bw-755c has been researched along with calcimycin in 36 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 29 (80.56) | 18.7374 |
1990's | 7 (19.44) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Lenti, L; Pasetto, N; Piccione, E; Pontieri, G; Ticconi, C; Zicari, A | 1 |
Amalsadvala, TM; Vaughn, DM | 1 |
Ishizaki, Y; Murota, S | 1 |
Hagiwara, M; Iwamura, S; Kobayashi, M; Mikami, T; Miyasaka, K; Miyazawa, K | 1 |
Razin, E; Shoam, H | 1 |
Boctor, AM; Pugsley, TA | 1 |
Miura, K; Nozawa, Y; Okano, Y; Yamada, K | 1 |
Chand, N; Diamantis, W; Pillar, J; Sofia, RD | 1 |
McCormack, DG; Paterson, NA | 1 |
Abraham, NG; Lutton, JD; Schwartzman, ML | 1 |
Bednar, MM; Hatala, MA; Kraemer, R; Mullane, KM | 1 |
Lefkowith, JB; Morrison, AR; Schreiner, GF | 1 |
Moncada, S; Salmon, JA; Tilling, LC | 1 |
Catt, KJ; Kiesel, L; Naor, Z; Vanderhoek, JY | 1 |
Ishitoya, J; Nagai, Y; Takenawa, T | 1 |
Aked, D; Foster, SJ; Howarth, A; McCormick, ME | 1 |
Carey, F; Forder, RA | 1 |
Dreyling, KW; Hoppe, U; Kozuschek, W; Morgenroth, K; Peskar, BA; Peskar, BM | 1 |
Mita, H; Shida, T; Yui, Y | 1 |
Edwards, RH; Jackson, MJ; Wagenmakers, AJ | 1 |
Nakashima, S; Nozawa, Y; Shirato, L; Takenaka, A; Tohmatsu, T | 1 |
Hartung, HP; Toyka, KV | 1 |
BĂ©liard, R; Bocquet, J; Bouakka, M; Jouis, V; Langris, M; Legendre, P; Loyau, G | 1 |
Brooks, RR; Doerr, IL; Kaufman, J | 1 |
Boeynaems, JM; Galand, N; Ketelbant, P | 1 |
Burka, JF | 1 |
Brune, K; Peskar, BA | 1 |
Hidaka, T; Hosoe, K; Katsumi, I; Takeo, K; Watanabe, K; Yamashita, T | 1 |
Johnson, KJ; Sulavik, MC; Ward, PA | 1 |
Palmer, RM; Salmon, JA; Simmons, PM | 1 |
Harvey, J; Osborne, DJ | 1 |
Galton, SA; Letts, LG; Piper, PJ | 1 |
Piper, PJ; Samhoun, MN | 1 |
Ho, TF; Lin, CN; Teng, CM; Wang, JP | 1 |
Murthy, M; Rao, GH; Reddy, S | 1 |
Becker, I; Huber, W; Peskar, BM; Schenck, U; Schepp, W; Trautmann, M | 1 |
36 other study(ies) available for bw-755c and calcimycin
Article | Year |
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Influence of labor and oxytocin on in vitro leukotriene release by human fetal membranes and uterine decidua at term gestation.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adult; Calcimycin; Culture Techniques; Cycloheximide; Decidua; Extraembryonic Membranes; Female; Humans; Labor, Obstetric; Leukotriene B4; Oxytocin; Pregnancy; SRS-A | 1992 |
Characterization of leukotriene B4 synthesis in canine polymorphonuclear leukocytes.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Benzeneacetamides; Calcimycin; Dogs; Dose-Response Relationship, Drug; Female; Hydroxamic Acids; In Vitro Techniques; Kinetics; Leukotriene B4; Lipoxygenase Inhibitors; Male; Neutrophils; Temperature | 1992 |
Arachidonic acid metabolism in cultured astrocytes: presence of 12-lipoxygenase activity in the intact cells.
