Page last updated: 2024-09-03

bw a868c and prostaglandin d2

bw a868c has been researched along with prostaglandin d2 in 33 studies

Compound Research Comparison

Studies
(bw a868c)
Trials
(bw a868c)
Recent Studies (post-2010)
(bw a868c)
Studies
(prostaglandin d2)
Trials
(prostaglandin d2)
Recent Studies (post-2010) (prostaglandin d2)
470113,45478751

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-19903 (9.09)18.7374
1990's12 (36.36)18.2507
2000's10 (30.30)29.6817
2010's8 (24.24)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abramovitz, M; Boie, Y; Metters, KM; Sawyer, N; Slipetz, DM1
Hirata, M; Kiriyama, M; Kobayashi, T; Narumiya, S; Sugimoto, Y; Ushikubi, F1
Abramovitz, M; Ford-Hutchinson, AW; Metters, KM; Wright, DH1
Alvarez, R; Artis, DR; Bruno, JJ; Chang, LF; Eglen, RM; Kluge, AF; Whiting, RL1
Hamid-Bloomfield, S; Payne, AN; Petrovic, AA; Whittle, BJ1
Collins, BA; Kelly, MG; Robertson, AD; Trist, DG; Wood, J1
Hamid-Bloomfield, S; Whittle, BJ1
Bolofo, ML; Giles, H; Kelly, MG; Leff, P; Robertson, AD1
Betti, PA; Prior, ET; Rangachari, PK; Roberts, LJ1
Loi, RK; Warren, JB; Wilson, AJ1
Hawley, SB; Nieves, AL; Protzman, CE; Spada, CS; Williams, LS; Woodward, DF1
Hayaishi, O; Ito, S; Minami, T; Mori, H; Okuda-Ashitaka, E1
Leff, P; Lydford, SJ; McKechnie, KC1
Eguchi, N; Hayaishi, O; Ito, S; Kanaoka, Y; Minami, T; Nagata, A; Shirafuji, N; Tanaka, T; Urade, Y; Yoshida, N1
Crider, JY; Griffin, BW; Sharif, NA1
Davis, TL; Sharif, NA; Williams, GW1
Chadee, K; Ford-Hutchinson, AW; Metters, KM; Wright, DH1
Diamond, M; Gravel, S; Monneret, G; Powell, WS; Rokach, J1
Antoniou, J; de Brum-Fernandes, AJ; Gallant, MA; Hackett, JA; Parent, JL; Samadfam, R1
Ago, J; Inoue, T; Ishikawa, T; Kamei, C; Rahman, A1
Arai, I; Futaki, N; Hashimoto, Y; Honma, Y; Inoue, T; Koizumi, C; Nakaike, S; Nakanishi, Y; Ono, N; Sakurai, T; Sugimoto, M; Takahashi, N; Takaoka, A; Tanami, T; Yagi, M1
Ohinata, K; Usui, H; Yoshikawa, M; Zhao, H1
Heinemann, A; Peskar, BA; Prenn, C; Schuligoi, R1
Furuta, K; Hokamura, K; Ibaraki, K; Maeda, M; Suzuki, M; Thura, M; Umemura, K; Yamamoto, S1
Asakawa, A; Biyajima, K; Eguchi, N; Inui, A; Kaneko, K; Miyamoto, C; Ohinata, K; Takagi, K; Urade, Y; Yoshikawa, M1
Ebersberger, A; Eitner, A; Halbhuber, KJ; Natura, G; Rost, R; Schaible, HG1
Mak, OT; Wang, JJ1
Doi, H; Egawa, G; Hirabayashi, T; Kabashima, K; Miyachi, Y; Murakami, M; Nakahigashi, K; Otsuka, A; Tanizaki, H; Urade, Y; Zouboulis, CC1
Wu, X; Yu, S; Zhang, S1
Arai, T; Awata, A; Fujino, H; Murayama, T; Okura, I; Oyama, S; Regan, JW; Yamazaki, R1
Baird, AW; Collins, D; Medani, M; Mohan, HM; Walsh, E; Winter, DC1
de Verdier, PJ; Guan, NN; Gustafsson, LE; Svennersten, K; Wiklund, NP1
Hu, X; Ji, C; Kuang, S; Liang, G; Luo, Y; Ma, J; Mai, S; Tian, X; Wei, Y; Yang, J; Yang, Q; Yang, Y1

