caffeine has been researched along with gamma-aminobutyric acid in 79 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 15 (18.99) | 18.7374 |
1990's | 13 (16.46) | 18.2507 |
2000's | 19 (24.05) | 29.6817 |
2010's | 26 (32.91) | 24.3611 |
2020's | 6 (7.59) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Giralt, E; Malakoutikhah, M; Prades, R; Teixidó, M | 1 |
Bornstein, MB; Corrigall, WA; Crain, SM | 1 |
Markovich, VV; Molodavkin, GM; Ostrovskaia, RU | 1 |
Feltz, P; Mouginot, D; Schlichter, R | 1 |
Farb, DH; Friedman, L; Gibbs, TT; Roca, DJ; Rozenberg, I; Schiller, GD | 1 |
Missak, SS | 1 |
Boux, O; Desaulles, E; Feltz, P | 1 |
Dohi, T; Kitayama, S; Morita, K; Tsujimoto, A | 1 |
Costa, E; Guidotti, A | 1 |
Hosoda, K; Matsumoto, S; Shirakawa, J; Tanaka, C; Taniyama, K | 1 |
Farb, DH; Roca, DJ; Schiller, GD | 1 |
Amalric, M; Koob, GF; Swerdlow, NR; Vaccarino, FJ | 1 |
Ferrario, P; Mantegazza, P; Zambotti, F; Zecca, L; Zonta, N | 1 |
Gordon-Weeks, PR; Lockerbie, RO | 1 |
Chesielski, L; Kempf, E; Lehmann, A; Maitre, M; Mandel, P | 1 |
Berti, C; Nistri, A | 3 |
Paul, SM; Skolnick, P | 1 |
Hollins, C; Lloyd, H; Stone, TW | 1 |
Erickson, CK | 1 |
Akaike, N; Harata, N; Uneyama, H | 1 |
Alastra, AJ; Cohen, C; Goldberg, SR; Marley, RJ; Sannerud, CA; Serdikoff, SL | 1 |
Bingmann, D; Bonnet, U | 1 |
Charney, DS; Deutsch, DN; Krystal, JH | 1 |
Brussaard, AB; de Vlieger, TA; Kits, KS | 1 |
Mukhopadhyay, S; Poddar, MK | 2 |
Akopian, A; Gabriel, R; Witkovsky, P | 1 |
Das, M; Ganguly, DK; Gomes, A; Vedasiromoni, JR | 1 |
Fredholm, BB; Grandy, DK; Hanania, T; Kelly, MA; Larson, GA; Low, MJ; Mayfield, RD; Negri, CA; Rubinstein, M; Simosky, JK; Zahniser, NR | 1 |
Mendonça-Silva, DL; Noël, F; Quintas, LE | 1 |
Kim, SU; Krieger, C; Puil, E; Yokogawa, T | 1 |
Büyükokuroğlu, ME; Demirezer, LO; Güvenalp, Z | 1 |
Lasater, EM; Vigh, J | 1 |
Kiss, T; Molnár, G; Salánki, J | 1 |
An, J; Li, S; Li, ZW; Sun, CK | 1 |
Campusano, JM; Jiang, SA; O'Dowd, DK; Su, H | 1 |
Misgeld, U; Yanovsky, Y; Zhang, W | 1 |
Borges, S; Dalcino, D; Walters, C; Warrier, A; Wilson, M | 1 |
Fischer, W; Franke, H; Gröger-Arndt, H; Günther, A; Illes, P; Köfalvi, A; Madarász, E; Nörenberg, W; Schneider, D; Sperlágh, B; Vizi, ES; Wirkner, K | 1 |
Cao, LH; Yang, XL; Yu, YC | 1 |
Misgeld, U; Velte, S; Yanovsky, Y | 1 |
Coecke, S; Eskes, C; Hartung, T; Honegger, P; Linge, J; Morath, S; Rappsilber, J; van Vliet, E | 1 |
Correa, M; Font, L | 1 |
Grzelak, ME; Hodgson, RA; Hunter, JC; Parker, EM; Pond, AJ; Varty, GB | 1 |
Andrikoula, M; Prelevic, G | 1 |
Patil, T; Raffa, RB; Rawls, SM; Yuvasheva, E | 1 |
Abrams, JK; Hale, MW; Johnson, PL; Lowry, CA; Shekhar, A; Westerman, AM | 1 |
Erol, DD | 1 |
Baulieu, EE; Ghoumari, AM; Levenes, C; Rakotomamonjy, J; Schumacher, M | 1 |
Basurto Ona, X; Bonfill Cosp, X; Martínez García, L; Solà, I | 1 |
Chuang, CH; Ho, CT; Kuo, SC; Lee, MR; Li, YH; Lin, HY; Lin, JN; Way, TD; Yang, NS | 1 |
John, J; Kodama, T; Siegel, JM | 1 |
de Mello, FG; Ferreira, DD; Kubrusly, RC; Reis, RA; Stutz, B | 1 |
Basurto Ona, X; Bonfill Cosp, X; Osorio, D | 1 |
Ge, Y; Huang, Y; Li, Y; Ma, W; Zhao, W | 1 |
Batisti, AP; Daruge-Neto, E; Emer, AA; Martins, DF; Mazzardo-Martins, L; Piovezan, AP; Prado, MR; Santos, AR | 1 |
Bisagno, V; Garcia-Rill, E; Gingrich, JA; Goitia, B; Rivero-Echeto, MC; Urbano, FJ; Weisstaub, NV | 1 |
Bagga, P; Chugani, AN; Patel, AB | 1 |
Hong, KB; Park, Y; Suh, HJ | 1 |
Isokawa, M | 1 |
