caffeine and bicuculline

caffeine has been researched along with bicuculline in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19907 (25.93)18.7374
1990's9 (33.33)18.2507
2000's8 (29.63)29.6817
2010's2 (7.41)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Bornstein, MB; Corrigall, WA; Crain, SM1
Markovich, VV; Molodavkin, GM; Ostrovskaia, RU1
Bitran, D; Kellogg, CK; Primus, RJ1
Dohi, T; Kitayama, S; Morita, K; Tsujimoto, A1
Ferrario, P; Hafner, B; Mantegazza, P; Tammiso, R; Zambotti, F; Zonta, N1
Henry, JL; Salter, MW1
Kharlamov, AN; Raevskiĭ, KS1
Lee, EK; Ross, RJ; Walters, JR; Waszczak, BL1
Dunham, L; Guillet, R1
Bingmann, D; Bonnet, U1
Brussaard, AB; de Vlieger, TA; Kits, KS1
Fredholm, BB; Georgiev, V; Johansson, B; Kuosmanen, T1
Mukhopadhyay, S; Poddar, MK1
Kuribara, H; Maruyama, Y; Stavinoha, WB1
Akopian, A; Gabriel, R; Witkovsky, P1
Dixon, AK; Freeman, TC; Lee, K; Preston, Z; Richardson, PJ; Widdowson, L1
Kim, SU; Krieger, C; Puil, E; Yokogawa, T1
Lasater, EM; Vigh, J1
Chopde, CT; Hirani, K; Jain, NS1
Fischer, W; Franke, H; Gröger-Arndt, H; Günther, A; Illes, P; Köfalvi, A; Madarász, E; Nörenberg, W; Schneider, D; Sperlágh, B; Vizi, ES; Wirkner, K1
Kubová, H; Mares, P; Tchekalarova, J1
Chen, JF; Coelho, JE; Fredholm, BB; Fu, Y; Karaoz, U; Tillman, A; Weng, Z; Yu, L; Zhang, X1
Morimoto, Y; Takita, K1
Vargas, RA1
Ahn, Y; Cho, HJ; Jo, K; Kwak, WK; Min, B; Suh, HJ1

Other Studies

27 other study(ies) available for caffeine and bicuculline

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Electrophysiological studies of fetal mouse olifactory bulb explants during development of synaptic functions in culture.
    Journal of neurobiology, 1976, Volume: 7, Issue:6

    Topics: Action Potentials; Animals; Bicuculline; Caffeine; Evoked Potentials; Fetus; gamma-Aminobutyric Acid; Mice; Neural Inhibition; Neurons; Olfactory Bulb; Organ Culture Techniques; Picrotoxin; Synapses; Time Factors; Tubocurarine

1976
[The effect of substnaces altering gamma-aminobutyric acid metabolism on the recovery cycle of the interzonal response of the cat motor cortex].
    Biulleten' eksperimental'noi biologii i meditsiny, 1975, Volume: 79, Issue:2

    Topics: Aminobutyrates; Animals; Arecoline; Bemegride; Benactyzine; Bicuculline; Caffeine; Cats; Drug Interactions; Electrophysiology; gamma-Aminobutyric Acid; Motor Cortex; Receptors, Drug; Semicarbazides; Somatosensory Cortex; Sulfhydryl Compounds; Valproic Acid

1975
Gestational exposure to diazepam increases sensitivity to convulsants that act at the GABA/benzodiazepine receptor complex.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Bicuculline; Caffeine; Carbolines; Cerebral Cortex; Chlorides; Convulsants; Diazepam; Female; GABA-A Receptor Antagonists; Male; Picrotoxin; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A; Seizures; Strychnine; Synaptosomes

1991
Enhancement by GABA of the stimulation-evoked catecholamine release from cultured bovine adrenal chromaffin cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:5

    Topics: Acetylcholine; Adrenal Glands; Animals; Bicuculline; Caffeine; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Muscimol; Nicotine; Picrotoxin; Potassium; Receptors, GABA-A; Veratridine

1990
Reversal of the effect of centrally-administered diazepam on morphine antinociception by specific (Ro 15-1788 and Ro 15-3505) and non-specific (bicuculline and caffeine) benzodiazepine antagonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:1

    Topics: Animals; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Flumazenil; Injections, Intraventricular; Male; Morphine; Pain; Rats; Rats, Inbred Strains

1986
Evidence that adenosine mediates the depression of spinal dorsal horn neurons induced by peripheral vibration in the cat.
    Neuroscience, 1987, Volume: 22, Issue:2

    Topics: Adenosine; Animals; Bicuculline; Blood Pressure; Caffeine; Cats; Dipyridamole; Injections, Intravenous; Iontophoresis; Naloxone; Neurons; Spinal Cord; Strychnine; Theophylline; Vibration

