caffeine and flunitrazepam

caffeine has been researched along with flunitrazepam in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19906 (50.00)18.7374
1990's2 (16.67)18.2507
2000's3 (25.00)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Farb, DH; Friedman, L; Gibbs, TT; Roca, DJ; Rozenberg, I; Schiller, GD1
Farb, DH; Roca, DJ; Schiller, GD1
Chweh, AY; Swinyard, EA; Ulloque, RA1
Aguilar, JS; Lowenstein, PR; Sabato, UC1
Dijkhuis, IC1
Airaksinen, MM; Saano, V1
Hruska, RE; Weir, RL1
Blandl, T; Kardos, J1
Mendonça-Silva, DL; Noël, F; Quintas, LE1

Other Studies

12 other study(ies) available for caffeine and flunitrazepam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
gamma-Aminobutyric acidA receptor regulation in culture: altered allosteric interactions following prolonged exposure to benzodiazepines, barbiturates, and methylxanthines.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Allosteric Regulation; Animals; Barbital; Barbiturates; Brain; Caffeine; Cells, Cultured; Chick Embryo; Flumazenil; Flunitrazepam; Flurazepam; gamma-Aminobutyric Acid; Kinetics; Neurons; Pentobarbital; Receptors, GABA-A; Tetrodotoxin; Theophylline; Veratridine

1990
Chronic caffeine or theophylline exposure reduces gamma-aminobutyric acid/benzodiazepine receptor site interactions.
    Molecular pharmacology, 1988, Volume: 33, Issue:5

    Topics: Allosteric Regulation; Animals; Caffeine; Chick Embryo; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Receptors, GABA-A; Theophylline; Time Factors

1988
Benzodiazepine inhibition of [3H]flunitrazepam binding and caffeine-induced seizures in mice.
    European journal of pharmacology, 1986, Mar-18, Volume: 122, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding, Competitive; Caffeine; Flumazenil; Flunitrazepam; Male; Mice; Receptors, GABA-A; Seizures

1986
Effects of the methylxanthine derivative pentoxifylline on benzodiazepine and muscarinic binding sites in rat cerebral cortex.
    Acta physiologica et pharmacologica latinoamericana : organo de la Asociacion Latinoamericana de Ciencias Fisiologicas y de la Asociacion Latinoamericana de Farmacologia, 1985, Volume: 35, Issue:4

    Topics: Animals; Binding, Competitive; Caffeine; Cerebral Cortex; Female; Flunitrazepam; Pentoxifylline; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Muscarinic; Theobromine

1985
Quality control in therapeutic drug monitoring.
    Pharmaceutisch weekblad. Scientific edition, 1988, Aug-19, Volume: 10, Issue:4

    Topics: Caffeine; Flunitrazepam; Gentamicins; Humans; Laboratories; Netherlands; Pharmaceutical Preparations; Quality Control; Reference Values; Theophylline; Thiopental; United States

1988
Binding of beta-carbolines and caffeine on benzodiazepine receptors: correlations to convulsions and tremor.
    Acta pharmacologica et toxicologica, 1982, Volume: 51, Issue:4

    Topics: Animals; Brain; Caffeine; Carbolines; Flunitrazepam; Harmaline; Harmine; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Tremor

1982
Interaction between methylxanthines and the benzodiazepine receptor.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 265, Issue:1

    Topics: Animals; Brain; Caffeine; Flunitrazepam; In Vitro Techniques; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Theophylline

1983
Inhibition of a gamma aminobutyric acid A receptor by caffeine.
    Neuroreport, 1994, Jun-02, Volume: 5, Issue:10

    Topics: Animals; Caffeine; Cerebral Cortex; Chlorides; Chlorine; Dantrolene; Flunitrazepam; GABA-A Receptor Antagonists; In Vitro Techniques; Kinetics; Male; Membranes; Radioisotopes; Rats; Rats, Wistar

1994
Radioligand binding assays in the drug discovery process: potential pitfalls of high throughput screenings.
    Arzneimittel-Forschung, 2001, Volume: 51, Issue:2

    Topics: Animals; Binding, Competitive; Caffeine; Central Nervous System Stimulants; Drug Evaluation, Preclinical; Excitatory Amino Acid Agonists; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kainic Acid; Membranes; Microsomes; Myocardium; Pharmacology; Radioligand Assay; Rats; Rats, Wistar; Ryanodine; Spermine

2001