Andres-Mach, M; Chrościńska-Krawczyk, M; Czuczwar, SJ; Jargiełło-Baszak, M; Łuszczki, JJ | 1 |
Vargas, RA | 1 |
Bernard, C; Esclapez, M; Fazeli, W; Grendel, J; Isbrandt, D; Marguet, SL; Zappettini, S | 1 |
Bendix, I; Bührer, C; Endesfelder, S; Schiller, C; Sifringer, M; Weichelt, U | 1 |
Hew, SA; Ly, J; McKendrick, AM; Nguyen, BN; Shin, HY; Wong, JC; Yeung, E | 1 |
Ahn, SH; Han, SH; Hong, KB; Ko, BS; Noh, DO; Suh, HJ | 1 |
Cheng, S; Guo, Z; He, X; Hu, D; Lu, J; Wang, H; Xu, D; Zhang, C | 1 |
Jonuscheit, M; Lanzman, RS; Oeltzschner, G; Schnitzler, A; Wittsack, HJ; Zöllner, HJ | 1 |
Gilbert, N | 1 |
Deng, Y; Dong, C; Hua, J; Jiang, Y; Li, J; Wang, J; Yang, Y; Yao, Y; Yuan, H; Zhou, Q | 1 |
Borges-Martins, VPP; da Rosa Valli, T; de Melo Reis, RA; de Moura, P; Dos Santos Pereira, M; Ferreira, DDP; Ferreira, GC; Ferreira, MNMR; Kubrusly, RCC; Manhães, AC; Martins, RS; Sathler, MF | 1 |
Ahn, Y; Cho, HJ; Jo, K; Kwak, WK; Min, B; Suh, HJ | 1 |
Kim, H; Kim, YI; Park, BG; Park, I; Park, K; Park, S | 1 |
Dai, S; Guo, Z; He, X; Hu, Z; Jiao, Z; Lu, M; Wang, H; Xu, D | 1 |
Georgiyants, V; Kayal, WE; Mishchenko, M; Severina, H; Shtrygol, D; Shtrygol, S; Zalevskyi, S | 1 |
Ahmad, MF; Akbor, MS; Araújo, IM; Bappi, MH; Coutinho, HDM; Elbendary, EY; Gonçalves, SA; Han, H; Islam, MT; Kamli, H; Lho, LH; Prottay, AAS; Raposo, A; Shaikh, A; Sonia, FA | 1 |
7 review(s) available for caffeine and gamma-aminobutyric acid
Article | Year |
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Endogenous ligands for benzodiazepine recognition sites.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Caffeine; Carrier Proteins; Chlorides; Conflict, Psychological; Diazepam Binding Inhibitor; Flumazenil; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; Hypoxanthine; Hypoxanthines; Inosine; Ion Channels; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neuroglia; Neurons; Niacinamide; Organic Anion Transporters; Peptides; Phosphorylation; Protein Conformation; Protein Precursors; Receptors, GABA-A; Synaptic Membranes; Tissue Distribution; Trypsin | 1985 |
The neural substrates for the motor-activating properties of psychostimulants: a review of recent findings.
Topics: Animals; Apomorphine; Brain; Brain Mapping; Caffeine; Central Nervous System Stimulants; Corticotropin-Releasing Hormone; Dextroamphetamine; Dopamine; Endorphins; gamma-Aminobutyric Acid; Heroin; Mesencephalon; Motor Activity; Neural Pathways; Nucleus Accumbens; Preoptic Area; Rats; Receptors, Dopamine; Substantia Innominata; Synaptic Transmission | 1986 |
The mechanism(s) of action of the benzodiazepines.
Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Caffeine; Carbolines; Cats; Cattle; Diazepam; gamma-Aminobutyric Acid; Humans; Molecular Weight; Muscle Relaxation; Neurotransmitter Agents; Niacinamide; Purines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Sleep Wake Disorders | 1981 |
The biological basis of panic disorder.
Topics: Brain; Caffeine; Carbon Dioxide; gamma-Aminobutyric Acid; Humans; Lactates; Norepinephrine; Panic Disorder; Piperazines; Serotonin; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon | 1996 |
Menopausal hot flushes revisited.
Topics: Acupuncture Therapy; Adult; Alcohol Drinking; Amines; Caffeine; Cyclohexanecarboxylic Acids; Estrogen Replacement Therapy; Estrogens; Exercise; Female; Gabapentin; gamma-Aminobutyric Acid; Hot Flashes; Humans; Menopause; Middle Aged; Phytoestrogens; Smoking | 2009 |
Drug therapy for treating post-dural puncture headache.
