caffeine and nicardipine

caffeine has been researched along with nicardipine in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.70)18.7374
1990's13 (35.14)18.2507
2000's14 (37.84)29.6817
2010's8 (21.62)24.3611
2020's1 (2.70)2.80

Authors

AuthorsStudies
Coassolo, P; Lavé, T; Schneider, G1
Topliss, JG; Yoshida, F1
Jolivette, LJ; Ward, KW1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1
Somasundaram, B; Tregear, RT; Trentham, DR1
Chang, CC; Hong, SJ; Huang, CY1
Hatae, J; Kawata, H1
Fujino, M; Sato, Y1
Chapunoff, D; Herman, CA; Romero, MA; Schulmeister, K; Skarda, S; Torres, OA1
Ogihara, M1
Gerthoffer, WT; Publicover, NG; Sanders, KM; Sato, K1
Hata, S; Ishii, K; Ishiro, H; Nakayama, K; Tanaka, Y1
Advenier, C; Candenas, ML; Martin, JD; Moreau, J; Naline, E; Norte, M; Palette, C; Pays, M1
Itoh, T; Kanmura, Y; Ohashi, M; Shiraishi, Y; Yamaguchi, S; Yoshimura, N1
Hiraoka, M; Kawano, S; Kuruma, A1
Thayer, SA; Usachev, YM1
Guan, Z; Saqr, HE; Stokes, BT; Yates, AJ1
Cameron, JS; Coyne, MD; Gwathmey, JK; Kim, CS1
Nobe, H; Nobe, K; Obara, K; Paul, RJ1
Nishi, K; Tokutomi, N; Tokutomi, Y1
Jin, NG; Li, L; Li, Y; Li, ZL; Piao, L; Xu, WX1
Fujita, A; Hata, F; Hirayama, N; Kitayama, M; Sumiyoshi, M; Takeuchi, T1
Hong, SJ; Liang, HC; Shen, CJ1
Cho, MC; Choi, MY; Choi, W; Hwang, KK; Kim, KW; Kim, YC; Lee, SJ; Lim, SW; Park, JK; Sim, JH1
Fleming, NW; Hennig, GW; Keef, KD; Lee, HT; Sanders, KM; Smith, TK; Spencer, NJ; Ward, SM1
Hashitani, H; Suzuki, H1
Callison, CR; Kumar, AB; Miller, M1
Lopatin, AN; Moench, I1

Reviews

2 review(s) available for caffeine and nicardipine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022

Other Studies

35 other study(ies) available for caffeine and nicardipine

ArticleYear
Combining in vitro and in vivo pharmacokinetic data for prediction of hepatic drug clearance in humans by artificial neural networks and multivariate statistical techniques.
    Journal of medicinal chemistry, 1999, Dec-16, Volume: 42, Issue:25

    Topics: Animals; Biological Availability; Dogs; Humans; Least-Squares Analysis; Liver; Multivariate Analysis; Neural Networks, Computer; Pharmacokinetics; Rats

1999
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Extrapolation of human pharmacokinetic parameters from rat, dog, and monkey data: Molecular properties associated with extrapolative success or failure.
    Journal of pharmaceutical sciences, 2005, Volume: 94, Issue:7

    Topics: Algorithms; Animals; Dogs; Haplorhini; Humans; Pharmaceutical Preparations; Pharmacokinetics; Rats; Species Specificity; Tissue Distribution

2005
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
GTP gamma S causes contraction of skinned frog skeletal muscle via the DHP-sensitive Ca2+ channels of sealed T-tubules.
    Pflugers Archiv : European journal of physiology, 1991, Volume: 418, Issue:1-2

    Topics: Animals; Binding Sites; Binding, Competitive; Caffeine; Calcium Channels; Dihydropyridines; Egtazic Acid; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Microtubules; Muscle Contraction; Nicardipine; Pertussis Toxin; Photolysis; Rana pipiens; Rana temporaria; Virulence Factors, Bordetella