Topics: 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid; 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonate 12-Lipoxygenase; Arachidonic Acid; Astrocytes; Calcimycin; Cells, Cultured; Chromatography, High Pressure Liquid; Female; Hydroxyeicosatetraenoic Acids; Indomethacin; Pregnancy; Rats; Rats, Inbred Strains; Spectrophotometry, Ultraviolet | 1991 |
Effects of TZI-41127, a novel selective 5-lipoxygenase inhibitor, on A23187-induced pleurisy in rats.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Calcimycin; Chromatography, High Pressure Liquid; Cyclooxygenase Inhibitors; Dinoprostone; Indoles; Leukocytes; Leukotrienes; Lipoxygenase Inhibitors; Male; Pleura; Pleurisy; Radioimmunoassay; Rats; Rats, Inbred Strains | 1991 |
BW755C inhibits the 5-lipoxygenase in E-mast cells without affecting degranulation.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; beta-N-Acetylhexosaminidases; Bone Marrow Cells; Calcimycin; Cytoplasmic Granules; Dose-Response Relationship, Drug; Hexosaminidases; Histamine Release; Hydroxyeicosatetraenoic Acids; Immunoglobulin E; Lipoxygenase Inhibitors; Male; Mast Cells; Mice; Mice, Inbred BALB C; Pyrazoles; SRS-A | 1985 |
Effect of CI-922, a potential new antiallergy agent, on arachidonic acid metabolism in vitro.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adult; Animals; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arachidonic Acids; Azoles; Calcimycin; Cattle; Histamine Release; Humans; Hydroxyeicosatetraenoic Acids; In Vitro Techniques; Indoles; Indomethacin; Leukocytes; Male; Masoprocol; Pyrazoles; Seminal Vesicles; Tetrazoles | 1986 |
Arachidonic acid release in BW755C-pretreated rat peritoneal mast cells stimulated with A23187, concanavalin A and compound 48/80.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Concanavalin A; Cyclooxygenase Inhibitors; Histamine Release; In Vitro Techniques; Lipoxygenase Inhibitors; Mast Cells; p-Methoxy-N-methylphenethylamine; Pyrazoles; Rats; Rats, Inbred Strains | 1987 |
Modulation of allergic and nonallergic histamine secretion by lipoxygenase inhibitors.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 5,8,11,14-Eicosatetraynoic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcimycin; Catechols; Fatty Acids, Unsaturated; Histamine Release; Hypersensitivity; Kinetics; Lipoxygenase Inhibitors; Masoprocol; Mast Cells; Pyrazoles; Rabbits; Rats; Rats, Inbred Strains | 1987 |
The contrasting influence of two lipoxygenase inhibitors on hypoxic pulmonary vasoconstriction in anesthetized pigs.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Angiotensin II; Animals; Calcimycin; Epoprostenol; Female; Histamine Release; Hypoxia; Lipoxygenase Inhibitors; Lung; Male; Pulmonary Circulation; Pyrazoles; SRS-A; Swine; Vascular Resistance; Vasoconstriction | 1989 |
Cytochrome P450 dependent arachidonic acid metabolism in hemopoietic cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cells, Cultured; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Erythropoiesis; Hematopoietic Stem Cells; Humans; Indomethacin; Lipoxygenase Inhibitors; Mice; NADP; Neutrophils; Pyridines | 1989 |
A neutrophil-derived cytochrome P450-dependent metabolite of arachidonic acid modulates neutrophil behavior.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Cell Adhesion; Cell Aggregation; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Dogs; Leukotriene B4; Mixed Function Oxygenases; Neutrophils; Pyrazoles; Superoxides | 1987 |
Murine glomerular leukotriene B4 synthesis. Manipulation by (n-6) fatty acid deprivation and cellular origin.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Calcimycin; Chromatography, High Pressure Liquid; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids; Indomethacin; Kidney Glomerulus; Leukotriene B4; Mice; Pyrazoles; Radioimmunoassay; Rats; Rats, Inbred Lew | 1988 |
Evaluation of inhibitors of eicosanoid synthesis in leukocytes: possible pitfall of using the calcium ionophore A23187 to stimulate 5' lipoxygenase.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonate Lipoxygenases; Calcimycin; Humans; Leukotriene B4; Lipoxygenase; Neutrophils; Propionates; Pyrazoles; Thromboxane B2; Zymosan | 1985 |
Mechanism of action of gonadotropin releasing hormone: role of lipoxygenase products of arachidonic acid in luteinizing hormone release.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonate Lipoxygenases; Arachidonic Acid; Arachidonic Acids; Calcimycin; Catechols; Cells, Cultured; Gonadotropin-Releasing Hormone; Hydroxyeicosatetraenoic Acids; Leukotriene B4; Lipoxygenase; Luteinizing Hormone; Masoprocol; Pituitary Gland; Pyrazoles; Rats; SRS-A | 1985 |
Inhibitory effect of prostaglandin E2, forskolin, and dibutyryl cAMP on arachidonic acid release and inositol phospholipid metabolism in guinea pig neutrophils.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Bucladesine; Calcimycin; Catechols; Colforsin; Dinoprostone; Fatty Acids, Nonesterified; Guinea Pigs; Lysosomes; Masoprocol; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphatidylinositols; Prostaglandins E; Pyrazoles; Superoxides | 1986 |