Topics: Adrenocorticotropic Hormone; Amines; Analgesics; Caffeine; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Humans; Hydrocortisone; Male; Pain Measurement; Post-Dural Puncture Headache; Randomized Controlled Trials as Topic; Spinal Puncture; Sumatriptan; Theophylline; Treatment Outcome | 2011 |
Drug therapy for treating post-dural puncture headache.
Topics: Adrenocorticotropic Hormone; Adult; Amines; Analgesics; Blood Patch, Epidural; Caffeine; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Humans; Hydrocortisone; Male; Middle Aged; Pain Measurement; Post-Dural Puncture Headache; Randomized Controlled Trials as Topic; Spinal Puncture; Sumatriptan; Theophylline; Treatment Outcome | 2015 |
1 trial(s) available for caffeine and gamma-aminobutyric acid
Article | Year |
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The analgesic and antiemetic efficacy of gabapentin or ergotamine/caffeine for the treatment of postdural puncture headache.
Topics: Adult; Amines; Analgesics, Non-Narcotic; Antiemetics; Caffeine; Cyclohexanecarboxylic Acids; Drug Combinations; Ergotamine; Female; Gabapentin; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Post-Dural Puncture Headache | 2011 |
71 other study(ies) available for caffeine and gamma-aminobutyric acid
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
N-methyl phenylalanine-rich peptides as highly versatile blood-brain barrier shuttles.
Topics: Aminolevulinic Acid; Animals; Animals, Newborn; Astrocytes; Biological Transport; Blood Vessels; Blood-Brain Barrier; Brain; Cattle; Cell Membrane Permeability; Cells, Cultured; Chromatography, High Pressure Liquid; Coculture Techniques; Drug Carriers; Endothelial Cells; gamma-Aminobutyric Acid; Mass Spectrometry; Molecular Structure; Nipecotic Acids; Oligopeptides; Phenylalanine; Rats | 2010 |
Electrophysiological studies of fetal mouse olifactory bulb explants during development of synaptic functions in culture.
Topics: Action Potentials; Animals; Bicuculline; Caffeine; Evoked Potentials; Fetus; gamma-Aminobutyric Acid; Mice; Neural Inhibition; Neurons; Olfactory Bulb; Organ Culture Techniques; Picrotoxin; Synapses; Time Factors; Tubocurarine | 1976 |
[The effect of substnaces altering gamma-aminobutyric acid metabolism on the recovery cycle of the interzonal response of the cat motor cortex].
Topics: Aminobutyrates; Animals; Arecoline; Bemegride; Benactyzine; Bicuculline; Caffeine; Cats; Drug Interactions; Electrophysiology; gamma-Aminobutyric Acid; Motor Cortex; Receptors, Drug; Semicarbazides; Somatosensory Cortex; Sulfhydryl Compounds; Valproic Acid | 1975 |
Modulation of GABA-gated chloride currents by intracellular Ca2+ in cultured porcine melanotrophs.
Topics: Animals; Caffeine; Calcium; Calcium Channels; Cells, Cultured; Chlorides; Electrophysiology; Female; gamma-Aminobutyric Acid; Ion Channel Gating; Pituitary Gland; Pyrrolidonecarboxylic Acid; Swine; Thyrotropin-Releasing Hormone | 1991 |
gamma-Aminobutyric acidA receptor regulation in culture: altered allosteric interactions following prolonged exposure to benzodiazepines, barbiturates, and methylxanthines.
Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Allosteric Regulation; Animals; Barbital; Barbiturates; Brain; Caffeine; Cells, Cultured; Chick Embryo; Flumazenil; Flunitrazepam; Flurazepam; gamma-Aminobutyric Acid; Kinetics; Neurons; Pentobarbital; Receptors, GABA-A; Tetrodotoxin; Theophylline; Veratridine | 1990 |
Exploring the role of an endogenous caffeine-like substance in the pathogenesis of schizophrenia.
Topics: Brain; Caffeine; Female; gamma-Aminobutyric Acid; Humans; Pregnancy; Pregnancy Complications; Receptors, Dopamine; Schizophrenia | 1991 |
Caffeine-induced Ca2+ release inhibits GABAA responsiveness in rat identified native primary afferents.
Topics: Action Potentials; Animals; Caffeine; Calcium; Electric Stimulation; gamma-Aminobutyric Acid; Ganglia, Spinal; In Vitro Techniques; Neurons, Afferent; Rats; Rats, Inbred Strains; Ryanodine | 1991 |
Enhancement by GABA of the stimulation-evoked catecholamine release from cultured bovine adrenal chromaffin cells.
Topics: Acetylcholine; Adrenal Glands; Animals; Bicuculline; Caffeine; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Nicotine; Picrotoxin; Potassium; Receptors, GABA-A; Veratridine | 1990 |
gamma-Aminobutyric acid-A receptor-mediated suppression of 5-hydroxytryptamine-induced guinea-pig basilar artery smooth muscle contractility.
