bw a868c has been researched along with hydantoins in 44 studies
Studies (bw a868c) | Trials (bw a868c) | Recent Studies (post-2010) (bw a868c) | Studies (hydantoins) | Trials (hydantoins) | Recent Studies (post-2010) (hydantoins) |
---|---|---|---|---|---|
47 | 0 | 11 | 3,404 | 80 | 435 |
Protein | Taxonomy | bw a868c (IC50) | hydantoins (IC50) |
---|---|---|---|
Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 0.062 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (6.82) | 18.7374 |
1990's | 15 (34.09) | 18.2507 |
2000's | 15 (34.09) | 29.6817 |
2010's | 11 (25.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chen, J; Woodward, DF | 1 |
Ebisui, O; Fukata, J; Imura, H; Kasting, NW; Mori, K; Murakami, N; Naito, Y; Nakai, Y; Shindo, K; Tominaga, T | 1 |
Alvarez, R; Artis, DR; Bruno, JJ; Chang, LF; Eglen, RM; Kluge, AF; Whiting, RL | 1 |
Hamid-Bloomfield, S; Payne, AN; Petrovic, AA; Whittle, BJ | 1 |
Collins, BA; Kelly, MG; Robertson, AD; Trist, DG; Wood, J | 1 |
Hamid-Bloomfield, S; Whittle, BJ | 1 |
Bolofo, ML; Giles, H; Kelly, MG; Leff, P; Robertson, AD | 1 |
Betti, PA; Prior, ET; Rangachari, PK; Roberts, LJ | 1 |
Loi, RK; Warren, JB; Wilson, AJ | 1 |
Giles, H; Kageyama, M; Matsugi, T; Nishimura, K; Shirasawa, E | 1 |
Gonzalez, AP; Menger, MD; Otto, G; Palma, P; Post, S; Rentsch, M | 1 |
Hawley, SB; Nieves, AL; Protzman, CE; Spada, CS; Williams, LS; Woodward, DF | 1 |
Blackham, A; Jackson, DM; Liu, YJ | 1 |
Blackham, A; Jackson, DM; Leff, P; Liu, YJ | 1 |
Hayaishi, O; Ito, S; Minami, T; Mori, H; Okuda-Ashitaka, E | 1 |
Leff, P; Lydford, SJ; McKechnie, KC | 1 |
Eguchi, N; Hayaishi, O; Ito, S; Kanaoka, Y; Minami, T; Nagata, A; Shirafuji, N; Tanaka, T; Urade, Y; Yoshida, N | 1 |
Crider, JY; Griffin, BW; Sharif, NA | 1 |
Crankshaw, DJ; Oliveira, L; Stallwood, NA | 1 |
Davis, TL; Sharif, NA; Williams, GW | 1 |
Chadee, K; Ford-Hutchinson, AW; Metters, KM; Wright, DH | 1 |
Hu, DN; McCormick, SA; Woodward, DF | 1 |
Diamond, M; Gravel, S; Monneret, G; Powell, WS; Rokach, J | 1 |
Antoniou, J; de Brum-Fernandes, AJ; Gallant, MA; Hackett, JA; Parent, JL; Samadfam, R | 1 |
Ago, J; Inoue, T; Ishikawa, T; Kamei, C; Rahman, A | 1 |
Arai, I; Futaki, N; Hashimoto, Y; Honma, Y; Inoue, T; Koizumi, C; Nakaike, S; Nakanishi, Y; Ono, N; Sakurai, T; Sugimoto, M; Takahashi, N; Takaoka, A; Tanami, T; Yagi, M | 1 |
Inoue, T; Ishikawa, T; Kamei, C; Ohtsu, H; Rahman, MA; Yatsuzuka, R | 1 |
Ohinata, K; Usui, H; Yoshikawa, M; Zhao, H | 1 |
Heinemann, A; Peskar, BA; Prenn, C; Schuligoi, R | 1 |
Heinemann, A; Lippe, IT; Peskar, BA; Schuligoi, R; Sedej, M; Sturm, EM; Vukoja, A; Waldhoer, M | 1 |
Ohinata, K; Yoshikawa, M; Zhao, H | 1 |
Furuta, K; Hokamura, K; Ibaraki, K; Maeda, M; Suzuki, M; Thura, M; Umemura, K; Yamamoto, S | 1 |
Asakawa, A; Biyajima, K; Eguchi, N; Inui, A; Kaneko, K; Miyamoto, C; Ohinata, K; Takagi, K; Urade, Y; Yoshikawa, M | 1 |
Ebersberger, A; Eitner, A; Halbhuber, KJ; Natura, G; Rost, R; Schaible, HG | 1 |
