Page last updated: 2024-09-05

bw a522 and adenosine

bw a522 has been researched along with adenosine in 5 studies

Compound Research Comparison

Studies
(bw a522)
Trials
(bw a522)
Recent Studies (post-2010)
(bw a522)
Studies
(adenosine)
Trials
(adenosine)
Recent Studies (post-2010) (adenosine)
100032,5361,0758,930

Protein Interaction Comparison

ProteinTaxonomybw a522 (IC50)adenosine (IC50)
high affinity choline transporter 1 isoform aHomo sapiens (human)0.3851
Sodium/nucleoside cotransporter 1Homo sapiens (human)5.5
Sodium/nucleoside cotransporter 2Homo sapiens (human)5.5
Adenosine receptor A3Homo sapiens (human)0.0011
Adenosine receptor A1Homo sapiens (human)0.0023
Equilibrative nucleoside transporter 1Homo sapiens (human)63
Solute carrier family 28 member 3Homo sapiens (human)3.3

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fozard, JR; Hannon, JP1
Bai, TR; Jacobson, MA; Knight, DA; Salvatore, CA; Walker, BA; Weir, T; Zhou, D1
Jones, CA; Reeves, JJ; Sheehan, MJ; Vardey, CJ; Whelan, CJ1
Auchampach, JA; Caughey, GH; Jin, X; Linden, J; Wan, TC1
Bril, A; Broadley, KJ; Gardner, NM; Khandoudi, N; Maddock, HL1

Other Studies

5 other study(ies) available for bw a522 and adenosine

ArticleYear
BW-A522 blocks adenosine A3 receptor-mediated hypotensive responses in the rat.
    European journal of pharmacology, 1994, Feb-03, Volume: 252, Issue:2

    Topics: Adenosine; Animals; Blood Pressure; Depression, Chemical; Dose-Response Relationship, Drug; Male; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Theophylline; Xanthines

1994
Adenosine A3 receptor expression and function in eosinophils.
    American journal of respiratory cell and molecular biology, 1997, Volume: 16, Issue:5

    Topics: Adenosine; Animals; Bronchi; Cells, Cultured; Chemotaxis, Leukocyte; Eosinophils; Gene Expression Regulation; Humans; Hypersensitivity, Immediate; Iodobenzenes; Lung; Lung Diseases, Obstructive; Mesoderm; Molecular Sequence Data; Platelet Activating Factor; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; RNA, Messenger; Sheep; Xanthines

1997
Adenosine A3 receptors promote degranulation of rat mast cells both in vitro and in vivo.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1997, Volume: 46, Issue:5

    Topics: Adenosine; Administration, Cutaneous; Animals; Blood Proteins; Cell Degranulation; Cyproheptadine; Dinitrophenols; Female; Humans; In Vitro Techniques; Injections, Intravenous; Male; Mast Cells; Mice; p-Methoxy-N-methylphenethylamine; Pleura; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Rats; Rats, Wistar; Receptors, Purinergic P1; Serotonin; Serotonin Antagonists; Serum Albumin; Skin; Theophylline; Triazoles; Xanthines

1997
Canine mast cell adenosine receptors: cloning and expression of the A3 receptor and evidence that degranulation is mediated by the A2B receptor.
    Molecular pharmacology, 1997, Volume: 52, Issue:5

    Topics: Adenine; Adenosine; Amino Acid Sequence; Animals; Base Sequence; beta-N-Acetylhexosaminidases; Calcium; Chlorocebus aethiops; COS Cells; Dinucleoside Phosphates; DNA, Complementary; Dogs; Mast Cells; Mast-Cell Sarcoma; Molecular Sequence Data; Neoplasm Proteins; Norbornanes; Receptor, Adenosine A3; Receptors, Purinergic P1; RNA, Messenger; Sequence Alignment; Sequence Homology, Amino Acid; Xanthines

1997
Protection from myocardial stunning by ischaemia and hypoxia with the adenosine A3 receptor agonist, IB-MECA.
    European journal of pharmacology, 2003, Sep-23, Volume: 477, Issue:3

    Topics: Adenosine; Adenosine A3 Receptor Agonists; Animals; Coronary Circulation; Endothelium, Vascular; Guinea Pigs; Heart Atria; Hypoxia; Male; Myocardial Ischemia; Myocardial Stunning; Oxygen; Papillary Muscles; Perfusion; Receptor, Adenosine A3; Reperfusion Injury; Time Factors; Xanthines

2003