Topics: Animals; Basilar Artery; Caffeine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Receptors, GABA-A; Serotonin | 1989 |
Chronic caffeine or theophylline exposure reduces gamma-aminobutyric acid/benzodiazepine receptor site interactions.
Topics: Allosteric Regulation; Animals; Caffeine; Chick Embryo; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Receptors, GABA-A; Theophylline; Time Factors | 1988 |
Effects of 2-chloroadenosine on hippocampal GABA content and turnover.
Topics: 2-Chloroadenosine; 4-Aminobutyrate Transaminase; Adenosine; Aminooxyacetic Acid; Animals; Caffeine; gamma-Aminobutyric Acid; Hippocampus; Injections, Intraventricular; Kinetics; Male; Rats; Rats, Inbred Strains | 1986 |
Further characterization of [3H]gamma-aminobutyric acid release from isolated neuronal growth cones: role of intracellular Ca2+ stores.
Topics: Animals; Antimycin A; Brain; Caffeine; Calcium; Gallopamil; gamma-Aminobutyric Acid; Mitochondria; Neurons; Potassium; Rats; Subcellular Fractions; Time Factors | 1986 |
Protective effect of adenosine and nicotinamide against audiogenic seizure.
Topics: Acoustic Stimulation; Adenosine; Adenosine Triphosphate; Animals; Blood Pressure; Brain Chemistry; Caffeine; Dose-Response Relationship, Drug; Electroencephalography; Epilepsy; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Mice; Mice, Inbred Strains; NAD; Niacinamide; Norepinephrine; Phosphocreatine; Phosphorus Radioisotopes; Time Factors | 1974 |
GABA-induced depolarizing responses of the frog spinal cord can be either enhanced or antagonized by the benzodiazepine midazolam and the methylxanthine caffeine.
Topics: Animals; Benzodiazepines; Caffeine; Culture Techniques; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Midazolam; Neural Inhibition; Ranidae; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord; Stimulation, Chemical; Synaptic Transmission | 1984 |
Methylxanthines modulate adenosine release from slices of cerebral cortex.
Topics: 1-Methyl-3-isobutylxanthine; Adenine; Adenosine; Adenosine Triphosphatases; Aminophylline; Animals; Caffeine; Cerebral Cortex; Cyclic AMP; gamma-Aminobutyric Acid; Male; Mice; Ouabain; Theophylline; Xanthines | 1981 |
Influence of caffeine and midazolam on gamma-aminobutyric acid-evoked responses in the frog spinal cord.
Topics: Animals; Benzodiazepines; Caffeine; Drug Synergism; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Midazolam; Rana temporaria; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord | 1983 |
Caffeine-induced potentiation of GABA effects on frog spinal cord: an electrophysiological study.
Topics: Animals; Caffeine; Drug Synergism; Electric Conductivity; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Spinal; Motor Neurons; Rana temporaria; Spinal Cord | 1983 |
Requirements for an ideal alcohol antagonist.
Topics: Alcoholic Intoxication; Animals; Caffeine; Cats; Dextroamphetamine; Disease Models, Animal; Dogs; Ethanol; gamma-Aminobutyric Acid; Humans; Maleates; Naloxone; Pentylenetetrazole; Rabbits; Strychnine | 1980 |
Caffeine and related compounds block inhibitory amino acid-gated Cl- currents in freshly dissociated rat hippocampal neurones.
Topics: Amino Acids; Animals; Caffeine; Chloride Channels; Egtazic Acid; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; In Vitro Techniques; Ion Channel Gating; Ion Channels; Membrane Proteins; N-Methylaspartate; Neurons; Rats; Rats, Wistar; Xanthines | 1993 |
Tolerance to the behavioral effects of chlordiazepoxide: pharmacological and biochemical selectivity.
Topics: Amphetamine; Animals; Behavior, Animal; Caffeine; Carbolines; Chlordiazepoxide; Chlorides; Chlorine; Dose-Response Relationship, Drug; Drug Tolerance; Flumazenil; gamma-Aminobutyric Acid; Male; Midazolam; Morphine; Pentobarbital; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sensitivity and Specificity; Stimulation, Chemical | 1993 |
GABA-responses of CA3 neurones at epileptogenic threshold concentrations of convulsants.
Topics: Action Potentials; Animals; Bicarbonates; Bicuculline; Caffeine; Chlorides; Convulsants; Epilepsy; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Penicillins; Pentylenetetrazole; Synapses | 1993 |
Postsynaptic mechanism of depression of GABAergic synapses by oxytocin in the supraoptic nucleus of immature rat.
Topics: Age Factors; Animals; Bicuculline; Caffeine; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Enzyme Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine 5'-O-(3-Thiotriphosphate); Neural Inhibition; Neurons; Oxytocin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Oxytocin; Supraoptic Nucleus; Synapses; Synaptic Transmission; Thapsigargin; Vasoconstrictor Agents; Vasopressins | 1996 |
Is GABA involved in the development of caffeine tolerance?