1987
[Tranquilizing effect of n-dipropylacetate and other GABA-ergic substances in conflict situations].
    Biulleten' eksperimental'noi biologii i meditsiny, 1980, Volume: 89, Issue:7

    Topics: Acetates; Aminooxyacetic Acid; Animals; Bicuculline; Caffeine; Conflict, Psychological; Male; Models, Psychological; Pantothenic Acid; Pentylenetetrazole; Piracetam; Pyrrolidinones; Rats; Tranquilizing Agents; Valproic Acid

1980
Effects of benzodiazepines on single unit activity in the substantia nigra pars reticulata.
    Life sciences, 1982, Sep-06, Volume: 31, Issue:10

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Dose-Response Relationship, Drug; Electric Conductivity; Flumazenil; Flurazepam; Male; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Substantia Nigra; Theophylline

1982
Neonatal caffeine exposure and seizure susceptibility in adult rats.
    Epilepsia, 1995, Volume: 36, Issue:8

    Topics: Animals; Animals, Newborn; Bicuculline; Brain; Caffeine; Female; Kainic Acid; Male; Pentylenetetrazole; Picrotoxin; Rats; Receptors, Purinergic P1; Seizures; Sex Factors; Strychnine

1995
GABA-responses of CA3 neurones at epileptogenic threshold concentrations of convulsants.
    Neuroreport, 1993, Volume: 4, Issue:6

    Topics: Action Potentials; Animals; Bicarbonates; Bicuculline; Caffeine; Chlorides; Convulsants; Epilepsy; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Penicillins; Pentylenetetrazole; Synapses

1993
Postsynaptic mechanism of depression of GABAergic synapses by oxytocin in the supraoptic nucleus of immature rat.
    The Journal of physiology, 1996, Dec-01, Volume: 497 ( Pt 2)

    Topics: Age Factors; Animals; Bicuculline; Caffeine; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Enzyme Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine 5'-O-(3-Thiotriphosphate); Neural Inhibition; Neurons; Oxytocin; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Oxytocin; Supraoptic Nucleus; Synapses; Synaptic Transmission; Thapsigargin; Vasoconstrictor Agents; Vasopressins

1996
Long-term treatment with some methylxanthines decreases the susceptibility to bicuculline- and pentylenetetrazol-induced seizures in mice. Relationship to c-fos expression and receptor binding.
    The European journal of neuroscience, 1996, Volume: 8, Issue:12

    Topics: Animals; Autoradiography; Behavior, Animal; Bicuculline; Brain; Caffeine; Disease Susceptibility; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Proto-Oncogene Proteins c-fos; Receptors, GABA-A; Receptors, Purinergic P1; RNA, Messenger; Seizures; Time Factors; Xanthines

1996
Is GABA involved in the development of caffeine tolerance?
    Neurochemical research, 1998, Volume: 23, Issue:1

    Topics: 4-Aminobutyrate Transaminase; Animals; Bicuculline; Brain; Caffeine; Cerebellum; Cerebral Cortex; Corpus Striatum; Drug Tolerance; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Medulla Oblongata; Motor Activity; Muscimol; Pons; Rats

1998
Behavioural pharmacological characteristics of honokiol, an anxiolytic agent present in extracts of Magnolia bark, evaluated by an elevated plus-maze test in mice.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:7

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Bicuculline; Biphenyl Compounds; Caffeine; Central Nervous System Depressants; Central Nervous System Stimulants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Injections, Subcutaneous; Lignans; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Tetragastrin; Therapeutic Equivalency

1998
Calcium released from intracellular stores inhibits GABAA-mediated currents in ganglion cells of the turtle retina.
    Journal of neurophysiology, 1998, Volume: 80, Issue:3

    Topics: Alkaline Phosphatase; Animals; Bicuculline; Caffeine; Calcineurin; Calcium; Calcium Channels; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Imidazoles; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Membrane Potentials; Phosphodiesterase Inhibitors; Phosphoric Monoester Hydrolases; Pyridazines; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Retinal Ganglion Cells; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin; Turtles

1998
Adenosine receptor expression and function in rat striatal cholinergic interneurons.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Acetylcholine; Adenosine; Adenosine Deaminase; Animals; Baclofen; Bicuculline; Caffeine; Cholinergic Fibers; Corpus Striatum; Dose-Response Relationship, Drug; GABA Antagonists; Gene Expression; Male; Membrane Potentials; Naloxone; Narcotic Antagonists; Neurons; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; RNA, Messenger; Tritium; Xanthines

2000
Analysis of GABA(A)- and GABA(B)-receptor mediated effects on intracellular Ca(2+) in DRG hybrid neurones.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: Acrylates; Adenosine Triphosphate; Animals; Bicuculline; Caffeine; Calcium; Capsaicin; Cell Line; Diazepam; Dihydropyridines; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Hybrid Cells; Mice; Mice, Inbred BALB C; Neurons; Potassium Chloride; Receptors, GABA-A; Receptors, GABA-B; Thapsigargin; Time Factors