Mak, OT; Wang, JJ | 1 |
Doi, H; Egawa, G; Hirabayashi, T; Kabashima, K; Miyachi, Y; Murakami, M; Nakahigashi, K; Otsuka, A; Tanizaki, H; Urade, Y; Zouboulis, CC | 1 |
Miyamoto, C; Mizushige, T; Ohinata, K; Yoshida, M; Yoshikawa, M | 1 |
Wu, X; Yu, S; Zhang, S | 1 |
Arai, T; Awata, A; Fujino, H; Murayama, T; Okura, I; Oyama, S; Regan, JW; Yamazaki, R | 1 |
Baird, AW; Collins, D; Medani, M; Mohan, HM; Walsh, E; Winter, DC | 1 |
Jones, RL; Syed, NI | 1 |
de Verdier, PJ; Guan, NN; Gustafsson, LE; Svennersten, K; Wiklund, NP | 1 |
Hu, X; Ji, C; Kuang, S; Liang, G; Luo, Y; Ma, J; Mai, S; Tian, X; Wei, Y; Yang, J; Yang, Q; Yang, Y | 1 |
Hirai, R; Masuko, S; Murata, T; Nagata, N; Nakamura, T; Tachibana, Y | 1 |
44 other study(ies) available for bw a868c and hydantoins
Article | Year |
---|---|
Prostanoid-induced relaxation of precontracted cat ciliary muscle is mediated by EP2 and DP receptors.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cats; Ciliary Body; Female; Hydantoins; Isometric Contraction; Male; Muscle Relaxation; Muscle, Smooth; Platelet Aggregation Inhibitors; Prostaglandins; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Prostaglandin E | 1992 |
Effects of interleukins on plasma arginine vasopressin and oxytocin levels in conscious, freely moving rats.
Topics: Animals; Arginine Vasopressin; Aspirin; Blood Pressure; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Humans; Hydantoins; Interleukin-1; Interleukin-6; Male; Oxytocin; Platelet Aggregation Inhibitors; Rats; Rats, Inbred Strains; Recombinant Proteins; Reference Values | 1991 |
Stimulation of prostaglandin D2 receptors on human platelets by analogs of prostacyclin.
Topics: Adenosine Diphosphate; Adenylyl Cyclases; Alprostadil; Blood Platelets; Bridged-Ring Compounds; Dose-Response Relationship, Drug; Epoprostenol; Female; Humans; Hydantoins; Molecular Conformation; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Stereoisomerism | 1991 |
The role of prostanoid TP- and DP-receptors in the bronchoconstrictor effect of inhaled PGD2 in anaesthetized guinea-pigs: effect of the DP-antagonist BW A868C.
Topics: Administration, Inhalation; Anesthesia; Animals; Benzeneacetamides; Bronchi; Cyclooxygenase Inhibitors; Guinea Pigs; Hydantoins; Hydroxamic Acids; Indomethacin; Lipoxygenase Inhibitors; Male; Platelet Aggregation Inhibitors; Prostaglandin D2; Prostaglandins D; Receptors, Prostaglandin; Respiratory Function Tests; Sulfonamides; Thromboxane A2; Vagotomy | 1990 |
The antagonism by BW A868C of PGD2 and BW245C activation of human platelet adenylate cyclase.
Topics: Adenylyl Cyclases; Blood Platelets; Enzyme Activation; Epoprostenol; Humans; Hydantoins; Iloprost; In Vitro Techniques; Platelet Aggregation; Prostaglandin D2; Receptors, Prostaglandin | 1989 |
Antagonism of PGD2 vasodepressor responses in the rat in vivo by the novel, selective antagonist, BW A868C.