Other Studies

33 other study(ies) available for bw a868c and prostaglandin d2

ArticleYear
Molecular cloning and characterization of the human prostanoid DP receptor.
    The Journal of biological chemistry, 1995, Aug-11, Volume: 270, Issue:32

    Topics: Amino Acid Sequence; Base Sequence; Blotting, Northern; Calcium; Cells, Cultured; Cloning, Molecular; Cyclic AMP; Humans; Molecular Sequence Data; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin

1995
Ligand binding specificities of the eight types and subtypes of the mouse prostanoid receptors expressed in Chinese hamster ovary cells.
    British journal of pharmacology, 1997, Volume: 122, Issue:2

    Topics: Animals; CHO Cells; Cricetinae; Ligands; Mice; Prostaglandins; Receptors, Prostaglandin; Transfection

1997
Characterization of the recombinant human prostanoid DP receptor and identification of L-644,698, a novel selective DP agonist.
    British journal of pharmacology, 1998, Volume: 123, Issue:7

    Topics: Adenine Nucleotides; Benzoates; Binding, Competitive; Cell Line; Cyclic AMP; Dinoprostone; Guanine Nucleotides; Humans; Kinetics; Receptors, Immunologic; Receptors, Prostaglandin; Recombinant Proteins; Thiazoles; Thiazolidines; Tritium

1998
Stimulation of prostaglandin D2 receptors on human platelets by analogs of prostacyclin.
    Prostaglandins, 1991, Volume: 42, Issue:2

    Topics: Adenosine Diphosphate; Adenylyl Cyclases; Alprostadil; Blood Platelets; Bridged-Ring Compounds; Dose-Response Relationship, Drug; Epoprostenol; Female; Humans; Hydantoins; Molecular Conformation; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Stereoisomerism

1991
The role of prostanoid TP- and DP-receptors in the bronchoconstrictor effect of inhaled PGD2 in anaesthetized guinea-pigs: effect of the DP-antagonist BW A868C.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Administration, Inhalation; Anesthesia; Animals; Benzeneacetamides; Bronchi; Cyclooxygenase Inhibitors; Guinea Pigs; Hydantoins; Hydroxamic Acids; Indomethacin; Lipoxygenase Inhibitors; Male; Platelet Aggregation Inhibitors; Prostaglandin D2; Prostaglandins D; Receptors, Prostaglandin; Respiratory Function Tests; Sulfonamides; Thromboxane A2; Vagotomy

1990
The antagonism by BW A868C of PGD2 and BW245C activation of human platelet adenylate cyclase.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Adenylyl Cyclases; Blood Platelets; Enzyme Activation; Epoprostenol; Humans; Hydantoins; Iloprost; In Vitro Techniques; Platelet Aggregation; Prostaglandin D2; Receptors, Prostaglandin

1989
Antagonism of PGD2 vasodepressor responses in the rat in vivo by the novel, selective antagonist, BW A868C.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Animals; Blood Pressure; Epoprostenol; Hydantoins; Infusions, Intravenous; Male; Prostaglandin D2; Rats; Rats, Inbred Strains; Receptors, Prostaglandin; Sulfonamides

1989
The classification of prostaglandin DP-receptors in platelets and vasculature using BW A868C, a novel, selective and potent competitive antagonist.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Blood Platelets; Blood Vessels; Guinea Pigs; Humans; Hydantoins; In Vitro Techniques; Jugular Veins; Male; Muscle Contraction; Platelet Aggregation; Prostaglandin D2; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Prostaglandin; Sulfonamides; Trachea

1989
Effects of a selective DP receptor agonist (BW 245C) and antagonist (BW A868C) on the canine colonic epithelium: an argument for a different DP receptor?
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Colon; Dogs; Electrophysiology; Female; Hydantoins; In Vitro Techniques; Intestinal Mucosa; Male; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin

