caffeine and nitrendipine

caffeine has been researched along with nitrendipine in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-19903 (9.09)18.7374
1990's9 (27.27)18.2507
2000's10 (30.30)29.6817
2010's10 (30.30)24.3611
2020's1 (3.03)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Coassolo, P; Lavé, T; Schneider, G1
Topliss, JG; Yoshida, F1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Campillo, NE; Guerra, A; Páez, JA1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Sen, S; Sinha, N1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Barber, S; Dew, TP; Farrell, TL; Poquet, L; Williamson, G1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1
Biguad, M; Julou-Schaeffer, G; Parratt, JR; Stoclet, JC1
Fesce, R; Malgaroli, A; Meldolesi, J1
Baró, I; Escande, D1
Billing, B; Bratel, T; Dahlqvist, R1
Chapunoff, D; Herman, CA; Romero, MA; Schulmeister, K; Skarda, S; Torres, OA1
Cohen, ML; Cox, DA1
Andriantsitohaina, R; Lagaud, GJ; Stoclet, JC1
López, JR; Terzic, A1
Dayanithi, G; Scamps, F; Valentin, S; Valmier, J1
Guan, Z; Saqr, HE; Stokes, BT; Yates, AJ1
Anselmi, E; Bermejo, A; Cabedo, N; Catret, M; Cortes, D; D'Ocon, P; Elorriaga, M; Ivorra, MD; Magraner, J; Tur, R1
Buchan, AM; Meloche, RM; Ring, M; Squires, PE1
Camello, PJ; Gomez-Pinilla, PJ; Pozo, MJ1
Barnes, WS; Kim, JH; Kwak, HB; Lawler, JM1
Brightling, CE; Challiss, RA; Gomez, E; Hollins, F; Saunders, R; Sweeney, D1

Reviews

1 review(s) available for caffeine and nitrendipine

ArticleYear
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022

Other Studies

32 other study(ies) available for caffeine and nitrendipine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Combining in vitro and in vivo pharmacokinetic data for prediction of hepatic drug clearance in humans by artificial neural networks and multivariate statistical techniques.
    Journal of medicinal chemistry, 1999, Dec-16, Volume: 42, Issue:25

    Topics: Animals; Biological Availability; Dogs; Humans; Least-Squares Analysis; Liver; Multivariate Analysis; Neural Networks, Computer; Pharmacokinetics; Rats

1999
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Predicting phenolic acid absorption in Caco-2 cells: a theoretical permeability model and mechanistic study.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:2

    Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Cinnamates; Enterocytes; Humans; Hydrophobic and Hydrophilic Interactions; Intestinal Absorption; Kinetics; Models, Biological; Molecular Conformation; Osmolar Concentration; Phenols

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Endotoxin-induced impairment of vascular smooth muscle contractions elicited by different mechanisms.
    European journal of pharmacology, 1990, Nov-06, Volume: 190, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Caffeine; Calcimycin; Calcium; Clonidine; Endothelium, Vascular; Endotoxins; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitrendipine; Phenylephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Sarcoplasmic Reticulum

1990
Spontaneous [Ca2+]i fluctuations in rat chromaffin cells do not require inositol 1,4,5-trisphosphate elevations but are generated by a caffeine- and ryanodine-sensitive intracellular Ca2+ store.
    The Journal of biological chemistry, 1990, Feb-25, Volume: 265, Issue:6

    Topics: Adrenal Medulla; Alkaloids; Bradykinin; Caffeine; Calcium; Egtazic Acid; Histamine; Inositol 1,4,5-Trisphosphate; Kinetics; Membrane Potentials; Neomycin; Nitrendipine; Ryanodine; Spectrometry, Fluorescence

1990
A long lasting Ca2+-activated outward current in guinea-pig atrial myocytes.
    Pflugers Archiv : European journal of physiology, 1989, Volume: 415, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Apamin; Atrial Function; Caffeine; Calcium; Calcium Channels; Cobalt; Electric Conductivity; Guinea Pigs; Heart; Kinetics; Nitrendipine; Potassium Channels; Quinine; Ryanodine

1989
Felodipine reduces the absorption of theophylline in man.
    European journal of clinical pharmacology, 1989, Volume: 36, Issue:5

    Topics: Adult; Blood Pressure; Caffeine; Calcium Channel Blockers; Drug Interactions; Felodipine; Humans; Intestinal Absorption; Male; Nitrendipine; Theophylline

1989
Leukotriene C4-stimulated contractions in bullfrog lung are affected by cold acclimation and calcium antagonists.
    Prostaglandins, 1995, Volume: 49, Issue:2

    Topics: Acclimatization; Animals; Caffeine; Calcium Channel Blockers; Calcium-Transporting ATPases; Cold Temperature; Contracture; Egtazic Acid; Eicosapentaenoic Acid; Female; Hot Temperature; Leukotriene C4; Lung; Male; Nicardipine; Nifedipine; Nitrendipine; Rana catesbeiana; SRS-A; Terpenes; Thapsigargin; Verapamil

1995
5-Hydroxytryptamine2B receptor signaling in rat stomach fundus: role of voltage-dependent calcium channels, intracellular calcium release and protein kinase C.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:1