Topics: Animals; Blood Pressure; Epoprostenol; Hydantoins; Infusions, Intravenous; Male; Prostaglandin D2; Rats; Rats, Inbred Strains; Receptors, Prostaglandin; Sulfonamides | 1989 |
The classification of prostaglandin DP-receptors in platelets and vasculature using BW A868C, a novel, selective and potent competitive antagonist.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Blood Platelets; Blood Vessels; Guinea Pigs; Humans; Hydantoins; In Vitro Techniques; Jugular Veins; Male; Muscle Contraction; Platelet Aggregation; Prostaglandin D2; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Prostaglandin; Sulfonamides; Trachea | 1989 |
Effects of a selective DP receptor agonist (BW 245C) and antagonist (BW A868C) on the canine colonic epithelium: an argument for a different DP receptor?
Topics: Animals; Colon; Dogs; Electrophysiology; Female; Hydantoins; In Vitro Techniques; Intestinal Mucosa; Male; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin | 1995 |
PGD2 is an intermediate in agonist-stimulated nitric oxide release in rabbit skin microcirculation.
Topics: Acetylcholine; Adenosine Triphosphate; Amino Acid Oxidoreductases; Animals; Arachidonic Acid; Arginine; Bradykinin; Dinoprostone; Hydantoins; Indomethacin; Male; Microcirculation; Models, Cardiovascular; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Platelet Aggregation Inhibitors; Prostaglandin D2; Rabbits; Regional Blood Flow; Skin | 1994 |
Selective prostaglandin D2 receptor stimulation elicits ocular hypotensive effects in rabbits and cats.
Topics: Animals; Butyrates; Cats; Hydantoins; Imidazoles; Intraocular Pressure; Male; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin | 1995 |
Role of eicosanoids in reperfusion injury in rat liver transplantation.
Topics: Animals; Eicosanoids; Hydantoins; Indoles; Leukotriene Antagonists; Liver Transplantation; Male; Methacrylates; Platelet Aggregation Inhibitors; Rats; Rats, Inbred Lew; Receptors, Thromboxane; Reperfusion Injury; Thromboxane A2; Thromboxane-A Synthase | 1993 |
Further studies on ocular responses to DP receptor stimulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Capillary Permeability; Cats; Conjunctiva; Dinoprost; Dinoprostone; Eye; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Intraocular Pressure; Male; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin | 1993 |
Effects of BW A868C, a selective prostaglandin DP receptor antagonist, in dog isolated vascular preparations.
Topics: Animals; Dogs; Female; Hydantoins; In Vitro Techniques; Male | 1996 |
Partial agonist effects of BW A868C, a selective DP receptor antagonist, on Cl- secretion in dog tracheal epithelium.
Topics: Animals; Chlorides; Dogs; Drug Interactions; Epithelium; Female; Hydantoins; In Vitro Techniques; Male; Models, Biological; Prostaglandins D; Receptors, Prostaglandin; Trachea | 1996 |
Prostaglandin D2 inhibits prostaglandin E2-induced allodynia in conscious mice.
Topics: Adrenergic Agonists; Animals; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glycine; Hydantoins; Male; Mice; N-Methylaspartate; Pain; Prostaglandin D2; Spinal Cord; Wakefulness | 1996 |
Interaction of BW A868C, a prostanoid DP-receptor antagonist, with two receptor subtypes in the rabbit isolated saphenous vein.
Topics: Animals; Anti-Arrhythmia Agents; Biphenyl Compounds; Dinoprostone; Dose-Response Relationship, Drug; Hydantoins; Male; Potassium Chloride; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Saphenous Vein | 1996 |
Lack of tactile pain (allodynia) in lipocalin-type prostaglandin D synthase-deficient mice.