1995
PGD2 is an intermediate in agonist-stimulated nitric oxide release in rabbit skin microcirculation.
    The American journal of physiology, 1994, Volume: 266, Issue:5 Pt 2

    Topics: Acetylcholine; Adenosine Triphosphate; Amino Acid Oxidoreductases; Animals; Arachidonic Acid; Arginine; Bradykinin; Dinoprostone; Hydantoins; Indomethacin; Male; Microcirculation; Models, Cardiovascular; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Platelet Aggregation Inhibitors; Prostaglandin D2; Rabbits; Regional Blood Flow; Skin

1994
Further studies on ocular responses to DP receptor stimulation.
    European journal of pharmacology, 1993, Jan-19, Volume: 230, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Capillary Permeability; Cats; Conjunctiva; Dinoprost; Dinoprostone; Eye; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Intraocular Pressure; Male; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin

1993
Prostaglandin D2 inhibits prostaglandin E2-induced allodynia in conscious mice.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:3

    Topics: Adrenergic Agonists; Animals; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glycine; Hydantoins; Male; Mice; N-Methylaspartate; Pain; Prostaglandin D2; Spinal Cord; Wakefulness

1996
Interaction of BW A868C, a prostanoid DP-receptor antagonist, with two receptor subtypes in the rabbit isolated saphenous vein.
    Prostaglandins, 1996, Volume: 52, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Biphenyl Compounds; Dinoprostone; Dose-Response Relationship, Drug; Hydantoins; Male; Potassium Chloride; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Saphenous Vein

1996
Lack of tactile pain (allodynia) in lipocalin-type prostaglandin D synthase-deficient mice.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Jan-19, Volume: 96, Issue:2

    Topics: Anesthesia; Animals; Bicuculline; Central Nervous System; Dinoprost; Dinoprostone; GABA Antagonists; Gene Targeting; Hydantoins; Hyperalgesia; Immunohistochemistry; Intramolecular Oxidoreductases; Lipocalins; Mice; Mice, Knockout; Molecular Sequence Data; Pain; Prostaglandin D2; Receptors, Prostaglandin

1999
Prostaglandin DP receptors positively coupled to adenylyl cyclase in embryonic bovine tracheal (EBTr) cells: pharmacological characterization using agonists and antagonists.
    British journal of pharmacology, 1999, Volume: 127, Issue:1

    Topics: Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cattle; Cells, Cultured; Cyclic AMP; Embryo, Mammalian; Enzyme Inhibitors; Hydantoins; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Stimulation, Chemical; Trachea; Xanthenes; Xanthones

1999
Pharmacology and autoradiography of human DP prostanoid receptors using [(3)H]-BWA868C, a DP receptor-selective antagonist radioligand.
    British journal of pharmacology, 2000, Volume: 131, Issue:6

    Topics: Autoradiography; Blood Platelets; Cell Membrane; Eye; Humans; Hydantoins; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin

2000
The human prostanoid DP receptor stimulates mucin secretion in LS174T cells.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Benzoates; Binding, Competitive; Cell Membrane; Colon; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Humans; Hydantoins; In Situ Hybridization; Mucins; Prostaglandin D2; Radioligand Assay; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger; Thiazoles; Thiazolidines; Transcription, Genetic; Tritium; Tumor Cells, Cultured

2000
Prostaglandin D2 is a potent chemoattractant for human eosinophils that acts via a novel DP receptor.
    Blood, 2001, Sep-15, Volume: 98, Issue:6

    Topics: Actins; Cells, Cultured; Chemotactic Factors; Chemotaxis, Leukocyte; Cyclic AMP; Dose-Response Relationship, Drug; Eosinophils; Humans; Hydantoins; L-Selectin; Macrophage-1 Antigen; Models, Biological; Neutrophils; Prostaglandin D2; Prostaglandins; Receptors, Immunologic; Receptors, Prostaglandin

