Page last updated: 2024-09-03

bw 373u86 and enkephalin, leucine-2-alanine

bw 373u86 has been researched along with enkephalin, leucine-2-alanine in 2 studies

Compound Research Comparison

Studies
(bw 373u86)
Trials
(bw 373u86)
Recent Studies (post-2010)
(bw 373u86)
Studies
(enkephalin, leucine-2-alanine)
Trials
(enkephalin, leucine-2-alanine)
Recent Studies (post-2010) (enkephalin, leucine-2-alanine)
80041,5812374

Protein Interaction Comparison

ProteinTaxonomybw 373u86 (IC50)enkephalin, leucine-2-alanine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0915
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0017
Kappa-type opioid receptorMus musculus (house mouse)0.009
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0419
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)1.4691
Mu-type opioid receptorMus musculus (house mouse)0.009

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Befort, K; Kieffer, BL; Tabbara, L1
Becketts, K; Bilsky, EJ; Calderon, SN; Davis, P; Flippen-Anderson, JL; Horvath, R; Kayakiri, H; Porreca, F; Rice, KC; Rothman, RB; Smith, LE; Xu, H1

Other Studies

2 other study(ies) available for bw 373u86 and enkephalin, leucine-2-alanine

ArticleYear
[35S]GTP gamma S binding: a tool to evaluate functional activity of a cloned opioid receptor transiently expressed in COS cells.
    Neurochemical research, 1996, Volume: 21, Issue:11

    Topics: Animals; Benzamides; CHO Cells; Cloning, Molecular; COS Cells; Cricetinae; Enkephalin, Leucine-2-Alanine; Guanosine 5'-O-(3-Thiotriphosphate); Mice; Naloxone; Piperazines; Receptors, Opioid, delta; Recombinant Proteins; Signal Transduction; Sulfur Radioisotopes; Transfection

1996
Probes for narcotic receptor mediated phenomena. 23. Synthesis, opioid receptor binding, and bioassay of the highly selective delta agonist (+)-4-[(alpha R)-alpha-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]- N,N-diethylbenzamide (SNC 80)
    Journal of medicinal chemistry, 1997, Feb-28, Volume: 40, Issue:5

    Topics: Animals; Benzamides; Binding, Competitive; Brain; Crystallography, X-Ray; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; Magnetic Resonance Spectroscopy; Male; Mice; Molecular Conformation; Molecular Structure; Muscle Contraction; Piperazines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Stereoisomerism; Vas Deferens

1997