Topics: Anesthesia; Animals; Bicuculline; Central Nervous System; Dinoprost; Dinoprostone; GABA Antagonists; Gene Targeting; Hydantoins; Hyperalgesia; Immunohistochemistry; Intramolecular Oxidoreductases; Lipocalins; Mice; Mice, Knockout; Molecular Sequence Data; Pain; Prostaglandin D2; Receptors, Prostaglandin | 1999 |
Prostaglandin DP receptors positively coupled to adenylyl cyclase in embryonic bovine tracheal (EBTr) cells: pharmacological characterization using agonists and antagonists.
Topics: Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cattle; Cells, Cultured; Cyclic AMP; Embryo, Mammalian; Enzyme Inhibitors; Hydantoins; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Stimulation, Chemical; Trachea; Xanthenes; Xanthones | 1999 |
Effects of some isoprostanes on the human umbilical artery in vitro.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Arachidonic Acids; Dinoprostone; Endocannabinoids; Enzyme Inhibitors; Female; Humans; Hydantoins; In Vitro Techniques; Isometric Contraction; Isoprostanes; Muscle Contraction; NG-Nitroarginine Methyl Ester; Polyunsaturated Alkamides; Pregnancy; Prostaglandins F; Prostaglandins, Synthetic; Receptors, Prostaglandin; Structure-Activity Relationship; Umbilical Arteries | 2000 |
Pharmacology and autoradiography of human DP prostanoid receptors using [(3)H]-BWA868C, a DP receptor-selective antagonist radioligand.
Topics: Autoradiography; Blood Platelets; Cell Membrane; Eye; Humans; Hydantoins; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin | 2000 |
The human prostanoid DP receptor stimulates mucin secretion in LS174T cells.
Topics: Benzoates; Binding, Competitive; Cell Membrane; Colon; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Humans; Hydantoins; In Situ Hybridization; Mucins; Prostaglandin D2; Radioligand Assay; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger; Thiazoles; Thiazolidines; Transcription, Genetic; Tritium; Tumor Cells, Cultured | 2000 |
A functional study on prostanoid receptors involved in cultured human iridal melanocyte stimulation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Cell Count; Cells, Cultured; Cyclic AMP; Dinoprostone; Epoprostenol; Fibroblast Growth Factor 2; Humans; Hydantoins; Iris; Melanins; Melanocytes; Prostaglandin Antagonists; Prostanoic Acids; Receptors, Prostaglandin | 2001 |
Prostaglandin D2 is a potent chemoattractant for human eosinophils that acts via a novel DP receptor.
Topics: Actins; Cells, Cultured; Chemotactic Factors; Chemotaxis, Leukocyte; Cyclic AMP; Dose-Response Relationship, Drug; Eosinophils; Humans; Hydantoins; L-Selectin; Macrophage-1 Antigen; Models, Biological; Neutrophils; Prostaglandin D2; Prostaglandins; Receptors, Immunologic; Receptors, Prostaglandin | 2001 |
Production of prostaglandin D(2) by human osteoblasts and modulation of osteoprotegerin, RANKL, and cellular migration by DP and CRTH2 receptors.
Topics: Bone and Bones; Carrier Proteins; Chemotaxis; Cyclic AMP; Glycoproteins; Growth Substances; Humans; Hydantoins; Insulin-Like Growth Factor I; Interleukin-1; Membrane Glycoproteins; Osteoblasts; Osteoprotegerin; Prostaglandin D2; RANK Ligand; Receptor Activator of Nuclear Factor-kappa B; Receptors, Cytoplasmic and Nuclear; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Tumor Necrosis Factor; Tumor Necrosis Factor-alpha; Vascular Endothelial Growth Factor A | 2005 |
Interactive effect of histamine and prostaglandin D2 on nasal allergic symptoms in rats.
Topics: Administration, Intranasal; Administration, Oral; Animals; Carbazoles; Chlorpheniramine; Cyproheptadine; Dose-Response Relationship, Drug; Drug Synergism; Histamine; Histamine Agents; Histamine H1 Antagonists; Hydantoins; Injections, Intravenous; Nasal Mucosa; Prostaglandin D2; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Rhinitis; Sneezing; Sulfonamides | 2007 |
Effects of TS-022, a newly developed prostanoid DP1 receptor agonist, on experimental pruritus, cutaneous barrier disruptions and atopic dermatitis in mice.
