Page last updated: 2024-09-03

bw 373u86 and naltrindole

bw 373u86 has been researched along with naltrindole in 14 studies

Compound Research Comparison

Studies
(bw 373u86)
Trials
(bw 373u86)
Recent Studies (post-2010)
(bw 373u86)
Studies
(naltrindole)
Trials
(naltrindole)
Recent Studies (post-2010) (naltrindole)
80048010139

Protein Interaction Comparison

ProteinTaxonomybw 373u86 (IC50)naltrindole (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0007
Delta-type opioid receptorHomo sapiens (human)0.0006

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (64.29)18.2507
2000's4 (28.57)29.6817
2010's1 (7.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bernard, D; Coop, A; MacKerell, AD1
Moerschbaecher, JM; Pakarinen, ED; Woods, JH1
Butelman, ER; Chang, KJ; DeCosta, B; Negus, SS; Winger, G; Woods, JH1
Borsodi, A; Chang, KJ; Fang, L; McNutt, RW; Porreca, F; Toth, G; Wild, KD; Yamamura, HI1
Chang, KJ; Dykstra, LA; McNutt, R; Schoenbaum, GM; Yarbrough, J1
Cook, CD; Morgan, D; Negus, SS; Picker, MJ1
Cozzolino, A; Di Chiara, G; Giagheddu, M; Marrosu, F; Puligheddu, M1
Kapusta, DR; Kenigs, VA; Sezen, SF1
Cadoni, C; Di Chiara, G; Longoni, R; Mulas, A; Spina, L1
Chang, KJ; McNutt, RW; Su, YF1
Fiore, P; Gannon, RL; Tierno, A1
Folk, JE; Isgor, C; Rice, KC; Torregrossa, MM; Watson, SJ; Woods, JH1
Jutkiewicz, EM; Ko, MC; Rice, KC; Shi, YG; Torregrossa, MM; Watson, SJ; Woods, JH; Zhang, H1
Chai, W; Ding, Q; Gao, C; Sun, M; Sun, X; Yang, L; Yao, L; Yu, D; Zhao, X1

Other Studies

14 other study(ies) available for bw 373u86 and naltrindole

ArticleYear
Quantitative conformationally sampled pharmacophore for delta opioid ligands: reevaluation of hydrophobic moieties essential for biological activity.
    Journal of medicinal chemistry, 2007, Apr-19, Volume: 50, Issue:8

    Topics: Animals; Cell Line, Tumor; Enkephalin, Leucine; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Molecular Conformation; Phenylalanine; Quantitative Structure-Activity Relationship; Rats; Receptors, Opioid, delta

2007
Repeated acquisition of behavioral chains in squirrel monkeys: comparisons of a mu, kappa and delta opioid agonist.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzamides; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Morphine; Naltrexone; Piperazines; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri

1995
Behavioral effects of the systemically active delta opioid agonist BW373U86 in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Benzamides; Female; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Piperazines; Receptors, Opioid, delta; Respiration

1994
Binding of BW 373U86, a non-peptidic delta opioid receptor agonist, is not regulated by guanine nucleotides and sodium.
    European journal of pharmacology, 1993, Aug-15, Volume: 246, Issue:3

    Topics: Animals; Benzamides; Binding, Competitive; Brain; Guanine Nucleotides; Male; Membranes; Mice; Mice, Inbred ICR; Naltrexone; Narcotic Antagonists; Piperazines; Radioligand Assay; Receptors, Opioid, delta; Sodium; Vas Deferens

1993
A novel delta opioid agonist, BW373U86, in squirrel monkeys responding under a schedule of shock titration.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Amino Acid Sequence; Animals; Behavior, Animal; Benzamides; Drug Interactions; Drug Tolerance; Electroshock; Male; Methadone; Molecular Sequence Data; Naltrexone; Narcotic Antagonists; Nociceptors; Piperazines; Receptors, Opioid, delta; Receptors, Opioid, mu; Saimiri