2001
Production of prostaglandin D(2) by human osteoblasts and modulation of osteoprotegerin, RANKL, and cellular migration by DP and CRTH2 receptors.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2005, Volume: 20, Issue:4

    Topics: Bone and Bones; Carrier Proteins; Chemotaxis; Cyclic AMP; Glycoproteins; Growth Substances; Humans; Hydantoins; Insulin-Like Growth Factor I; Interleukin-1; Membrane Glycoproteins; Osteoblasts; Osteoprotegerin; Prostaglandin D2; RANK Ligand; Receptor Activator of Nuclear Factor-kappa B; Receptors, Cytoplasmic and Nuclear; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Tumor Necrosis Factor; Tumor Necrosis Factor-alpha; Vascular Endothelial Growth Factor A

2005
Interactive effect of histamine and prostaglandin D2 on nasal allergic symptoms in rats.
    European journal of pharmacology, 2007, Jan-12, Volume: 554, Issue:2-3

    Topics: Administration, Intranasal; Administration, Oral; Animals; Carbazoles; Chlorpheniramine; Cyproheptadine; Dose-Response Relationship, Drug; Drug Synergism; Histamine; Histamine Agents; Histamine H1 Antagonists; Hydantoins; Injections, Intravenous; Nasal Mucosa; Prostaglandin D2; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Rhinitis; Sneezing; Sulfonamides

2007
Effects of TS-022, a newly developed prostanoid DP1 receptor agonist, on experimental pruritus, cutaneous barrier disruptions and atopic dermatitis in mice.
    European journal of pharmacology, 2007, Feb-05, Volume: 556, Issue:1-3

    Topics: Acetates; Animals; Antipruritics; Concanavalin A; Cyclohexanes; Cytokines; Dermatitis, Atopic; Dexamethasone; Humans; Hydantoins; Immunosuppressive Agents; Inflammation; Male; Mice; Platelet Aggregation; Prostaglandin D2; Pruritus; Receptors, Immunologic; Receptors, Prostaglandin; Skin; Sulfhydryl Compounds; Tacrolimus; Wound Healing

2007
Met-Arg-Trp derived from Rubisco lowers blood pressure via prostaglandin D(2)-dependent vasorelaxation in spontaneously hypertensive rats.
    Peptides, 2008, Volume: 29, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Blood Pressure; Drug Administration Schedule; Hydantoins; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Peptides; Prostaglandin D2; Rats; Rats, Inbred SHR; Ribulose-Bisphosphate Carboxylase; Transcription Factor DP1; Vasodilation

2008
CRTH2 is not involved in the anti-enteropooling effect of PGD2 in the small intestine.
    Pharmacology, 2008, Volume: 81, Issue:3

    Topics: 16,16-Dimethylprostaglandin E2; Animals; Female; Hydantoins; Intestinal Secretions; Intestine, Small; Prostaglandin D2; Rats; Rats, Sprague-Dawley; Receptors, Immunologic; Receptors, Prostaglandin

2008
GIF-0173 protects against cerebral infarction through DP1 receptor activation.
    Experimental neurology, 2009, Volume: 219, Issue:2

    Topics: Animals; Brain Infarction; Calcium; Cell Death; Cells, Cultured; Cerebral Cortex; Cerebrovascular Circulation; Dantrolene; Disease Models, Animal; Dose-Response Relationship, Drug; Glutamic Acid; Hydantoins; Infarction, Middle Cerebral Artery; Intracellular Fluid; Lactones; Laser-Doppler Flowmetry; Male; N-Methylaspartate; Neurons; Neuroprotective Agents; Platelet Aggregation Inhibitors; Prostaglandin D2; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Sesquiterpenes; Severity of Illness Index; Tetrazolium Salts

2009
Complement C5a stimulates food intake via a prostaglandin D(2)- and neuropeptide Y-dependent mechanism in mice.
    Prostaglandins & other lipid mediators, 2009, Volume: 90, Issue:3-4

