Page last updated: 2024-09-03

bw 245c and iloprost

bw 245c has been researched along with iloprost in 10 studies

Compound Research Comparison

Studies
(bw 245c)
Trials
(bw 245c)
Recent Studies (post-2010)
(bw 245c)
Studies
(iloprost)
Trials
(iloprost)
Recent Studies (post-2010) (iloprost)
963102,150271462

Protein Interaction Comparison

ProteinTaxonomybw 245c (IC50)iloprost (IC50)
Prostacyclin receptorHomo sapiens (human)0.0112

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's2 (20.00)18.2507
2000's6 (60.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Collins, BA; Kelly, MG; Robertson, AD; Trist, DG; Wood, J1
Brink, C; de Montpreville, V; Gascard, JP; Labat, C; Norel, X; Walch, L1
Brink, C; Dulmet, E; Gascard, JP; Labat, C; Norel, X; Walch, L1
Cao, J; Kitazawa, T; Shayibuzhati, M; Tajima, T; Taneike, T1
Heinemann, A; Holzer, P; Peskar, BA; Shahbazian, A1
Sharif, NA; Xu, SX1
Jones, RL; Kan, KK; Ngan, MP; Rudd, JA1
Kinsella, BT; O'Meara, SJ1
Bing, N; Cox, RF; Gauthier, J; Jensen, D; Johnson, EN; Kostura, M; Murray, DL; Sorensen, SD; Vanderwall, D; Wang, P; Xu, Z1
Devillier, P; Grassin-Delyle, S; Mechiche, H; Nazeyrollas, P; Robinet, A1

Other Studies

10 other study(ies) available for bw 245c and iloprost

ArticleYear
The antagonism by BW A868C of PGD2 and BW245C activation of human platelet adenylate cyclase.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Adenylyl Cyclases; Blood Platelets; Enzyme Activation; Epoprostenol; Humans; Hydantoins; Iloprost; In Vitro Techniques; Platelet Aggregation; Prostaglandin D2; Receptors, Prostaglandin

1989
Prostanoid receptors involved in the relaxation of human pulmonary vessels.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Female; Humans; Hydantoins; Iloprost; In Vitro Techniques; Male; Middle Aged; Norepinephrine; Prostaglandin D2; Prostaglandins E; Pulmonary Artery; Pulmonary Veins; Receptors, Prostaglandin; Vasodilation

1999
Prostanoid receptors involved in the relaxation of human bronchial preparations.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Aged; Bronchi; Female; Humans; Hydantoins; Iloprost; In Vitro Techniques; Male; Middle Aged; Muscle Relaxation; Prostaglandin D2; Prostaglandins E; Receptors, Prostaglandin

1999
In vitro pharmacological characterization of the prostanoid receptor population in the non-pregnant porcine myometrium.
    European journal of pharmacology, 2002, May-03, Volume: 442, Issue:1-2

    Topics: Animals; Cloprostenol; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Epoprostenol; Female; Hydantoins; Iloprost; In Vitro Techniques; Muscle Contraction; Myometrium; Prostaglandin D2; Receptors, Prostaglandin; Swine

2002
Differential peristaltic motor effects of prostanoid (DP, EP, IP, TP) and leukotriene receptor agonists in the guinea-pig isolated small intestine.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alprostadil; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; Iloprost; In Vitro Techniques; Intestine, Small; Leukotriene Antagonists; Leukotriene D4; Male; Oxazepines; Peristalsis; Prostaglandin D2; Prostaglandins A; Receptors, Leukotriene; Receptors, Prostaglandin; Xanthenes; Xanthones; Yohimbine

2002
Pharmacological characterization and identification of EP3 prostanoid receptor binding sites in hamster uterus homogenates.
    The Journal of pharmacy and pharmacology, 2004, Volume: 56, Issue:2

    Topics: Animals; Binding Sites; Biphenyl Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cloprostenol; Cricetinae; Dinoprost; Dinoprostone; Enprostil; Epoprostenol; Fatty Acids, Unsaturated; Female; Hydantoins; Hydrazines; Iloprost; Latanoprost; Misoprostol; Prostaglandins; Prostaglandins E, Synthetic; Prostaglandins F, Synthetic; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP3 Subtype; Tritium; Uterus

2004
Excitatory action of prostanoids on the ferret isolated vagus nerve preparation.
    European journal of pharmacology, 2004, Apr-26, Volume: 491, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Biguanides; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Electrophysiology; Epoprostenol; Ferrets; Hydantoins; Iloprost; In Vitro Techniques; Male; Prostaglandins; Prostaglandins F, Synthetic; Serotonin; Vagus Nerve

2004
Effect of the statin atorvastatin on intracellular signalling by the prostacyclin receptor in vitro and in vivo.
    British journal of pharmacology, 2004, Volume: 143, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenylyl Cyclases; Animals; Atorvastatin; Blood Platelets; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cell Line; Cell Line, Tumor; Cholesterol; Clinical Trials as Topic; Cyclic AMP; Drug Evaluation, Preclinical; Fatty Acids, Unsaturated; Female; Heptanoic Acids; Humans; Hydantoins; Hydrazines; Iloprost; Ireland; Lipids; Male; Mice; Middle Aged; Propanolamines; Protein Prenylation; Pyrroles; Radioligand Assay; Receptor Cross-Talk; Receptors, Epoprostenol; Receptors, Immunologic; Receptors, Prostaglandin; Signal Transduction; Tritium

2004
Functional antagonism of IL-1alpha induced gene expression profiles define the cAMP/PKA pathway as a unique regulator of IL-1alpha signaling networks.
    Journal of receptor and signal transduction research, 2009, Volume: 29, Issue:5

    Topics: Alprostadil; Anti-Ulcer Agents; Calcium; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Fibroblasts; Gene Expression Profiling; Humans; Hydantoins; I-kappa B Kinase; Iloprost; Interleukin-1alpha; JNK Mitogen-Activated Protein Kinases; Lung; MAP Kinase Kinase Kinases; Misoprostol; Oligonucleotide Array Sequence Analysis; p38 Mitogen-Activated Protein Kinases; Platelet Aggregation Inhibitors; Prostaglandins E, Synthetic; Receptors, G-Protein-Coupled; Receptors, Prostaglandin; Signal Transduction

2009
Prostanoid receptors involved in regulation of the beating rate of neonatal rat cardiomyocytes.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Animals, Newborn; Blotting, Western; Cells, Cultured; Cloprostenol; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Epoprostenol; Hydantoins; Iloprost; Latanoprost; Myocytes, Cardiac; Prostaglandin D2; Prostaglandins F, Synthetic; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Thromboxane

2012