1991
Organic calcium channel antagonists provoke acetylcholine receptor autodesensitization on train stimulation of motor nerve.
    Neuroscience, 1990, Volume: 38, Issue:3

    Topics: Animals; Bungarotoxins; Caffeine; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Diaphragm; Egtazic Acid; Electric Stimulation; Electrophysiology; Mice; Motor Endplate; Muscle Contraction; Neostigmine; Nicardipine; Phrenic Nerve; Receptors, Cholinergic; Theophylline

1990
Dependence of contractile responses by some calcium antagonists on external calcium in the skeletal muscle.
    The Japanese journal of physiology, 1990, Volume: 40, Issue:3

    Topics: Animals; Caffeine; Calcium; Membrane Potentials; Muscle Contraction; Muscles; Nicardipine; Ranidae; Verapamil

1990
Inhibition of excitation-contraction coupling by a Ca channel blocker nicardipine at low temperature in frog twitch fibers.
    The Japanese journal of physiology, 1987, Volume: 37, Issue:1

    Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Cold Temperature; Electrophysiology; Muscle Contraction; Nicardipine; Potassium; Ranidae

1987
Leukotriene C4-stimulated contractions in bullfrog lung are affected by cold acclimation and calcium antagonists.
    Prostaglandins, 1995, Volume: 49, Issue:2

    Topics: Acclimatization; Animals; Caffeine; Calcium Channel Blockers; Calcium-Transporting ATPases; Cold Temperature; Contracture; Egtazic Acid; Eicosapentaenoic Acid; Female; Hot Temperature; Leukotriene C4; Lung; Male; Nicardipine; Nifedipine; Nitrendipine; Rana catesbeiana; SRS-A; Terpenes; Thapsigargin; Verapamil

1995
Nifedipine and nicardipine potentiate glucagon-stimulated glycogenolysis in primary cultures of rat hepatocytes.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:9

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Caffeine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Glucagon; Glycogen; Liver; Male; Nicardipine; Nifedipine; Papaverine; Rats; Rats, Wistar

1993
Sources of calcium utilized in cholinergic responses in canine colonic smooth muscle.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 1

    Topics: Acetylcholine; Animals; Caffeine; Calcium; Colon; Dogs; Female; Male; Muscle Contraction; Muscle, Smooth; Nicardipine; Ryanodine

1994
Stretching releases Ca2+ from intracellular storage sites in canine cerebral arteries.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:1

    Topics: Animals; Basilar Artery; Caffeine; Calcium; Calcium Channel Blockers; Carbamates; Cholera Toxin; Dogs; Female; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Phenylcarbamates; Ryanodine; Temperature; Type C Phospholipases; Virulence Factors, Bordetella

1994
Effects of okadaic acid on the human isolated bronchus.
    European journal of pharmacology, 1994, May-02, Volume: 256, Issue:3

    Topics: Acetylcholine; Bronchi; Cadmium; Cadmium Compounds; Caffeine; Dose-Response Relationship, Drug; Ethers, Cyclic; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Nicardipine; Okadaic Acid; Papaverine; Phosphatidylinositols; Potassium Chloride; Sulfates; Vasoconstrictor Agents

1994
Possible mechanisms underlying the midazolam-induced relaxation of the noradrenaline-contraction in rabbit mesenteric resistance artery.
    British journal of pharmacology, 1997, Volume: 121, Issue:6

    Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; Midazolam; Muscle Contraction; Muscle Relaxation; Nicardipine; Norepinephrine; Potassium; Rabbits; Vascular Resistance; Vasodilator Agents

1997
Activation of Ca2+-sensitive Cl- current by reverse mode Na+/Ca2+ exchange in rabbit ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 1998, Volume: 436, Issue:6

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Caffeine; Calcium; Chloride Channels; Electric Conductivity; Female; Heart; Heart Ventricles; Kinetics; Male; Nicardipine; Patch-Clamp Techniques; Rabbits; Ryanodine; Sarcoplasmic Reticulum; Sodium; Sodium-Calcium Exchanger; Thapsigargin; Ventricular Function