Topics: 4-Aminobutyrate Transaminase; Animals; Bicuculline; Brain; Caffeine; Cerebellum; Cerebral Cortex; Corpus Striatum; Drug Tolerance; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Medulla Oblongata; Motor Activity; Muscimol; Pons; Rats | 1998 |
Calcium released from intracellular stores inhibits GABAA-mediated currents in ganglion cells of the turtle retina.
Topics: Alkaline Phosphatase; Animals; Bicuculline; Caffeine; Calcineurin; Calcium; Calcium Channels; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Membrane Potentials; Phosphodiesterase Inhibitors; Phosphoric Monoester Hydrolases; Pyridazines; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Retinal Ganglion Cells; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin; Turtles | 1998 |
Proconvulsive effect of tea (Camellia sinensis) in mice.
Topics: Animals; Brain Chemistry; Caffeine; Convulsants; Electroshock; Female; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred BALB C; Phosphodiesterase Inhibitors; Seizures; Strychnine; Tea; Tissue Extracts | 1999 |
Functional uncoupling of adenosine A(2A) receptors and reduced responseto caffeine in mice lacking dopamine D2 receptors.
Topics: Animals; Basal Ganglia Diseases; Caffeine; Cyclic AMP; Female; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Male; Mice; Mice, Congenic; Mice, Knockout; Motor Activity; Neostriatum; Neural Pathways; Proto-Oncogene Proteins c-fos; Receptor, Adenosine A2A; Receptors, Dopamine D2; Receptors, Purinergic P1; RNA, Messenger | 2000 |
Long-term caffeine inhibits Ehrlich ascites carcinoma cell-induced induction of central GABAergic activity.
Topics: Animals; Caffeine; Carcinoma, Ehrlich Tumor; Female; GABA Antagonists; gamma-Aminobutyric Acid; Mice; Neoplasm Transplantation | 2000 |
Radioligand binding assays in the drug discovery process: potential pitfalls of high throughput screenings.
Topics: Animals; Binding, Competitive; Caffeine; Central Nervous System Stimulants; Drug Evaluation, Preclinical; Excitatory Amino Acid Agonists; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kainic Acid; Membranes; Microsomes; Myocardium; Pharmacology; Radioligand Assay; Rats; Rats, Wistar; Ryanodine; Spermine | 2001 |
Analysis of GABA(A)- and GABA(B)-receptor mediated effects on intracellular Ca(2+) in DRG hybrid neurones.
Topics: Acrylates; Adenosine Triphosphate; Animals; Bicuculline; Caffeine; Calcium; Capsaicin; Cell Line; Diazepam; Dihydropyridines; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Hybrid Cells; Mice; Mice, Inbred BALB C; Neurons; Potassium Chloride; Receptors, GABA-A; Receptors, GABA-B; Thapsigargin; Time Factors | 2001 |
Sedative, anticonvulsant and behaviour modifying effects of Centranthus longiflorus ssp. longiflorus: a study of comparison to diazepam.
Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Depression; Diazepam; Female; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Mice; Plant Extracts; Plants, Medicinal; Rats; Rats, Sprague-Dawley; Seizures; Sleep; Swimming; Thiopental; Turkey; Valerianaceae | 2002 |
Intracellular calcium release resulting from mGluR1 receptor activation modulates GABAA currents in wide-field retinal amacrine cells: a study with caffeine.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amacrine Cells; Animals; Anticoagulants; Bicuculline; Caffeine; Calcium; Calcium Channels; Carps; Cells, Cultured; Central Nervous System Stimulants; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Conductivity; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heparin; Immunohistochemistry; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Kainic Acid; Membrane Potentials; Methoxyhydroxyphenylglycol; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retina; Ryanodine | 2003 |
Cadmium inhibits GABA-activated ion currents by increasing intracellular calcium level in snail neurons.
Topics: Animals; Cadmium; Caffeine; Calcium; Calcium Signaling; Central Nervous System Stimulants; Chloride Channels; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Ion Channels; Lymnaea; Microinjections; Neurons; Pertussis Toxin; Signal Transduction; Suramin | 2004 |
[Inhibitory effect of caffeine on GABA-activated current in acutely isolated rat dorsal root ganglion neurons].
Topics: Animals; Animals, Newborn; Caffeine; Cell Separation; Cells, Cultured; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2004 |
Drosophila mushroom body Kenyon cells generate spontaneous calcium transients mediated by PLTX-sensitive calcium channels.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Age Factors; Analysis of Variance; Animals; Caffeine; Calcium; Calcium Channels; Cells, Cultured; Chlorine; Cobalt; Curare; Diagnostic Imaging; Dose-Response Relationship, Radiation; Drosophila; Drug Combinations; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fura-2; GABA Antagonists; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Iodine; Mushroom Bodies; Neurons; Nicotine; Nicotinic Antagonists; Patch-Clamp Techniques; Phenols; Picrotoxin; Pupa; Salicylates; Spider Venoms; Tetrodotoxin; Thapsigargin; Time Factors; Valine | 2005 |
Two pathways for the activation of small-conductance potassium channels in neurons of substantia nigra pars reticulata.