Topics: Acetates; Animals; Antipruritics; Concanavalin A; Cyclohexanes; Cytokines; Dermatitis, Atopic; Dexamethasone; Humans; Hydantoins; Immunosuppressive Agents; Inflammation; Male; Mice; Platelet Aggregation; Prostaglandin D2; Pruritus; Receptors, Immunologic; Receptors, Prostaglandin; Skin; Sulfhydryl Compounds; Tacrolimus; Wound Healing | 2007 |
Involvement of chemical mediators in nasal allergic responses of HDC-KO mice.
Topics: Animals; Behavior, Animal; Chlorpheniramine; Histamine H1 Antagonists; Histidine Decarboxylase; Hydantoins; Immunization; Immunoglobulin E; Inflammation Mediators; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Immunologic; Receptors, Prostaglandin; Rhinitis, Allergic, Seasonal; Sneezing; Substance P | 2007 |
Met-Arg-Trp derived from Rubisco lowers blood pressure via prostaglandin D(2)-dependent vasorelaxation in spontaneously hypertensive rats.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Blood Pressure; Drug Administration Schedule; Hydantoins; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Peptides; Prostaglandin D2; Rats; Rats, Inbred SHR; Ribulose-Bisphosphate Carboxylase; Transcription Factor DP1; Vasodilation | 2008 |
CRTH2 is not involved in the anti-enteropooling effect of PGD2 in the small intestine.
Topics: 16,16-Dimethylprostaglandin E2; Animals; Female; Hydantoins; Intestinal Secretions; Intestine, Small; Prostaglandin D2; Rats; Rats, Sprague-Dawley; Receptors, Immunologic; Receptors, Prostaglandin | 2008 |
Prostaglandin H2 induces the migration of human eosinophils through the chemoattractant receptor homologous molecule of Th2 cells, CRTH2.
Topics: Basophils; Blood Proteins; Calcium; Carbazoles; Cations, Divalent; Cell Degranulation; Cell Line; Chemotaxis; Collagen; Eosinophils; Humans; Hydantoins; Intramolecular Oxidoreductases; Lipocalins; Neutrophils; Piperidines; Prostaglandin H2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides | 2009 |
Central prostaglandin D(2) exhibits anxiolytic-like activity via the DP(1) receptor in mice.
Topics: Adenosine A2 Receptor Antagonists; Animals; Anti-Anxiety Agents; Bicuculline; GABA-A Receptor Antagonists; Hydantoins; Male; Maze Learning; Mice; Prostaglandins D; Receptor, Adenosine A2A; Receptors, GABA-A; Receptors, Prostaglandin | 2009 |
GIF-0173 protects against cerebral infarction through DP1 receptor activation.
Topics: Animals; Brain Infarction; Calcium; Cell Death; Cells, Cultured; Cerebral Cortex; Cerebrovascular Circulation; Dantrolene; Disease Models, Animal; Dose-Response Relationship, Drug; Glutamic Acid; Hydantoins; Infarction, Middle Cerebral Artery; Intracellular Fluid; Lactones; Laser-Doppler Flowmetry; Male; N-Methylaspartate; Neurons; Neuroprotective Agents; Platelet Aggregation Inhibitors; Prostaglandin D2; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Sesquiterpenes; Severity of Illness Index; Tetrazolium Salts | 2009 |
Complement C5a stimulates food intake via a prostaglandin D(2)- and neuropeptide Y-dependent mechanism in mice.
Topics: Animals; Complement C5a; Cyclooxygenase 1; Cyclooxygenase 2; Eating; Hydantoins; Hypothalamus; Male; Mice; Neuropeptide Y; Prostaglandin D2; Receptors, Prostaglandin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2009 |
Effects of prostaglandin D2 on tetrodotoxin-resistant Na+ currents in DRG neurons of adult rat.
