bw a868c has been researched along with dinoprostone in 12 studies
Studies (bw a868c) | Trials (bw a868c) | Recent Studies (post-2010) (bw a868c) | Studies (dinoprostone) | Trials (dinoprostone) | Recent Studies (post-2010) (dinoprostone) |
---|---|---|---|---|---|
47 | 0 | 11 | 29,105 | 1,346 | 6,357 |
Protein | Taxonomy | bw a868c (IC50) | dinoprostone (IC50) |
---|---|---|---|
Prostaglandin E2 receptor EP1 subtype | Homo sapiens (human) | 0.0155 | |
Prostaglandin E2 receptor EP4 subtype | Homo sapiens (human) | 0.0031 | |
Prostaglandin E2 receptor EP4 subtype | Rattus norvegicus (Norway rat) | 0.0021 | |
Prostaglandin E2 receptor EP3 subtype | Homo sapiens (human) | 0.002 | |
Prostaglandin E2 receptor EP2 subtype | Homo sapiens (human) | 0.0087 | |
Prostacyclin receptor | Homo sapiens (human) | 0.26 | |
Prostaglandin E2 receptor EP2 subtype | Rattus norvegicus (Norway rat) | 0.0052 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (66.67) | 18.2507 |
2000's | 3 (25.00) | 29.6817 |
2010's | 1 (8.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Abramovitz, M; Boie, Y; Metters, KM; Sawyer, N; Slipetz, DM | 1 |
Hirata, M; Kiriyama, M; Kobayashi, T; Narumiya, S; Sugimoto, Y; Ushikubi, F | 1 |
Abramovitz, M; Ford-Hutchinson, AW; Metters, KM; Wright, DH | 1 |
Loi, RK; Warren, JB; Wilson, AJ | 1 |
Hawley, SB; Nieves, AL; Protzman, CE; Spada, CS; Williams, LS; Woodward, DF | 1 |
Hayaishi, O; Ito, S; Minami, T; Mori, H; Okuda-Ashitaka, E | 1 |
Leff, P; Lydford, SJ; McKechnie, KC | 1 |
Eguchi, N; Hayaishi, O; Ito, S; Kanaoka, Y; Minami, T; Nagata, A; Shirafuji, N; Tanaka, T; Urade, Y; Yoshida, N | 1 |
Crankshaw, DJ; Oliveira, L; Stallwood, NA | 1 |
Chadee, K; Ford-Hutchinson, AW; Metters, KM; Wright, DH | 1 |
Hu, DN; McCormick, SA; Woodward, DF | 1 |
Arai, T; Awata, A; Fujino, H; Murayama, T; Okura, I; Oyama, S; Regan, JW; Yamazaki, R | 1 |
12 other study(ies) available for bw a868c and dinoprostone
Article | Year |
---|---|
Molecular cloning and characterization of the human prostanoid DP receptor.
Topics: Amino Acid Sequence; Base Sequence; Blotting, Northern; Calcium; Cells, Cultured; Cloning, Molecular; Cyclic AMP; Humans; Molecular Sequence Data; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin | 1995 |
Ligand binding specificities of the eight types and subtypes of the mouse prostanoid receptors expressed in Chinese hamster ovary cells.
Topics: Animals; CHO Cells; Cricetinae; Ligands; Mice; Prostaglandins; Receptors, Prostaglandin; Transfection | 1997 |
Characterization of the recombinant human prostanoid DP receptor and identification of L-644,698, a novel selective DP agonist.
Topics: Adenine Nucleotides; Benzoates; Binding, Competitive; Cell Line; Cyclic AMP; Dinoprostone; Guanine Nucleotides; Humans; Kinetics; Receptors, Immunologic; Receptors, Prostaglandin; Recombinant Proteins; Thiazoles; Thiazolidines; Tritium | 1998 |
PGD2 is an intermediate in agonist-stimulated nitric oxide release in rabbit skin microcirculation.
Topics: Acetylcholine; Adenosine Triphosphate; Amino Acid Oxidoreductases; Animals; Arachidonic Acid; Arginine; Bradykinin; Dinoprostone; Hydantoins; Indomethacin; Male; Microcirculation; Models, Cardiovascular; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Platelet Aggregation Inhibitors; Prostaglandin D2; Rabbits; Regional Blood Flow; Skin | 1994 |
Further studies on ocular responses to DP receptor stimulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Capillary Permeability; Cats; Conjunctiva; Dinoprost; Dinoprostone; Eye; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Intraocular Pressure; Male; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin | 1993 |
Prostaglandin D2 inhibits prostaglandin E2-induced allodynia in conscious mice.
Topics: Adrenergic Agonists; Animals; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glycine; Hydantoins; Male; Mice; N-Methylaspartate; Pain; Prostaglandin D2; Spinal Cord; Wakefulness | 1996 |
Interaction of BW A868C, a prostanoid DP-receptor antagonist, with two receptor subtypes in the rabbit isolated saphenous vein.
Topics: Animals; Anti-Arrhythmia Agents; Biphenyl Compounds; Dinoprostone; Dose-Response Relationship, Drug; Hydantoins; Male; Potassium Chloride; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Saphenous Vein | 1996 |
Lack of tactile pain (allodynia) in lipocalin-type prostaglandin D synthase-deficient mice.
Topics: Anesthesia; Animals; Bicuculline; Central Nervous System; Dinoprost; Dinoprostone; GABA Antagonists; Gene Targeting; Hydantoins; Hyperalgesia; Immunohistochemistry; Intramolecular Oxidoreductases; Lipocalins; Mice; Mice, Knockout; Molecular Sequence Data; Pain; Prostaglandin D2; Receptors, Prostaglandin | 1999 |
Effects of some isoprostanes on the human umbilical artery in vitro.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Arachidonic Acids; Dinoprostone; Endocannabinoids; Enzyme Inhibitors; Female; Humans; Hydantoins; In Vitro Techniques; Isometric Contraction; Isoprostanes; Muscle Contraction; NG-Nitroarginine Methyl Ester; Polyunsaturated Alkamides; Pregnancy; Prostaglandins F; Prostaglandins, Synthetic; Receptors, Prostaglandin; Structure-Activity Relationship; Umbilical Arteries | 2000 |
The human prostanoid DP receptor stimulates mucin secretion in LS174T cells.
Topics: Benzoates; Binding, Competitive; Cell Membrane; Colon; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Humans; Hydantoins; In Situ Hybridization; Mucins; Prostaglandin D2; Radioligand Assay; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger; Thiazoles; Thiazolidines; Transcription, Genetic; Tritium; Tumor Cells, Cultured | 2000 |
A functional study on prostanoid receptors involved in cultured human iridal melanocyte stimulation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Cell Count; Cells, Cultured; Cyclic AMP; Dinoprostone; Epoprostenol; Fibroblast Growth Factor 2; Humans; Hydantoins; Iris; Melanins; Melanocytes; Prostaglandin Antagonists; Prostanoic Acids; Receptors, Prostaglandin | 2001 |
A novel indole compound, AWT-489, inhibits prostaglandin D2-induced CD55 expression by acting on DP prostanoid receptors as an antagonist in LS174T human colon cancer cells.
Topics: Carcinogenesis; CD55 Antigens; Cell Line, Tumor; Colonic Neoplasms; Cyclic AMP; Dinoprostone; Drug Design; Gene Expression Regulation, Neoplastic; Humans; Hydantoins; Indoles; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger | 2014 |