Topics: Action Potentials; Animals; Animals, Newborn; Apamin; Caffeine; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Neurons; Nickel; omega-Conotoxins; Rats; Rats, Wistar; Ryanodine; Signal Transduction; Small-Conductance Calcium-Activated Potassium Channels; Substantia Nigra; Time Factors | 2005 |
Calcium from internal stores triggers GABA release from retinal amacrine cells.
Topics: Amacrine Cells; Animals; Boron Compounds; Caffeine; Calcium; Calcium Channels; Calcium-Binding Proteins; Central Nervous System Stimulants; Chick Embryo; Diagnostic Imaging; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Endoplasmic Reticulum; Evoked Potentials; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Glycine; Heparin; Immunohistochemistry; Inositol 1,4,5-Trisphosphate Receptors; Membrane Potentials; Microscopy, Confocal; Organic Chemicals; Patch-Clamp Techniques; Phenylacetates; Receptors, Cytoplasmic and Nuclear; Retina; Ryanodine; Ryanodine Receptor Calcium Release Channel; Time Factors | 2005 |
Supersensitivity of P2X receptors in cerebrocortical cell cultures after in vitro ischemia.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine Triphosphate; Anesthetics, Local; Animals; Bicuculline; Caffeine; Calcium; Cell Count; Cells, Cultured; Cerebral Cortex; Deoxyadenosines; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fura-2; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Ischemia; Membrane Potentials; Microscopy, Confocal; Microtubule-Associated Proteins; Neurons; Patch-Clamp Techniques; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrodotoxin; Time Factors; Triazines; Tritium; Xanthines | 2005 |
Modulation by brain natriuretic peptide of GABA receptors on rat retinal ON-type bipolar cells.
Topics: Animals; Atrial Natriuretic Factor; Caffeine; Calcium; Calcium Channels; Calcium Signaling; Calcium-Transporting ATPases; Calmodulin; Carbazoles; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Guanylate Cyclase; Heparin; Imidazoles; Indoles; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Male; Membrane Potentials; Natriuretic Peptide, Brain; Oxazoles; Patch-Clamp Techniques; Peptide Fragments; Peptides, Cyclic; Polysaccharides; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Atrial Natriuretic Factor; Receptors, Cytoplasmic and Nuclear; Receptors, GABA; Receptors, GABA-A; Retinal Bipolar Cells; Ruthenium Red; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin | 2006 |
Ca2+ release-dependent hyperpolarizations modulate the firing pattern of juvenile GABA neurons in mouse substantia nigra pars reticulata in vitro.
Topics: Action Potentials; Animals; Animals, Newborn; Benzimidazoles; Caffeine; Calcium; Calcium Channel Agonists; Central Nervous System Stimulants; Electric Stimulation; Electrophysiology; gamma-Aminobutyric Acid; Indoles; Mice; Mice, Inbred C57BL; Neurons; Small-Conductance Calcium-Activated Potassium Channels; Substantia Nigra; Time Factors | 2006 |
A novel in vitro metabolomics approach for neurotoxicity testing, proof of principle for methyl mercury chloride and caffeine.
Topics: Animals; Caffeine; Cell Survival; Cells, Cultured; Central Nervous System Stimulants; Choline; Creatine; Dose-Response Relationship, Drug; Embryo, Mammalian; gamma-Aminobutyric Acid; Glutamine; Kidney; L-Lactate Dehydrogenase; Liver; Mercuric Chloride; Neurons; Neurotoxins; Principal Component Analysis; Rats; Spermine; Tandem Mass Spectrometry; Telencephalon | 2008 |
Is there a major role for adenosine A2A receptors in anxiety?
Topics: Adenosine A2 Receptor Antagonists; Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Anxiety; Caffeine; Disease Models, Animal; Ethanol; gamma-Aminobutyric Acid; Humans; Hydrocortisone; Receptor, Adenosine A1; Receptor, Adenosine A2A; Stress, Psychological | 2008 |
The effects of adenosine A2A receptor antagonists on haloperidol-induced movement disorders in primates.
Topics: Adenosine A2 Receptor Antagonists; Animals; Antipsychotic Agents; Caffeine; Catalepsy; Cebus; Corpus Striatum; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Globus Pallidus; Haloperidol; Neurologic Examination; Purines; Pyrimidines; Receptor, Adenosine A2A; Saimiri; Triazoles; Xanthines | 2008 |
First evidence that drugs of abuse produce behavioral sensitization and cross sensitization in planarians.
Topics: Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Cocaine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glutamic Acid; Hypnotics and Sedatives; Methamphetamine; Motor Activity; Muscarinic Antagonists; Planarians; Scopolamine; Substance Withdrawal Syndrome; Substance-Related Disorders | 2010 |
Multiple anxiogenic drugs recruit a parvalbumin-containing subpopulation of GABAergic interneurons in the basolateral amygdala.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Brain; Caffeine; Carbolines; Cell Count; gamma-Aminobutyric Acid; Gene Expression Regulation; Interneurons; Male; Parvalbumins; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Time Factors; Yohimbine | 2010 |
Novel protective effect of mifepristone on detrimental GABAA receptor activity to immature Purkinje neurons.