1998
Ca2+ influx in resting rat sensory neurones that regulates and is regulated by ryanodine-sensitive Ca2+ stores.
    The Journal of physiology, 1999, Aug-15, Volume: 519 Pt 1

    Topics: Action Potentials; Animals; Animals, Newborn; Biological Transport; Caffeine; Calcium; Calcium Channel Blockers; Cells, Cultured; Ganglia, Spinal; Membrane Potentials; Neurons, Afferent; Nicardipine; Nimodipine; Patch-Clamp Techniques; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Ryanodine; Ryanodine Receptor Calcium Release Channel

1999
Mechanisms through which PDGF alters intracellular calcium levels in U-1242 MG human glioma cells.
    Neurochemistry international, 1999, Volume: 35, Issue:6

    Topics: Becaplermin; Brain Neoplasms; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Elapid Venoms; Endoplasmic Reticulum; Enzyme Inhibitors; Flufenamic Acid; Glioma; Humans; Imidazoles; Ion Transport; Masoprocol; Neoplasm Proteins; Nicardipine; Nimodipine; Nitrendipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Peptides; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Ryanodine; Thapsigargin; Tumor Cells, Cultured; Verapamil

1999
Effects of temperature and calcium availability on ventricular myocardium from rainbow trout.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 278, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Adrenergic beta-Agonists; Animals; Body Temperature; Cadmium; Caffeine; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Central Nervous System Stimulants; Cold Temperature; Heart Ventricles; Isometric Contraction; Isoproterenol; Myocardial Contraction; Myocardium; Nicardipine; Oncorhynchus mykiss; Oxygen Consumption; Patch-Clamp Techniques; Ryanodine; Sarcolemma; Ventricular Function

2000
Preferential role of intracellular Ca2+ stores in regulation of isometric force in NIH 3T3 fibroblast fibres.
    The Journal of physiology, 2000, Dec-15, Volume: 529 Pt 3

    Topics: 3T3 Cells; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Cattle; Drug Synergism; Endoplasmic Reticulum; Enzyme Inhibitors; Estrenes; Fibroblasts; Indoles; Intracellular Membranes; Mice; Nicardipine; Potassium Chloride; Pyrrolidinones; Ryanodine; Thapsigargin; Type C Phospholipases

2000
The properties of ryanodine-sensitive Ca(2+) release in mouse gastric smooth muscle cells.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: Animals; Bucladesine; Caffeine; Calcium; Carbachol; Cells, Cultured; Dose-Response Relationship, Drug; Electric Conductivity; Fura-2; Gastric Mucosa; In Vitro Techniques; Ion Channel Gating; Isometric Contraction; Large-Conductance Calcium-Activated Potassium Channels; Mice; Mice, Inbred BALB C; Muscle Relaxation; Muscle, Smooth; Nicardipine; Potassium; Potassium Channels; Potassium Channels, Calcium-Activated; Potassium Chloride; Ryanodine; Stomach; Tetraethylammonium

2001
The involvement of calcium mobilization in the calcium-activated potassium currents activated by hyposmotic swelling in gastric antral circular myocytes of the guinea-pig.
    The Japanese journal of physiology, 2001, Volume: 51, Issue:2

    Topics: Animals; Caffeine; Calcium Channel Blockers; Central Nervous System Stimulants; Female; Gadolinium; Guinea Pigs; Male; Muscle, Smooth; Myocardium; Nicardipine; Osmotic Pressure; Patch-Clamp Techniques; Potassium Channels; Pyloric Antrum; Ryanodine; Stomach

2001
Origin of Ca2+ necessary for carbachol-induced contraction in longitudinal muscle of the proximal colon of rats.
    Japanese journal of pharmacology, 2001, Volume: 87, Issue:4