Leukocyte recruitment in the subcutaneous sponge implant model of acute inflammation in the rat is not mediated by leukotriene B1.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acute Disease; Animals; Blood Proteins; Calcimycin; Chemotaxis, Leukocyte; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Flurbiprofen; Indomethacin; Inflammation; Leukocytes; Leukotriene B4; Lipoxygenase Inhibitors; Male; Prostaglandins E; Pyrazoles; Pyrazolones; Rats; Rats, Inbred Strains; Skin | 1986 |
Radioimmunoassay of LTB4 and 6-trans LTB4: analytical and pharmacological characterisation of immunoreactive LTB4 in ionophore stimulated human blood.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Antibodies; Antibody Specificity; Calcimycin; Catechols; Chromatography, High Pressure Liquid; Cross Reactions; Dose-Response Relationship, Drug; Female; Humans; Leukotriene B4; Male; Masoprocol; Pyrazoles; Pyrazolones; Rabbits; Radioimmunoassay; Thromboxane B2; Time Factors | 1986 |
Leukotriene synthesis by human gastrointestinal tissues.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Adenocarcinoma; Arachidonic Acid; Arachidonic Acids; Calcimycin; Chromatography, High Pressure Liquid; Colonic Neoplasms; Digestive System; Dinoprostone; Gastric Mucosa; Humans; In Vitro Techniques; Intestinal Mucosa; Leukotriene B4; Masoprocol; Muscle, Smooth; Prostaglandins E; Pyrazoles; SRS-A | 1986 |
Effect of AA-861, a 5-lipoxygenase inhibitor, on leukotriene synthesis in human polymorphonuclear leukocytes and on cyclooxygenase and 12-lipoxygenase activities in human platelets.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Blood Platelets; Calcimycin; Diethylcarbamazine; Humans; Leukotriene B4; Lipoxygenase Inhibitors; Neutrophils; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Quinones; SRS-A | 1986 |
Effect of inhibitors of arachidonic acid metabolism on efflux of intracellular enzymes from skeletal muscle following experimental damage.
Topics: 2,4-Dinitrophenol; 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonate Lipoxygenases; Arachidonic Acid; Arachidonic Acids; Calcimycin; Creatine Kinase; Cyclooxygenase Inhibitors; Dinitrophenols; Female; In Vitro Techniques; Masoprocol; Muscles; Muscular Diseases; Phenylacetates; Prostaglandins; Pyrazoles; Rats; Rats, Inbred Strains | 1987 |
Neomycin is a potent agent for arachidonic acid release in human platelets.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcimycin; Calcium; Cell Membrane Permeability; Humans; Neomycin; Phospholipases A; Phospholipases A2; Pyrazoles; Saponins; Serotonin; Thrombin | 1987 |
Leukotriene production by cultured astroglial cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Astrocytes; Calcimycin; Carcinogens; Cells, Cultured; Kinetics; Phorbol Esters; Pyrazoles; Rats; SRS-A; Tetradecanoylphorbol Acetate | 1987 |
Calcium ionophore and phorbol myristate acetate synergistically inhibited proteoglycan biosynthesis in articular chondrocytes by prostaglandin independent mechanism.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acids; Calcimycin; Cartilage, Articular; Diglycerides; Dinoprostone; Drug Synergism; Indomethacin; Prostaglandins E; Proteoglycans; Pyrazoles; Rabbits; Tetradecanoylphorbol Acetate | 1988 |
Effects of orpanoxin on arachidonic acid metabolism of human polymorphonuclear leucocytes and platelets in vitro.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcimycin; Chromatography, High Pressure Liquid; Female; Humans; In Vitro Techniques; Indicators and Reagents; Indomethacin; Male; Neutrophils; Propionates | 1988 |
Prostacyclin production by the deendothelialized rabbit aorta.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 6-Ketoprostaglandin F1 alpha; Animals; Aorta; Arachidonic Acid; Arachidonic Acids; Calcimycin; Endothelium; Epoprostenol; Indomethacin; Kinetics; Male; Pyrazoles; Rabbits | 1985 |
Pharmacological modulation of responses of guinea-pig airways contracted with antigen and calcium ionophore A23187.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonate Lipoxygenases; Calcimycin; Catechols; Chromones; Drug Interactions; Epoprostenol; Guinea Pigs; Indomethacin; Lipoxygenase Inhibitors; Lung; Male; Masoprocol; Muscle Contraction; Ovalbumin; Pyrazoles; Pyrazolones; Trachea | 1985 |
Modulation by drugs of leukotriene and prostaglandin production from mouse peritoneal macrophages.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acetaminophen; Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Calcimycin; Dinoprostone; Dipyrone; Indomethacin; Macrophages; Male; Mice; Propionates; Prostaglandins E; Pyrazoles; Pyrazolones; SRS-A | 1985 |
Inhibition of polymorphonuclear leukocyte 5-lipoxygenase and platelet cyclooxygenase by alpha-(3,5-di-tert-butyl-4-hydroxybenzylidene)-gamma-butyrolacto ne (KME-4), a new anti-inflammatory drug.