Topics: Action Potentials; Animals; Carbazoles; Cells, Cultured; Dose-Response Relationship, Drug; Ganglia, Spinal; Hydantoins; Male; Membrane Potentials; Patch-Clamp Techniques; Platelet Aggregation Inhibitors; Prostaglandin D2; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Prostaglandin; Sensory Receptor Cells; Sodium Channel Blockers; Sulfonamides; Tetrodotoxin | 2011 |
Induction of apoptosis in non-small cell lung carcinoma A549 cells by PGD₂ metabolite, 15d-PGJ₂.
Topics: Apoptosis; Carbazoles; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cell Survival; Chromatography, High Pressure Liquid; Cytochromes c; Cytosol; DNA Fragmentation; Humans; Hydantoins; Mitochondria; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides | 2011 |
PGD2 induces eotaxin-3 via PPARγ from sebocytes: a possible pathogenesis of eosinophilic pustular folliculitis.
Topics: Anilides; Carbazoles; Cell Line; Cells, Cultured; Chemokine CCL26; Chemokines, CC; Eosinophilia; Eosinophils; Fibroblasts; Folliculitis; Humans; Hydantoins; Keratinocytes; PPAR gamma; Prostaglandin D2; Receptors, Prostaglandin; RNA, Messenger; RNA, Small Interfering; Sebaceous Glands; Skin Diseases, Vesiculobullous; Sulfonamides; Transfection | 2012 |
Complement C5a exhibits anxiolytic-like activity via the prostaglandin D2-DP1 receptor system coupled to adenosine A2A and GABAA receptors.
Topics: Animals; Anti-Anxiety Agents; Bicuculline; Complement C5a; Hydantoins; Indomethacin; Male; Mice; Receptor, Adenosine A2A; Receptors, GABA-A; Receptors, Immunologic; Receptors, Prostaglandin | 2012 |
Prostaglandin D2 receptor D-type prostanoid receptor 2 mediates eosinophil trafficking into the esophagus.
Topics: Animals; Carbazoles; Cell Movement; Eosinophil Major Basic Protein; Eosinophilic Esophagitis; Eosinophils; Epithelium; Esophagus; Guinea Pigs; Hydantoins; Male; Mast Cells; Ovalbumin; Prostaglandin Antagonists; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; Sulfonamides | 2014 |
A novel indole compound, AWT-489, inhibits prostaglandin D2-induced CD55 expression by acting on DP prostanoid receptors as an antagonist in LS174T human colon cancer cells.
Topics: Carcinogenesis; CD55 Antigens; Cell Line, Tumor; Colonic Neoplasms; Cyclic AMP; Dinoprostone; Drug Design; Gene Expression Regulation, Neoplastic; Humans; Hydantoins; Indoles; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger | 2014 |
Prostaglandin D2 regulates human colonic ion transport via the DP1 receptor.
Topics: Calcium; Cells, Cultured; Chlorides; Colon; Cyclic AMP; Humans; Hydantoins; Ion Transport; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Prostaglandin | 2015 |
Assessing the agonist profiles of the prostacyclin analogues treprostinil and naxaprostene, particularly their DP₁ activity.
Topics: Animals; Epoprostenol; Hydantoins; Indoles; Male; Mice; Mice, Inbred C57BL; Molecular Structure; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin; Structure-Activity Relationship | 2015 |
Receptors involved in the modulation of guinea pig urinary bladder motility by prostaglandin D2.
Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Prostaglandin D2; Receptors, Prostaglandin; Receptors, Thromboxane; Urinary Bladder | 2015 |
Effect of the PGD2-DP signaling pathway on primary cultured rat hippocampal neuron injury caused by aluminum overload.
Topics: Animals; Calcium; Carbazoles; Cells, Cultured; Hippocampus; Hydantoins; L-Lactate Dehydrogenase; Neurons; Organometallic Compounds; Prostaglandin D2; Pyrones; Rats; Receptors, Prostaglandin; Signal Transduction; Sulfonamides | 2016 |
Therapeutic potential of D prostanoid receptor 1 signal enhancement in a murine model of food allergy.
Topics: Animals; Disease Models, Animal; Female; Food Hypersensitivity; Hydantoins; Intestines; Mast Cells; Mice, Inbred BALB C; Receptors, Prostaglandin | 2019 |