Topics: Animals; Caffeine; Chlorides; gamma-Aminobutyric Acid; Imidazoles; Mice; Mifepristone; Muscimol; p38 Mitogen-Activated Protein Kinases; Purkinje Cells; Pyrimidines; Receptors, GABA-A | 2011 |
Chemical constituents and anticancer activity of yellow camellias against MDA-MB-231 human breast cancer cells.
Topics: Amino Acids; Antineoplastic Agents, Phytogenic; Antioxidants; Breast Neoplasms; Caffeine; Camellia; Catechin; Cell Line, Tumor; Cell Survival; Chromatography, High Pressure Liquid; Chromatography, Liquid; Female; Flavonoids; Flowers; gamma-Aminobutyric Acid; Glucosides; Humans; Kaempferols; Monosaccharides; Plant Extracts; Plant Leaves; Polyphenols; Quercetin; Tandem Mass Spectrometry | 2013 |
Caffeine promotes glutamate and histamine release in the posterior hypothalamus.
Topics: Animals; Behavior, Animal; Biosensing Techniques; Caffeine; Central Nervous System Stimulants; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Glutamic Acid; Histamine Release; Hypothalamus, Posterior; Male; Microdialysis; Neurons; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Time Factors; Wakefulness | 2014 |
Caffeine potentiates the release of GABA mediated by NMDA receptor activation: Involvement of A1 adenosine receptors.
Topics: Animals; Caffeine; Central Nervous System Stimulants; Chick Embryo; Cyclic AMP-Dependent Protein Kinases; D-Aspartic Acid; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Receptor, Adenosine A1; Receptors, N-Methyl-D-Aspartate; Retina; Signal Transduction | 2014 |
A study on quality components and sleep-promoting effects of GABA black tea.
Topics: Animals; Caffeine; Catechin; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Male; Mice; Pentobarbital; Plant Extracts; Polyphenols; Sleep; Tea | 2015 |
Caffeine prevents antihyperalgesic effect of gabapentin in an animal model of CRPS-I: evidence for the involvement of spinal adenosine A1 receptor.
Topics: Amines; Analgesics; Animals; Caffeine; Cyclohexanecarboxylic Acids; Disease Models, Animal; Gabapentin; gamma-Aminobutyric Acid; Hyperalgesia; Male; Mice; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A1; Reflex Sympathetic Dystrophy; Spinal Cord | 2015 |
Modulation of GABA release from the thalamic reticular nucleus by cocaine and caffeine: role of serotonin receptors.
Topics: Action Potentials; Animals; Cadmium Chloride; Caffeine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Mice; Mice, Knockout; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Agents; Thalamic Nuclei; Type C Phospholipases | 2016 |
Neuroprotective effects of caffeine in MPTP model of Parkinson's disease: A (13)C NMR study.
Topics: Amino Acids; Animals; Behavior, Animal; Brain; Caffeine; gamma-Aminobutyric Acid; Glucose; Hand Strength; Inositol; Magnetic Resonance Spectroscopy; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neostriatum; Neuroprotective Agents | 2016 |
Sleep-promoting effects of a GABA/5-HTP mixture: Behavioral changes and neuromodulation in an invertebrate model.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Drosophila melanogaster; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Motor Activity; Neurotransmitter Agents; Receptor, Serotonin, 5-HT1A; Receptors, GABA-B; Signal Transduction; Sleep | 2016 |
Caffeine-Induced Suppression of GABAergic Inhibition and Calcium-Independent Metaplasticity.
Topics: Animals; Caffeine; Calcium Signaling; Cells, Cultured; gamma-Aminobutyric Acid; Hippocampus; Inhibitory Postsynaptic Potentials; Neuronal Plasticity; Pyramidal Cells; Rats | 2016 |
Influence of caffeine on the protective activity of gabapentin and topiramate in a mouse model of generalized tonic-clonic seizures.
Topics: Amines; Animals; Anticonvulsants; Caffeine; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Fructose; Gabapentin; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Memory, Long-Term; Mice; Motor Skills; Seizures; Topiramate | 2016 |
Effects of GABA, Neural Regulation, and Intrinsic Cardiac Factors on Heart Rate Variability in Zebrafish Larvae.
Topics: Acetylcholine; Animals; Bicuculline; Caffeine; Central Nervous System Depressants; Central Nervous System Stimulants; Cholinergic Agonists; Dopamine; Dopamine Agents; Ethanol; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Heart; Heart Rate; Larva; Lidocaine; Methacholine Chloride; Muscarinic Agonists; Muscimol; Zebrafish | 2017 |
Early-life exposure to caffeine affects the construction and activity of cortical networks in mice.