2001
Intracellular calcium release resulting from mGluR1 receptor activation modulates GABAA currents in wide-field retinal amacrine cells: a study with caffeine.
    The European journal of neuroscience, 2003, Volume: 17, Issue:11

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amacrine Cells; Animals; Anticoagulants; Bicuculline; Caffeine; Calcium; Calcium Channels; Carps; Cells, Cultured; Central Nervous System Stimulants; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Conductivity; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heparin; Immunohistochemistry; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Kainic Acid; Membrane Potentials; Methoxyhydroxyphenylglycol; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retina; Ryanodine

2003
Reversal of caffeine-induced anxiety by neurosteroid 3-alpha-hydroxy-5-alpha-pregnane-20-one in rats.
    Neuropharmacology, 2005, Volume: 48, Issue:5

    Topics: Adrenalectomy; Analysis of Variance; Anesthetics; Animals; Anxiety; Bicuculline; Caffeine; Central Nervous System Stimulants; Corticotropin-Releasing Hormone; Diazepam; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; Hormone Antagonists; Injections, Intraventricular; Male; Maze Learning; Muscimol; Peptide Fragments; Pregnanolone; Progestins; Rats; Rats, Sprague-Dawley; Reaction Time

2005
Supersensitivity of P2X receptors in cerebrocortical cell cultures after in vitro ischemia.
    Journal of neurochemistry, 2005, Volume: 95, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine Triphosphate; Anesthetics, Local; Animals; Bicuculline; Caffeine; Calcium; Cell Count; Cells, Cultured; Cerebral Cortex; Deoxyadenosines; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fura-2; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Ischemia; Membrane Potentials; Microscopy, Confocal; Microtubule-Associated Proteins; Neurons; Patch-Clamp Techniques; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrodotoxin; Time Factors; Triazines; Tritium; Xanthines

2005
Effects of postnatal caffeine exposure on seizure susceptibility in developing rats.
    Brain research, 2007, May-30, Volume: 1150

    Topics: Age Factors; Aminophylline; Animals; Animals, Newborn; Behavior, Animal; Bicuculline; Caffeine; Central Nervous System Stimulants; Disease Models, Animal; Disease Susceptibility; Drug Interactions; Pentylenetetrazole; Picrotoxin; Rats; Rats, Wistar; Reaction Time; Seizures; Severity of Illness Index

2007
Uncovering multiple molecular targets for caffeine using a drug target validation strategy combining A 2A receptor knockout mice with microarray profiling.
    Physiological genomics, 2009, May-13, Volume: 37, Issue:3

    Topics: Animals; Bicuculline; Caffeine; Central Nervous System Stimulants; Cluster Analysis; Dose-Response Relationship, Drug; Female; GABA Antagonists; Gene Expression Profiling; Gene Expression Regulation; Male; Mice; Mice, Knockout; Neostriatum; Oligonucleotide Array Sequence Analysis; Phosphodiesterase Inhibitors; Receptor, Adenosine A2A; Reverse Transcriptase Polymerase Chain Reaction; Rolipram

2009
Nociceptin/orphanin FQ slows inspiratory rhythm via its direct effects on the pre-Bötzinger complex.
    Respiratory physiology & neurobiology, 2015, Feb-01, Volume: 207

    Topics: Action Potentials; Analysis of Variance; Animals; Animals, Newborn; Bicuculline; Caffeine; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Electric Stimulation; GABA-A Receptor Antagonists; In Vitro Techniques; Neurons; Nociceptin; Opioid Peptides; Patch-Clamp Techniques; Periodicity; Potassium; Rats; Rats, Wistar; Respiratory Center; Xanthines

2015
Effects of GABA, Neural Regulation, and Intrinsic Cardiac Factors on Heart Rate Variability in Zebrafish Larvae.
    Zebrafish, 2017, Volume: 14, Issue:2

    Topics: Acetylcholine; Animals; Bicuculline; Caffeine; Central Nervous System Depressants; Central Nervous System Stimulants; Cholinergic Agonists; Dopamine; Dopamine Agents; Ethanol; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Heart; Heart Rate; Larva; Lidocaine; Methacholine Chloride; Muscarinic Agonists; Muscimol; Zebrafish

2017
GABA
    Molecules (Basel, Switzerland), 2021, Nov-24, Volume: 26, Issue:23

    Topics: Acids; Animals; Bicuculline; Caffeine; Cyclohexenes; Disease Models, Animal; Electroencephalography; Flavonoids; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Humulus; Hypnotics and Sedatives; Mice; Picrotoxin; Propiophenones; Receptors, GABA-A; Sleep; Sleep Initiation and Maintenance Disorders; Terpenes

2021