1993
Effects of the delta opioid against BW373U86 in pigeons trained to discriminate fentanyl, bremazocine and water in a three-choice drug discrimination procedure.
    Psychopharmacology, 1996, Volume: 126, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Columbidae; Discrimination, Psychological; Female; Fentanyl; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Piperazines; Receptors, Opioid, delta

1996
Hippocampal theta activity after systemic administration of a non-peptide delta-opioid agonist in freely-moving rats: relationship to D1 dopamine receptors.
    Brain research, 1997, Nov-21, Volume: 776, Issue:1-2

    Topics: Animals; Benzamides; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Hippocampus; Locomotion; Naltrexone; Narcotic Antagonists; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Opioid, delta; Theta Rhythm

1997
Renal excretory responses produced by the delta opioid agonist, BW373U86, in conscious rats.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzamides; Denervation; Infusions, Intravenous; Kidney; Male; Naltrexone; Oligopeptides; Opioid Peptides; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta

1998
Dopamine-dependent behavioural stimulation by non-peptide delta opioids BW373U86 and SNC 80: 2. Place-preference and brain microdialysis studies in rats.
    Behavioural pharmacology, 1998, Volume: 9, Issue:1

    Topics: Animals; Behavior, Animal; Benzamides; Benzazepines; Brain Chemistry; Caudate Nucleus; Conditioning, Operant; Dopamine; Dopamine Antagonists; Extracellular Space; Male; Microdialysis; Naltrexone; Narcotic Antagonists; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley

1998
Delta-opioid ligands reverse alfentanil-induced respiratory depression but not antinociception.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:3

    Topics: Alfentanil; Analgesics, Opioid; Animals; Benzamides; Hypercapnia; Ligands; Male; Naltrexone; Narcotic Antagonists; Narcotics; Oligopeptides; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Respiration; Respiratory Insufficiency; Somatostatin

1998
Delta opioid inhibition of light-induced phase advances in hamster circadian activity rhythms.
    Brain research, 2002, May-24, Volume: 937, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzamides; Biological Clocks; Circadian Rhythm; Cricetinae; Enkephalins; Light; Male; Mesocricetus; Morphine; Motor Activity; Naltrexone; Narcotic Antagonists; Nerve Tissue Proteins; Opioid Peptides; Piperazines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Suprachiasmatic Nucleus

2002
The delta-opioid receptor agonist (+)BW373U86 regulates BDNF mRNA expression in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:4

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Antidepressive Agents; Behavior, Animal; Benzamides; Brain; Brain-Derived Neurotrophic Factor; Bupropion; Desipramine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Drug Tolerance; Gene Expression Regulation; Immobilization; In Situ Hybridization; Male; Midazolam; Naltrexone; Narcotic Antagonists; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, trkB; Receptors, Opioid, delta; RNA, Messenger; Swimming; Time Factors; Up-Regulation

2004
Endogenous opioids upregulate brain-derived neurotrophic factor mRNA through delta- and micro-opioid receptors independent of antidepressant-like effects.
    The European journal of neuroscience, 2006, Volume: 23, Issue:4

    Topics: Analgesics, Opioid; Analysis of Variance; Animals; Autoradiography; Behavior, Animal; Benzamides; Brain-Derived Neurotrophic Factor; Dose-Response Relationship, Drug; Drug Interactions; Freezing Reaction, Cataleptic; In Situ Hybridization; Injections, Intraventricular; Male; Naltrexone; Narcotics; Opioid Peptides; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Swimming; Up-Regulation

2006
Delta opioid receptor agonist BW373U86 attenuates post-resuscitation brain injury in a rat model of asphyxial cardiac arrest.
    Resuscitation, 2014, Volume: 85, Issue:2

    Topics: Animals; Asphyxia; Benzamides; Blotting, Western; Brain Damage, Chronic; Cardiopulmonary Resuscitation; CREB-Binding Protein; Disease Models, Animal; Heart Arrest; Immunoenzyme Techniques; Male; Naltrexone; Neuroprotective Agents; Piperazines; Rats, Sprague-Dawley

2014