    Topics: Animals; Caffeine; Calcium; Calcium Channels; Carbachol; Gastrointestinal Motility; In Vitro Techniques; Indoles; Male; Maleimides; Membrane Potentials; Muscle Contraction; Nitrendipine; Protein Kinase C; Rats; Rats, Wistar; Receptors, Serotonin; Ryanodine; Serotonin; Signal Transduction; Stomach

1995
Calcium handling and purinoceptor subtypes involved in ATP-induced contraction in rat small mesenteric arteries.
    The Journal of physiology, 1996, May-01, Volume: 492 ( Pt 3)

    Topics: Adenosine Triphosphate; Animals; Caffeine; Calcium; Calcium Channel Blockers; Imidazoles; Male; Mesenteric Arteries; Muscle Contraction; Nitrendipine; Pertussis Toxin; Platelet Aggregation Inhibitors; Purinergic Agonists; Purinergic Antagonists; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Purinergic; Terpenes; Thapsigargin; Vascular Resistance; Virulence Factors, Bordetella

1996
Inositol 1,4,5-trisphosphate-induced Ca2+ release is regulated by cytosolic Ca2+ in intact skeletal muscle.
    Pflugers Archiv : European journal of physiology, 1996, Volume: 432, Issue:5

    Topics: Animals; Caffeine; Calcium; Cytosol; Dantrolene; Heparin; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Magnesium; Membrane Potentials; Microinjections; Muscle, Skeletal; Nitrendipine; Rana temporaria; Ruthenium Red

1996
Calcium channel subtypes responsible for voltage-gated intracellular calcium elevations in embryonic rat motoneurons.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Central Nervous System Stimulants; Electric Stimulation; Fetus; Ion Channel Gating; Membrane Potentials; Motor Neurons; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; Patch-Clamp Techniques; Peptides; Potassium Chloride; Rats; Rats, Sprague-Dawley; Ryanodine; Spider Venoms

1998
Mechanisms through which PDGF alters intracellular calcium levels in U-1242 MG human glioma cells.
    Neurochemistry international, 1999, Volume: 35, Issue:6

    Topics: Becaplermin; Brain Neoplasms; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Elapid Venoms; Endoplasmic Reticulum; Enzyme Inhibitors; Flufenamic Acid; Glioma; Humans; Imidazoles; Ion Transport; Masoprocol; Neoplasm Proteins; Nicardipine; Nimodipine; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Peptides; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Ryanodine; Thapsigargin; Tumor Cells, Cultured; Verapamil

1999
Mechanism of vascular relaxation by thaligrisine: functional and binding assays.
    Life sciences, 2000, Aug-18, Volume: 67, Issue:13

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkaloids; Animals; Aorta, Thoracic; Arteries; Binding Sites; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Cortex; Diltiazem; Female; In Vitro Techniques; Membranes; Muscle Relaxation; Muscle, Smooth, Vascular; Nitrendipine; Norepinephrine; Potassium Chloride; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tail; Trees; Tritium; Vasoconstrictor Agents

2000
Mechanism of action of the calcium-sensing receptor in human antral gastrin cells.
    Gastroenterology, 2001, Volume: 120, Issue:5

    Topics: Adenine; Caffeine; Calcium; Calcium Channel Blockers; Cells, Cultured; Cyclic AMP; DNA Primers; Enzyme Inhibitors; Gastric Mucosa; Gastrins; Gene Expression; Humans; Indoles; Maleimides; Nitrendipine; ortho-Aminobenzoates; Phosphodiesterase Inhibitors; Protein Kinase C; Pyloric Antrum; Receptors, Calcium-Sensing; Receptors, Cell Surface; RNA, Messenger; Signal Transduction

2001
Protective effect of melatonin on Ca2+ homeostasis and contractility in acute cholecystitis.
    Journal of pineal research, 2008, Volume: 44, Issue:3

    Topics: Acalculous Cholecystitis; Animals; Caffeine; Calcium; Cholecystitis, Acute; Common Bile Duct; Disease Models, Animal; Gallbladder; Guinea Pigs; Homeostasis; Ligation; Lipid Peroxidation; Male; Melatonin; Muscle Contraction; Nitrendipine; Pinacidil; Thapsigargin

2008
Redox modulation of diaphragm contractility: Interaction between DHPR and RyR channels.
    Free radical biology & medicine, 2010, Dec-15, Volume: 49, Issue:12

    Topics: Animals; Antioxidants; Caffeine; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Diaphragm; Dithiothreitol; In Vitro Techniques; Male; Muscle Contraction; Nitrendipine; Organometallic Compounds; Oxidation-Reduction; Oxidative Stress; Procaine; Rats; Rats, Inbred F344; Reactive Oxygen Species; Reducing Agents; Ruthenium Red; Ryanodine Receptor Calcium Release Channel; Salicylates; Xanthine Oxidase

2010
[Ca2+]i oscillations in ASM: relationship with persistent airflow obstruction in asthma.
    Respirology (Carlton, Vic.), 2014, Volume: 19, Issue:5

    Topics: Adult; Aged; Asthma; Biopsy; Caffeine; Calcium Signaling; Case-Control Studies; Female; Forced Expiratory Volume; Humans; Male; Middle Aged; Muscle, Smooth; Nitrendipine; Pulmonary Disease, Chronic Obstructive; Respiratory Muscles; Severity of Illness Index; Verapamil; Vital Capacity

2014