Smad Proteins; Transforming Growth Factor beta1; Up-Regulation

2014
Blockade of phosphodiesterase 4 reverses morphine-induced ventilatory disturbance without loss of analgesia.
    Life sciences, 2015, Apr-15, Volume: 127

    Topics: Analgesics, Opioid; Animals; Caffeine; Male; Morphine; Pain Measurement; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Phrenic Nerve; Rats; Rats, Wistar; Respiration Disorders; Respiratory Mechanics; Rolipram; Vagotomy

2015
Characterisation of the mechanisms underlying the special sensitivity of the CA2 hippocampal area to adenosine receptor antagonists.
    Neuropharmacology, 2019, Volume: 144

    Topics: Adenylyl Cyclases; Animals; CA1 Region, Hippocampal; CA2 Region, Hippocampal; Caffeine; Colforsin; Excitatory Postsynaptic Potentials; Male; Phosphodiesterase Inhibitors; Purinergic Agonists; Purinergic P1 Receptor Antagonists; Rats, Sprague-Dawley; Receptor, Adenosine A1; Rolipram; Synapses; Tissue Culture Techniques; Xanthines

2019