Topics: Animals; Animals, Newborn; Caffeine; Central Nervous System Stimulants; Cerebral Cortex; Dendrites; Electrophysiological Phenomena; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neocortex; Nerve Net; Pregnancy; Prenatal Exposure Delayed Effects; Seizures, Febrile; Somatostatin; Visual Cortex | 2017 |
Caffeine Protects Against Anticonvulsant-Induced Neurotoxicity in the Developing Rat Brain.
Topics: Animals; Animals, Newborn; Anticonvulsants; Apoptosis; Brain; Caffeine; Cytokines; gamma-Aminobutyric Acid; Gene Expression; Nerve Degeneration; Neuroprotective Agents; Phenobarbital; Random Allocation; Rats, Wistar; Receptors, Purinergic P1; Time Factors | 2017 |
Acute caffeine ingestion affects surround suppression of perceived contrast.
Topics: Adult; Caffeine; Contrast Sensitivity; Discrimination, Psychological; Female; gamma-Aminobutyric Acid; Humans; Male; Neurotransmitter Agents; Photic Stimulation; Sensory Thresholds; Visual Perception; Young Adult | 2018 |
Effect of explosion-puffed coffee on locomotor activity and behavioral patterns in Drosophila melanogaster.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Caffeine; Chlorogenic Acid; Coffee; Drosophila melanogaster; Food Handling; gamma-Aminobutyric Acid; Locomotion; Male; RNA, Messenger | 2017 |
High expression of hippocampal glutamic acid decarboxylase 67 mediates hypersensitivity of the hypothalamic-pituitary-adrenal axis in response to prenatal caffeine exposure in rats.
Topics: Adrenocorticotropic Hormone; Animals; Caffeine; Cells, Cultured; Corticosterone; Female; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Hippocampus; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar | 2018 |
J-difference-edited MRS measures of γ-aminobutyric acid before and after acute caffeine administration.
Topics: Adult; Algorithms; Aspartic Acid; Brain Mapping; Caffeine; Central Nervous System Stimulants; Creatine; gamma-Aminobutyric Acid; Glutamic Acid; Glutamine; Healthy Volunteers; Humans; Image Processing, Computer-Assisted; Inositol; Magnetic Resonance Spectroscopy; Male; Neurotransmitter Agents; Normal Distribution; Young Adult | 2018 |
The science of tea's mood-altering magic.
Topics: Adenosine; Affect; Alpha Rhythm; Animals; Antioxidants; Behavior; Beta Rhythm; Blood-Brain Barrier; Caffeine; Catechin; Cognition; Dementia; Depression; Exercise; gamma-Aminobutyric Acid; Glutamates; Humans; Hydrocortisone; Life Style; Mental Health; Middle Aged; Stress, Psychological; Tea; Theta Rhythm | 2019 |
Rutin, γ-Aminobutyric Acid, Gallic Acid, and Caffeine Negatively Affect the Sweet-Mellow Taste of Congou Black Tea Infusions.
Topics: Caffeine; Camellia sinensis; Female; Gallic Acid; gamma-Aminobutyric Acid; Humans; Male; Rutin; Taste; Tea | 2019 |
Caffeine Improves GABA Transport in the Striatum of Spontaneously Hypertensive Rats (SHR).
Topics: Animals; Blotting, Western; Caffeine; Central Nervous System Stimulants; Corpus Striatum; Female; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred SHR; Rats, Wistar | 2021 |
GABA
Topics: Acids; Animals; Bicuculline; Caffeine; Cyclohexenes; Disease Models, Animal; Electroencephalography; Flavonoids; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Humulus; Hypnotics and Sedatives; Mice; Picrotoxin; Propiophenones; Receptors, GABA-A; Sleep; Sleep Initiation and Maintenance Disorders; Terpenes | 2021 |
The Positive Effects of
Topics: Animals; Caffeine; gamma-Aminobutyric Acid; Mice; Mice, Inbred ICR; Plant Extracts; Quality of Life; Rats; Rats, Sprague-Dawley; Sleep; Sleep Initiation and Maintenance Disorders; Sleep Quality; Wolfiporia | 2022 |
The upregulation of glutamate decarboxylase 67 against hippocampal excitability damage in male fetal rats by prenatal caffeine exposure.
Topics: Adenylyl Cyclases; Animals; Brain-Derived Neurotrophic Factor; Caffeine; Colforsin; Female; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Hippocampus; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Receptor, Adenosine A2A; Up-Regulation | 2022 |
Promising anticonvulsant N-[(2,4-dichlorophenyl) methyl]-2-(2,4-dioxo-1H-quinazolin-3-yl) acetamide: dose-dependent study and evaluation of anticonvulsant action spectrum in vivo and in silico.
Topics: Acetamides; Action Spectrum; Animals; Anticonvulsants; Caffeine; gamma-Aminobutyric Acid; Mice; Molecular Docking Simulation; Pentylenetetrazole; Picrotoxin; Seizures; Strychnine | 2022 |
Sclareol exerts synergistic antidepressant effects with quercetin and caffeine, possibly suppressing GABAergic transmission in chicks.
Topics: Caffeine; gamma-Aminobutyric Acid; Humans; Quercetin; Receptors, GABA-A | 2023 |