Page last updated: 2024-09-05

bw 501c and ketanserin

bw 501c has been researched along with ketanserin in 4 studies

Compound Research Comparison

Studies
(bw 501c)
Trials
(bw 501c)
Recent Studies (post-2010)
(bw 501c)
Studies
(ketanserin)
Trials
(ketanserin)
Recent Studies (post-2010) (ketanserin)
17003,094335283

Protein Interaction Comparison

ProteinTaxonomybw 501c (IC50)ketanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.015
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.015
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.265
5-hydroxytryptamine receptor 1BHomo sapiens (human)6.5
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0184
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0027
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.29
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.015
D(2) dopamine receptorRattus norvegicus (Norway rat)1.8
Synaptic vesicular amine transporterHomo sapiens (human)0.18
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.001

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19903 (75.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Leysen, JE; Schotte, A1
De Clerck, F; Janssen, PA; Tollenaere, JP; Xhonneux, B1
McLennan, PL; Taylor, DA1
Knowles, ID; Ramage, AG1

Other Studies

4 other study(ies) available for bw 501c and ketanserin

ArticleYear
Identification of 5-HT2 receptors, alpha 1-adrenoceptors and amine release sites in rat brain by autoradiography with [125I]7-amino-8-iodo-ketanserin.
    European journal of pharmacology, 1989, May-11, Volume: 172, Issue:2

    Topics: Amidines; Amines; Animals; Autoradiography; Binding, Competitive; Brain; Brain Chemistry; Female; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists; Tetrabenazine

1989
Dependence of the antagonism at human platelet 5-HT2 receptors by ketanserin on the reaction pH.
    Thrombosis research, 1985, Dec-01, Volume: 40, Issue:5

    Topics: Amidines; Blood Platelets; Butyrophenones; Cyproheptadine; Female; Humans; Hydrogen-Ion Concentration; Ketanserin; Kinetics; Male; Piperidines; Platelet Aggregation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone

1985
Antagonism by ketanserin of 5-HT-induced vasoconstriction unmasks a 5-HT-induced vasodilation.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: Amidines; Animals; Antihypertensive Agents; Blood Pressure; Hypertension; In Vitro Techniques; Ketanserin; Male; Norepinephrine; Piperidines; Rats; Serotonin; Serotonin Antagonists; Vasoconstriction; Vasodilation

1984
Evidence that activation of central 5-HT(2B) receptors causes renal sympathoexcitation in anaesthetized rats.
    British journal of pharmacology, 2000, Volume: 129, Issue:1

    Topics: Amidines; Anesthesia; Animals; Blood Pressure; Heart Rate; Indoles; Injections, Intraventricular; Ketanserin; Kidney; Male; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Stimulation, Chemical; Sulfonamides; Sympathetic Nervous System; Thiophenes

2000