    Topics: Animals; Complement C5a; Cyclooxygenase 1; Cyclooxygenase 2; Eating; Hydantoins; Hypothalamus; Male; Mice; Neuropeptide Y; Prostaglandin D2; Receptors, Prostaglandin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2009
Effects of prostaglandin D2 on tetrodotoxin-resistant Na+ currents in DRG neurons of adult rat.
    Pain, 2011, Volume: 152, Issue:5

    Topics: Action Potentials; Animals; Carbazoles; Cells, Cultured; Dose-Response Relationship, Drug; Ganglia, Spinal; Hydantoins; Male; Membrane Potentials; Patch-Clamp Techniques; Platelet Aggregation Inhibitors; Prostaglandin D2; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Sensory Receptor Cells; Sodium Channel Blockers; Sulfonamides; Tetrodotoxin

2011
Induction of apoptosis in non-small cell lung carcinoma A549 cells by PGD₂ metabolite, 15d-PGJ₂.
    Cell biology international, 2011, Volume: 35, Issue:11

    Topics: Apoptosis; Carbazoles; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cell Survival; Chromatography, High Pressure Liquid; Cytochromes c; Cytosol; DNA Fragmentation; Humans; Hydantoins; Mitochondria; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides

2011
PGD2 induces eotaxin-3 via PPARγ from sebocytes: a possible pathogenesis of eosinophilic pustular folliculitis.
    The Journal of allergy and clinical immunology, 2012, Volume: 129, Issue:2

    Topics: Anilides; Carbazoles; Cell Line; Cells, Cultured; Chemokine CCL26; Chemokines, CC; Eosinophilia; Eosinophils; Fibroblasts; Folliculitis; Humans; Hydantoins; Keratinocytes; PPAR gamma; Prostaglandin D2; Receptors, Prostaglandin; RNA, Messenger; RNA, Small Interfering; Sebaceous Glands; Skin Diseases, Vesiculobullous; Sulfonamides; Transfection

2012
Prostaglandin D2 receptor D-type prostanoid receptor 2 mediates eosinophil trafficking into the esophagus.
    Diseases of the esophagus : official journal of the International Society for Diseases of the Esophagus, 2014, Volume: 27, Issue:6

    Topics: Animals; Carbazoles; Cell Movement; Eosinophil Major Basic Protein; Eosinophilic Esophagitis; Eosinophils; Epithelium; Esophagus; Guinea Pigs; Hydantoins; Male; Mast Cells; Ovalbumin; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides

2014
A novel indole compound, AWT-489, inhibits prostaglandin D2-induced CD55 expression by acting on DP prostanoid receptors as an antagonist in LS174T human colon cancer cells.
    Archives of biochemistry and biophysics, 2014, Jan-01, Volume: 541

    Topics: Carcinogenesis; CD55 Antigens; Cell Line, Tumor; Colonic Neoplasms; Cyclic AMP; Dinoprostone; Drug Design; Gene Expression Regulation, Neoplastic; Humans; Hydantoins; Indoles; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger

2014
Prostaglandin D2 regulates human colonic ion transport via the DP1 receptor.
    Life sciences, 2015, Feb-01, Volume: 122

    Topics: Calcium; Cells, Cultured; Chlorides; Colon; Cyclic AMP; Humans; Hydantoins; Ion Transport; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Prostaglandin

2015
Receptors involved in the modulation of guinea pig urinary bladder motility by prostaglandin D2.
    British journal of pharmacology, 2015, Volume: 172, Issue:16

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Prostaglandin D2; Receptors, Prostaglandin; Receptors, Thromboxane; Urinary Bladder

2015
Effect of the PGD2-DP signaling pathway on primary cultured rat hippocampal neuron injury caused by aluminum overload.
    Scientific reports, 2016, Apr-19, Volume: 6

    Topics: Animals; Calcium; Carbazoles; Cells, Cultured; Hippocampus; Hydantoins; L-Lactate Dehydrogenase; Neurons; Organometallic Compounds; Prostaglandin D2; Pyrones; Rats; Receptors, Prostaglandin; Signal Transduction; Sulfonamides

2016