    Topics: Aminobenzoates; Animals; Caffeine; Calcium; Calcium Channel Blockers; Carbachol; Chlorobenzoates; Cinnamates; Colon; Enzyme Inhibitors; Gastrointestinal Motility; Male; Muscle Contraction; Muscle, Smooth; Nicardipine; ortho-Aminobenzoates; Parasympathomimetics; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Thapsigargin

2001
Alteration of cyclopiazonic acid-mediated contracture of mouse diaphragm after denervation.
    Pharmacology, 2005, Volume: 73, Issue:4

    Topics: Action Potentials; Animals; Biological Assay; Boron Compounds; Caffeine; Cromakalim; Crotalid Venoms; Diaphragm; Electric Stimulation; Estrenes; Female; Glyburide; Indoles; Male; Membrane Potentials; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle Denervation; Nicardipine; Phrenic Nerve; Pyrrolidinones; Sarcoplasmic Reticulum

2005
Regulation of membrane excitability by intracellular pH (pHi) changers through Ca2+-activated K+ current (BK channel) in single smooth muscle cells from rabbit basilar artery.
    Pflugers Archiv : European journal of physiology, 2007, Volume: 454, Issue:2

    Topics: Ammonium Chloride; Animals; Basilar Artery; Caffeine; Calcium; Calcium Channel Blockers; Calcium Signaling; Cytoplasm; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Hydrogen-Ion Concentration; Isometric Contraction; Large-Conductance Calcium-Activated Potassium Channels; Membrane Potentials; Myocytes, Smooth Muscle; Nicardipine; Rabbits; Sodium Acetate; Tetraethylammonium

2007
The mechanism and spread of pacemaker activity through myenteric interstitial cells of Cajal in human small intestine.
    Gastroenterology, 2007, Volume: 132, Issue:5

    Topics: Adult; Biological Clocks; Caffeine; Calcium; Calcium Channel Blockers; Central Nervous System Stimulants; Electrophysiology; Female; Humans; In Vitro Techniques; Inositol 1,4,5-Trisphosphate Receptors; Intestinal Mucosa; Jejunum; Male; Middle Aged; Myenteric Plexus; Myocytes, Smooth Muscle; Nicardipine

2007
Properties of spontaneous Ca2+ transients recorded from interstitial cells of Cajal-like cells of the rabbit urethra in situ.
    The Journal of physiology, 2007, Sep-01, Volume: 583, Issue:Pt 2

    Topics: Adrenergic alpha-Agonists; Animals; Boron Compounds; Caffeine; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Signaling; Calcium-Transporting ATPases; Enzyme Inhibitors; Indoles; Inositol 1,4,5-Trisphosphate Receptors; Male; Membrane Potentials; Molsidomine; Muscle Contraction; Myocytes, Smooth Muscle; Nicardipine; Nitric Oxide; Nitric Oxide Donors; Phenylephrine; Rabbits; Receptors, Adrenergic, alpha; Ryanodine; Ryanodine Receptor Calcium Release Channel; Time Factors; Urethra

2007
Refractory caffeine and ergot-induced cervico-cerebral vasospasm and stroke treated with combined medical and endovascular approach.
    Neuroradiology, 2012, Volume: 54, Issue:1

    Topics: Adult; Caffeine; Cerebral Angiography; Dihydroergotamine; Drug Therapy, Combination; Female; Humans; Magnetic Resonance Angiography; Migraine Disorders; Nicardipine; Phosphodiesterase Inhibitors; Stents; Stroke; Vasoconstrictor Agents; Vasodilator Agents; Vasospasm, Intracranial

2012
Ca(2+) homeostasis in sealed t-tubules of mouse ventricular myocytes.
    Journal of molecular and cellular cardiology, 2014, Volume: 72

    Topics: Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cells, Cultured; Cytoplasm; Dinitrophenols; Heart Ventricles; Homeostasis; Ion Transport; Membrane Potentials; Mice; Myocytes, Cardiac; Nicardipine; Potassium; Sarcolemma; Uncoupling Agents

2014