Topics: 4-Butyrolactone; 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Anti-Inflammatory Agents; Arachidonate Lipoxygenases; Blood Platelets; Calcimycin; Chromatography, Thin Layer; Cyclooxygenase Inhibitors; Furans; Guinea Pigs; In Vitro Techniques; Indomethacin; Lipoxygenase Inhibitors; Male; Neutrophils; Pyrazoles; Rabbits | 1985 |
Rat neutrophil activation and effects of lipoxygenase and cyclooxygenase inhibitors.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Antigen-Antibody Complex; Antioxidants; Calcimycin; Catechols; Cyclooxygenase Inhibitors; Cytochalasin B; Ibuprofen; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Muramidase; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Piroxicam; Pyrazoles; Pyrazolones; Rats; Superoxides; Tetradecanoylphorbol Acetate; Thiazines; Zymosan | 1984 |
Release of leukotriene B4 from human neutrophils measured by specific radioimmunoassay.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Anti-Inflammatory Agents; Calcimycin; Cytochalasin B; Dinoprostone; Humans; Indomethacin; Kinetics; Leukotriene B4; N-Formylmethionine; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oligopeptides; Prostaglandins E; Pyrazoles; Radioimmunoassay; Thromboxane B2 | 1983 |
A rapid method for detecting inhibitors of both cyclo-oxygenase lipoxygenase metabolites of arachidonic acid.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Anti-Inflammatory Agents; Antioxidants; Arachidonic Acid; Arachidonic Acids; Ascitic Fluid; Biotransformation; Calcimycin; Catechols; Chromatography, High Pressure Liquid; Chromatography, Thin Layer; Cyclooxygenase Inhibitors; Gas Chromatography-Mass Spectrometry; Guinea Pigs; Indomethacin; Lipoxygenase Inhibitors; Male; Masoprocol; Neutrophils; Oxygenases; Propionates; Pyrazoles | 1983 |
Generation of a leukotriene-like substance from porcine vascular and other tissues.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Anti-Inflammatory Agents; Arteries; Calcimycin; Heart; Heart Ventricles; Myocardium; Organ Specificity; Pyrazoles; SRS-A; Swine | 1983 |
Actions and interactions of lipoxygenase and cyclo-oxygenase products in respiratory and vascular tissues.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bronchi; Calcimycin; Chromones; Coronary Vessels; Guinea Pigs; Humans; Lipoxygenase; Lung; Prostaglandin-Endoperoxide Synthases; Pulmonary Artery; Pyrazoles; SRS-A | 1984 |
Effect of norathyriol, isolated from Tripterospermum lanceolatum, on A23187-induced pleurisy and analgesia in mice.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Analgesia; Animals; Calcimycin; Dinoprostone; Female; Indomethacin; Kinetics; Leukocyte Count; Leukotriene B4; Mice; Neutrophils; Pleurisy; Radioimmunoassay; Xanthenes | 1994 |
Differential effects of phorbol 12-myristate 13-acetate and diacylglycerols on thromboxane A2-independent phospholipase A2 activation in collage-stimulated human platelets.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Blood Platelets; Calcimycin; Calcium; Collagen; Diglycerides; Enzyme Activation; Humans; Phospholipases A; Phospholipases A1; Phospholipases A2; Tetradecanoylphorbol Acetate; Thromboxane A2 | 1994 |
Leukotriene B4 and C4 production in isolated rat gastric mucosal cells.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Bucladesine; Calcimycin; Cell Separation; Colforsin; Diglycerides; Female; Gastric Mucosa; Histamine; In Vitro Techniques; Interleukin-1; Interleukin-2; Kinetics; Leukotriene B4; Leukotriene C4; Lipoxygenase Inhibitors; N-Formylmethionine Leucyl-Phenylalanine; Pentagastrin; Phenothiazines; Platelet Activating Factor; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1993 |